Title:
FLUORINATION OF ORGANIC COMPOUNDS
Document Type and Number:
WIPO Patent Application WO/2010/059943
Kind Code:
A3
Abstract:
Methods for fluorinating organic compounds are described herein.
Inventors:
RITTER TOBIAS (US)
FURUYA TAKERU (US)
TANG PINGPING (US)
FURUYA TAKERU (US)
TANG PINGPING (US)
Application Number:
PCT/US2009/065339
Publication Date:
September 10, 2010
Filing Date:
November 20, 2009
Export Citation:
Assignee:
HARVARD COLLEGE (US)
RITTER TOBIAS (US)
FURUYA TAKERU (US)
TANG PINGPING (US)
RITTER TOBIAS (US)
FURUYA TAKERU (US)
TANG PINGPING (US)
International Classes:
C07C17/093; A61K31/566; C07B39/00
Other References:
MARCUS A. TIUS ET AL.: "The Reaction of XeF2 with Trialkylvinylstannanes: Scope and Some Mechanistic Observations", TETRAHEDRON, vol. 51, no. 14, 1995, pages 3997 - 4010
MATTHEW TREDWELL ET AL.: "Electrophilic fluorination of organosilanes", ORG. BIOMOL. CHEM., vol. 4, 2005, pages 26 - 32
TAKERU FURUYA ET AL.: "Palladium-Mediated Fluorination of Arylboronic acids", ANGEW. CHEM. INT. ED., vol. 47, 4 July 2008 (2008-07-04), pages 5993 - 5996, XP009115959
RAJENDRA P. SINGH ET AL.: "Recent Highlights in Electrophilic Fluorination with 1-Chloromethyl-4-fluoro-1.4-diazoniabicyclo[2.2.2]octane Bis(tetrafluoroborate)", ACC. CHEM. RES., vol. 37, 2004, pages 31 - 44
MATTHEW TREDWELL ET AL.: "Electrophilic fluorination of organosilanes", ORG. BIOMOL. CHEM., vol. 4, 2005, pages 26 - 32
TAKERU FURUYA ET AL.: "Palladium-Mediated Fluorination of Arylboronic acids", ANGEW. CHEM. INT. ED., vol. 47, 4 July 2008 (2008-07-04), pages 5993 - 5996, XP009115959
RAJENDRA P. SINGH ET AL.: "Recent Highlights in Electrophilic Fluorination with 1-Chloromethyl-4-fluoro-1.4-diazoniabicyclo[2.2.2]octane Bis(tetrafluoroborate)", ACC. CHEM. RES., vol. 37, 2004, pages 31 - 44
Attorney, Agent or Firm:
MCCARTY, Catherine, M. (LLPOne Main Street, Eleventh Floo, Cambridge MA, US)
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