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Title:
AMIDINOPHENYLPYRUVIC ACID DERIVATIVE
Document Type and Number:
WIPO Patent Application WO/2001/042199
Kind Code:
A1
Abstract:
An amidinophenylpyruvic acid derivative represented by the following formula, its analogs and pharmaceutically acceptable salts thereof which have an excellent effect of inhibiting activated blood coagulation factor VII.

Inventors:
SUGIKI MASAYUKI (JP)
SAGI KAZUYUKI (JP)
FUJITA KOHICHI (JP)
KAYAHARA TAKASHI (JP)
TAKEHANA SHUNJI (JP)
SAKURAI KUNIYA (JP)
TASHIRO KAZUMI (JP)
Application Number:
PCT/JP2000/008569
Publication Date:
June 14, 2001
Filing Date:
December 04, 2000
Export Citation:
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Assignee:
AJINOMOTO KK (JP)
SUGIKI MASAYUKI (JP)
SAGI KAZUYUKI (JP)
FUJITA KOHICHI (JP)
KAYAHARA TAKASHI (JP)
TAKEHANA SHUNJI (JP)
SAKURAI KUNIYA (JP)
TASHIRO KAZUMI (JP)
International Classes:
A61P7/02; A61P9/10; A61P43/00; C07C257/18; C07C279/14; C07C279/18; C07C279/22; C07D213/56; C07D213/73; C07D215/48; C07D233/60; C07D235/08; C07D235/30; C07D239/84; C07D277/64; C07D277/82; C07D307/79; C07D333/24; C07D333/38; C07D401/04; C07D521/00; (IPC1-7): C07C257/18; C07C279/14; C07C279/22; C07D215/48; C07D235/30; C07D235/08; C07D333/40; C07D333/24; C07D215/58; C07D213/74; C07D401/04; C07D277/82; C07D277/64; C07D233/60; C07D239/84; A61K31/166; A61K31/197; A61K31/47; A61K31/4184; A61K31/381; A61K31/44; A61K31/4453; A61K31/4545; A61K31/428; A61K31/4164; A61K31/517; A61P43/00; A61P7/02; A61P9/10
Domestic Patent References:
WO1998031661A11998-07-23
WO1999064392A11999-12-16
Other References:
See also references of EP 1236712A4
Attorney, Agent or Firm:
Nakamura, Minoru (Shin-Tokyo Bldg 3-1 Marunouchi 3-Chome Chiyoda-Ku, Tokyo, JP)
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