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Title:
GLUCOPYRANOSYL DERIVATIVE AND USE THEREOF
Document Type and Number:
WIPO Patent Application WO/2019/144864
Kind Code:
A1
Abstract:
Provided are a glucopyranosyl derivative as a sodium-dependent glucose transporters inhibitor, especially as a SGLT1 inhibitor, a pharmaceutically acceptable salt or a stereoisomer thereof, a pharmaceutical composition thereof, and the uses of the compound and pharmaceutical composition thereof in the preparation of drugs for the treatment of diabetes and diabetes-related diseases.

Inventors:
GU ZHENG (CN)
WU WUYONG (CN)
QU TONG (CN)
KANG PANPAN (CN)
ZHANG ZONGYUAN (CN)
HUANG WEIMING (CN)
LIU JIANYU (CN)
ZHANG YINGJUN (CN)
Application Number:
PCT/CN2019/072666
Publication Date:
August 01, 2019
Filing Date:
January 22, 2019
Export Citation:
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Assignee:
SUNSHINE LAKE PHARMA CO LTD (CN)
International Classes:
A61K31/351; C07D309/10; A61P3/10
Domestic Patent References:
WO2010095768A12010-08-26
WO2007136116A22007-11-29
WO2010095768A12010-08-26
WO2007136116A22007-11-29
WO2012023582A12012-02-23
WO2006035967A12006-04-06
Foreign References:
CN107519161A2017-12-29
US20110218159A12011-09-08
US20110218159A12011-09-08
CN107519161A2017-12-29
US20110218159A12011-09-08
Other References:
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See also references of EP 3743412A4
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