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Title:
HERBICIDAL PYRIMIDINE COMPOUNDS
Document Type and Number:
WIPO Patent Application WO/2018/019574
Kind Code:
A1
Abstract:
The present invention relates to the pyrimidine compounds of formula (I), or their agriculturally acceptable salts or derivatives as herbicides, wherein the variables are defined according to the description, use of pyrimidine compounds of formula (I) as herbicide, compositions comprising them and their use as herbicides, i.e. for controlling harmful plants, and also a method for controlling unwanted vegetation which comprises allowing a herbicidal effective amount of at least one pyrimidine compounds of the formula (I) to act on plants, their seed and/or their habitat.

Inventors:
VOGT FLORIAN (DE)
WITSCHEL MATTHIAS (DE)
SEISER TOBIAS (DE)
LOPEZ CARRILLO VERONICA (DE)
SEITZ THOMAS (DE)
KRAEMER GERD (DE)
NEWTON TREVOR WILLIAM (DE)
Application Number:
PCT/EP2017/067423
Publication Date:
February 01, 2018
Filing Date:
July 11, 2017
Export Citation:
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Assignee:
BASF SE (DE)
International Classes:
A01N43/54; C07D403/04; C07D409/04; C07D413/04; C07D419/04; C07D419/14
Domestic Patent References:
WO2013178585A12013-12-05
WO2005063721A12005-07-14
WO2000073278A22000-12-07
WO2013186229A12013-12-19
WO2014202493A12014-12-24
WO2009013462A12009-01-29
WO2011154327A12011-12-15
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WO2007096576A12007-08-30
WO2002015701A22002-02-28
WO1993007278A11993-04-15
WO1995034656A11995-12-21
WO2003018810A22003-03-06
WO2003052073A22003-06-26
WO2003018810A22003-03-06
Foreign References:
EP0374753A21990-06-27
EP0427529A11991-05-15
EP0451878A11991-10-16
EP0392225A21990-10-17
Other References:
KAMEI ET AL., TETRAHEDRON LETT., vol. 55, 2014, pages 4245 - 4247
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, vol. 36, 2013, pages 8083
"Farm Chemicals Handbook", vol. 86, 2000, MEISTER PUBLISHING COMPANY
B. HOCK; C. FEDTKE; R. R. SCHMIDT: "Herbizide [Herbicides", 1995, GEORG THIEME VERLAG
W. H. AHRENS: "Herbicide Handbook", 1994, WEED SCIENCE SOCIETY OF AMERICA
K. K. HATZIOS: "Herbicide Handbook", 1998, WEED SCIENCE SOCIETY OF AMERICA
"Technical Monograph No. 2", May 2008, CROPLIFE INTERNATIONAL, article "Catalogue of pesticide formulation types and international coding system"
MOLLET; GRUBEMANN: "Formulation technology", 2001, WILEY VCH
KNOWLES: "Agrow Reports DS243", 2005, T&F INFORMA, article "New developments in crop protection product formulation"
MCCUTCHEON'S: "Emulsifiers & Detergents, McCutcheon's Directories", vol. 1, 2008
KNOWLES: "Agrow Reports DS256", 2006, T&F INFORMA UK, article "Adjuvants, and additives"
PEST MANAGEMENT SCIENCE, vol. 61, 2005, pages 246
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AUSTRALIAN JOURNAL OF AGRICULTURAL RESEARCH, vol. 58, 2007, pages 708
SCIENCE, vol. 316, 2007, pages 1185
Attorney, Agent or Firm:
BASF IP ASSOCIATION (DE)
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Claims:
Claims

1. The pyrimidine compounds of formula (I)

wherein

the dotted line (----- ) is a single bond or a double bond;

R1 is Ci-Ce-alkyl, C1-C6-haloalkyl, HO-C1-C6-alkyl, C3-C6-alkenyl, C3-C6-haloalkenyl, C2- C6-alkynyl, C3-C6-haloalkynyl, C1-C6-alkoxy-C1-C6-alkyl, C1-C6-alkoxy, C3-C6- alkenyloxy, C3-C6-haloalkenyloxy, C3-C6-alkynyloxy, C3-C6-haloalkynyloxy, C1-C6- haloalkoxy, C3-C6-cycloalkoxy, C3-C6-halocycloalkoxy, C3-C6-cycloalkenyloxy, C3-C6- halocycloalkenyloxy, C1-C6-alkylthio, C1-C6-haloalkylthio, (C1-C6-alkyl)amino, di(Ci- C6-alkyl)amino, C1-C6-alkylsulfinyl, C1-C6-alkylsulfonyl, C3-C6-cycloalkyl, C3-C6-cyclo- alkenyl, C3-C6-halocycloalkyl, C3-C6-halocycloalkenyl, [1-(C1-C6-alkyl)]-C3-C6-cyclo- alkyl, [1-(C3-C6-alkenyl)]-C3-C6-cycloalkyl, [1-(C2-C6-alkynyl)]-C3-C6-cycloalkyl, [1- (C1-C6-haloalkyl)]-C3-C6-cycloalkyl, [1-(C3-C6-haloalkenyl)]-C3-C6-cycloalkyl, [1-(C3-

C6-haloalkynyl)]-C3-C6-cycloalkyl, C3-C6-cycloalkyl-C1-C6-alkyl, C3-C6-cycloalkyl-Ci- C6-haloalkyl, C3-C6-cycloalkyl-C1-C6-alkoxy, C3-C6-cycloalkyl-C1-C6-haloalkoxy, phenyl, 5- or 6-membered heteroaryl, or 3- to 6-membered heterocyclyl; wherein the cyclic groups of R1 are unsubstituted or substituted by Ra;

R2 is Ci-Ce-alkyl, C1-C6-haloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C1-C6-alkoxy-C2-C6- alkenyl, C1-C6-alkoxy-C2-C6-haloalkenyl, C1-C6-haloalkoxy-C2-C6-alkenyl, C1-C6- haloalkoxy-C2-C6-haloalkenyl, C2-C6-alkynyl, C2-C6-haloalkynyl, C1-C6-alkoxy-C2-C6- alkynyl, C1-C6-alkoxy-C3-C6-haloalkynyl, C1-C6-haloalkoxy-C2-C6-alkynyl, C1-C6- haloalkoxy-C3-C6-haloalkynyl, C3-C6-cycloalkyl, C3-C6-halocycloalkyl, C3-C6- cycloalkenyl, C3-C6-halocycloalkenyl, C3-C6-cycloalkyl-CrC6-alkyl, C3-C6-cycloalkyl- C1-C6-haloalkyl, C3-C6-halocycloalkyl-C1-C6-alkyl, C3-C6-halocycloalkyl-C1-C6- haloalkyl, C3-C6-cycloalkenyl-C1-C6-alkyl, C3-C6-cycloalkenyl-C1-C6-haloalkyl, C3-C6- halocycloalkenyl-C1-C6-alkyl, C3-C6-halocycloalkenyl-C1-C6-haloalkyl, C3-C6- cycloalkyl- C2-C6-alkenyl, C3-C6-cycloalkyl-C2-C6-haloalkenyl, C3-C6-halocycloalkyl- C2-C6-alkenyl, C3-C6-halocycloalkyl-C2-C6-haloalkenyl, C3-C6-cycloalkenyl-C2-C6- alkenyl, C3-C6-cycloalkenyl-C2-C6-haloalkenyl, C3-C6-halocycloalkenyl-C2-C6-alkenyl, C3-C6-halocycloalkenyl-C2-C6-haloalkenyl, C3-C6-cycloalkyl-C2-C6-alkynyl, C3-C6- cycloalkyl-C3-C6-haloalkynyl, C3-C6-halocycloalkyl-C2-C6-alkynyl, C3-C6- halocycloalkyl-C3-C6-haloalkynyl, C3-C6-cycloalkenyl-C2-C6-alkynyl, C3-C6- cycloalkenyl-C3-C6-haloalkynyl, C3-C6-halocycloalkenyl-C2-C6-alkynyl, C3-C6- halocycloalkenyl-C3-C6-haloalkynyl, C3-C6-cycloalkyl-C1-C6-alkylidenyl, C3-C6- cycloalkyl-C2-C6-haloalkylidenyl, C3-C6-halocycloalkyl-C1-C6-alkylidenyl, C3-C6- halocycloalkyl-C2-C6-haloalkylidenyl, C3-C6-cycloalkenyl-C1-C6-alkylidenyl, C3-C6- cycloalkenyl-C2-C6-haloalkylidenyl, C3-C6-halocycloalkenyl-C1-C6-alkylidenyl, C3-C6- halocycloalkenyl-C2-C6-haloalkylidenyl, heterocyclyl-C1-C6-alkylidenyl, heterocyclyl- C2-C6-haloalkylidenyl, C3-C6-hydroxycycloalkyl-C1-C6-alkyl, C3-C6-hydroxycycloalkyl- C1-C6-haloalkyl, C3-C6-hydroxycycloalkenyl-C1-C6-alkyl, C3-C6-hydroxycycloalkenyl- C1-C6-haloalkyl, C1-C6-hydroxyalkyl, C2-C6-hydroxyhaloalkyl, C3-C6-hydroxyalkenyl, C3-C6-hydroxyhaloalkenyl, C3-C6-hydroxyalkynyl, C4-C6-hydroxyhaloalkynyl, C3-C6- hydroxycycloalkyl, C3-C6-hydroxyhalocycloalkyl, C3-C6-hydroxycycloalkenyl, C3-C6- hydroxyhalocycloalkenyl, C3-C6-cycloalkyl-C1-C6-hydroxyalkyl, C3-C6-cycloalkyl-C2- C6-hydroxyhaloalkyl, C3-C6-halocycloalkyl-C1-C6-hydroxyalkyl, C3-C6-halocycloalkyl- C2-C6-hydroxyhaloalkyl, C3-C6-cycloalkenyl-C1-C6-hydroxyalkyl, C3-C6-cycloalkenyl- C2-C6-hydroxyhaloalkyl, C3-C6-halocycloalkenyl-C1-C6-hydroxyalkyl, C3-C6- halocycloalkenyl-C2-C6-hydroxyhaloalkyl, C3-C6-cycloalkyl-C3-C6-hydroxyalkenyl, C3- C6-cycloalkyl-C3-C6-hydroxyhaloalkenyl, C3-C6-halocycloalkyl-C3-C6-hydroxyalkenyl, C3-C6-halocycloalkyl-C3-C6-hydroxyhaloalkenyl, C3-C6-cycloalkenyl-C3-C6- hydroxyalkenyl, C3-C6-cycloalkenyl-C3-C6-hydroxyhaloalkenyl, C3-C6- halocycloalkenyl-C3-C6-hydroxyalkenyl, C3-C6-halocycloalkenyl-C3-C6- hydroxyhaloalkenyl, C3-C6-cycloalkyl-C3-C6-hydroxyalkynyl, C3-C6-halocycloalkyl-C3- C6-hydroxyalkynyl, C3-C6-cycloalkenyl-C3-C6-hydroxyalkynyl, C3-C6- halocycloalkenyl-C3-C6-hydroxyalkynyl, C3-C6-cycloalkyl-C2-C6-hydroxyalkylidenyl, C3-C6-halocycloalkyl-C2-C6-hydroxyalkylidenyl, C3-C6-cycloalkenyl-C2-C6- hydroxyalkylidenyl, C3-C6-halocycloalkyl-C2-C6-hydroxyalkylidenyl, heterocyclyl-C2- C6-hydroxyalkylidenyl, hydroxycarbonyl-C1-C6-hydroxyalkyl, hydroxycarbonyl-C1-C6- alkyl, hydroxycarbonyl-C1-C6-haloalkyl, C1-C6-alkoxycarbonyl-C1-C6-hydroxyalkyl, C1-C6-haloalkoxycarbonyl-C1-C6-hydroxyalkyl, C1-C6-alkoxycarbonyl-C1-C6-haloalkyl, C1-C6-haloalkoxycarbonyl-C1-C6-haloalkyl, CrC6-alkoxycarbonyl-C1-C6-alkyl, C1-C6- haloalkoxycarbonyl-C1-C6-alkyl, C3-C6-hydroxycycloalkyl-C1-C6-hydroxyalkyl, C3-C6- hydroxycycloalkenyl-C1-C6-hydroxyalkyl, C3-C6-hydroxycycloalkyl-C3-C6- hydroxyalkenyl, C3-C6-hydroxycycloalkenyl-C3-C6-hydroxyalkenyl, C3-C6- hydroxycycloalkyl-C3-C6-hydroxyalkynyl, C3-C6-hydroxycycloalkenyl-C3-C6- hydroxyalkenyl, C2-C6-dihydroxyalkyl, C3-C6-dihydroxyhaloalkyl, C4-C6- dihydroxyalkenyl, C4-C6-dihydroxyhaloalkenyl, C4-C6-dihydroxyalkynyl, C5-C6- dihydroxyhaloalkynyl, C4-C6-dihydroxycycloalkyl, C4-C6-dihydroxyhalocycloalkyl, C4- C6-dihydroxycycloalkenyl, C4-C6-dihydroxyhalocycloalkenyl, C3-C6-cycloalkyl-C2-C6- dihydroxyalkyl, C3-C6-halocycloalkyl-C2-C6-dihydroxyalkyl, C3-C6-cycloalkenyl-C2-C6- dihydroxyalkyl, C3-C6-halocycloalkenyl-C2-C6-dihydroxyalkyl, C3-C6-cycloalkyl-C3-C6- dihydroxyalkenyl, C3-C6-halocycloalkyl-C3-C6-dihydroxyalkenyl, C3-C6-cycloalkenyl- C3-C6-dihydroxyalkenyl, C3-C6-halocycloalkenyl-C3-C6-dihydroxyalkenyl, C3-C6- cycloalkyl-C4-C6-dihydroxyalkynyl, C3-C6-halocycloalkyl-C4-C6-dihydroxyalkynyl, C3- C6-cycloalkenyl-C4-C6-dihydroxyalkynyl, C3-C6-halocycloalkyl-C4-C6- dihydroxyalkynyl, C3-C6-cycloalkyl-C3-C6-dihydroxyalkylidenyl, C3-C6-halocycloalkyl- C3-C6-dihydroxyalkylidenyl, heterocyclyl-C3-C6-dihydroxyalkylidenyl,

hydroxycarbonyl-C2-C6-dihydroxyalkyl, hydroxycarbonyl-C3-C6-dihydroxyhaloalkyl, C1-C6-alkoxycarbonyl-C2-C6-dihydroxyalkyl, C1-C6-haloalkoxycarbonyl-C2-C6- dihydroxyalkyl, C1-C6-haloalkoxycarbonyl-C3-C6-dihydroxyhaloalkyl, C3-C6- dihydroxycycloalkyl- C1-C6-alkyl, C3-C6-dihydroxycycloalkyl- C1-C6-haloalkylC3-C6- dihydroxycycloalkyl- C2-C6-alkenyl, C3-C6-dihydroxycycloalkyl- C2-C6-haloalkenyl, C3-C6-dihydroxycycloalkyl- C2-C6-alkynyl, C3-C6-dihydroxycycloalkyl- C3-C6- haloalkynyl, C1-C6-alkylcarbonyl-C1-C6-alkyl, C1-C6-haloalkylcarbonyl-C1-C6-alkyl, C1-C6-alkylcarbonyl-C1-C6-haloalkyl, C1-C6-haloalkylcarbonyl-C1-C6-haloalkyl, hydroxycarbonyl-C2-C6-alkenyl, hydroxycarbonyl-C2-C6-haloalkenyl, C1-C6-alkoxy- carbonyl-C2-C6-alkenyl, C1-C6-haloalkoxycarbonyl-C2-C6-alkenyl, C1-C6-alkoxy- carbonyl-C2-C6-haloalkenyl, C1-C6-haloalkoxycarbonyl-C2-C6-haloalkenyl, hydroxycarbonyl-C2-C6-alkynyl, hydroxycarbonyl-C3-C6-haloalkynyl, C1-C6-alkoxy- carbonyl-C2-C6-alkynyl, C1-C6-haloalkoxycarbonyl-C2-C6-alkynyl, C1-C6-alkoxy- carbonyl-C3-C6-haloalkynyl, C1-C6-haloalkoxycarbonyl-C3-C6-haloalkynyl, C1-C6- cyanoalkyl, C2-C6-cyanohaloalkyl, C1-C6-dicyanoalkyl, C2-C6-dicyanohaloalkyl, di(hydroxycarbonyl)-C1-C6-alkyl, di(hydroxycarbonyl)-C1-C6-haloalkyl, di(C1-C6- alkoxycarbonyl)-C1-C6-alkyl, di(C1-C6-haloalkoxycarbonyl)-C1-C6-alkyl, di(C1-C6- alkoxycarbonyl)-C1-C6-haloalkyl, di(C1-C6-haloalkoxycarbonyl)-C1-C6-haloalkyl, di(C1-C6-alkoxyl)phosphoryl-C1-C6-alkyl, di(C1-C6-haloalkoxyl)phosphoryl-C1-C6- alkyl, di(C1-C6-alkoxyl)phosphoryl-C1-C6-haloalkyl, di(C1-C6-haloalkoxyl)phosphoryl- C1-C6-haloalkyl, phosphoryl-C1-C6-alkyl , phosphoryl-C1-C6-haloalkyl , di[di(C1-C6- alkoxyl)phosphoryl-)]C1-C6-alkyl, di[di(C1-C6-haloalkoxyl)phosphoryl-)]CrC6-alkyl, di[di(C1-C6-alkoxyl)phosphoryl-)]C1-C6-haloalkyl, di[di(C1-C6-haloalkoxyl)phosphoryl- )]C1-C6-haloalkyl, diphosphoryl-C1-C6-alkyl , diphosphoryl-C1-C6-haloalkyl, C1-C6- alkylthio-Ci-Ce-alkyl, Ci-Ce-haloalkylthio-Ci-Ce-alkyl, Ci-Ce-alkylthio-Ci-Ce-haloalkyl, Ci-Ce-haloalkylthio-Ci-Ce-haloalkyl, Ci-Ce-alkylsulfinly-Ci-Ce-alkyl, C1-C6- haloalkylsulfinly-C1-C6-alkyl, C1-C6-alkylsulfinly-C1-C6-haloalkyl, C1-C6- haloalkylsulfinly-C1-C6-haloalkyl, C1-C6-alkylsulfonyl-C1-C6-alkyl, C1-C6- haloalkylsulfonyl-C1-C6-alkyl, C1-C6-haloalkylsulfonyl-C1-C6-haloalkyl, phenyl, 5- or 6-membered heteroaryl, 3- to 6-membered heterocyclyl;

wherein hydroxy groups of R2 are unsubstituted or substituted by Rb;

cyclic groups of R2 are unsubstituted or substituted by Rc; and

acyclic aliphatic groups of R2 are unsubstituted or substituted by Rd;

Rb is Ci-Ce-alkyl, C1-C6-haloalkyl, C3-C6-alkenyl, C3-C6-haloalkenyl, C3-C6-alkynyl, C3- C6-haloalkynyl, C3-C6-cycloalkyl, C3-C6-halocycloalkyl, C4-C6-cycloalkenyl, C3-C6- halocycloalkenyl, CrC6-alkoxycarbonyl-C1-C6-alkyl, CrC6-haloalkoxycarbonyl-Ci- C6-alkyl, C1-C6-alkoxycarbonyl-CrC6-haloalkyl, C1-C6-haloalkoxycarbonyl-CrC6- haloalkyl, C1-C6-alkylcarbonyl, C1-C6-haloalkylcarbonyl, hydroxycarbonyl-C1-C6-alkyl, hydroxycarbonyl-C1-C6-haloalkyl, C1-C6-alkyloxycarbonyl, C1-C6- haloalkyloxycarbonyl, C1-C6-alkylthiocarbonyl, C1-C6-haloalkylthiocarbonyl, C1-C6- alkylaminocarbonyl, C1-C6-haloalkylaminocarbonyl, C1-C6-dialkylaminocarbonyl, Ci- C6-dihaloalkylaminocarbonyl, C1-C6-alkylsulfonyl, C1-C6-haloalkylsulfonyl, C1-C6- alkoxy-C1-C6-alkyl, C1-C6-haloalkoxy-C1-C6-alkyl, C1-C6-alkoxy-C1-C6-haloalkyl, Ci- C6-haloalkoxy-CrC6-haloalkyl, phenyl-C1-C6-alkyl, or phenyl-C1-C6-haloalkyl;

