Title:
CRYSTAL OF 1,3,5-TRIAZINE DERIVATIVE OR SOLVATE THEREOF AND METHOD FOR PRODUCING SAME
Document Type and Number:
WIPO Patent Application WO/2021/054421
Kind Code:
A1
Abstract:
Provided are: a crystal of a 1,3,5-triazine derivative or a solvate thereof; and a method for producing the same. The present invention pertains to a crystal of a compound represented by formula (I) or a solvate thereof, and a pharmaceutical composition containing the same. The present invention also pertains to a method for producing a crystal of a compound represented by formula (I) or a solvate thereof.
Inventors:
KAI HIROYUKI (JP)
MAKI TOSHIKATSU (JP)
ODA SHINICHI (JP)
BAN KAZUNORI (JP)
TSUBONE KOICHI (JP)
HOSOYA MASAHIRO (JP)
MURAKAMI YUKI (JP)
MAKI TOSHIKATSU (JP)
ODA SHINICHI (JP)
BAN KAZUNORI (JP)
TSUBONE KOICHI (JP)
HOSOYA MASAHIRO (JP)
MURAKAMI YUKI (JP)
Application Number:
PCT/JP2020/035378
Publication Date:
March 25, 2021
Filing Date:
September 18, 2020
Export Citation:
Assignee:
SHIONOGI & CO (JP)
International Classes:
C07D401/12; A61K31/53; A61P9/12; A61P11/00; A61P13/02; A61P25/04; A61P43/00; C07C227/08; C07C227/18; C07C229/08; C07C229/14
Domestic Patent References:
| WO2014200078A1 | 2014-12-18 | |||
| WO2020071530A1 | 2020-04-09 | |||
| WO2002094767A2 | 2002-11-28 | |||
| WO2006012639A2 | 2006-02-02 | |||
| WO2010149578A2 | 2010-12-29 | |||
| WO2015027212A1 | 2015-02-26 | |||
| WO2017058645A1 | 2017-04-06 | |||
| WO2010092966A1 | 2010-08-19 | |||
| WO2012020749A1 | 2012-02-16 | |||
| WO2013089212A1 | 2013-06-20 | |||
| WO2014200078A1 | 2014-12-18 | |||
| WO2020071530A1 | 2020-04-09 |
Other References:
HIRAYAMA NORIAKI: "Handbook of organic compounds crystallization - principles and know-how", 25 July 2008, XX , JP , ISBN: 978-4-621-07991-1, article HIRAYAMA NORIAKI: "Handbook of organic compounds crystallization - principles and know-how", pages: 57 - 84, XP008183996
NORIYUKI TAKATA: "Soyaku Dankai ni Okeru Gen'yaku Form Screening to Sentaku - API form screening and selection in drug discovery stage", PHARM STAGE, vol. 6, no. 10, 1 January 2007 (2007-01-01), JP , pages 20 - 25, XP008145548, ISSN: 1346-3918
SHUSTOV, G. V. ET AL.: "3-Methylazetidin-2-one and Its Precursors: Optical Resolution and Absolute Configurations", TETRAHEDRON : ASYMMETRY, vol. 7, no. 3, 1996, pages 699 - 708, XP004188762, DOI: 10.1016/0957-4166(96)00065-1
NEUROSCIENTIST, vol. 11, 2005, pages 345 - 356
J. PHYSIOL., vol. 567, no. 2, 2005, pages 621 - 639
EXPERT OPIN.THER.PATENS, vol. 16, no. 8, 2006, pages 1113 - 1127
J. PHYSIOL., vol. 553, no. 3, 2003, pages 683 - 694
PFLUNGERS ARCH EUR J PHYSIOL, vol. 452, 2006, pages 513 - 537
PNAS, vol. 99, no. 26, 2002, pages 17179 - 17184
BROUNS ET AL., AM J RESPIR CELL MOL BIOL, vol. 23, 2000, pages 52 - 61
BASOGLU ET AL., CHEST, vol. 128, no. 4, 2005, pages 1905 - 9
ADRIAENSEN ET AL., THE ANATOMICAL RECORD, vol. 270A, 2003, pages 25 - 40
LANCET, vol. 385, 2015, pages 1198 - 205
NAT MED, vol. 22, 2016, pages 1151 - 1159
AM J PHYSIOL GASTROINTEST LIVER PHYSIOL, vol. 308, 2015, pages 710 - 719
PLOS ONE, vol. 12, no. 9, 2017
INTERNATIONAL JOURNAL OF NANOMEDICINE, vol. 12, 2017, pages 8171 - 8183
TETRAHEDRON ASYMMETRY, vol. 7, no. 3, 1996, pages 699 - 708
TOSHIO SAKURAI: "X-sen Kozo Kaiseki no Tebiki (Guide to X-ray Structural Analysis", 1983, SHOKABO CO., LTD.
STOUTJENSEN: "X-Ray Structure Determination: A Practical Guide", 1968, MACMILLAN CO.
NORIYUKI TAKATA: "Soyaku Dankai ni Okeru Gen'yaku Form Screening to Sentaku - API form screening and selection in drug discovery stage", PHARM STAGE, vol. 6, no. 10, 1 January 2007 (2007-01-01), JP , pages 20 - 25, XP008145548, ISSN: 1346-3918
SHUSTOV, G. V. ET AL.: "3-Methylazetidin-2-one and Its Precursors: Optical Resolution and Absolute Configurations", TETRAHEDRON : ASYMMETRY, vol. 7, no. 3, 1996, pages 699 - 708, XP004188762, DOI: 10.1016/0957-4166(96)00065-1
NEUROSCIENTIST, vol. 11, 2005, pages 345 - 356
J. PHYSIOL., vol. 567, no. 2, 2005, pages 621 - 639
EXPERT OPIN.THER.PATENS, vol. 16, no. 8, 2006, pages 1113 - 1127
J. PHYSIOL., vol. 553, no. 3, 2003, pages 683 - 694
PFLUNGERS ARCH EUR J PHYSIOL, vol. 452, 2006, pages 513 - 537
PNAS, vol. 99, no. 26, 2002, pages 17179 - 17184
BROUNS ET AL., AM J RESPIR CELL MOL BIOL, vol. 23, 2000, pages 52 - 61
BASOGLU ET AL., CHEST, vol. 128, no. 4, 2005, pages 1905 - 9
ADRIAENSEN ET AL., THE ANATOMICAL RECORD, vol. 270A, 2003, pages 25 - 40
LANCET, vol. 385, 2015, pages 1198 - 205
NAT MED, vol. 22, 2016, pages 1151 - 1159
AM J PHYSIOL GASTROINTEST LIVER PHYSIOL, vol. 308, 2015, pages 710 - 719
PLOS ONE, vol. 12, no. 9, 2017
INTERNATIONAL JOURNAL OF NANOMEDICINE, vol. 12, 2017, pages 8171 - 8183
TETRAHEDRON ASYMMETRY, vol. 7, no. 3, 1996, pages 699 - 708
TOSHIO SAKURAI: "X-sen Kozo Kaiseki no Tebiki (Guide to X-ray Structural Analysis", 1983, SHOKABO CO., LTD.
STOUTJENSEN: "X-Ray Structure Determination: A Practical Guide", 1968, MACMILLAN CO.
Attorney, Agent or Firm:
SUGITA Ken-ichi et al. (JP)
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