Title:
ASCORBIC ACID DERIVATIVE AND GLYCOSIDE PRODUCTION METHOD USING SAME
Document Type and Number:
WIPO Patent Application WO/2016/063896
Kind Code:
A1
Abstract:
Provided is an ascorbic acid derivative that can be used to obtain a glycoside of which ascorbic acid is the aglycone. The abovementioned derivative is the compound represented by formula (A) (i.e., 2,3,6-tri-O-acyl-ascorbic acid). (In the formula, R1 indicates an acyl group.)
Inventors:
SHIMAMOTO KEIKO (JP)
MATSUOKA TATSUO (JP)
MATSUOKA TATSUO (JP)
Application Number:
PCT/JP2015/079662
Publication Date:
April 28, 2016
Filing Date:
October 21, 2015
Export Citation:
Assignee:
SUNTORY HOLDINGS LTD (JP)
International Classes:
C07D307/62; A23L33/15; A61K8/60; A61K31/7048; A61Q5/02; A61Q5/12; A61Q19/00; A61Q19/10; C07H17/04
Domestic Patent References:
WO2011030816A1 | 2011-03-17 | |||
WO2014050894A1 | 2014-04-03 | |||
WO2014013744A1 | 2014-01-23 | |||
WO2014013743A1 | 2014-01-23 | |||
WO2005000319A1 | 2005-01-06 |
Foreign References:
JPS435885B1 | ||||
JPS439216B1 | ||||
JPS5030864A | 1975-03-27 | |||
JPS601175A | 1985-01-07 | |||
JPS6023307A | 1985-02-05 | |||
JPS6185308A | 1986-04-30 | |||
JPS6270366A | 1987-03-31 | |||
JPS6270367A | 1987-03-31 | |||
JPS6281307A | 1987-04-14 | |||
JPS62164609A | 1987-07-21 | |||
JPS6485907A | 1989-03-30 | |||
JPH11217380A | 1999-08-10 | |||
JPS63316743A | 1988-12-26 | |||
JP2012527433A | 2012-11-08 | |||
CN102250168A | 2011-11-23 | |||
CN101671376A | 2010-03-17 | |||
US20080220140A1 | 2008-09-11 | |||
JPH06263790A | 1994-09-20 | |||
JP2005518401A | 2005-06-23 |
Other References:
HIROYOSHI TANAKA ET AL.: "Pharmaceutucal Studies on Ascorbic Acid Derivatives. I", JOURNAL OF THE PHARMACEUTICAL SOCIETY OF JAPAN, vol. 86, no. 5, 1966, pages 376 - 383, XP002236531
TAKAHASHI MAREYUKI ET AL.: "Oxidation of lipids. XIV. Inhibition of oxidation of methyl linoleate by fatty acid esters of L-ascorbic acid", BULLETIN OF THE CHEMICAL SOCIETY OF JAPAN, vol. 59, no. 10, 1986, pages 3179 - 3183, XP055275404
YOSHIKO TOYODA-ONO ET AL: "2-O-(β-d-Glucopyranosyl)ascorbic Acid, a Novel Ascorbic Acid Analogue Isolated from Lycium Fruit", JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, vol. 52, no. 7, 2004, pages 2092 - 2096, XP055275408
GREENE, THEODORA W. ET AL: "Greene's PROTECTIVE GROUPS IN ORGANIC SYNTHESIS", article THEODORA W. GREENE: "THE ROLE OF PROTECTIVE GROUPS IN ORGANIC SYNTHESIS", pages: 10 - 14, XP055275414
TAKAHASHI MAREYUKI ET AL.: "Oxidation of lipids. XIV. Inhibition of oxidation of methyl linoleate by fatty acid esters of L-ascorbic acid", BULLETIN OF THE CHEMICAL SOCIETY OF JAPAN, vol. 59, no. 10, 1986, pages 3179 - 3183, XP055275404
YOSHIKO TOYODA-ONO ET AL: "2-O-(β-d-Glucopyranosyl)ascorbic Acid, a Novel Ascorbic Acid Analogue Isolated from Lycium Fruit", JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, vol. 52, no. 7, 2004, pages 2092 - 2096, XP055275408
GREENE, THEODORA W. ET AL: "Greene's PROTECTIVE GROUPS IN ORGANIC SYNTHESIS", article THEODORA W. GREENE: "THE ROLE OF PROTECTIVE GROUPS IN ORGANIC SYNTHESIS", pages: 10 - 14, XP055275414
Attorney, Agent or Firm:
IWATANI, Ryo (JP)
Tatsu Iwatani (JP)
Tatsu Iwatani (JP)
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