Title:
FLUORINATED PYRIMIDINE COMPOUND AND METHOD FOR MANUFACTURING SAME
Document Type and Number:
WIPO Patent Application WO/2021/085550
Kind Code:
A1
Abstract:
A fluorinated pyrimidine compound represented by general formula (1), (2), or (3). (In general formulas (1)-(3): R represents a C1-12 hydrocarbon group; X and Y each independently represent a hydrogen atom, a halogen atom, a C1-10 hydrocarbon group, -CnF2n+1, a nitro group, a boric acid group, -OA1, -SOmA1, -NA1A2, -COOA1, or -CONA1A2; Z represents CW or N; W represents a hydrogen atom, a halogen atom, a C1-10 hydrocarbon group, -CnF2n+1, a nitro group, a boric acid group, -OA1, -SOmA1, -NA1A2, -COOA1, or -CONA1A2; n is an integer from 1 to 10; m is an integer from 0 to 3; and A1 and A2 each independently represent a hydrogen atom or a C1-10 hydrocarbon group.)
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Inventors:
SEINO JUNYA (JP)
AOTSU RIE (JP)
KOKIN KEISUKE (JP)
AOTSU RIE (JP)
KOKIN KEISUKE (JP)
Application Number:
PCT/JP2020/040682
Publication Date:
May 06, 2021
Filing Date:
October 29, 2020
Export Citation:
Assignee:
UNIMATEC CO LTD (JP)
International Classes:
C07D409/04; A01N43/54; A01P3/00; A61K31/506; A61P9/12; A61P25/00; A61P25/04; A61P25/24; A61P31/04; A61P31/06; A61P31/12; A61P31/16; A61P35/00; C07D417/04
Domestic Patent References:
| WO2020116926A1 | 2020-06-11 | |||
| WO2011019405A1 | 2011-02-17 | |||
| WO2013086131A1 | 2013-06-13 | |||
| WO2009129905A1 | 2009-10-29 | |||
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Other References:
YOSHIO INOUYE, YOICHI HIGUCHI: "A facile one-pot preparation of 2-methyl-and 2-phenyl-4- fluoro-5-trifluoromethyl-6-methoxypyrimidine from methyl 2-hydryl-2-(-methyl)--propyl ether", JOURNAL OF FLUORINE CHEMISTRY, ELSEVIER, NL, vol. 27, no. 2, 1 February 1985 (1985-02-01), NL , pages 231 - 236, XP055717031, ISSN: 0022-1139, DOI: 10.1016/S0022-1139(00)84991-X
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ACS CATALYSIS, vol. 8, 2018, pages 2839 - 2843
ANGEWANDTE CHEMIE INTERNATIONAL EDITION, vol. 57, 2018, pages 6926 - 6929
DAS SIVA PRASAD; BORUAH JEENA JYOTI; CHETRY HIRAN; ISLAM NASHREEN S.: "Selective oxidation of organic sulfides by mononuclear and dinuclear peroxotungsten(VI) complexes", TETRAHEDRON LETTERS, vol. 53, no. 9, 1 January 1900 (1900-01-01), Amsterdam , NL , pages 1163 - 1168, XP028887804, ISSN: 0040-4039, DOI: 10.1016/j.tetlet.2011.12.105
JEYAKUMAR, K. ; CHAKRAVARTHY, R.D. ; CHAND, D.K.: "Simple and efficient method for the oxidation of sulfides to sulfones using hydrogen peroxide and a Mo(VI) based catalyst", CATALYSIS COMMUNICATIONS, vol. 10, no. 14, 25 August 2009 (2009-08-25), AMSTERDAM, NL , pages 1948 - 1951, XP026470090, ISSN: 1566-7367, DOI: 10.1016/j.catcom.2009.07.009
DAS SIVA PRASAD; BORUAH JEENA JYOTI; CHETRY HIRAN; ISLAM NASHREEN S.: "Selective oxidation of organic sulfides by mononuclear and dinuclear peroxotungsten(VI) complexes", TETRAHEDRON LETTERS, vol. 53, no. 9, 1 January 1900 (1900-01-01), Amsterdam , NL , pages 1163 - 1168, XP028887804, ISSN: 0040-4039, DOI: 10.1016/j.tetlet.2011.12.105
JEYAKUMAR, K. ; CHAKRAVARTHY, R.D. ; CHAND, D.K.: "Simple and efficient method for the oxidation of sulfides to sulfones using hydrogen peroxide and a Mo(VI) based catalyst", CATALYSIS COMMUNICATIONS, vol. 10, no. 14, 25 August 2009 (2009-08-25), AMSTERDAM, NL , pages 1948 - 1951, XP026470090, ISSN: 1566-7367, DOI: 10.1016/j.catcom.2009.07.009
TETRAHEDRON, vol. 72, 2016, pages 3250 - 3255
ACS CATALYSIS, vol. 8, 2018, pages 2839 - 2843
ANGEWANDTE CHEMIE INTERNATIONAL EDITION, vol. 57, 2018, pages 6926 - 6929
DAS SIVA PRASAD; BORUAH JEENA JYOTI; CHETRY HIRAN; ISLAM NASHREEN S.: "Selective oxidation of organic sulfides by mononuclear and dinuclear peroxotungsten(VI) complexes", TETRAHEDRON LETTERS, vol. 53, no. 9, 1 January 1900 (1900-01-01), Amsterdam , NL , pages 1163 - 1168, XP028887804, ISSN: 0040-4039, DOI: 10.1016/j.tetlet.2011.12.105
JEYAKUMAR, K. ; CHAKRAVARTHY, R.D. ; CHAND, D.K.: "Simple and efficient method for the oxidation of sulfides to sulfones using hydrogen peroxide and a Mo(VI) based catalyst", CATALYSIS COMMUNICATIONS, vol. 10, no. 14, 25 August 2009 (2009-08-25), AMSTERDAM, NL , pages 1948 - 1951, XP026470090, ISSN: 1566-7367, DOI: 10.1016/j.catcom.2009.07.009
DAS SIVA PRASAD; BORUAH JEENA JYOTI; CHETRY HIRAN; ISLAM NASHREEN S.: "Selective oxidation of organic sulfides by mononuclear and dinuclear peroxotungsten(VI) complexes", TETRAHEDRON LETTERS, vol. 53, no. 9, 1 January 1900 (1900-01-01), Amsterdam , NL , pages 1163 - 1168, XP028887804, ISSN: 0040-4039, DOI: 10.1016/j.tetlet.2011.12.105
JEYAKUMAR, K. ; CHAKRAVARTHY, R.D. ; CHAND, D.K.: "Simple and efficient method for the oxidation of sulfides to sulfones using hydrogen peroxide and a Mo(VI) based catalyst", CATALYSIS COMMUNICATIONS, vol. 10, no. 14, 25 August 2009 (2009-08-25), AMSTERDAM, NL , pages 1948 - 1951, XP026470090, ISSN: 1566-7367, DOI: 10.1016/j.catcom.2009.07.009
Attorney, Agent or Firm:
EINSEL Felix-Reinhard et al. (JP)
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