Title:
BENZOTHIAZOLE AND QUINOLINE DERIVATIVES AND THEIR USE
Document Type and Number:
WIPO Patent Application WO/2022/063153
Kind Code:
A1
Abstract:
Provided are compounds of Formula (I) or (II) and related compositions and methods for their use as inhibitors of alpha-kinase 1 (ALPK1).
Inventors:
LIU DANYANG (CN)
XU CONG (CN)
MELVIN LAWRENCE S (CN)
WEI XIONG (CN)
LI TONGRUEI RAYMOND (CN)
FAN JIEQING (CN)
PAN YANFANG (CN)
DANG HUAIXIN (CN)
LICHENSTEIN HENRI (CN)
XU TIAN (CN)
XU CONG (CN)
MELVIN LAWRENCE S (CN)
WEI XIONG (CN)
LI TONGRUEI RAYMOND (CN)
FAN JIEQING (CN)
PAN YANFANG (CN)
DANG HUAIXIN (CN)
LICHENSTEIN HENRI (CN)
XU TIAN (CN)
Application Number:
PCT/CN2021/119802
Publication Date:
March 31, 2022
Filing Date:
September 23, 2021
Export Citation:
Assignee:
SHANGHAI YAO YUAN BIOTECHNOLOGY CO LTD (CN)
International Classes:
C07D277/82; A61K31/428; A61K31/47; A61P25/00; A61P35/00; A61P37/00; C07D215/38; C07D217/06; C07D401/12; C07D417/02
Domestic Patent References:
WO2005037845A1 | 2005-04-28 | |||
WO2017223514A1 | 2017-12-28 |
Foreign References:
CN101830855A | 2010-09-15 | |||
CN86102102A | 1987-01-07 | |||
CN103006645A | 2013-04-03 | |||
KR20160124373A | 2016-10-27 |
Other References:
CORBO FILOMENA, CAROCCI ALESSIA, ARMENISE DOMENICO, DE LAURENTIS NICOLINO, LAGHEZZA ANTONIO, LOIODICE FULVIO, ANCONA PATRIZIA, MUR: "Antiproliferative Activity Evaluation of a Series of N -1,3-Benzothiazol-2-ylbenzamides as Novel Apoptosis Inducers", JOURNAL OF CHEMISTRY, vol. 2016, 1 January 2016 (2016-01-01), US , pages 1 - 5, XP055913926, ISSN: 2090-9063, DOI: 10.1155/2016/4267564
Attorney, Agent or Firm:
WU, FENG & ZHANG (CN)
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