Rc is halogen, CN, N02, C1-C6-alkyl, C1-C6-haloalkyl, OH, C1-C6-alkoxy or C1-C6- haloalkoxy, C1-C6-alkylthio, C1-C6-alkylsulfinyl, or C1-C6-alkylsulfonyl;

Rd is phenyl, 5- or 6-membered heteroaryl, or 3- to 6-membered heterocyclyl;

wherein the substituent Rd is unsubstituted or substituted by Re; Re is halogen, CN, N02, C1-C6-alkyl, C1-C6-haloalkyl, OH, C1-C6-alkoxy or C1-C6- haloalkoxy, C1-C6-alkylsulfonyl;

A is CR3 or NR3A;

Z is a 5 or 6 membered heteroaryl ring comprising A;

R3 is halogen, CN, N02, CHO, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkylcarbonyl, C3-C6- alkenyl, C3-C6-haloalkenyl, C2-C6-alkynyl, C3-C6-haloalkynyl, C1-C6-alkoxy, C1-C6- haloalkoxy, C3-C6-alkenyloxy, C3-C6-haloalkenyloxy, C3-C6-alkynyloxy, C3-C6-ha- loalkynyloxy, C1-C6-alkoxy-C1-C6-alkoxy, hydroxycarbonyl, C1-C6-alkoxycarbonyl, C1-C6-alkylthio, C1-C6-haloalkylthio, NH2, (C1-C6-alkyl)amino, di(C1-C6-alkyl)amino, (C1-C6-alkyl)sulfinyl, (C1-C6-alkyl)sulfonyl, C3-C6-cycloalkyl, (C3-C6-cycloalkyl)oxy, or phenyl;

wherein the cyclic groups of R3are unsubstituted or substituted by substituents Ra;

R3A is H, Ci-Ce-alkyl, C1-C6-haloalkyl, C1-C6-alkylcarbonyl, C3-C6-alkenyl, C3-C6- haloalkenyl, C2-C6-alkynyl, C3-C6-haloalkynyl, C1-C6-alkoxy, C1-C6-haloalkoxy, C3- C6-alkenyloxy, C3-C6-haloalkenyloxy, C3-C6-alkynyloxy, C3-C6-haloalkynyloxy, C1-C6- alkoxy-C1-C6-alkoxy, C1-C6-alkoxycarbonyl, C1-C6-alkylthio, C1-C6-haloalkylthio, NH2, (C1-C6-alkyl)amino, di(C1-C6-alkyl)amino, (C1-C6-alkyl)sulfinyl, (C1-C6-alkyl)sulfonyl, C3-C6-cycloalkyl, (C3-C6-cycloalkyl)oxy, or phenyl;

wherein the cyclic groups of R3A are unsubstituted or substituted by Ra;

R4 is halogen, CN, N02, CHO, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkylcarbonyl, C3-C6- alkenyl, C3-C6-haloalkenyl, C3-C6-alkenyl, C3-C6-haloalkenyl, C1-C6-alkoxy, C1-C6- haloalkoxy, C3-C6-alkenyloxy, C3-C6-haloalkenyloxy, C3-C6-alkenyloxy, C3-C6- haloalkenyloxy, C1-C6-alkoxy-C1-C6-alkoxy, hydroxycarbonyl, C1-C6-alkoxycarbonyl, C1-C6-alkylthio, C1-C6-haloalkylthio, NH2, (C1-C6-alkyl)amino, di(C1-C6-alkyl)amino, (C1-C6-alkyl)sulfinyl, (C1-C6-alkyl)sulfonyl, C3-C6-cycloalkyl, (C3-C6-cycloalkyl)oxy, or phenyl;

wherein the cyclic groups of R4 are unsubstituted or substituted by Ra;

Ra is halogen, CN, N02, Ci-Ce-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, or C1-C6- haloalkoxy;

m is 0, 1 , 2, or 3;

including agriculturally acceptable salts or derivatives of compounds of formula (I) having an acidic functionality.

The pyrimidine compounds of formula (I) according to claim 1 , wherein the heteroaryl ring Z is selected from rings A to G,

wherein

R3 is halogen, CHO, CN, C1-C6-alkyl, C1-C6-haloalkyl, or C1-C6-alkoxy;

m is 0 or 1 ;

R4 is halogen, CHO, CN, C1-C6-alkyl, C1-C6-haloalkyl, or C1-C6-alkoxy;

X is O, S, or NR3A;

R3A is H, Ci-Ce-alkyl, C1-C6-haloalkyl, C1-C6-alkylcarbonyl, C3-C6-alkenyl, C3-C6- haloalkenyl, C3-C6-alkenyl, C3-C6-haloalkenyl, or C3-C6-cycloalkyl;

# denotes the point of attachment to the pyrimidine ring.

The pyrimidine compounds of formula (I) according to claim 1 or 2, wherein

R1 is C1-C6-alkyl, C1-C6-alkoxy, C1-C6-haloalkoxy, C3-C6-alkenyloxy, C3-C6- haloalkenyloxy C3-C6-alkynyloxy, C3-C6-haloalkynyloxy, C1-C6-alkylthio, or C3-C6- cycloalkyl, wherein the cycloalkyl substituent is unsubstituted.

The pyrimidine compounds of formula (I) according to any of claims 1 to 3, wherein R2 is C2-C6-alkenyl, C2-C6-haloalkenyl, CrC6-alkoxy-C2-C6-alkenyl, C2-C6-alkynyl, C3-C6- cycloalkenyl, C3-C6-cycloalkenyl-C1-C6-alkyl, C3-C6-cycloalkyl-C1-C6-alkylidenyl, C3- C6-halocycloalkyl-C1-C6-alkylidenyl, C3-C6-cycloalkenyl-C1-C6-alkylidenyl, C3-C6- hydroxycycloalkyl-C1-C6-alkyl, C3-C6-hydroxycycloalkenyl-C1-C6-alkyl, C1-C6- hydroxyalkyl, C3-C6-cycloalkyl-C2-C6-hydroxyalkylidenyl, hydroxycarbonyl-C1-C6- alkyl, hydroxycarbonyl-C1-C6-haloalkyl, C1-C6-alkoxycarbonyl-C1-C6-alkyl, C3-C6- hydroxycycloalkyl-C1-C6-hydroxyalkyl, C2-C6-dihydroxyalkyl, C3-C6-cycloalkyl-C3-C6- dihydroxyalkylidenyl, hydroxycarbonyl-C2-C6-dihydroxyalkyl, C1-C6-alkoxycarbonyl- C2-C6-dihydroxyalkyl, C1-C6-dicyanoalkyl, or 5- or 6-membered heteroaryl;

wherein OH groups of R2 are unsubstituted or substituted by Rb;

cyclic groups of R2 are unsubstituted or substituted by Rc; and

acyclic aliphatic groups of R2 are unsubstituted or substituted by Rd;

Rb is Ci-Ce-alkyl, C1-C6-haloalkyl, C3-C6-alkenyl, C3-C6-haloalkenyl, C3-C6-alkynyl, C3- C6-haloalkynyl, C3-C6-cycloalkyl, C3-C6-halocycloalkyl, C4-C6-cycloalkenyl, C3-C6- halocycloalkenyl, C1-C6-alkoxycarbonyl-C1-C6-alkyl, C1-C6-haloalkoxycarbonyl-Ci- C6-alkyl, C1-C6-alkoxycarbonyl-C1-C6-haloalkyl, C1-C6-haloalkoxycarbonyl-C1-C6- haloalkyl, C1-C6-alkylcarbonyl, C1-C6-haloalkylcarbonyl, hydroxycarbonyl-C1-C6- alkyl, hydroxycarbonyl-C1-C6-haloalkyl, C1-C6-alkyloxycarbonyl, C1-C6- haloalkyloxycarbonyl, C1-C6-alkylthiocarbonyl, C1-C6-haloalkylthiocarbonyl, C1-C6- alkylaminocarbonyl, C1-C6-haloalkylaminocarbonyl, C1-C6-dialkylaminocarbonyl, C1-C6-dihaloalkylaminocarbonyl, C1-C6-alkylsulfonyl, C1-C6-haloalkylsulfonyl, Ci- C6-alkoxy-C1-C6-alkyl, C1-C6-haloalkoxy-C1-C6-alkyl, C1-C6-alkoxy-C1-C6- haloalkyl, C1-C6-haloalkoxy-C1-C6-haloalkyl, phenyl-C1-C6-alkyl, or phenyl-C1-C6- haloalkyl;

Rc is halogen, CN, N02, C1-C6-alkyl, C1-C6-haloalkyl, OH, C1-C6-alkoxy or C1-C6- haloalkoxy, C1-C6-alkylthio, C1-C6-alkylsulfinyl, or C1-C6-alkylsulfonyl;

Rd is phenyl, 5- or 6- membered heteroaryl, or 3- to 6-membered heterocyclyl;

wherein the substituent Rd is unsubstituted or substituted by Re; Re is halogen, CN, N02, C1-C6-alkyl, C1-C6-haloalkyl, OH, C1-C6-alkoxy or C1-C6- haloalkoxy, C1-C6-alkylsulfonyl.

The pyrimidine compounds of formula (I) according to any of claims 1 to 4, wherein R1 is c-C3H5;

R2 is Ci-Ce-alkyl, C2-C6-alkenyl, C3-C6-cycloalkyl-Ci-Ce-alkyl, C3-C6-cycloalkenyl-Ci-Ce- alkyl, C3-C6-cycloalkyl-C1-C6-alkylidenyl, C1-C6-hydroxyalkyl, hydroxycarbonyl-C1-C6- alkyl, hydroxycarbonyl-C1-C6-haloalkyl, C1-C6-alkoxycarbonyl-CrC6-alkyl, C1-C6- alkoxycarbonyl-CrC6-haloalkyl, or 5- membered heteroaryl;

wherein OH groups of R2 are unsubstituted or substituted by Rb,

cyclic groups of R2 are unsubstituted or substituted by Rc, and

acyclic aliphatic groups of R2 are unsubstituted or substituted by Rd;

Rb is Ci-Ce-alkyl;

Rc is Ci-Ce-alkyl or OH;

Rd is phenyl or 5- or 6- membered heteroaryl;

wherein the substituent Rd is unsubstituted or substituted by Re;

Re is halogen, CN, N02, C1-C6-alkyl, C1-C6-haloalkyl, OH, C1-C6-alkoxy, C1-C6- haloalkoxy, C1-C6-alkylsulfonyl;

Z is A, E, F, or G;

X is S;

R3 is CI, Br, F, I, CH3, or OCF3;

m is 0 or 1 ;

R4 is Br.

A use of pyrimidine compounds of formula (I), including agriculturally acceptable salts or derivatives of compounds of formula (I) having an acidic functionality, according to any of claims 1 to 5, as herbicide.

A herbicidal composition comprising:

A) at least one pyrimidine compound of formula I, including agriculturally acceptable salts or derivatives of compounds of formula (I) having an acidic functionality, according to any of claims 1 to 5;

and

B) herbicides of class b1 ) to b15):

b1 ) lipid biosynthesis inhibitors;

b2) acetolactate synthase inhibitors (ALS inhibitors);

b3) photosynthesis inhibitors;

b4) protoporphyrinogen-IX oxidase inhibitors,

b5) bleacher herbicides;

b6) enolpyruvyl shikimate 3-phosphate synthase inhibitors (EPSP inhibitors); b7) glutamine synthetase inhibitors;

b8) 7,8-dihydropteroate synthase inhibitors (DHP inhibitors);

b9) mitosis inhibitors;

b10) inhibitors of the synthesis of very long chain fatty acids (VLCFA inhibitors);

b11) cellulose biosynthesis inhibitors;

b12) decoupler herbicides;

b13) auxinic herbicides;

b14) auxin transport inhibitors; and

b15) other herbicides selected from the group consisting of bromobutide, chlorflurenol, chlorflurenol-methyl, cinmethylin, cumyluron, dalapon, dazomet, difenzoquat, difenzoquat-metilsulfate, dimethipin, DSMA, dymron, endothal and its salts, etobenzanid, flamprop, flamprop- isopropyl, flamprop-methyl, flamprop-M-isopropyl, flamprop-M-methyl, flurenol, flurenol-butyl, flurprimidol, fosamine, fosamine-ammonium, indanofan, indaziflam, maleic hydrazide, mefluidide, metam, methiozolin (CAS 403640-27-7), methyl azide, methyl bromide, methyl-dymron, methyl iodide, MSMA, oleic acid, oxaziclomefone, pelargonic acid, pyributicarb, quinoclamine, triaziflam, tridiphane and 6-chloro-3-(2- cyclopropyl-6-methylphenoxy)-4-pyridazinol, and its salts and esters; including their agriculturally acceptable salts or derivatives.

8. A herbicidal composition comprising the herbicidal composition according to claim 7, and safeners.

9. The herbicidal composition according to claim 7 or 8, wherein the herbicidal

composition comprises at least one herbicide B selected from herbicides of class b1 , b2, b3, b4, b5, b6, b9, b10, b13 and b14.

10. The herbicidal composition according to any of claims 7 to 9, wherein the herbicidal composition comprises at least one herbicide B selected from herbicides of class b1 , b2, b4, b5, b9, b10, b13 and b14. 11. The herbicidal composition according to any of claim 7 to 10, wherein the weight ratio of component A to component B is in the range of from 1 :500 to 500:1.

12. A herbicidal composition comprising a herbicidal active amount of at least one

pyrimidine compound of formula (I) including agriculturally acceptable salts or derivatives of compounds of formula (I) having an acidic functionality, according to any of claims 1 to 5, and at least one inert liquid and/or solid carrier and, if appropriate, at least one surface-active substance.

13. A herbicidal composition comprising a herbicidal composition according to any of claims 7 to 11 , and at least one inert liquid and/or solid carrier and, if appropriate, at least one surface-active substance.

14. A method of controlling undesired vegetation, which comprises allowing a herbicidal active amount of at least one pyrimidine compound of formula (I) including agriculturally acceptable salts or derivatives of compounds of formula (I) having an acidic functionality, according to any of claims 1 to 5 or a composition according to any of claims 7 to 13 to act on plants, their environment or on seed. 15. A use of the herbicidal compositions according to any of claims 7 to 13 as herbicides.

Description:
Herbicidal pyrimidine compounds

The present invention relates to pyrimidine compounds of the general formula (I) defined below and to their use as herbicides. Moreover, the invention relates to compositions for crop protection and to a method for controlling unwanted vegetation.

Description:

Compounds having a 5-phenyl pyrimidine moiety are known in the art. WO 2000/073278 describes such compounds being antagonists of the Neurokinin 1 receptor and thus having pharmaceutical properties.

In agriculture, there is a constant demand to develop novel active ingredients, which complement or outperform present methods of treatment regarding activity, selectivity and environmental safety.

These and further objects are achieved by pyrimidine compounds of formula (I), defined below, and by their agriculturally suitable salts.

Accordingly, the present invention provides the pyrimidine compounds of formula (I)

the dotted line (----- ) is a single bond or a double bond;

R 1 is Ci-Ce-alkyl, C 1 -C 6 -haloalkyl, HO-C 1 -C 6 -alkyl, C 3 -C 6 -alkenyl, C 3 -C 6 -haloalkenyl, C 2 -C 6 - alkynyl, C 3 -C 6 -haloalkynyl, C 1 -C 6 -alkoxy-C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, C 3 -C 6 -alkenyloxy, C3- C6-haloalkenyloxy, C 3 -C 6 -alkynyloxy, C 3 -C 6 -haloalkynyloxy, C 1 -C 6 -haloalkoxy, C 3 -C 6 - cycloalkoxy, C 3 -C 6 -halocycloalkoxy, C 3 -C 6 -cycloalkenyloxy, C 3 -C 6 -halocycloalkenyloxy, C 1 -C 6 -alkylthio, C 1 -C 6 -haloalkylthio, (C 1 -C 6 -alkyl)amino, di(C 1 -C 6 -alkyl)amino, C 1 -C 6 -alkyl- sulfinyl, C 1 -C 6 -alkylsulfonyl, C 3 -C 6 -cycloalkyl, C 3 -C 6 -cycloalkenyl, C 3 -C 6 -halocycloalkyl, C3- Ce-halocycloalkenyl, [1-( C 1 -C 6 -alkyl)]-C 3 -C 6 -cycloalkyl, [1-(C 3 -C6-alkenyl)]-C 3 -C6-cycloalkyl, [1-(C 2 -C 6 -alkynyl)]-C 3 -C 6 -cycloalkyl, [1-(C 1 -C 6 -haloalkyl)]-C 3 -C 6 -cycloalkyl, [1-(C 3 -C 6 -halo- alkenyl)]-C 3 -C 6 -cycloalkyl, [1-(C 3 -C 6 -haloalkynyl)]-C 3 -C 6 -cycloalkyl, C 3 -C 6 -cycloalkyl-C 1 -C 6 - alkyl, C 3 -C 6 -cycloalkyl-C 1 -C 6 -haloalkyl, C 3 -C 6 -cycloalkyl-C 1 -C 6 -alkoxy, C 3 -C 6 -cycloalkyl-Ci- C6-haloalkoxy, phenyl, 5- or 6-membered heteroaryl, or 3- to 6-membered heterocyclyl; wherein the cyclic groups of R 1 are unsubstituted or substituted by R a ;

