FUSICOCCIN COMPOUND

WIPO Patent Application WO/2018/143140

A1

Through the fusicoccin compound according to the present invention represented by general formula (1A), PPI stabilization effect can be enhanced. [In the formula, Y represents a carbonyl group, a sulfonyl group, or a substituted or unsubstituted alkylene group; R1 and R2 are the same or different and represent a hydrogen atom or a hydroxyl group; R3 represents a hydrogen atom, a substituted or unsubstituted aminoalkyl group, or a group represented by general formula (2) (In general formula (2), R5 represents a hydrogen atom or a substituted or unsubstituted alkyl group; R6 represents a hydrogen atom; R5 and R6 may be bonded and form a substituted or unsubstituted alkylene group; and the symbol * represents a bond.); R4a represents a substituted or unsubstituted alkyl group, a substituted or unsubstituted (hetero)cycloalkyl group, a substituted or unsubstituted alkoxy group, a substituted or unsubstituted (hetero)aryl group, or a substituted or unsubstituted amino group; and the case of R4a representing an epoxy group is excluded when Y is a carbonyl group, R1 is a hydroxyl group, R2 is a hydrogen atom, and R3 is a group represented by general formula (2).]

JP4020961	Amphiphilic compounds with at least 2 hydrophilic groups and at least 2 hydrophobic groups based on diol ethers, oligool ethers or polyol ethers
JP2624901	NOVEL DERIVATIVE HAVING NAPHTHALENE STRUCTURE, PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME
JPS6154	PHENYLACETAMIDE AS ANTIALLERGIC, ANTIASTHMATIC AND ANTIINFLAMMATORY

HIGUCHI YUSUKE (JP)
KATO NOBUO (JP)
HAN LING (JP)

PCT/JP2018/002825

August 09, 2018

January 30, 2018

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UNIV OSAKA (JP)

C07C233/17; A01G7/06; A01N45/02; A01N47/12; A01N47/28; A01N53/12; A01P21/00; A61K31/704; A61P35/00; C07H15/24

WO2013031975A1	2013-03-07
WO2010090234A1	2010-08-12
WO2008010324A1	2008-01-24

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SAEGUSA & PARTNERS (JP)

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