R 2 is Ci-Ce-alkyl, C 1 -C 6 -haloalkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -haloalkenyl, C 1 -C 6 -alkoxy-C2-C 6 - alkenyl, C 1 -C 6 -alkoxy-C 2 -C 6 -haloalkenyl, C 1 -C 6 -haloalkoxy-C 2 -C 6 -alkenyl, C 1 -C 6 - haloalkoxy-C 2 -C 6 -haloalkenyl, C 2 -C 6 -alkynyl, C 2 -C 6 -haloalkynyl, C 1 -C 6 -alkoxy-C 2 -C 6 - alkynyl, C 1 -C 6 -alkoxy-C 3 -C 6 -haloalkynyl, C 1 -C 6 -haloalkoxy-C 2 -C 6 -alkynyl, C 1 -C 6 - haloalkoxy-C 3 -C 6 -haloalkynyl, C 3 -C 6 -cycloalkyl, C 3 -C 6 -halocycloalkyl, C 3 -C 6 -cycloalkenyl, C 3 -C 6 -halocycloalkenyl, C 3 -C 6 -cycloalkyl- C 1 -C 6 -alkyl, C 3 -C 6 -cycloalkyl-CrC 6 -haloalkyl, C3- C6-halocycloalkyl-C 1 -C 6 -alkyl, C 3 -C 6 -halocycloalkyl-C 1 -C 6 -haloalkyl, C 3 -C 6 -cycloalkenyl-Ci- C6-alkyl, C 3 -C 6 -cycloalkenyl-C 1 -C 6 -haloalkyl, C 3 -C 6 -halocycloalkenyl-C 1 -C 6 -alkyl, C 3 -C 6 - halocycloalkenyl-C 1 -C 6 -haloalkyl, C 3 -C 6 -cycloalkyl- C 2 -C 6 -alkenyl, C 3 -C 6 -cycloalkyl-C 2 -C 6 - haloalkenyl, C 3 -C 6 -halocycloalkyl-C 2 -C 6 -alkenyl, C 3 -C 6 -halocycloalkyl-C 2 -C 6 -haloalkenyl, C 3 -C 6 -cycloalkenyl-C 2 -C 6 -alkenyl, C 3 -C 6 -cycloalkenyl-C 2 -C 6 -haloalkenyl, C 3 -C 6 - halocycloalkenyl-C 2 -C 6 -alkenyl, C 3 -C 6 -halocycloalkenyl-C 2 -C 6 -haloalkenyl, C 3 -C 6 - cycloalkyl-C 2 -C 6 -alkynyl, C 3 -C 6 -cycloalkyl-C 3 -C 6 -haloalkynyl, C 3 -C 6 -halocycloalkyl-C 2 -C 6 - alkynyl, C 3 -C 6 -halocycloalkyl-C 3 -C 6 -haloalkynyl, C 3 -C 6 -cycloalkenyl-C 2 -C 6 -alkynyl, C 3 -C 6 - cycloalkenyl-C 3 -C 6 -haloalkynyl, C 3 -C 6 -halocycloalkenyl-C 2 -C 6 -alkynyl, C 3 -C 6 - halocycloalkenyl-C 3 -C 6 -haloalkynyl, C 3 -C 6 -cycloalkyl-C 1 -C 6 -alkylidenyl, C 3 -C 6 -cycloalkyl- C 2 -C 6 -haloalkylidenyl, C 3 -C 6 -halocycloalkyl-C 1 -C 6 -alkylidenyl, C 3 -C 6 -halocycloalkyl-C 2 -C 6 - haloalkylidenyl, C 3 -C 6 -cycloalkenyl-C 1 -C 6 -alkylidenyl, C 3 -C 6 -cycloalkenyl-C 2 -C 6 - haloalkylidenyl, C 3 -C 6 -halocycloalkenyl-C 1 -C 6 -alkylidenyl, C 3 -C 6 -halocycloalkenyl-C 2 -C 6 - haloalkylidenyl, heterocyclyl-C 1 -C 6 -alkylidenyl, heterocyclyl-C 2 -C 6 -haloalkylidenyl, C 3 -C 6 - hydroxycycloalkyl-C 1 -C 6 -alkyl, C 3 -C 6 -hydroxycycloalkyl-C 1 -C 6 -haloalkyl, C 3 -C 6 - hydroxycycloalkenyl-C 1 -C 6 -alkyl, C 3 -C 6 -hydroxycycloalkenyl-C 1 -C 6 -haloalkyl, C 1 -C 6 - hydroxyalkyl, C 2 -C 6 -hydroxyhaloalkyl, C 3 -C 6 -hydroxyalkenyl, C 3 -C 6 -hydroxyhaloalkenyl, C 3 -C 6 -hydroxyalkynyl, C4-C6-hydroxyhaloalkynyl, C 3 -C 6 -hydroxycycloalkyl, C 3 -C 6 - hydroxyhalocycloalkyl, C 3 -C 6 -hydroxycycloalkenyl, C 3 -C 6 -hydroxyhalocycloalkenyl, C 3 -C 6 - cycloalkyl-CrC6-hydroxyalkyl, C 3 -C 6 -cycloalkyl-C 2 -C 6 -hydroxyhaloalkyl, C 3 -C 6 - halocycloalkyl-C 1 -C 6 -hydroxyalkyl, C 3 -C 6 -halocycloalkyl-C 2 -C 6 -hydroxyhaloalkyl, C 3 -C 6 - cycloalkenyl-C 1 -C 6 -hydroxyalkyl, C 3 -C 6 -cycloalkenyl-C 2 -C 6 -hydroxyhaloalkyl, C 3 -C 6 - halocycloalkenyl-C 1 -C 6 -hydroxyalkyl, C 3 -C 6 -halocycloalkenyl-C 2 -C 6 -hydroxyhaloalkyl, C3-

C6-cycloalkyl-C 3 -C 6 -hydroxyalkenyl, C 3 -C 6 -cycloalkyl-C 3 -C 6 -hydroxyhaloalkenyl, C 3 -C 6 - halocycloalkyl-C 3 -C 6 -hydroxyalkenyl, C 3 -C 6 -halocycloalkyl-C 3 -C 6 -hydroxyhaloalkenyl, C3- C6-cycloalkenyl-C 3 -C 6 -hydroxyalkenyl, C 3 -C 6 -cycloalkenyl-C 3 -C 6 -hydroxyhaloalkenyl, C3- C6-halocycloalkenyl-C 3 -C 6 -hydroxyalkenyl, C 3 -C 6 -halocycloalkenyl-C 3 -C 6 - hydroxyhaloalkenyl, C 3 -C 6 -cycloalkyl-C 3 -C 6 -hydroxyalkynyl, C 3 -C 6 -halocycloalkyl-C 3 -C 6 - hydroxyalkynyl, C 3 -C 6 -cycloalkenyl-C 3 -C 6 -hydroxyalkynyl, C 3 -C 6 -halocycloalkenyl-C 3 -C 6 - hydroxyalkynyl, C 3 -C 6 -cycloalkyl-C 2 -C 6 -hydroxyalkylidenyl, C 3 -C 6 -halocycloalkyl-C 2 -C 6 - hydroxyalkylidenyl, C 3 -C 6 -cycloalkenyl-C 2 -C 6 -hydroxyalkylidenyl, C 3 -C 6 -halocycloalkyl-C2- C6-hydroxyalkylidenyl, heterocyclyl-C 2 -C 6 -hydroxyalkylidenyl, hydroxycarbonyl-C 1 -C 6 - hydroxyalkyl, hydroxycarbonyl-C 1 -C 6 -alkyl, hydroxycarbonyl-C 1 -C 6 -haloalkyl, C 1 -C 6 - alkoxycarbonyl-CrC6-hydroxyalkyl, C 1 -C 6 -haloalkoxycarbonyl-CrC6-hydroxyalkyl, C 1 -C 6 - alkoxycarbonyl-CrC6-haloalkyl, CrC6-haloalkoxycarbonyl-C 1 -C 6 -haloalkyl, C 1 -C 6 - alkoxycarbonyl-C 1 -C 6 -alkyl, C 1 -C 6 -haloalkoxycarbonyl-C 1 -C 6 -alkyl, C 3 -C 6 - hydroxycycloalkyl-C 1 -C 6 -hydroxyalkyl, C 3 -C 6 -hydroxycycloalkenyl-C 1 -C 6 -hydroxyalkyl, C3- C6-hydroxycycloalkyl-C 3 -C 6 -hydroxyalkenyl, C 3 -C 6 -hydroxycycloalkenyl-C 3 -C 6 - hydroxyalkenyl, C 3 -C 6 -hydroxycycloalkyl-C 3 -C 6 -hydroxyalkynyl, C 3 -C 6 - hydroxycycloalkenyl-C 3 -C 6 -hydroxyalkenyl, C 2 -C 6 -dihydroxyalkyl, C 3 -C 6 - dihydroxyhaloalkyl, C4-C6-dihydroxyalkenyl, C4-C6-dihydroxyhaloalkenyl, C4-C6- dihydroxyalkynyl, Cs-Ce-dihydroxyhaloalkynyl, C4-C6-dihydroxycycloalkyl, C4-C6- dihydroxyhalocycloalkyl, C 4 -C6-dihydroxycycloalkenyl, C4-C6-dihydroxyhalocycloalkenyl, C 3 -C 6 -cycloalkyl-C 2 -C 6 -dihydroxyalkyl, C 3 -C 6 -halocycloalkyl-C 2 -C 6 -dihydroxyalkyl, C 3 -C 6 - cycloalkenyl-C 2 -C 6 -dihydroxyalkyl, C 3 -C 6 -halocycloalkenyl-C 2 -C 6 -dihydroxyalkyl, C 3 -C 6 - cycloalkyl-C 3 -C 6 -dihydroxyalkenyl, C 3 -C 6 -halocycloalkyl-C 3 -C 6 -dihydroxyalkenyl, C 3 -C 6 - cycloalkenyl-C 3 -C 6 -dihydroxyalkenyl, C 3 -C 6 -halocycloalkenyl-C 3 -C 6 -dihydroxyalkenyl, C3- C6-cycloalkyl-C4-C6-dihydroxyalkynyl, C 3 -C 6 -halocycloalkyl-C4-C6-dihydroxyalkynyl, C 3 -C 6 - cycloalkenyl-C4-C6-dihydroxyalkynyl, C 3 -C 6 -halocycloalkyl-C4-C6-dihydroxyalkynyl, C 3 -C 6 - cycloalkyl-C 3 -C 6 -dihydroxyalkylidenyl, C 3 -C 6 -halocycloalkyl-C 3 -C 6 -dihydroxyalkylidenyl, heterocyclyl-C 3 -C 6 -dihydroxyalkylidenyl, hydroxycarbonyl-C 2 -C 6 -dihydroxyalkyl, hydroxycarbonyl-C 3 -C 6 -dihydroxyhaloalkyl, C 1 -C 6 -alkoxycarbonyl-C 2 -C 6 -dihydroxyalkyl, C 1 -C 6 -haloalkoxycarbonyl-C 2 -C 6 -dihydroxyalkyl, C 1 -C 6 -haloalkoxycarbonyl-C 3 -C 6 - dihydroxyhaloalkyl, C 3 -C 6 -dihydroxycycloalkyl- C 1 -C 6 -alkyl, C 3 -C 6 -dihydroxycycloalkyl- Ci- C6-haloalkylC 3 -C 6 -dihydroxycycloalkyl- C 2 -C 6 -alkenyl, C 3 -C 6 -dihydroxycycloalkyl- C 2 -C 6 - haloalkenyl, C 3 -C 6 -dihydroxycycloalkyl- C 2 -C 6 -alkynyl, C 3 -C 6 -dihydroxycycloalkyl- C 3 -C 6 - haloalkynyl, C 1 -C 6 -alkylcarbonyl-C 1 -C 6 -alkyl, C 1 -C 6 -haloalkylcarbonyl-C 1 -C 6 -alkyl, C 1 -C 6 - alkylcarbonyl-C 1 -C 6 -haloalkyl, C 1 -C 6 -haloalkylcarbonyl-C 1 -C 6 -haloalkyl, hydroxycarbonyl- C 2 -C 6 -alkenyl, hydroxycarbonyl-C 2 -C 6 -haloalkenyl, C 1 -C 6 -alkoxycarbonyl-C 2 -C 6 -alkenyl, C 1 -C 6 -haloalkoxycarbonyl-C 2 -C 6 -alkenyl, C 1 -C 6 -alkoxycarbonyl-C 2 -C 6 -haloalkenyl, C 1 -C 6 - haloalkoxycarbonyl-C 2 -C 6 -haloalkenyl, hydroxycarbonyl-C 2 -C 6 -alkynyl, hydroxycarbonyl- C 3 -C 6 -haloalkynyl, C 1 -C 6 -alkoxycarbonyl-C 2 -C 6 -alkynyl, C 1 -C 6 -haloalkoxycarbonyl-C 2 -C 6 - alkynyl, C 1 -C 6 -alkoxycarbonyl-C 3 -C 6 -haloalkynyl, C 1 -C 6 -haloalkoxycarbonyl-C 3 -C 6 - haloalkynyl, C 1 -C 6 -cyanoalkyl, C 2 -C 6 -cyanohaloalkyl, C 1 -C 6 -dicyanoalkyl, C 2 -C 6 - dicyanohaloalkyl, di(hydroxycarbonyl)-C 1 -C 6 -alkyl, di(hydroxycarbonyl)-C 1 -C 6 -haloalkyl, di(C 1 -C 6 -alkoxycarbonyl)-C 1 -C 6 -alkyl, di(C 1 -C 6 -haloalkoxycarbonyl)-C 1 -C 6 -alkyl, di(C 1 -C 6 - alkoxycarbonyl)-C 1 -C 6 -haloalkyl, di(C 1 -C 6 -haloalkoxycarbonyl)-C 1 -C 6 -haloalkyl, di(C 1 -C 6 - alkoxyl)phosphoryl-C 1 -C 6 -alkyl, di(C 1 -C 6 -haloalkoxyl)phosphoryl-C 1 -C 6 -alkyl, di(C 1 -C 6 - alkoxyl)phosphoryl-C 1 -C 6 -haloalkyl, di(C 1 -C 6 -haloalkoxyl)phosphoryl-C 1 -C 6 -haloalkyl, phosphoryl-C 1 -C 6 -alkyl , phosphoryl-C 1 -C 6 -haloalkyl , di[di(C 1 -C 6 -alkoxyl)phosphoryl-)]Ci- C6-alkyl, di[di(C 1 -C 6 -haloalkoxyl)phosphoryl-)]C 1 -C 6 -alkyl, di[di(C 1 -C 6 -alkoxyl)phosphoryl- )]C 1 -C 6 -haloalkyl, di[di(C 1 -C 6 -haloalkoxyl)phosphoryl-)]C 1 -C 6 -haloalkyl, diphosphoryl-Ci-

C6-alkyl , diphosphoryl-C 1 -C 6 -haloalkyl, C 1 -C 6 -alkylthio-C 1 -C 6 -alkyl, C 1 -C 6 -haloalkylthio-Ci- Ce-alkyl, Ci-Ce-alkylthio-Ci-Ce-haloalkyl, Ci-Ce-haloalkylthio-Ci-Ce-haloalkyl, C 1 -C 6 - alkylsulfinly-C 1 -C 6 -alkyl, C 1 -C 6 -haloalkylsulfinly-C 1 -C 6 -alkyl, C 1 -C 6 -alkylsulfinly-C 1 -C 6 - haloalkyl, C 1 -C 6 -haloalkylsulfinly-C 1 -C 6 -haloalkyl, C 1 -C 6 -alkylsulfonyl-C 1 -C 6 -alkyl, C 1 -C 6 - haloalkylsulfonyl-C 1 -C 6 -alkyl, C 1 -C 6 -haloalkylsulfonyl-C 1 -C 6 -haloalkyl, phenyl, 5- or 6- membered heteroaryl, 3- to 6-membered heterocyclyl, ;

wherein hydroxy groups of R 2 are unsubstituted or substituted by R b ;

cyclic groups of R 2 are unsubstituted or substituted by R c ; and

acyclic aliphatic groups of R 2 are unsubstituted or substituted by R d .

R b is Ci-Ce-alkyl, C 1 -C 6 -haloalkyl, C 3 -C 6 -alkenyl, C 3 -C 6 -haloalkenyl, C 3 -C 6 -alkynyl, C 3 -C 6 - haloalkynyl, C 3 -C 6 -cycloalkyl, C 3 -C 6 -halocycloalkyl, C4-C6-cycloalkenyl, C 3 -C 6 - halocycloalkenyl, C 1 -C 6 -alkoxycarbonyl-C 1 -C 6 -alkyl, C 1 -C 6 -haloalkoxycarbonyl-C 1 -C 6 -alkyl, C 1 -C 6 -alkoxycarbonyl-C 1 -C 6 -haloalkyl, C 1 -C 6 -haloalkoxycarbonyl-C 1 -C 6 -haloalkyl, C 1 -C 6 - alkylcarbonyl, CrC 6 -haloalkylcarbonyl, hydroxycarbonyl-C 1 -C 6 -alkyl, hydroxycarbonyl-Ci- C6-haloalkyl, CrC 6 -alkyloxycarbonyl, C 1 -C 6 -haloalkyloxycarbonyl, C 1 -C 6 -alkylthiocarbonyl, C 1 -C 6 -haloalkylthiocarbonyl, C 1 -C 6 -alkylaminocarbonyl, C 1 -C 6 -haloalkylaminocarbonyl, Ci- C6-dialkylaminocarbonyl, C 1 -C 6 -dihaloalkylaminocarbonyl, C 1 -C 6 -alkylsulfonyl, C 1 -C 6 - haloalkylsulfonyl, C 1 -C 6 -alkoxy-C 1 -C 6 -alkyl, C 1 -C 6 -haloalkoxy-C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy-Ci- C6-haloalkyl, CrC 6 -haloalkoxy-C 1 -C 6 -haloalkyl, phenyl-C 1 -C 6 -alkyl, or phenyl-C 1 -C 6 - haloalkyl;

R c is halogen, CN, N0 2 , Ci-Ce-alkyl, C 1 -C 6 -haloalkyl, OH, C 1 -C 6 -alkoxy or C 1 -C 6 - haloalkoxy, C 1 -C 6 -alkylthio, C 1 -C 6 -alkylsulfinyl, or C 1 -C 6 -alkylsulfonyl;

R d is phenyl, 5- or 6-membered heteroaryl, or 3- to 6-membered heterocyclyl;

wherein the substituent R d is unsubstituted or substituted by R e ;

R e is halogen, CN, N0 2 , Ci-Ce-alkyl, C 1 -C 6 -haloalkyl, OH, C 1 -C 6 -alkoxy or C 1 -C 6 - haloalkoxy, C 1 -C 6 -alkylsulfonyl;

A is CR 3 or NR 3A ;

Z is a 5 or 6 membered heteroaryl ring comprising A;

R 3 is halogen, CN, N0 2 , CHO, Ci-Ce-alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkylcarbonyl, C 3 -C 6 - alkenyl, C 3 -C 6 -haloalkenyl, C 2 -C 6 -alkynyl, C 3 -C 6 -haloalkynyl, C 1 -C 6 -alkoxy, C 1 -C 6 - haloalkoxy, C 3 -C 6 -alkenyloxy, C 3 -C 6 -haloalkenyloxy, C 3 -C 6 -alkynyloxy, C 3 -C 6 -ha- loalkynyloxy, C 1 -C 6 -alkoxy-C 1 -C 6 -alkoxy, hydroxycarbonyl, C 1 -C 6 -alkoxycarbonyl, C 1 -C 6 - alkylthio, C 1 -C 6 -haloalkylthio, NH2, (C 1 -C 6 -alkyl)amino, di(C 1 -C 6 -alkyl)amino, (C 1 -C 6 - alkyl)sulfinyl, (C 1 -C 6 -alkyl)sulfonyl, C 3 -C 6 -cycloalkyl, (C 3 -C 6 -cycloalkyl)oxy, or phenyl; wherein the cyclic groups of R 3 are unsubstituted or substituted by substituents R a ;

R 3A is H, Ci-Ce-alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkylcarbonyl, C 3 -C 6 -alkenyl, C 3 -C 6 -haloalkenyl, C 2 -C 6 -alkynyl, C 3 -C 6 -haloalkynyl, C 1 -C 6 -alkoxy, C 1 -C 6 -haloalkoxy, C 3 -C 6 -alkenyloxy, C 3 -C 6 - haloalkenyloxy, C 3 -C 6 -alkynyloxy, C 3 -C 6 -haloalkynyloxy, C 1 -C 6 -alkoxy-C 1 -C 6 -alkoxy, Ci-

C6-alkoxycarbonyl, C 1 -C 6 -alkylthio, C 1 -C 6 -haloalkylthio, NH2, (C 1 -C 6 -alkyl)amino, di(C 1 -C 6 - alkyl)amino, (C 1 -C 6 -alkyl)sulfinyl, (C 1 -C 6 -alkyl)sulfonyl, C 3 -C 6 -cycloalkyl, (C 3 -C 6 - cycloalkyl)oxy, or phenyl;

wherein the cyclic groups of R 3A are unsubstituted or substituted by R a ;

R 4 is halogen, CN, N0 2 , CHO, Ci-Ce-alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkylcarbonyl, C 3 -C 6 - alkenyl, C 3 -C 6 -haloalkenyl, C 3 -C 6 -alkenyl, C 3 -C 6 -haloalkenyl, C 1 -C 6 -alkoxy, C 1 -C 6 - haloalkoxy, C 3 -C 6 -alkenyloxy, C 3 -C 6 -haloalkenyloxy, C 3 -C 6 -alkenyloxy, C 3 -C 6 - haloalkenyloxy, C 1 -C 6 -alkoxy-C 1 -C 6 -alkoxy, hydroxycarbonyl, C 1 -C 6 -alkoxycarbonyl, Ci- C6-alkylthio, C 1 -C 6 -haloalkylthio, NH2, (C 1 -C 6 -alkyl)amino, di(C 1 -C 6 -alkyl)amino, (C 1 -C 6 - alkyl)sulfinyl, (C 1 -C 6 -alkyl)sulfonyl, C 3 -C 6 -cycloalkyl, (C 3 -C 6 -cycloalkyl)oxy, or phenyl; wherein the cyclic groups of R 4 are unsubstituted or substituted by R a ;

R a is halogen, CN, NO2, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkoxy, or C 1 -C 6 -haloalkoxy; m is 0, 1 , 2, or 3;

including agriculturally acceptable salts or derivatives of compounds of formula (I) having an acidic functionality.

The present invention also provides use of the pyrimidine compounds of formula (I) as described herein including agriculturally acceptable salts or derivatives of compounds of formula (I) having an acidic functionality, as herbicide.

The pyrimidine compounds of formula (I) according to the invention can be prepared by standard processes of organic chemistry, e.g. by the following processes:

Process A: The pyrimidines of formula (II) can be obtained by reacting respective pyrimidines of formula (I), R 2 = CH3, (prepared analogous to known procedures like e.g. in WO 2013186229) with base and an electrophile, e.g. a carbonyl compound (III):

The reaction of the pyrimidine (I) with the electrophile (III), with R independent of each other equals hydrogen, alkyl, cycloalkyl, halocycloalkyl, haloalkyl, cycloalkenyl, halocycloalkenyl, alkenyl, haloalkenyl, alkynyl, phenyl, heterocyclyl, heteroaryl or both R form together a carbocycle or a heterocycle, is usually carried out at temperatures of from -100 °C to the boiling point of the reaction mixture, preferably from -80 °C to 20 °C, particularly preferably from -80 °C to -20 °C, in an inert organic solvent in the presence of a base.

Suitable solvents are aliphatic hydrocarbons, such as pentane, hexane, cyclohexane and mixtures of Cs-Ce-alkanes, aromatic hydrocarbons, such as toluene, 0-, m- and p-xylene, ethers, such as diethyl ether, diisopropyl ether, tert-butyl methyl ether (TBME), dioxane, anisole and tetrahydrofuran (THF), and also dimethyl sulfoxide (DMSO), dimethylformamide (DMF) and Ν,Ν-dimethylacetamide (DMAC), particularly diethyl ether, dioxane and THF.

It is also possible to use mixtures of the solvents mentioned.

Suitable bases are, in general, inorganic compounds, such as alkali metal and alkaline earth metal anhydrides, such as lithium hydride (LiH), sodium hydride (NaH), potassium hydride (KH) and calcium hydride (CaH), alkali metal amides, such as lithium hexamethyidisilazide (LHMDS) and lithium diisopropylamide (LDA), organometallic compounds, in particular alkali metal alkyls, such as methyllithium (MeLi), butyllithium (BuLi) and phenyllithium (PhLi), and also alkali metal and alkaline earth metal alkoxides, such as sodium methoxide (NaOChb), sodium ethoxide (NaOC2H5), potassium ethoxide (KOC2H5), potassium tert-butoxide (/BuOK), potassium tert- pentoxide and dimethoxymagnesium, moreover organic bases, e.g. tertiary amines, such as trimethylamine (TMA), triethylamine (TEA), diisopropylethylamine (DIPEA) and N- methylpiperidine, pyridine, substituted pyridines, such as collidine, lutidine and 4- dimethylaminpyridine, and also bicyclic amines. Particular preference is given to NaH, LHMDS and lithium diisopropylamide (LDA).

The bases are generally employed in equimolar amounts; however, they can also be employed in catalytic amounts, in excess or, if appropriate, as solvents.

The starting materials are generally reacted with one another in equimolar amounts. It may be advantageous to employ an excess of base and/or the electrophile, based on the pyrimidine compounds (I).

The elimination of the alcohol of the pyrimidine (II) is usually carried out at temperatures from -100 °C to the boiling point of the reaction mixture, preferably from 0 °C to 120 °C, particularly preferably from 20 °C to 100 °C, in an inert solvent optionally in the presence of an acid.

Suitable solvents are aliphatic hydrocarbons, such as pentane, hexane, cyclohexane and mixtures of Cs-Ce-alkanes, aromatic hydrocarbons, such as toluene, o-, m- and p-xylene, ethers, such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, and also DMSO, DMF and DMAC, particularly preferably toluene and o-xylene.

It is also possible to use mixtures of the solvents mentioned.

Suitable acids are inorganic acids, such as HCI, HBr, sulfuric acid; organic acids p- toluenesulfonic acid, benzene sulfonic acid, pyridinium p-toluol sulfonic acid, methanesulfonic acid, acetic acid; preferably p-toluenesulfonic acid and HCI.

The acids are generally employed in equimolar amounts; however, they can also be employed in catalytic amounts, in excess or, if appropriate, as solvents.

(IV)

The oxidation of the olefin (IV) to the diol (V) is usually carried out at temperatures of from -100 °C to the boiling point of the reaction mixture, preferably from 0 °C to 120 °C, particularly preferably from 20 °C to 100 °C, in an inert solvent.

The reaction may in principle be carried out in substance. However, preference is given to reacting the pyrimidines (IV) with the oxidant in an organic solvent with or without water as co- solvent.

Suitable in principle are all solvents which are capable of dissolving the pyrimidines (IV) and the oxidant at least partly and preferably fully under the reaction conditions.

Suitable solvents are aliphatic hydrocarbons, such as pentane, hexane, cyclohexane and mixtures of Cs-Ce-alkanes, aromatic hydrocarbons, such as toluene, o-, m- and p-xylene, ethers, such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, and also DMSO, DMF and DMAC, particularly preferably TBME, THF It is also possible to use mixtures of the solvents mentioned.

Suitable oxidants are e.g. potassium permanganate, potassium perruthenate, osmium tetroxide and other osmium salts, like potassium osmate. The oxidant can be used in equimolar amounts or in catalytic amounts together with a reoxidant like N-methylmorpholine-N-oxide or potassium hexacyanoferrate in stochiometric amounts or in excess.

Process B:

The halopyrimidines (VI) are known or can be prepared by known procedures (X=CI, Br, I). The boronic acids or esters required for the preparation of pyrimidine compounds of formula (VII) are commercially available, known from literature or can easily prepared analogously to published procedures (e.g. Kamei et al. Tetrahedron Lett. 2014, 55, 4245 - 4247).

The pyrimidine compounds of formula (VII) can obtained by reacting phenyl boronic acids or esters with halides of formula (VI) in which X equals CI, Br, or I in presence of a base and a catalyst in analogy to WO 2014202493.

The reaction may in principle be carried out in substance. However, preference is given to reacting the pyrimidines (VI) with the boronic acid or ester in an organic solvent with or without water as co-solvent.

Suitable in principle are all solvents which are capable of dissolving the pyrimidines (VI) and the boronic acid or ester at least partly and preferably fully under the reaction conditions.

Examples of suitable solvents are aromatic hydrocarbons such as benzene, chlorobenzene, toluene, cresols, o-, m- and p-xylene, ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, as well as dipolar aprotic solvents such as sulfolane,

dimethylsulfoxide, DMF, DMAC, DMI, Ν,Ν'-dimethylpropylene urea (DMPU), DMSO and 1 - methyl-2 pyrrolidinone (NMP).

It is also possible to use mixtures of the solvents mentioned.

Examples of suitable metal-containing bases are inorganic compounds including metal- containing bases such as alkali metal and alkaline earth metal hydroxides, and other metal hydroxides, such as LiOH, NaOH, KOH, Mg(OH) 2 , Ca(OH) 2 and AI(OH) 3 ; alkali metal and alkaline earth metal oxide, and other metal oxides, such as Li 2 O , Na20 , K 2 O, MgO , and CaO, Fe 2 O 3 , Ag20; alkali metal and alkaline earth metal carbonates such as L12CO 3 , Na2CO 3 , K2CO 3 , CS2CO 3 , MgCO 3 , and CaCO 3 , as well as alkali metal hydrogen carbonates (bi carbonates) such as LiHCO 3 , NaHCC>3, KHCO 3 ; alkali metal and alkaline earth metal phosphates such as potassium phosphate (K3PO4), calcium phosphate (Ca3(PO 4 )2); alkali metal and alkaline earth metal acetates such as sodium acetate or potassium acetate.

The term base as used herein also includes mixtures of two or more, preferably two of the above bases. Particular preference is given to the use of one base.

The bases are used preferably from 1 to 10 equivalents based on the pyrimidine (VI), more preferably from 1 .0 to 5.0 equivalents based on the pyrimidine (VI), most preferably from 1 .2 to 2.5 equivalents based on the pyrimidine (VI).

It may be advantageous to add the base offset over a period of time.

The reaction of the pyrimidines (VI) with the phenyl boronic acid or ester is carried out in the presence of a catalyst. Examples of suitable catalysts include e.g., palladium based catalysts like, e.g., Palladium(ll)acetate, tetrakis(triphenylphosphine)palladium(0),

bis(triphenylphosphine)palladium(ll)chloride, or (1 ,1.-bis(diphenylphosphino)ferrocene)- dichloropalladium(ll), and optionally suitable additives such as, e.g., phosphines like, e.g., P(o- tolyl)3, triphenylphosphine, or BINAP (2,2'-Bis(diphenylphospino)-1 ,1'-binaphthyl).

The amount of catalyst is usually 0.01 to 10 mol% (0.0001 to 0.1 equivalents) based on the pyrimidine (VI).

The pyrimidine compounds of formula (VIII) can be obtained by reacting respective pyrimidines of formula (VII) with base and an electrophile, e.g. a carbonyl compound (III): O ( )

The reaction of the pyrimidine (VII) with the electrophile (III), with R independent of each other equals hydrogen, alkyl, cycloalkyl, halocycloalkyl, haloalkyl, cycloalkenyl, halocycloalkenyl, alkenyl, haloalkenyl, alkynyl, phenyl, heterocyclyl, heteroaryl or both R form together a carbocycle or a heterocycle, is usually carried out at temperatures from -100 °C to the boiling point of the reaction mixture, preferably from -80 °C to 20 °C, particularly preferably from -80 °C to -20 °C, in an inert organic solvent in the presence of a base.

Suitable solvents are aliphatic hydrocarbons, such as pentane, hexane, cyclohexane and mixtures of Cs-Ce-alkanes, aromatic hydrocarbons, such as toluene, o-, m- and p-xylene, ethers, such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, and also dimethyl sulfoxide, DMF and DMAC, particularly preferably diethyl ether, dioxane and THF.

It is also possible to use mixtures of the solvents mentioned.

Suitable bases are, in general, inorganic compounds, such as alkali metal and alkaline earth metal anhydrides, such as LiH, NaH, KH and CaH, alkali metal amides, such as LDA, LHMDS, lithium 2,2,6,6-tetramethylpiperidide (LTMP), organometallic compounds, in particular alkali metal alkyls, such as MeLi, BuLi and PhLi, and also alkali metal and alkaline earth metal alkoxides, such as NaOCH 3 , NaOC2H 5 , KOC2H5, tBuOK, potassium tert-pentoxide and dimethoxymagnesium, moreover organic bases, e.g. tertiary amines, such as TMA, TEA, DIPEA and N-methylpiperidine, pyridine, substituted pyridines, such as collidine, lutidine and 4- dimethylaminpyridine, and also bicyclic amines. Particular preference is given to NaH, LTMP and LDA.

The bases are generally employed in equimolar amounts; however, they can also be employed in catalytic amounts, in excess or, if appropriate, as solvents.

The starting materials are generally reacted with one another in equimolar amounts. It may be advantageous to employ an excess of base and/or the electrophile, based on the pyrimidine

(VII).

Process C:

The pyrimidine compounds of formula (IX,) can be obtained by reacting respective

aminoketones of formula (X) with base and amidine (XI):

The reaction of the aminoketone (X) with the amidine (XI) is usually carried out at

temperatures of from -100 °C to the boiling point of the reaction mixture, preferably from 20 °C to the boiling point, particularly preferably from 40 °C to 120 °C, in an inert organic solvent in the presence of a base. The reaction may in principle be carried out in substance. However, preference is given to reacting the aminoketones (X) with the amidine (XI) in an organic solvent.

Suitable in principle are all solvents which are capable of dissolving the aminoketones (X) with the amidine (XI) at least partly and preferably fully under the reaction conditions.

Examples of suitable solvents are aromatic hydrocarbons such as benzene, chlorobenzene, toluene, cresols, o-, m- and p-xylene, halogenated hydrocarbons such as dichloromethane, 1 ,2- dichloroethane, chloroform, carbon tetrachloride and chlorobenzene, ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, esters such as ethyl acetate and butyl acetate; nitriles such as acetonitrile and propionitrile, alcohols such as methanol, ethanol, n-propanol, isopropanol, n-butanol and tert.-butanol, as well as dipolar aprotic solvents such as sulfolane, dimethylsulfoxide, DMF, DMAC, DMIDMI, DMPU, DMSO and NMP.

Preferred solvents are alcohols such as methanol and ethanol.

It is also possible to use mixtures of the solvents mentioned.

Suitable bases are, in general, inorganic compounds, such as alkali metal and alkaline earth metal anhydrides, such as LiH, NaH, KH and CaH, alkali metal amides, such as LDA, LHMDS, lithium 2,2,6,6-tetramethylpiperidide (LTMP), organometallic compounds, in particular alkali metal alkyls, such as MeLi, BuLi and PhLi, and also alkali metal and alkaline earth metal alkoxides, such as NaOCH3, NaOC2H5, KOC2H5, tBuOK, potassium tert-pentoxide and dimethoxymagnesium, moreover organic bases, e.g. tertiary amines, such as TMA, TEA, DIPEA and N-methylpiperidine, pyridine, substituted pyridines, such as collidine, lutidine and 4- dimethylaminpyridine, and also bicyclic amines. Particular preference is given to NaOCH3, NaOC2H5, KOC2H5, potassium tert-butoxide and potassium tert-pentoxide.

The bases are generally employed in equimolar amounts; however, they can also be employed in catalytic amounts, in excess or, if appropriate, as solvents.

The starting materials are generally reacted with one another in equimolar amounts. It may be advantageous to employ an excess of base and/or the amidine (XI), based on the aminoketone

Amidines (XI) known from literature or commercial available.

Preparation of compound (X)

The aminoketones (X) are prepared from the corresponding ketones (XII) with N,N-DMF dimethyl acetal (CAS 4637-24-5). The reaction is usually carried out at temperatures from -100 °C to the boiling point of the reaction mixture, preferably from 20 °C to 160 °C, particularly preferably from 50 °C to 130 °C. The reaction can optionally be catalyzed be an acid.

The reaction may be carried out in substance or in an organic solvent. Suitable in principle are all solvents which are capable of dissolving the ketones (XII) and Ν,Ν-DMF dimethyl acetal (CAS 4637-24-5) at least partly and preferably fully under the reaction conditions.

Examples of suitable solvents are aromatic hydrocarbons such as benzene, chlorobenzene, toluene, cresols, 0-, m- and p-xylene, halogenated hydrocarbons such as dichloromethane, 1 ,2- dichloroethane, chloroform, carbon tetrachloride and chlorobenzene, ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, esters such as ethyl acetate and butyl acetate; nitriles such as acetonitrile and propionitrile, as well as dipolar aprotic solvents such as sulfolane, DMSO, DMF, DMAC, DMIDMI, DMPU, DMSO and NMP; preferably DMF dimethyl acetal is used as solvent.

It is also possible to use mixtures of the solvents mentioned.

Suitable acids are inorganic acids, such as HCI, HBr, sulfuric acid; organic acids p- toluenesulfonic acid, benzene sulfonic acid, pyridinium p-toluol sulfonic acid, methanesulfonic acid, acetic acid; preferably p-toluenesulfonic acid and HCI. Most preferred, no acid is used. The acids are generally employed in equimolar amounts; however, they can also be employed in catalytic amounts, in excess or, if appropriate, as solvents.

(XII)

The ketones (XII) are prepared by reacting Grignard-reagent (XIII) with a carbonyl electrophile (XIV) (e.g. an acid halide (Q = F, CI or Br) or a Weinreb-Amide (Q = N(Me)OMe)). The reaction is usually carried out at temperatures of from -100 °C to the boiling point of the reaction mixture, preferably from -80 °C to 60 °C, particularly preferably from -80 °C to 20 °C, in an inert solvent.

Suitable in principle are all solvents which are capable of dissolving the Grignard-reagent (XIII) and the carbonyl-electrophile (XIV) at least partly and preferably fully under the reaction conditions.

Examples of suitable solvents are aliphatic aromatic hydrocarbons such as benzene, chlorobenzene, toluene, cresols, o-, m- and p-xylene, ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, esters such as ethyl acetate and butyl acetate; nitriles such as acetonitrile and propionitrile, as well as dipolar aprotic solvents such as sulfolane, DMSO, DMF, DMAC, DMIDMI, DMPU, DMSO and NMP. Preferred solvents are ethers such as TBME or THF.

It is also possible to use mixtures of the solvents mentioned.

The Grignard-reagents (XIII) are either commercial available or can be prepared from the corresponding halides by known methods.

The carbonyl electrophiles (XIV) are either commercial available or can be prepared from the corresponding carboxylic acid or carboxylic ester by known methods.

Ketones (XII) can as well be prepared from morpholinonitriles (XV) as described in the literature {European Journal of Organic Chemistry 36, 8083)

The morpholinonitriles (XV) are prepared from morpholinonitriles (XVI) and halides (XVII) in the presence of a base. The reaction is usually carried out at temperatures of from -100 °C to the boiling point of the reaction mixture, preferably from -80 °C to 60 °C, particularly preferably from -50 °C to 20 °C, in an inert organic solvent in the presence of a base.

Suitable in principle are all solvents which are capable of dissolving the morpholinonitriles (XVI) and the halides (XVII) at least partly and preferably fully under the reaction conditions.

Examples of suitable solvents are aromatic hydrocarbons such as benzene, chlorobenzene, toluene, cresols, o-, m- and p-xylene, halogenated hydrocarbons such as dichloromethane, 1 ,2- dichloroethane, chloroform, carbon tetrachloride and chlorobenzene, ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, esters such as ethyl acetate and butyl acetate; nitriles such as acetonitrile and propionitrile, as well as dipolar aprotic solvents such as sulfolane, DMSO, DMF, DMAC, DMIDMI, DMPU, DMSO and NMP. Preferred solvents are dipolar aprotic solvents such as sulfolane, dimethylsulfoxide, DMF, DMAC, DMIDMI, DMPU, DMSO and NMP.

It is also possible to use mixtures of the solvents mentioned.

Suitable bases are, in general, inorganic compounds, such as alkali metal and alkaline earth metal anhydrides, such as LiH, NaH, KH and CaH, alkali metal amides, such as LDA, LHMDS, lithium 2,2,6,6-tetramethylpiperidide (LTMP), organometallic compounds, in particular alkali metal alkyls, such as MeLi, BuLi and PhLi, and also alkali metal and alkaline earth metal alkoxides, such as NaOCH3, NaOC2H5, KOC2H5, tBuOK, potassium tert-pentoxide and dimethoxymagnesium, moreover organic bases, e.g. tertiary amines, such as TMA, TEA, DIPEA and N-methylpiperidine, pyridine, substituted pyridines, such as collidine, lutidine and 4- dimethylaminpyridine, and also bicyclic amines. Particular preference is given to NaH, LTMP and LDAThe bases are generally employed in equimolar amounts; however, they can also be employed in catalytic amounts, in excess or, if appropriate, as solvents.

The starting materials are generally reacted with one another in equimolar amounts. It may be advantageous to employ an excess of base and/or the halide (XVII), based on the

morpholinonitrile (XVI).

Halides (XVII) are commercially available and can easily prepared by methods known to a person skilled in the art.

(XVIII)

(XVI)

Morpholinonitriles (XVI) are prepared from the corresponding aldehydes (XVIII) as described in the literature (WO 2009/013462).

Aldehydes (XVIII) are commercial available. Process D:

Pyrimidine compounds (XIX), with R equals alkyl, haloalkyl, alkoxy, haloalkoxy, X is a leaving group and L is halogen, alkyl, haloalkyl, alkenyl and alkynyl, can be obtained by reacting respective pyrimidine compounds of formula (XX) with base and an electrophile (XXI).

Electrophile (XXI) can be an alkyl-, alkenyl- or alkynyl-halide, e.g. methyl iodide, allyl bromide or propargyl bromide, or a halogenating agent, e.g. C , Br2, 12, NCS (/V-Chlorosuccinimide), NBS (/V-Bromosuccinimide), NIS (/V-lodosuccinimide), NFSI (N-Fluorobenzenesulfonimide), Selectfluor (1-Chloromethyl-4-fluoro-1 ,4-diazoniabicyclo[2.2.2]octane bis(tetrafluoroborate)). The reaction of the pyrimidine (XX) with the electrophile is usually carried out at temperatures of from -100 °C to the boiling point of the reaction mixture, preferably from -80 °C to 80 °C, particularly preferably from -80 °C to 30 °C, in an inert organic solvent in the presence of a base.

Suitable in principle are all solvents which are capable of dissolving the pyrimidine (XX) and the electrophile (XXI) at least partly and preferably fully under the reaction conditions.

Examples of suitable solvents are aromatic hydrocarbons such as benzene, chlorobenzene, toluene, cresols, 0-, m- and p-xylene, ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, nitriles such as acetonitrile and propionitrile, as well as dipolar aprotic solvents such as sulfolane, dimethylsulfoxide, DMF, Ν,Ν-DMAC (DMAC), DMIDMI, DMPU, DMSO and NMP.

Preferred solvents are ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF and dipolar aprotic solvents such as sulfolane, dimethylsulfoxide, DMF, DMAC, DMIDMI, DMPU, DMSO and NMP.

More preferred solvents are ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF.

It is also possible to use mixtures of the solvents mentioned.

Suitable bases are, in general, inorganic compounds, such as alkali metal and alkaline earth metal anhydrides, such as LiH, NaH, KH and CaH, alkali metal amides, such as LDA, LHMDS, lithium 2,2,6,6-tetramethylpiperidide (LTMP), organometallic compounds, in particular alkali metal alkyls, such as MeLi, BuLi and PhLi, and also alkali metal and alkaline earth metal alkoxides, such as NaOCH3, NaOC2H5, KOC2H5, tBuOK, potassium tert-pentoxide and dimethoxymagnesium, moreover organic bases, e.g. tertiary amines, such as TMA, TEA, DIPEA and N-methylpiperidine, pyridine, substituted pyridines, such as collidine, lutidine and 4- dimethylaminpyridine, and also bicyclic amines. Particular preference is given to NaH, LTMP and LDA.

The bases are generally employed in equimolar amounts; however, they can also be employed in catalytic amounts, in excess or, if appropriate, as solvents.

The starting materials are generally reacted with one another in equimolar amounts. It may be advantageous to employ an excess of base and/or the electrophile (XXI), based on the pyrimidine (XX). The pyrimidine compounds of formula (XX) can be obtained by reacting respective pyrimidines of formula (I), R 2 = CH3, (prepared analogous to known procedures like e.g. in

WO 2013186229) with base and an electrophile (XXII), e.g. a dialkylcarbonate (X = R = alkoxy), an alkyl chloroformiate (X = halogene, R = alkoxy) or an acid halide (X = halogene, R = alkyl or haloalkyl) :

(XX)

The reaction of the pyrimidine (I) with the electrophile (XXII) is usually carried out at temperatures of from -100 °C to the boiling point of the reaction mixture, preferably from -80 °C to 80 °C, particularly preferably from -80 °C to 30 °C, in an inert organic solvent in the presence of a base.

Suitable in principle are all solvents which are capable of dissolving the pyrimidine (I) and the electrophile (XXII) at least partly and preferably fully under the reaction conditions.

Examples of suitable solvents are aromatic hydrocarbons such as benzene, chlorobenzene, toluene, cresols, 0-, m- and p-xylene, ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, as well as dipolar aprotic solvents such as sulfolane, DMSO, DMF, DMAC, DMIDMI, DMPU, DMSO and NMP.

It is also possible to use mixtures of the solvents mentioned.

Suitable bases are, in general, inorganic compounds, such as alkali metal and alkaline earth metal anhydrides, such as LiH, NaH, KH and CaH, alkali metal amides, such as LDA, LHMDS, lithium 2,2,6,6-tetramethylpiperidide (LTMP), organometallic compounds, in particular alkali metal alkyls, such as MeLi, BuLi and PhLi, and also alkali metal and alkaline earth metal alkoxides, such as NaOCH3, NaOC2H5, KOC2H5, tBuOK, potassium tert-pentoxide and dimethoxymagnesium, moreover organic bases, e.g. tertiary amines, such as TMA, TEA, DIPEA and N-methylpiperidine, pyridine, substituted pyridines, such as collidine, lutidine and 4- dimethylaminpyridine, and also bicyclic amines. Particular preference is given to NaH, LTMP and LDAThe bases are generally employed in equimolar amounts; however, they can also be employed in catalytic amounts, in excess or, if appropriate, as solvents.

The starting materials are generally reacted with one another in equimolar amounts. It may be advantageous to employ an excess of base and/or the electrophile (XXII), based on the pyrimidine (I).

Process E:

The pyrimidines of formula (XXIII) can be obtained by reacting respective pyrimidines of formula (XXIV) with boronic acids/esters of formula (XXV):

The reaction of pyrimidines (XXIV) with boronic acids/esters (XXV) is usually carried out from 0 °C to the boiling point of the reaction mixture, preferably from 15 °C to 110 °C, particularly preferably from 40 °C to 100 °C, in an inert organic solvent in the presence of a base and a catalyst.

The reaction may in principle be carried out in substance. However, preference is given to reacting the pyrimidines (XXIV) with the boronic acids/esters (XXV) in an organic solvent with or without water as co-solvent.

Suitable in principle are all solvents which are capable of dissolving the pyrimidines (XXIV) and the boronic acids (XXV) at least partly and preferably fully under the reaction conditions.

Examples of suitable solvents are aromatic hydrocarbons such as benzene, chlorobenzene, toluene, cresols, o-, m- and p-xylene, ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, as well as dipolar aprotic solvents such as sulfolane,

dimethylsulfoxide, DMF, DMAC, DMIDMI, DMPU, DMSO and NMP.

Preferred solvents are ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF and dipolar aprotic solvents such as sulfolane, DMSO, DMF, Ν,Ν-DMAC (DMAC), DMIDMI, DMPU, DMSO and NMP.

More preferred solvents are ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF.

It is also possible to use mixtures of the solvents mentioned.

Examples of suitable metal-containing bases are inorganic compounds including metal- containing bases such as alkali metal and alkaline earth metal hydroxides, and other metal hydroxides, such as LiOH, NaOH, KOH, Mg(OH) 2 , Ca(OH) 2 and AI(OH) 3 ; alkali metal and alkaline earth metal oxide, and other metal oxides, such as Li 2 O , Na20 , K 2 O, MgO , and CaO, Fe 2 O 3 , Ag20; alkali metal and alkaline earth metal carbonates such as L12CO 3 , Na2CO 3 , K2CO 3 , CS2CO 3 , MgCO 3 , and CaCO 3 , as well as alkali metal hydrogen carbonates (bi carbonates) such as LiHCO 3 , NaHCO 3 , KHCO 3 ; alkali metal and alkaline earth metal phosphates such as potassium phosphate (K3PO4), calcium phosphate (Ca3(PO 4 )2); alkali metal and alkaline earth metal acetates such as sodium acetate or potassium acetate.

The term base as used herein also includes mixtures of two or more, preferably two of the above bases. Particular preference is given to the use of one base.

The bases are used preferably from 1 to 10 equivalents based on the pyrimidine (XXIV), more preferably from 1.0 to 5.0 equivalents based on the pyrimidine (XXIV), most preferably from 1.2 to 2.5 equivalents based on the pyrimidine (XXIV).

It may be advantageous to add the base offset over a period of time.

The reaction of the pyrimidines (XXIV) with the boronic acids/esters (XXV) is carried out in the presence of a catalyst. Examples of suitable catalysts include e.g., palladium based catalysts like, e.g., palladium(ll)acetate, tetrakis(triphenylphosphine)- palladium(O),

bis(triphenylphosphine)palladium(ll)chloride or (1 ,1.-bis(diphenylphosphino)- ferrocene)- dichloropalladium(ll), and optionally suitable additives such as, e.g., phosphines like, e.g., P(o- tolyl)3, triphenylphosphine or BINAP (2,2'-Bis(diphenylphospino)-1 ,1'-binaphthyl).

The amount of catalyst is usually 0.01 to 20 mol % (0.0001 to 0.2 equivalents) based on the pyrimidine (XXIV).

The halopyrimidines XXIV are known from the literature (e.g. WO 2011154327), are commercially available or can be prepared by known procedures. The boronic acids/esters XXV required for the preparation of pyrimidines of formula (XVII) are commercially available, known from literature or can easily prepared analogously to published procedures (e.g. Kamei et al. Tetrahedron Lett. 2014, 55, 4245 - 4247).

The pyrimidines of formula (XXVI) can be obtained by reacting respective pyrimidines of formula (XXIII) with a reducing agent such as LAH or DIBAIH.

The reduction of pyrimidines (XXIII) is usually carried out from - 80 °C to the boiling point of the reaction mixture, preferably from -20 °C to 60 °C, particularly preferably from 0 °C to 25 °C, in an inert organic solvent.

Suitable solvents are aliphatic hydrocarbons, such as pentane, hexane, cyclohexane and mixtures of Cs-Ce-alkanes, aromatic hydrocarbons, such as toluene, o-, m- and p-xylene, ethers, such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, and also DMSO, DMF and DMAC, particularly preferably diethyl ether, dioxane and THF.

It is also possible to use mixtures of the solvents mentioned.

Examples of reducing agents for pyrimidines (XXIII) include LAH, DIBALH, LiBH 4 or Lithium triethylborohydride.

Preferred agents include LAH and DIBALH.

The hydride-source is used preferably from 1 to 10 equivalents based on the pyrimidine (XXIII), more preferably from 1.0 to 5.0 equivalents based on the pyrimidine (XXIII), most preferably from 1.2 to 2.5 equivalents based on the pyrimidine (XXIII).

Process F:

The pyrimidines of formula (XXVII) can be obtained by reacting respective pyrimidines of formula (XXIII) with a metal organic species like a Grignard reagent (R'MgX, X = CI, Br, I; R' = alkyl, haloalkyl, alkenyl, alkynyl, cycloalkyl, phenyl, heterocyclyl, or heteroaryl).

The reaction of pyrimidines (XXIII) with a metal organic species is usually carried out from - 80 °C to the boiling point of the reaction mixture, preferably from -20 °C to 60 °C, particularly preferably from -20 °C to 25 °C, in an inert organic solvent.

Suitable solvents are aliphatic hydrocarbons, such as pentane, hexane, cyclohexane and mixtures of Cs-Ce-alkanes, aromatic hydrocarbons, such as toluene, o-, m- and p-xylene, ethers, such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, and also DMSO, DMF and DMAC, particularly preferably diethyl ether, dioxane and THF.

It is also possible to use mixtures of the solvents mentioned.

Examples of metal organic species for the synthesis of (XXVII) Grignard reagents like R'MgCI, R'MgBr or R'Mgl, lithium organic species, aluminum organic species like R 3AI, R 2AIX and R'AIX2, titanium organic species like R' 4 Ti, R'aTiX, R'2TiX2 and RTiX3, Preferred agents include Grignard reagents and lithium organic species.

The metal organic species is used preferably from 2 to 10 equivalents based on the pyrimidine (XXIII), more preferably from 2.0 to 5.0 equivalents based on the pyrimidine (XXIII), most preferably from 2.0 to 3.0 equivalents based on the pyrimidine (XXIII).

Process G:

The pyrimidines of formula (XXVIII) can be obtained by reacting respective pyrimidines of formula (XXIX) with a metal organic species like a Grignard reagent (R'MgX, X = CI, Br, I; R' = alkyl, haloalkyl, alkenyl, alkynyl, cycloalkyl, phenyl, heterocyclyl or heteroaryl).

(XXIX) (xxviii)

The reaction of pyrimidines (XXIX) with a metal organic species is usually carried out from - 80 °C to the boiling point of the reaction mixture, preferably from -20 °C to 60 °C, particularly preferably from -20 °C to 25 °C in an inert organic solvent.

Suitable solvents are aliphatic hydrocarbons, such as pentane, hexane, cyclohexane and mixtures of Cs-Ce-alkanes, aromatic hydrocarbons, such as toluene, o-, m- and p-xylene, ethers, such as diethyl ether, diisopropyl ether, tert-butyl methyl ether, dioxane, anisole and

tetrahydrofuran, and also dimethyl sulfoxide, DMF and DMAC, particularly preferably diethyl ether, dioxane and tetrahydrofuran.

It is also possible to use mixtures of the solvents mentioned.

Examples of metal organic species for the synthesis of pyrimidines (XXVIII) are Grignard reagents like R'MgCI, R'MgBr or R'Mgl, lithium organic species, aluminum organic species like R'3AI, R' 2 AIX and R'AIX 2 , titanium organic species like R' 4 Ti, R' 3 TiX, R' 2 TiX2 and RTiX 3 ,

Preferred agents include Grignard reagents and lithium organic species.

The metal organic species is used preferably from 2 to 10 equivalents based on the pyrimidine (XXIX), more preferably from 2.0 to 5.0 equivalents based on the pyrimidine (XXIX), most preferably from 2.0 to 3.0 equivalents based on the pyrimidine (XXIX).

Process H:

The pyrimidines of formula (XXIX) can be obtained by oxidizing respective pyrimidines of formula (XXVI).

(XXIX)

(xxvi)

The oxidation of pyrimidines (XXVI) is usually carried out from - 80 °C to the boiling point of the reaction mixture, preferably from -20 °C to 100 °C, particularly preferably from 0 °C to 75 °C, in an inert organic solvent.

The reaction may in principle be carried out in substance. However, preference is given to reacting the pyrimidines (XXVI) in an organic solvent.

Suitable in principle are all solvents which are capable of dissolving the pyrimidines (XXVI) at least partly and preferably fully under the reaction conditions. Examples of suitable solvents are aromatic hydrocarbons such as benzene, chlorobenzene, toluene, cresols, o-, m- and p-xylene, halogenated hydrocarbons such as CH2CI2, CHCI3, CCH2CICH2CI or CCI 4 , ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, as well as dipolar aprotic solvents such as sulfolane, dimethylsulfoxide, DMF, N,N- DMAC (DMAC), DMIDMI, DMPU, DMSO and NMP.

Preferred solvents are halogenated hydrocarbons such as CH2CI2, CHCI3, CCH2CICH2CI or CCU, and dipolar aprotic solvents such as sulfolane, dimethylsulfoxide, DMF, DMAC, DMIDMI, Ν,Ν'-dimethyhpropylene urea (DMPU), DMSO and NMP.

More preferred solvents halogenated hydrocarbons such as CH2CI2, CHCI3, CCH2CICH2CI or ecu.

It is also possible to use mixtures of the solvents mentioned.

Examples of oxidizing agents for the synthesis of pyrimidines (XXIX) are metal oxides such as MnO 2 , KMnO 4 , CrO 3 or PCC, and non-metal oxides such as NaCIO, NalO 4 or pyridine/SO 3 - complex. In addition methods like the Swern oxidation or the TEMPO oxidation known to a person skilled in the art can be used to obtain pyridines of formula (XXIX).

Preferred agents include Μηθ2, KMnO 4 and PCC, more preferred is Mn02.

The oxidizing agent is used preferably from 1 to 50 equivalents based on the pyrimidine (XXVI), more preferably from 1.0 to 20.0 equivalents based on the pyrimidine (XXVI), most preferably from 1.0 to 10.0 equivalents based on the pyrimidine (XXVI).

Process I:

The pyrimidines of formula (XXX; Q = cycloalkyl, halocycloalkyl, alkyl, haloalkyl, alkenyl, alkynyl, phenyl, heteroaryl, heterocyclyl, alkylidenyl or halo alkylidenyl and R' = alkyl, haloalkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, alkoxycarbonylalkyl) can be obtained by reacting respective pyrimidines of formula (XXXI) with base and an electrophile.

Electrophiles can be an alkyl-, alkenyl- or alkynyl-halide, e.g. methyl iodide, allyl bromide propargyl bromide, ethyl iodide, propyl bromide, or ethyl 2-bromoacetate.

The reaction of the pyrimidine (XXXI) with the electrophile is usually carried out at

temperatures of from -100 °C to the boiling point of the reaction mixture, preferably from -20 °C to 100 °C, particularly preferably from -0 °C to 30 °C, in an inert organic solvent in the presence of a base.

Suitable in principle are all solvents which are capable of dissolving the pyrimidine (XXXI) and the electrophile at least partly and preferably fully under the reaction conditions.

Examples of suitable solvents are aromatic hydrocarbons such as benzene, chlorobenzene, toluene, cresols, 0-, m- and p-xylene, ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, nitriles such as acetonitrile and propionitrile, as well as dipolar aprotic solvents such as sulfolane, dimethylsulfoxide, DMF, Ν,Ν-DMAC (DMAC), DMIDMI, DMPU, DMSO and NMP. Preferred solvents are ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF and dipolar aprotic solvents such as sulfolane, dimethylsulfoxide, DMF, N,N-DMAC (DMAC), DMIDMI, DMPU, DMSO and NMP.

More preferred solvents are dipolar aprotic solvents such as dimethylsulfoxide, DMF, and NMP.

It is also possible to use mixtures of the solvents mentioned.

Suitable bases are, in general, inorganic compounds, such as alkali metal and alkaline earth metal anhydrides, such as lithium hydride, sodium hydride, potassium hydride and calcium hydride, alkali metal azides, such as lithium hexamethyidisilazide, organometallic compounds, in particular alkali metal alkyls, such as methyl lithium, butyllithium and phenyllithium, and also alkali metal and alkaline earth metal alkoxides, such as sodium methoxide, sodium ethoxide, potassium ethoxide, potassium tert-butoxide, potassium tert-pentoxide and

dimethoxymagnesium, moreover organic bases, e.g. tertiary amines, such as trimethylamine, triethylamine, diisopropylethylamine and N-methylpiperidine, pyridine, substituted pyridines, such as collidine, lutidine and 4-dimethylaminpyridine, and also bicyclic amines. Particular preference is given to sodium hydride, lithium hexamethyidisilazide and lithium

diisopropylamide.

The bases are generally employed in equimolar amounts; however, they can also be employed in catalytic amounts, in excess or, if appropriate, as solvents.

The starting materials are generally reacted with one another in equimolar amounts. It may be advantageous to employ an excess of base and/or the electrophile, based on the pyrimidine (XXXI).

Process J:

The pyrimidine compounds of formula (I) can in addition be obtained by reacting respective pyrimidine boronic acid esters of formula (XXXII) with halides of formula (XXXIII) in which X equals CI, Br, or I:

The reaction of the pyrimidine (XXXII) with halides of formula (XXXIII) is usually carried out from 0 °C to the boiling point of the reaction mixture, preferably from 15 °C to 110 °C, particularly preferably from 40 °C to 100 °C, in an inert organic solvent in the presence of a base and a catalyst.

The reaction may in principle be carried out in substance. However, preference is given to reacting the pyrimidines (XXXII) with halides of formula (XXXIII) in an organic solvent with or without water as co-solvent.

Suitable in principle are all solvents which are capable of dissolving the pyrimidines (XXXII) with halides of formula (XXXIII) at least partly and preferably fully under the reaction conditions.

Examples of suitable solvents are aromatic hydrocarbons such as benzene, chlorobenzene, toluene, cresols, o-, m- and p-xylene, ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, as well as dipolar aprotic solvents such as sulfolane,

dimethylsulfoxide, DMF, Ν,Ν-DMAC (DMAC), DMIDMI, DMPU, DMSO and NMP. Preferred solvents are ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF and dipolar aprotic solvents such as sulfolane, dimethylsulfoxide, DMF, N,N-DMAC (DMAC), DM I DM I, Ν,Ν'-dimethyhpropylene urea (DMPU), DMSO and NMP.

More preferred solvents are ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF.

It is also possible to use mixtures of the solvents mentioned.

Examples of suitable metal-containing bases are inorganic compounds including metal- containing bases such as alkali metal and alkaline earth metal hydroxides, and other metal hydroxides, such as LiOH, NaOH, KOH, Mg(OH) 2 , Ca(OH) 2 and AI(OH) 3 ; alkali metal and alkaline earth metal oxide, and other metal oxides, such as Li 2 O , Na 2 O , K 2 O, MgO , and CaO, Fe 2 O 3 , Ag20; alkali metal and alkaline earth metal carbonates such as Li 2 CO 3 , Na2CO 3 , K2CO 3 , CS2CO 3 , MgCO 3 , and CaCO 3 , as well as alkali metal hydrogen carbonates (bi carbonates) such as LiHCO 3 , NaHCC>3, KHCO 3 ; alkali metal and alkaline earth metal phosphates such as potassium phosphate (K3PO4), calcium phosphate (Ca3(PO 4 )2).

The term base as used herein also includes mixtures of two or more, preferably two of the above bases. Particular preference is given to the use of one base.

The bases are used preferably from 1 to 10 equivalents based on the pyrimidine (XXXII), more preferably from 1.0 to 5.0 equivalents based on the pyrimidine (XXXII), most preferably from 1.2 to 2.5 equivalents based on the pyrimidine (XXXII).

It may be advantageous to add the base offset over a period of time.

The reaction of the pyrimidines (XXXII) with halides of formula (XXXIII) is carried out in the presence of a catalyst. Examples of suitable catalysts include e.g., palladium based catalysts like, e.g., Palladium(ll)acetate, tetrakis(triphenylphosphine)palladium(0),

bis(triphenylphosphine)palladium(ll)chloride or (1 ,1.-bis(diphenylphosphino)ferrocene)- dichloropalladium(ll), and optionally suitable additives such as, e.g., phosphines like, e.g., P(o- tolyl)3, triphenylphosphine or BINAP (2,2'-Bis(diphenylphospino)-1 ,1'-binaphthyl).

The amount of catalyst is usually 0.01 to 20 mol% (0.0001 to 0.2 equivalents) based on the pyrimidine (XXXII).

The halides (XXXIII) required for the preparation of pyrimidine compounds of formula (I) are known from the literature or are commercially available.

The pyrimidines of formula (XXXII) can be obtained by reacting the respective pyrimidines (XXXIV) with Bis(pinacolato)diboron XXXV.

The reaction of the pyrimidine (XXXIV) with Bis(pinacolato)diboron XXXV is usually carried out from 0 °C to the boiling point of the reaction mixture, preferably from 15 °C to 110 °C, particularly preferably from 40 °C to 100 °C, in an inert organic solvent in the presence of a base and a catalyst.

The reaction may in principle be carried out in substance. However, preference is given to reacting the pyrimidines (XXXIV) with Bis(pinacolato)diboron XXXV in an organic solvent with or without water as co-solvent. Suitable in principle are all solvents which are capable of dissolving the pyrimidines (XXXIV) with Bis(pinacolato)diboron XXXV at least partly and preferably fully under the reaction conditions.

Examples of suitable solvents are aromatic hydrocarbons such as benzene, chlorobenzene, toluene, cresols, o-, m- and p-xylene, ethers such as diethyl ether, diisopropyl ether, TBME, dioxane, anisole and THF, as well as dipolar aprotic solvents such as sulfolane,

dimethylsulfoxide, DMF, DMAC, DMIDMI, DMPU, DMSO and NMP.

It is also possible to use mixtures of the solvents mentioned.

Examples of suitable metal-containing bases are inorganic compounds including metal- containing bases such as alkali metal and alkaline earth metal hydroxides, and other metal hydroxides, such as LiOH, NaOH, KOH, Mg(OH) 2 , Ca(OH) 2 and AI(OH) 3 ; alkali metal and alkaline earth metal oxide, and other metal oxides, such as Li 2 O , Na20 , K 2 O, MgO , and CaO, Fe 2 O 3 , Ag20; alkali metal and alkaline earth metal carbonates such as L12CO 3 , Na2CO 3 , K2CO 3 , CS2CO 3 , MgCO 3 , and CaCO 3 , as well as alkali metal hydrogen carbonates (bi carbonates) such as UHCO 3 , NaHCO 3 , KHCO 3 ; alkali metal and alkaline earth metal phosphates such as potassium phosphate (K3PO4), calcium phosphate (Ca3(PO 4 )2); alkali metal and alkaline earth metal acetates such as sodium acetate or potassium acetate.

The term base as used herein also includes mixtures of two or more, preferably two of the above bases. Particular preference is given to the use of one base.

The bases are used preferably from 1 to 10 equivalents based on the pyrimidine (XXXIV), more preferably from 1.0 to 5.0 equivalents based on the pyrimidine (XXXIV), most preferably from 1.2 to 2.5 equivalents based on the pyrimidine (XXXIV).

It may be advantageous to add the base offset over a period of time.

The reaction of the pyrimidines (XXXIV) with Bis(pinacolato)diboron XXXV is carried out in the presence of a catalyst. Examples of suitable catalysts include e.g., palladium based catalysts like, e.g., Palladium(ll)acetate, tetrakis(triphenylphosphine)palladium(0),

bis(triphenylphosphine)palladium(ll)chloride or (1 ,1.-bis(diphenylphosphino)ferrocene)- dichloropalladium(ll), and optionally suitable additives such as, e.g., phosphines like, e.g., P(o- tolyl)3, triphenylphosphine or BINAP (2,2'-Bis(diphenylphospino)-1 ,1'-binaphthyl).

The amount of catalyst is usually 0.01 to 20 mol% (0.0001 to 0.2 equivalents) based on the pyrimidine (XXXIV).

The halides (XXXIV) required for the preparation of pyrimidine compounds of formula (XXXII) are known from the literature or are commercially available.

The end of the reactions can easily be determined by the skilled worker by means of routine methods.

The reaction mixtures are worked up in a customary manner, e.g. by mixing with water, separation of the phases and, if appropriate, chromatographic purification of the crude product.

Some of the intermediates and end products are obtained in the form of viscous oils, which can be purified or freed from volatile components under reduced pressure and at moderately elevated temperature.

If the intermediates and the end products are obtained as solid, purification can also be carried out by recrystallization or digestion. The present invention also provides agrochemical compositions comprising at least one pyrimidine compounds of formula (I) and auxiliaries customary for formulating crop protection agents.

The present invention furthermore provides a method for controlling unwanted vegetation where a herbicidal effective amount of at least one pyrimidine compounds of formula (I) is allowed to act on plants, their seeds and/or their habitat. Application can be done before, during and/or after, preferably during and/or after, the emergence of the undesirable plants.

Further embodiments of the present invention are evident from the claims, the description and the examples. It is to be understood that the features mentioned above and still to be illustrated below of the subject matter of the invention can be applied not only in the combination given in each particular case but also in other combinations, without leaving the scope of the invention. As used herein, the terms "controlling" and "combating" are synonyms.

As used herein, the terms "undesirable vegetation" and "harmful plants" are synonyms.

If the pyrimidine compounds of formula (I) as described herein are capable of forming geometrical isomers, e.g. E/Z isomers, it is possible to use both, the pure isomers and mixtures thereof, in the compositions according to the invention.

If the pyrimidine compounds of formula (I) as described herein have one or more centres of chirality and, as a consequence, are present as enantiomers or diastereomers, it is possible to use both, the pure enantiomers and diastereomers and their mixtures, in the compositions according to the invention.

If the pyrimidine compounds of formula (I) as described herein have ionisable functional groups, preferably an acidic functionality, more preferably a carboxylic group or a sulphonic group, they can also be employed in the form of their agriculturally acceptable salts. Suitable are, in general, the salts of those cations and the acid addition salts of those acids whose cations and anions, respectively, have no adverse effect on the activity of the active

compounds.

Preferred cations are the ions of the alkali metals, preferably of lithium, sodium and potassium, of the alkaline earth metals, preferably of calcium and magnesium, and of the transition metals, preferably of manganese, copper, zinc and iron, further ammonium and substituted ammonium in which one to four H atoms are replaced by Ci-C 4 -alkyl, HO-Ci-C 4 -alkyl, Ci-C 4 -alkoxy-Ci-C 4 - alkyl, HO-Ci-C 4 -alkoxy-Ci-C 4 -alkyl, phenyl or benzyl, preferably ammonium, methyl-ammonium, isopropylammonium, dimethylammonium, diisopropylammonium, trimethylammonium, heptylammonium, dodecylammonium, tetradecylammonium, tetramethylammonium,

tetraethylamm-onium, tetrabutylammonium, 2-hydroxyethylammonium (olamine salt), 2-(2- hydroxyeth-1-oxy)eth-1-ylammonium (diglycolamine salt), di(2-hydroxyeth-1-yl)ammonium (diol- amine salt), tris(2-HO-ethyl)ammonium (trolamine salt), tris(2-hydroxypropyl)ammonium, ben- zyltrimethylammonium, benzyltriethylammonium, Ν,Ν,Ν-trimethylethanolammonium (choline salt), furthermore phosphon-ium ions, sulfonium ions, preferably tri(Ci-C 4 -alkyl)sulfonium, such as trimethylsulfonium, and sulfoxonium ions, preferably tri(Ci-C 4 -alkyl)sulfoxonium, and finally the salts of polybasic amines such as N,N-bis-(3-aminopropyl)methylamine and

diethylenetriamine.

Anions of useful acid addition salts are primarily chloride, bromide, fluoride, iodide, hydrogen- sulfate, methylsulfate, sulfate, dihydrogenphosphate, hydrogenphosphate, nitrate, bicarbonate, carbonate, hexafluorosilicate, hexafluorophosphate, benzoate and also the anions of C1-C4- alkanoic acids, preferably formate, acetate, propionate and butyrate.

Pyrimidine compounds of formula (I) as described herein having an acidic functionality, preferably a carboxylic group or a sulphonic group, can be employed, if applicable, in the form of the acid, in the form of an agriculturally suitable salt with the cations as defined above or else in the form of an agriculturally acceptable derivative, e.g. as amides, such as mono- and di-Ci- C6-alkylamides or arylamides, as esters, e.g. as allyl esters, propargyl esters, Ci-Cio-alkyl esters, alkoxyalkyl esters, tefuryl ((tetrahydrofuran-2-yl)methyl) esters and also as thioesters, e.g. as Ci-Cio-alkylthio esters. Preferred mono- and di-C 1 -C 6 -alkylamides are the CH3 and the dimethylamides. Preferred arylamides are, e.g., the anilides and the 2-chloroanilides. Preferred alkyl esters are, e.g., the methyl, ethyl, propyl, isopropyl, butyl, isobutyl, pentyl, mexyl

(1-methylhexyl), meptyl (1-methylheptyl), heptyl, octyl or isooctyl (2-ethylhexyl) esters. Preferred Ci-C4-alkoxy-Ci-C4-alkyl esters are the straight-chain or branched Ci-C 4 -alkoxy ethyl esters, e.g. the 2-methoxyethyl, 2-ethoxyethyl, 2-butoxyethyl (butotyl), 2-butoxypropyl or 3-butoxypropyl ester. An example of a straight-chain or branched Ci-Cio-alkylthio ester is the ethylthio ester. The organic moieties mentioned in the definition of the variables R 1 , R 2 , A, Z, R 3 , R 3A , and R 4 , are - like the term halogen - collective terms for individual enumerations of the individual group members. The term halogen denotes in each case F, CI, Br, or I. All hydrocarbon chains, e.g. all alkyl, alkenyl, alkynyl, alkoxy chains can be straight-chain or branched, the prefix C n -C m denoting in each case the possible number of carbon atoms in the group.

Examples of such meanings are:

- Ci-C 4 -alkyl: e.g. CH 3 , C2H5, n-propyl, CH(CH 3 ) 2 , n-butyl, CH(CH 3 )-C 2 H5, CH2-CH(CH 3 )2, and C(CH 3 ) 3 ;

C 1 -C 6 -alkyl: Ci-C 4 -alkyl as mentioned above, and also, e.g., n-pentyl, 1-methylbutyl, 2- methylbutyl, 3-methylbutyl, 2,2-dimethylpropyl, 1-ethylpropyl, n-hexyl, 1 ,1-dimethylpropyl, 1 ,2- dimethylpropyl, 1-methylpentyl, 2-methylpentyl, 3-methylpentyl, 4-methylpentyl, 1 ,1-di- methylbutyl, 1 ,2-dimethylbutyl, 1 ,3-dimethylbutyl, 2,2-dimethylbutyl, 2,3-dimethylbutyl, 3,3- dimethylbutyl, 1-ethylbutyl, 2-ethylbutyl, 1 ,1 ,2-trimethylpropyl, 1 ,2,2-trimethylpropyl, 1 -ethyl-1- methylpropyl or 1-ethyl-2-methylpropyl, preferably methyl, ethyl, n-propyl, 1-methylethyl, n- butyl, 1 ,1-dimethylethyl, n-pentyl, or n-hexyl;

Ci-C 4 -haloalkyl: Ci-C 4 -alkyl as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, e.g., chloromethyl, dichloromethyl, trichloromethyl, fluoromethyl, difluoromethyl, trifluoromethyl, chlorofluoromethyl, dichlorofluoromethyl, chlorodifluoromethyl, bromomethyl, iodomethyl, 2-fluoroethyl, 2-chloroethyl, 2-bromoethyl, 2- iodoethyl, 2,2-difluoroethyl, 2,2,2-trifluoroethyl, 2-chloro-2-fluoroethyl, 2-chloro-2,2-difluoroethyl, 2,2-dichloro-2-fluoroethyl, 2,2,2-trichloroethyl, pentafluoroethyl, 2-fluoropropyl, 3-fluoropropyl, 2,2-difluoropropyl, 2,3-difluoropropyl, 2-chloropropyl, 3-chloropropyl, 2,3-dichloropropyl, 2- bromopropyl, 3-bromopropyl, 3,3,3-trifluoropropyl, 3,3,3-trichloropropyl, 2,2,3,3,3- pentafluoropropyl, heptafluoro-propyl, 1-(fluoromethyl)-2-fluoroethyl, 1-(chloromethyl)-2- chloroethyl, 1-(bromomethyl)-2-bromo-ethyl, 4-fluorobutyl, 4-chlorobutyl, 4-bromobutyl, nonafluorobutyl, 1 ,1 ,2,2,-tetrafluoroethyl, and 1-trifluoromethyl-1 ,2,2,2-tetrafluoroethyl;

C 1 -C 6 -haloalkyl: Ci-C 4 -haloalkyl as mentioned above, and also, e.g., 5-fluoropentyl, 5- chloropentyl, 5-bromopentyl, 5-iodopentyl, undecafluoropentyl, 6-fluorohexyl, 6-chlorohexyl, 6-bromohexyl, 6-iodohexyl, and dodecafluorohexyl; C 3 -C 6 -cycloalkyl: monocyclic saturated hydrocarbons having 3 to 6 ring members, such as cyclopropyl, cyclobutyl, cyclopentyl, and cyclohexyl;

C 3 -C 6 -alkenyl: e.g. 1-propenyl, 2-propenyl, 1-methylethenyl, 1-butenyl, 2-butenyl, 3- butenyl, 1 -methyl- 1-propenyl, 2-methyl-1-propenyl, 1-methyl-2-propenyl, 2-methyl-2-propenyl, 1- pentenyl, 2-pentenyl, 3-pentenyl, 4-pentenyl, 1-methyl-1-butenyl, 2-methyl-1-butenyl, 3-methyl-

1- butenyl, 1-methyl-2-butenyl, 2-methyl-2-butenyl, 3-methyl-2-butenyl, 1-methyl-3-butenyl,

2- methyl-3-butenyl, 3-methyl-3-butenyl, 1 ,1-dimethyl-2-propenyl, 1 ,2-dimethyl-1-propenyl, 1 ,2- dimethyl-2-propenyl, 1-ethyl-1-propenyl, 1-ethyl-2-propenyl, 1-hexenyl, 2-hexenyl, 3-hexenyl, 4- hexenyl, 5-hexenyl, 1-methyl-1 -pentenyl, 2-methyl-1 -pentenyl, 3-methyl-1 -pentenyl, 4-methyl-1- pentenyl, 1-methyl-2-pentenyl, 2-methyl-2-pentenyl, 3-methyl-2-pentenyl, 4-methyl-2-pentenyl,

1- methyl-3-pentenyl, 2-methyl-3-pentenyl, 3-methyl-3-pentenyl, 4-methyl-3-pentenyl, 1-methyl- 4-pentenyl, 2-methyl-4-pentenyl, 3-methyl-4-pentenyl, 4-methyl-4-pentenyl, 1 ,1-dimethyl-2- butenyl, 1 ,1-dimethyl-3-butenyl, 1 ,2-dimethyl-1-butenyl, 1 ,2-dimethyl-2-butenyl, 1 ,2-dimethyl-3- butenyl, 1 ,3-dimethyl-1-butenyl, 1 ,3-dimethyl-2-butenyl, 1 ,3-dimethyl-3-butenyl, 2,2-dimethyl-3- butenyl, 2,3-dimethyl-1-butenyl, 2,3-dimethyl-2-butenyl, 2,3-dimethyl-3-butenyl, 3,3-dimethyl-1- butenyl, 3,3-dimethyl-2-butenyl, 1 -ethyl- 1-butenyl, 1-ethyl-2-butenyl, 1-ethyl-3-butenyl, 2-ethyl-1- butenyl, 2-ethyl-2-butenyl, 2-ethyl-3-butenyl, 1 ,1 ,2-trimethyl-2-propenyl, 1-ethyl-1-methyl-

2- propenyl, 1-ethyl-2-methyl-1-propenyl, and 1-ethyl-2-methyl-2-propenyl;

C 3 -C 6 -haloalkenyl: a C 3 -C 6 -alkenyl substituent as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, e.g. 2-chloroprop-2-en-1-yl, 3- chloroprop-2-en-1-yl, 2,3-dichloroprop-2-en-1-yl, 3,3-dichloroprop-2-en-1-yl, 2,3,3-trichloro-2-en-

1- yl, 2,3-dichlorobut-2-en-1-yl, 2-bromoprop-2-en-1-yl, 3-bromoprop-2-en-1-yl, 2,3-dibromoprop-

2- en-1-yl, 3,3-dibromoprop-2-en-1-yl, 2,3,3-tribromo-2-en-1-yl, or 2,3-dibromobut-2-en-1-yl;

C 3 -C 6 -alkynyl: e.g. 1-propynyl, 2-propynyl, 1-butynyl, 2-butynyl, 3-butynyl, 1-methyl-2- propynyl, 1-pentynyl, 2-pentynyl, 3-pentynyl, 4-pentynyl, 1-methyl-2-butynyl, 1-methyl-3-butynyl, 2-methyl-3-butynyl, 3-methyl- 1-butynyl, 1 ,1-dimethyl-2-propynyl, 1-ethyl-2-propynyl, 1-hexynyl, 2-hexynyl, 3-hexynyl, 4-hexynyl, 5-hexynyl, 1-methyl-2-pentynyl, 1-methyl-3-pentynyl, 1-methyl- 4-pentynyl, 2-methyl-3-pentynyl, 2-methyl-4-pentynyl, 3-methyl- 1-pentynyl, 3-methyl-4-pentynyl, 4-methyl- 1-pentynyl, 4-methyl-2-pentynyl, 1 ,1-dimethyl-2-butynyl, 1 ,1-dimethyl-3-butynyl, 1 ,2- dimethyl-3-butynyl, 2,2-dimethyl-3-butynyl, 3,3-dimethyl-1-butynyl, 1-ethyl-2-butynyl, 1-ethyl-3- butynyl, 2-ethyl-3-butynyl, and 1 -ethyl- 1-methyl-2-propynyl;

C 2 -C 6 -alkynyl: C 3 -C 6 -alkynyl as mentioned above and also ethynyl;

C 3 -C 6 -haloalkynyl: a C 3 -C 6 -alkynyl group as mentioned above which is partially or fully substituted by F, CI, Br and/or I, e.g. 1 ,1-difluoroprop-2-yn-1-yl, 3-chloroprop-2-yn-1-yl, 3- bromoprop-2-yn-1-yl, 3-iodoprop-2-yn-1-yl, 4-fluorobut-2-yn-1-yl, 4-chlorobut-2-yn-1-yl, 1 ,1- difluorobut-2-yn-1-yl, 4-iodobut-3-yn-1-yl, 5-fluoropent-3-yn-1-yl, 5-iodopent-4-yn-1-yl, 6- fluorohex-4-yn-1-yl, or 6-iodohex-5-yn-1-yl;

Ci-C 4 -alkoxy: e.g. methoxy, ethoxy, propoxy, 1-methylethoxy butoxy, 1-methylpropoxy, 2-methylpropoxy, and 1 ,1-dimethylethoxy;

- C 1 -C 6 -alkoxy: Ci-C 4 -alkoxy as mentioned above, and also, e.g., pentoxy, 1-methyl- butoxy, 2-methylbutoxy, 3-methoxyl butoxy, 1 ,1-dimethylpropoxy, 1 ,2-dimethylpropoxy, 2,2- dimethylpropoxy, 1-ethylpropoxy, hexoxy, 1-methylpentoxy, 2-methylpentoxy, 3-methylpentoxy, 4-methylpentoxy, 1 ,1-dimethylbutoxy, 1 ,2-dimethylbutoxy, 1 ,3-dimethylbutoxy,

2,2-dimethylbutoxy, 2,3-dimethylbutoxy, 3,3-dimethylbutoxy, 1-ethylbutoxy, 2-ethylbutoxy, 1 ,1 ,2- trimethylpropoxy, 1 ,2,2-trimethylpropoxy, 1-ethyl-1-methylpropoxy, and 1 -ethyl-2- methylpropoxy.

Ci-C 4 -haloalkoxy: a Ci-C 4 -alkoxy group as mentioned above which is partially or fully substituted by fluorine, chlorine, bromine and/or iodine, i.e., e.g., fluoromethoxy,

difluoromethoxy, trifluoromethoxy, chlorodifluoromethoxy, bromodifluoromethoxy, 2- fluoroethoxy, 2-chloroethoxy, 2-bromomethoxy, 2-iodoethoxy, 2,2-difluoroethoxy, 2,2,2- trifluoroethoxy, 2-chloro-2-fluoroethoxy, 2-chloro-2,2-difluoroethoxy, 2,2-dichloro-2-fluoroethoxy, 2,2,2-trichloroethoxy, pentafluoroethoxy, 2-fluoropropoxy, 3-fluoropropoxy, 2-chloropropoxy, 3- chloropropoxy, 2-bromopropoxy, 3-bromopropoxy, 2,2-difluoropropoxy, 2,3-difluoropropoxy, 2,3- dichloropropoxy, 3,3,3-trifluoropropoxy, 3,3,3-trichloropropoxy, 2,2,3,3,3-pentafluoropropoxy, heptafluoropropoxy, 1 -(fluoromethyl)-2-fluoroethoxy, 1 -(chloromethyl)-2-chloroethoxy, 1 -(bromo- methyl)-2-bromoethoxy, 4-fluorobutoxy, 4-chlorobutoxy, 4-bromobutoxy, and nonafluorobutoxy;

C 1 -C 6 -haloalkoxy: a Ci-C 4 -haloalkoxy as mentioned above, and also, e.g., 5- fluoropentoxy, 5-chloropentoxy, 5-bromopentoxy, 5-iodopentoxy, undecafluoropentoxy, 6-fluoro- hexoxy, 6-chlorohexoxy, 6-bromohexoxy, 6-iodohexoxy and dodecafluorohexoxy;

Ci-C 4 -alkylthio: e.g. methylthio, ethylthio, propylthio, 1-methylethylthio, butylthio, 1- methylpropylthio, 2-methylpropylthio, and 1 ,1-dimethylethylthio;

C 1 -C 6 -alkylthio: Ci-C 4 -alkylthio as mentioned above, and also, e.g., pentylthio, 1- methylbutylthio, 2-methylbutylthio, 3-methylbutylthio, 2,2-dimethylpropylthio, 1-ethylpropylthio, hexylthio, 1 ,1-dimethylpropylthio, 1 ,2-dimethylpropylthio, 1-methylpentylthio, 2-methylpentylthio, 3-methylpentylthio, 4-methylpentylthio, 1 ,1-dimethylbutylthio, 1 ,2-dimethylbutylthio, 1 ,3- dimethylbutylthio, 2,2-dimethylbutylthio, 2,3-dimethylbutylthio, 3,3-dimethylbutylthio, 1- ethylbutylthio, 2-ethylbutylthio, 1 ,1 ,2-trimethylpropylthio, 1 ,2,2-trimethylpropylthio, 1-ethyl-1- methyl propylthio, and 1- ethyl-2-methylpropylthio;

- (Ci-C 4 -alkyl)amino: e.g. methylamino, ethylamino, propylamino, 1-methylethylamino, butylamino, 1-methylpropylamino, 2-methylpropylamino, or 1 ,1-dimethylethylamino;

(C 1 -C 6 -alkyl)amino: (Ci-C 4 -alkylamino) as mentioned above, and also, e.g., pentylamino, 1-methylbutylamino, 2-methylbutylamino, 3-methylbutylamino, 2,2-dimethylpropylamino, 1-ethyl- propylamino, hexylamino, 1 ,1-dimethylpropylamino, 1 ,2-dimethylpropylamino, 1-methyl- pentylamino, 2-methylpentylamino, 3-methylpentylamino, 4-methylpentylamino, 1 ,1-dimethyl- butylamino, 1 ,2-dimethylbutylamino, 1 ,3-dimethylbutylamino, 2,2-dimethylbutylamino, 2,3- dimethylbutyl-amino 3,3-dimethylbutylamino, 1-ethylbutylamino, 2-ethylbutylamino, 1 ,1 ,2- trimethylpropylamino, 1 ,2,2-trimethyl-propylamino, 1-ethyl-1-methylpropylamino, or 1 -ethyl-2- methylpropylamino;

- di(Ci-C 4 -alkyl)amino: e.g. N,N-dimethylamino, Ν,Ν-diethylamino, N,N-di(1- methylethyl)amino, Ν,Ν-dipropylamino, N,N-dibutylamino, N,N-di(1-methylpropyl)amino, N,N- di(2-methylpropyl)amino, N,N-di(1 ,1-dimethylethyl)amino, N-ethyl-N-methylamino, N-methyl-N- propylamino, N-methyl-N-(1-methylethyl)amino, N-butyl-N-methylamino, N-methyl-N-(1- methylpropyl)amino, N-methyl-N-(2-methylpropyl)amino, N-(1 ,1-dimethylethyl)-N-methylamino, N-ethyl-N-propylamino, N-ethyl-N-(1-methylethyl)amino, N-butyl-N-ethylamino, N-ethyl-N-(1- methylpropyl)amino, N-ethyl-N-(2-methylpropyl)amino, N-ethyl-N-(1 ,1-dimethylethyl)amino, N- (l-methylethyl)-N-propylamino, N-butyl-N-propylamino, N-(1-methylpropyl)-N-propylamino, N-(2- methylpropyl)-N-propylamino, N-(1 ,1-dimethylethyl)-N-propylamino, N-butyl-N-(1- methylethyl)amino, N-(1 -methylethyl)-N-(1-methylpropyl)amino, N-(1-methylethyl)-N-(2-methyl- propyl)amino, N-(1 ,1-dimethylethyl)-N-(1-methylethyl)amino, N-butyl-N-(1 -methylpropyl)amino, N-butyl-N-(2-methylpropyl)amino, N-butyl-N-(1 ,1-dimethylethyl)amino, N-(1 -methylpropyl)-N-(2- methylpropyl)amino, N-(1 ,1-dimethylethyl)-N-(1-methylpropyl)amino, or N-(1 ,1-dimethylethyl)-N- (2-methylpropyl)amino;

di(C 1 -C 6 -alkyl)amino: di(Ci-C4-alkyl)amino as mentioned above, and also, e.g., N- methyl-N-pentylamino, N-methyl-N-(1-methylbutyl)amino, N-methyl-N-(2-methylbutyl)amino, N- methyl-N-(3-methylbutyl)amino, N-methyl-N-(2,2-dimethylpropyl)amino, N-methyl-N-(1- ethylpropyl)amino, N-methyl-N-hexylamino, N-methyl-N-(1 ,1 -dimethylpropyl)amino, N-methyl-N- (1 ,2-dimethylpropyl)amino, N-methyl-N-(1-methylpentyl)amino, N-methyl-N-(2- methylpentyl)amino, N-methyl-N-(3-methylpentyl)amino, N-methyl-N-(4-methylpentyl)amino, N- methyl-N-(1 ,1-dimethylbutyl)amino, N-methyl-N-(1 ,2-dimethylbutyl)amino, N-methyl-N-(1 ,3- dimethylbutyl)amino, N-methyl-N-(2,2-dimethylbutyl)amino, N-methyl-N-(2,3- dimethylbutyl)amino, N-methyl-N-(3,3-dimethylbutyl)amino, N-methyl-N- (l-ethylbutyl)amino, N- methyl-N-(2-ethylbutyl)amino, N-methyl-N-(1 ,1 ,2-trimethylpropyl)amino, N-methyl-N- (1 ,2,2- trimethylpropyl)amino, N-methyl-N-(1-ethyl-1 -methylpropyl)amino, N-methyl-N- (1-ethyl-2- methylpropyl)amino, N-ethyl-N-pentylamino, N-ethyl-N-(1-methylbutyl)amino, N-ethyl-N-(2- methylbutyl)amino, N-ethyl-N-(3-methylbutyl)amino, N-ethyl-N-(2,2-dimethylpropyl)amino, N- ethyl-N-(1 -ethylpropyl)amino, N-ethyl-N-hexylamino, N-ethyl-N-(1 ,1-dimethylpropyl)amino, N- ethyl-N-(1 ,2-dimethylpropyl)amino, N-ethyl-N-(1 -methylpentyl)amino, N-ethyl-N-(2-methyl- pentyl)amino, N-ethyl-N-(3-methylpentyl)amino, N-ethyl-N-(4-methylpentyl)amino, N-ethyl-N- (1 ,1-dimethylbutyl)amino, N-ethyl-N-(1 ,2-dimethylbutyl)amino, N-ethyl-N-(1 ,3- dimethylbutyl)amino, N-ethyl-N-(2,2-dimethylbutyl)amino, N-ethyl-N-(2,3-dimethylbutyl)amino, N-ethyl-N-(3,3-dimethylbutyl)amino, N-ethyl-N-(1 -ethylbutyl)amino, N-ethyl-N-(2- ethylbutyl)amino, N-ethyl-N-(1 ,1 ,2-trimethylpropyl)amino, N-ethyl-N-(1 ,2,2- trimethylpropyl)amino, N-ethyl-N-(1 -ethyl-1 -methylpropyl)amino, N-ethyl-N-(1 -ethyl-2- methylpropyl)amino, N-propyl-N-pentylamino, N-butyl-N-pentylamino, Ν,Ν-dipentylamino, N- propyl-N-hexylamino, N-butyl-N-hexylamino, N-pentyl-N-hexylamino, or N,N-dihexylamino;

C 1 -C 6 -alkylsulfinyl (C 1 -C 6 -Alkyl-S(=0)-): e.g. methylsulfinyl, ethylsulfinyl, propylsulfinyl, 1- methylethylsulfinyl, butylsulfinyl, 1 -methylpropylsulfinyl, 2-methylpropylsulfinyl, 1 ,1-di- methylethylsulfinyl, pentylsulfinyl, 1-methylbutylsulfinyl, 2-methylbutylsulfinyl, 3- methylbutylsulfinyl, 2,2-dimethylpropylsulfinyl, 1-ethylpropylsulfinyl, 1 ,1 -dimethylpropylsulfinyl, 1 ,2-dimethylpropyl-sulfinyl, hexylsulfinyl, 1 -methylpentylsulfinyl, 2-methylpentylsulfinyl, 3- methylpentylsulfinyl, 4-methylpentyl-sulfinyl, 1 ,1 -dimethylbutylsulfinyl, 1 ,2-dimethylbutylsulfinyl, 1 ,3-dimethylbutyl-sulfinyl, 2,2-dimethylbutylsulfinyl, 2,3-dimethylbutylsulfinyl, 3,3-dimethylbutyl- sulfinyl, 1 -ethyl buty Isu If i ny 1 , 2-ethyl butylsulfinyl, 1 ,1 ,2-tri methyl propylsulfinyl, 1 ,2,2- trimethylpropylsulfinyl, 1 -ethyl-1 -methylpropyl-sulfinyl, and 1 -ethyl-2-methylpropylsulfinyl;

C 1 -C 6 -alkylsulfonyl (C 1 -C 6 -alkyl-S(0)2-): e.g. methylsulfonyl, ethylsulfonyl, propylsulfonyl, 1-methylethylsulfonyl, butylsulfonyl, 1 -methylpropylsulfonyl, 2-methyl-propylsulfonyl, 1 ,1 - dimethylethylsulfonyl, pentylsulfonyl, 1-methylbutylsulfonyl, 2-methylbutylsulfonyl, 3- methyl butylsulfonyl, 1 ,1-dimethylpropylsulfonyl, 1 ,2-dimethylpropylsulfonyl, 2,2-dimethylpropyl- sulfonyl, 1 -ethyl propylsulfonyl, hexylsulfonyl, 1 -methylpentylsulfonyl, 2-methylpentylsulfonyl, 3- methylpentylsulfonyl, 4-methylpentylsulfonyl, 1 ,1 -dimethylbutylsulfonyl, 1 ,2-dimethylbutyl- sulfonyl, 1 ,3-dimethylbutylsulfonyl, 2,2-dimethylbutylsulfonyl, 2,3-dimethylbutylsulfonyl, 3,3- dimethylbutyl-sulfonyl, 1-ethylbutylsulfonyl, 2-ethylbutylsulfonyl, 1 ,1 ,2-trimethyl-propylsulfonyl, 1 ,2,2-trimethyl-propylsulfonyl, 1-ethyl-1-methylpropylsulfonyl, and 1 -ethyls- methyl propy Isu If ony I ;

C 3 -C 6 -cycloalkyl: a monocyclic saturated hydrocarbon having 3 to 6 ring members, such as cyclopropyl, cyclobutyl, cyclopentyl, and cyclohexyl;

C 3 -C 6 -cycloalkenyl: 1-cyclopropenyl, 2-cyclopropenyl, 1 -cyclobutenyl, 2-cyclobutenyl, 1 - cyclopentenyl, 2-cyclopentenyl, 1 ,3-cyclopentadienyl, 1 ,4-cyclopentadienyl, 2,4- cyclopentadienyl, 1-cyclohexenyl, 2-cyclohexenyl, 3-cyclohexenyl, 1 ,3-cyclohexadienyl, 1 ,4- cyclohexadienyl, or 2,5-cyclohexadienyl;

- heterocyclyl: a 3- to 6-membered heterocyclyl: a saturated or partial unsaturated cycle having three to six ring members which comprises apart from carbon atoms one to four nitrogen atoms, or one or two oxygen atoms, or one or two sulfur atoms, or one to three nitrogen atoms and an oxygen atom, or one to three nitrogen atoms and a sulfur atom, or one sulfur and one oxygen atom, e.g.

3- or 4-membered heterocycles like 2-oxiranyl, 2-aziridinyl, 2-thiiranyl, 2-oxetanyl, 3-oxetanyl,

2- thietanyl, 3-thietanyl, 1 -azetidinyl, 2-azetidinyl, 1-azetinyl, or 2-azetinyl;

5-membered saturated heterocycles like2-tetrahydrofuranyl, 3-tetrahydrofuranyl, 2- tetrahydrothienyl, 3-tetrahydrothienyl, 1-pyrrolidinyl,2-pyrrolidinyl, 3-pyrrolidinyl, 3-isoxazolidinyl,

4- isoxazolidinyl, 5-isoxazolidinyl, 2-isothiazolidinyl, 3-isothiazolidinyl, 4-isothiazolidinyl, 5- isothiazolidinyl, 1 -pyrazolidinyl, 3-pyrazolidinyl, 4-pyrazolidinyl, 5-pyrazolidinyl, 2-oxazolidinyl, 4- oxazolidinyl, 5-oxazolidinyl, 2-thiazolidinyl, 4-thiazolidinyl, 5-thiazolidinyl, 1 -imidazolidinyl, 2- imidazolidinyl, 4-imidazolidinyl, 3-oxazolidinyl, 1 ,2,4-oxadiazolidin-3-yl, 1 ,2,4-oxadiazolidin-5-yl,

3- thiazolidinyl, 1 ,2,4-thiadiazolidin-3-yl, 1 ,2,4-thiadiazolidin-5-yl, 1 ,2,4-triazolidin-3-yl, 1 ,2,4- oxadiazolidin-2-yl, 1 ,2,4-oxadiazolidin-4-yl, 1 ,3,4-oxadiazolidin-2-yl, 1 ,2,4-thiadiazolidin-2-yl, 1 ,2,4-thiadiazolidin-4-yl, 1 ,3,4-thiadiazolidin-2-yl, 1 ,2,4-triazolidin-1 -yl, or 1 ,3,4-triazolidin-2-yl; 5-membered partial unsaturated heterocycles like 2,3-dihydrofur-2-yl, 2,3-dihydrofur-3-yl, 2,4- dihydrofur-2-yl, 2,4-dihydrofur-3-yl, dioxolan-2-yl, 1 ,3-dioxol-2-yl, 2,3-dihydrothien-2-yl, 2,3- dihydrothien-3-yl, 2,4-dihydrothien-2-yl, 2,4-dihydrothien-3-yl, 4,5-dihydropyrrol-1 -yl, 4,5- dihydropyrrol-2-yl, 4,5-dihydropyrrol-3-yl, 2,5-dihydropyrrol-1-yl, 2,5-dihydropyrrol-2-yl, 2,5- dihydropyrrol-3-yl, 2,3-dihydroisoxazol-1-yl, 2,3-dihydroisoxazol-3-yl, 2,3-dihydroisoxazol-4-yl, 2 , 3-d i hyd roisoxazol-5-y 1 , 2 , 5-d i hyd roisoxazol-3-y 1 , 2 , 5-d i hyd roisoxazol-4-y 1 , 2 , 5-d i hyd roisoxazol-

5- yl, 4,5-dihydroisoxazol-2-yl, 4,5-dihydroisoxazol-3-yl, 4,5-dihydroisoxazol-4-yl, 4,5- dihydroisoxazol-5-yl, 2,3-dihydroisothiazol-1 -yl, 2,3-dihydroisothiazol-3-yl, 2,3-dihydroisothiazol-

4- yl, 2,3-dihydroisothiazol-5-yl, 2,5-dihydroisothiazol-3-yl, 2,5-dihydroisothiazol-4-yl, 2,5- dihydroisothiazol-5-yl, 4,5-dihydroisothiazol-1-yl, 4,5-dihydroisothiazol-3-yl, 4,5- dihydroisothiazol-4-yl, 4,5-dihydroisothiazol-5-yl, 2,3-dihydropyrazol-1-yl, 2,3-dihydropyrazol-2- yl, 2,3-dihydropyrazol-3-yl, 2,3-dihydropyrazol-4-yl, 2,3-dihydropyrazol-5-yl, 3,4-dihydropyrazol- 1 -yl, 3,4-dihydropyrazol-3-yl, 3,4-dihydropyrazol-4-yl, 3,4-dihydropyrazol-5-yl, 4,5- dihydropyrazol-1-yl, 4,5-dihydropyrazol-3-yl, 4,5-dihydropyrazol-4-yl, 4,5-dihydropyrazol-5-yl, 2,3-dihydroimidazol-1 -yl, 2,3-dihydroimidazol-2-yl, 2,3-dihydroimidazol-3-yl ,2,3-dihydroimidazol- 4-yl, 2,3-dihydroimidazol-5-yl, 4,5-dihydroimidazol-1 -yl, 4,5-dihydroimidazol-2-yl, 4,5- dihydroimidazol-4-yl, 4,5-dihydroimidazol-5-yl, 2,5-dihydroimidazol-1 -yl, 2,5-dihydroimidazol-2- yl, 2,5-dihydroimidazol-4-yl, 2,5-dihydroimidazol-5-yl, 2,3-dihydrooxazol-2-yl, 2,3-dihydrooxazol- 3-yl, 2,3-dihydrooxazol-4-yl, 2,3-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3- yl, 3,4-dihydrooxazol-4-yl, 3,4-dihydrooxazol-5-yl, 2,3-dihydrothiazol-2-yl, 2,3-dihydrothiazol-3- yl, 2,3-dihydrothiazol-4-yl, 2,3-dihydrothiazol-5-yl, 3,4-dihydrothiazol-2-yl, 3,4-dihydrothiazol-3- yl, 3,4-dihydrothiazol-4-yl, 3,4-dihydrothiazol-5-yl, 3,4-dihydrothiazol-2-yl, 3,4-dihydrothiazol-3- yl, or 3,4-dihydrothiazol-4-yl;

6-membered saturated heterocycles like 1-piperidinyl, 2-piperidinyl, 3-piperidinyl, 4-piperidinyl, 1 ,3-dioxan-5-yl, 1 ,4-dioxanyl, 1 ,3-dithian-5-yl, 1 ,3-dithianyl, 1 ,3-oxathian-5-yl, 1 ,4-oxathianyl, 2-tetrahydropyranyl, 3-tetrahydopyranyl, 4-tetrahydropyranyl, 2-tetrahydrothiopyranyl, 3- tetrahydrothiopyranyl,4-tetrahydrothiopyranyl, 1-hexahydropyridazinyl, 3-hexahydropyridazinyl, 4-hexahydropyridazinyl, 1-hexahydropyrimidinyl, 2-hexahydropyrimidinyl, 4- hexahydropyrimidinyl, 5-hexahydropyrimidinyl, 1-piperazinyl, 2-piperazinyl, 1 ,3,5- hexahydrotriazin-1-yl, 1 ,3,5-hexahydrotriazin-2-yl, 1 ,2,4-hexahydrotriazin-1-yl, 1 ,2,4- hexahydrotriazin-3-yl, tetrahydro-1 ,3-oxazin-1-yl, tetrahydro-1 ,3-oxazin-2-yl, tetrahydro-1 ,3- oxazin-6-yl, 1-morpholinyl, or 2-morpholinyl, 3-morpholinyl;

6-membered partial unsaturated heterocycles like 2H-pyran-2-yl, 2H-pyran-3-yl, 2H-pyran-4-yl, 2H-pyran-5-yl, 2H-pyran-6-yl, 2H-thiopyran-2-yl, 2H-thiopyran-3-yl, 2H-thiopyran-4-yl, 2H- thiopyran-5-yl, 2H-thiopyran-6-yl, or 5,6-dihydro-4H-1 ,3-oxazin-2-yl.

heteroaryl: a 5- or 6-membered heteroaryl: monocyclic aromatic heteroaryl having 5 to 6 ring members which, in addition to carbon atoms and independent of their position in the ring, contains 1 to 4 nitrogen atoms, or 1 to 3 nitrogen atoms and an oxygen or sulfur atom, or an oxygen or a sulfur atom, e.g. 5-membered aromatic rings like furyl (e.g. 2-furyl, 3-furyl), thienyl (e.g. 2-thienyl, 3-thienyl), pyrrolyl (e.g. pyrrol-2-yl, pyrrol-3-yl), pyrazolyl (e.g. pyrazol-3-yl, pyrazol-4-yl), isoxazolyl (e.g. isoxazol-3-yl, isoxazol-4-yl, isoxazol-5-yl), isothiazolyl (e.g.

isothiazol-3-yl, isothiazol-4-yl, isothiazol-5-yl), imidazolyl (e.g. imidazole-2-yl, imidazole-4-yl), oxazolyl (e.g. oxazol-2-yl, oxazol-4-yl, oxazol-5-yl), thiazolyl (e.g. thiazol-2-yl, thiazol-4-yl, thiazol-5-yl), oxadiazolyl (e.g. 1 ,2,3-oxadiazol-4-yl, 1 ,2,3-oxadiazol-5-yl, 1 ,2,4-oxadiazol-3-yl, 1 ,2,4-oxadiazol-5-yl, 1 ,3,4-oxadiazol-2-yl), thiadiazolyl (e.g. 1 ,2,3-thiadiazol-4-yl, 1 ,2,3- thiadiazol-5-yl, 1 ,2,4-thiadiazol-3-yl, 1 ,2,4-thiadiazol-5-yl, 1 ,3,4-thiadiazolyl-2-yl), triazolyl (e.g. 1 ,2,3-triazol-4-yl, 1 ,2,4-triazol-3-yl); 1-tetrazolyl; 6-membered aromatic rings like pyridyl (e.g. pyridine-2-yl, pyridine-3-yl, pyridine-4-yl), pyrazinyl (e.g. pyridazin-3-yl, pyridazin-4-yl), pyrimidinyl (e.g. pyrimidin-2-yl, pyrimidin-4-yl, pyrimidin-5-yl), pyrazin-2-yl, triazinyl (e.g. 1 ,3,5- triazin-2-yl, or 1 ,2,4— triazin-3-yl, 1 ,2,4-triazin-5-yl, 1 ,2,4-triazin-6-yl).

The term "substituted" if not specified otherwise refers to substituted by 1 , 2 or maximum possible number of substituents. If substituents as defined in compounds of formula I are more than one then they are independently from each other are same or different if not mentioned otherwise.

The term "acidic functionality" if not specified otherwise refers to a functionality capable of donating a hydrogen (proton or hydrogen ion H + ), such as a carboxylic group or a sulphonic group, or, alternatively, capable of forming a covalent bond with an electron pair.

The terms "compounds of formula (I)", "Pyrimidine compounds of formula (I)", "Compounds I" and "compounds of invention" are synonyms.

The term "cyclic groups" comprises aliphatic cyclic groups such as cycloalkyl, cycloalkenyl and heterocyclyl and aromatic cyclic groups such as heteroaryl and phenyl.

The preferred embodiments of the invention mentioned herein below have to be understood as being preferred either independently from each other or in combination with one another. In general, pyrimidine compounds of formula (I) are suitable as herbicides.

According to a preferred embodiment of the invention preference is given pyrimidine compounds of formula (I), and their use as herbicides, wherein the variables, either

independently of one another or in combination with one another, have the following meanings: Preferred R 1 is C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, C 1 -C 6 -haloalkoxy, C 3 -C 6 -alkenyloxy, C 3 -C 6 - haloalkenyloxy C 3 -C 6 -alkynyloxy, C 4 -C6-haloalkynyloxy, C 1 -C 6 -alkylthio, C 3 -C 6 -cycloalkyl, wherein the cycloalkyl substituent is unsubstituted;

particularly preferred R 1 is C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, or C 3 -C 6 -cycloalkyl, wherein the cycloalkyl substituent is unsubstituted;

especially preferred R 1 is C 3 -C 6 -cycloalkyl, wherein the cycloalkyl substituent is unsubstituted; also especially preferred R 1 is C2H5, 1-C3H7, i-C 4 Hc>, OCH3, C-C3H5, or c-C 4 H9;

more preferred R 1 is C2H5, OCH3, or C-C3H5;

most preferred R 1 is C-C3H5.

Preferred R 2 is C 2 -C 6 -alkenyl, C 2 -C 6 -haloalkenyl, C 1 -C 6 -alkoxy-C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 6 -cycloalkenyl, C 3 -C 6 -cycloalkenyl-C 1 -C 6 -alkyl, C 3 -C 6 -cycloalkyl-C 1 -C 6 -alkylidenyl, C 3 -C 6 - halocycloalkyl-C 1 -C 6 -alkylidenyl, C 3 -C 6 -cycloalkenyl-C 1 -C 6 -alkylidenyl, C 3 -C 6 -hydroxycycloalkyl- C 1 -C 6 -alkyl, C 3 -C 6 -hydroxycycloalkenyl-C 1 -C 6 -alkyl, C 1 -C 6 -hydroxyalkyl, C 3 -C 6 -cycloalkyl-C 2 -C 6 - hydroxyalkylidenyl, hydroxycarbonyl-C 1 -C 6 -alkyl, hydroxycarbonyl-C 1 -C 6 -haloalkyl, C 1 -C 6 - alkoxycarbonyl-C 1 -C 6 -alkyl, C 3 -C 6 -hydroxycycloalkyl-C 1 -C 6 -hydroxyalkyl, C 2 -C 6 -dihydroxyalkyl, C 3 -C 6 -cycloalkyl-C 3 -C 6 -dihydroxyalkylidenyl, hydroxycarbonyl-C 2 -C 6 -dihydroxyalkyl, C 1 -C 6 - alkoxycarbonyl-C 2 -C 6 -dihydroxyalkyl, C 1 -C 6 -dicyanoalkyl, or 5- or 6-membered heteroaryl;

wherein hydroxy groups of R 2 are unsubstituted or substituted by R b ,

cyclic groups of R 2 are unsubstituted or substituted by R c , and

and acyclic aliphatic groups of R 2 are unsubstituted or substituted by R d .

particularly preferred R 2 is C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 6 -cycloalkenyl, C 3 -C 6 -cycloalkyl- C 1 -C 6 -alkylidenyl, C 3 -C 6 -halocycloalkyl-C 1 -C 6 -alkylidenyl, C 3 -C 6 -hydroxycycloalkyl-C 1 -C 6 -alkyl, C 3 -C 6 -hydroxycycloalkyl-C 1 -C 6 -hydroxyalkyl, C 2 -C 6 -dihydroxyalkyl, or 5- or 6-membered heteroaryl;

also particularly preferred R 2 is C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 6 -cycloalkenyl-C 1 -C 6 -alkyl, C 3 -C 6 -cycloalkyl-C 1 -C 6 -alkylidenyl, C 1 -C 6 -hydroxyalkyl, C 1 -C 6 -alkoxycarbonyl-C 1 -C 6 -alkyl, C 2 -C 6 - dihydroxyalkyl, C 1 -C 6 -dicyanoalkyl, 5- or 6-membered heteroaryl;

wherein hydroxy groups of R 2 are unsubstituted or substituted by R b ,

cyclic groups of R 2 are unsubstituted or substituted by R c , and

acyclic aliphatic groups of R 2 are unsubstituted or substituted by R d .

especially preferred R 2 is R 2 is C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 6 -cycloalkyl-C 1 -C 6 -alkylidenyl, C 3 -C 6 -hydroxycycloalkyl-C 1 -C 6 -alkyl, and 5- or 6-membered heteroaryl;

also especially preferred R 2 is C 2 -C 6 -alkenyl, C 1 -C 6 -hydroxyalkyl, C 3 -C 6 -cycloalkyl-C 1 -C 6 - alkylidenyl, C 2 -C 6 -dihydroxyalkyl, C 1 -C 6 -dicyanoalkyl and 5- or 6-membered heteroaryl;

also especially preferred R 2 is C 2 -C 6 -alkenyl, , C 3 -C 6 -cycloalkyl-C 1 -C 6 -alkylidenyl, C 1 -C 6 - hydroxyalkyl, C 2 -C 6 -dihydroxyalkyl, or 5- or 6-membered heteroaryl;

wherein hydroxy groups of R 2 are unsubstituted or substituted by R b ,

cyclic groups of R 2 are unsubstituted or substituted by R c , and

and acyclic aliphatic groups of R 2 are unsubstituted or substituted by R d . more preferred R 2 is C 2 -C 6 -alkenyl, C 3 -C 6 -cycloalkyl-C 1 -C 6 -alkylidenyl, or 5- or 6-membered heteroaryl;

also more preferred R 2 is C 1 -C 6 -hydroxyalkyl, C 2 -C 6 -dihydroxyalkyl, C 3 -C 6 -cycloalkyl-C 1 -C 6 - alkylidenyl, or 5- or 6-membered heteroaryl;

wherein OH groups of R 2 are unsubstituted or substituted by R b ,

cyclic groups of R 2 are unsubstituted or substituted by R c , and

acyclic aliphatic groups of R 2 are unsubstituted or substituted by R d .

most preferred R 2 is C 2 -C 6 -alkenyl;

also most preferred R 2 is C 3 -C 6 -cycloalkyl-C 1 -C 6 -alkylidenyl;

also most preferred R 2 is 5- or 6-membered heteroaryl;

also most preferred R 2 is 5-membered heteroaryl;

also most preferred R 2 is C 1 -C 6 -hydroxyalkyl;

also most preferred R 2 is C 2 -C 6 -dihydroxyalkyl;

wherein OH groups of R 2 are unsubstituted or substituted by R b ,

cyclic groups of R 2 are unsubstituted or substituted by R c , and

acyclic aliphatic groups of R 2 are unsubstituted or substituted by R d .

also more preferred R 2 is CH=CH-CH 3 , CH=C(CH 2 ) 3 , or CH=C(CH 2 ) 4 ;

also more preferred R 2 is 2-furyl, 3-furyl, 2-methyl-3-furyl, or 3-methyl-2-furyl;

also most preferred R 2 is CH=CH-CH 3 , CH=C(CH 2 )3, 2-furyl, 3-furyl, or 4-methyloxazol-5-yl; also most preferred R 2 is CHOH-CHOH-C 6 H 5 , CHOH-CHOH-2-furyl, CHOH-CHOH-CH 3 , or 4- methyl-5-oxazolyl.

also most preferred R 2 is CHOH-CHOH-C 6 H 5 , CHOH-CHOH-2-furyl, CHOH-CHOH-CH3, or 4- methyloxazol-5-yl;

also most preferred R 2 is selected from R 2 -1 to R 2 -16 as shown below,

wherein # denotes attachment to the pyrimidine ring, X and Y denotes R c which independently of each other are identical or different;

preferred R 2 is R 2 -1 , R 2 -2, R 2 -3, R 2 -4, R 2 -5, R 2 -6, R 2 -7, or R 2 -8;

also preferred R 2 is R 2 -9, R 2 -10, R 2 -1 1 , R 2 -13, R 2 -14, or R 2 -15;

more preferred R 2 is R 2 -9, R 2 -10, or R 2 -15;

most preferred R 2 is R 2 -9; preferred X is H, halogen, CN, C 1 -C 6 -alkyl, CrC6-haloalkyl, OH, C 1 -C 6 -alkoxy, C 1 -C 6 - haloalkoxy, or C 1 -C 6 -alkylthio;

particularrly preferred X is H, halogen, CN, C 1 -C 6 -alkyl, OH, C 1 -C 6 -alkoxy, or C 1 -C 6 -alkylthio; also particularrly preferred X is H, halogen, CN, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkoxy, or C 1 -C 6 -haloalkoxy;

especially preferred X is H, halogen, CN, Ci-C 4 -alkyl, OH, Ci-C 4 -alkoxy, or Ci-C 4 -alkylthio; more preferred X is H, CH3, C2H5, n-propyl, iso-propyl, iso-butyl, n-butyl, OH, OCH3, SCH3, F, CI, Br, or I;

most preferred X is H, CH 3 , C 2 H 5 , OH, or OCH 3 ;

also most preferred X is H, CH3, C2H5, or SCH3;

also most preferred X is H, CH3, C2H5, F, CI, Br, or I.

Preferred Y is H, halogen, CN, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, OH, C 1 -C 6 -alkoxy, C 1 -C 6 - haloalkoxy, or C 1 -C 6 -alkylthio;

particularrly preferred Y is H, halogen, CN, C 1 -C 6 -alkyl, OH, C 1 -C 6 -alkoxy, or C 1 -C 6 -alkylthio; also particularrly preferred Y is H, halogen, CN, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkoxy, or C 1 -C 6 -haloalkoxy;

especially preferred Y is H, halogen, CN, Ci-C 4 -alkyl, Ci-C2-fluoroalkyl, OH, Ci-C 4 -alkoxy, or Ci-C -alkylthio;

more preferred Y is H, CH3, C2H5, n- propyl, iso-propyl, iso-butyl, n-butyl, 2-butyl, t-butyl, OH, OCH3, SCH 3 , F, CI, Br, or I;

most preferred Y is H, CH3, C2H5, n- propyl, iso-propyl, iso-butyl, n-butyl, 2-butyl, OH, or OCH3; also most preferred Y is H, CH3, C2H5, n-propyl, iso-propyl, OH, OCH3, or SCH3;

also most preferred Y is H, CH 3 , C2H5, n-propyl, iso-propyl, F, CI, Br, or I.

Particulalrly preferred R 2 is 4-methyl-5-oxazolyl, 4-ethyl-5-oxazolyl, 2,4-dimethyl-5-oxazolyl, 2- ethyl-4-methyl-5-oxazolyl, 2-methyl-4-ethyl-5-oxazolyl, or 2,4-diethyl-5-oxazolyl.

Examples of particularly preferred R 2 are provided in Table R 2 -9, Table R 2 -10, and Table R 2 - 15.

Table R 2 -9: examples of particularly preferred R 2 are R 2 -9.1 to R 2 -9.676 wherein R 2 is R 2 -9 and combinitions of variables X and Y are as defined in each row of table R2, numbering of each compound e.g. R 2 -9.1 means R 2 is R 2 -9 wherein X and Y are as defined in row 1 of table R2;

Table R 2 -10: examples of particularly preferred R 2 are R 2 -10.1 to R 2 -10.676 wherein R 2 is R 2 - 10 and combinitions of variables X and Y are as defined in each row of table R2, numbering of each compound e.g. R 2 -10.1 means R 2 is R 2 -10 wherein X and Y are as defined in row 1 of table R2;

Table R 2 -15: examples of particularly preferred R 2 are R 2 -15.1 to R 2 -15.676 wherein R 2 is R 2 - 15 and combinitions of variables X and Y are as defined in each row of table R2, numbering of each compound e.g. R 2 -15.1 means R 2 is R 2 -15 wherein X and Y are as defined in row 1 of table R2.

Table R2:

Preferred A is CR 3 or NR 3A ;

most preferred A is CR 3;

also most preferred A is NR 3A .

Preferred Z is 6-membered heteroaryl ring, preferably triazine, pyrimidine, or pyridine; particularly preferred Z is pyrimidine or pyridine;

especially preferred Z is pyridine.

Also preferred Z is 5-membered heteroaryl ring, preferably thiadiazole, oxadiazole, triazole, thiazole, isothiazole, oxazole, isoxazole, pyrazole, imidazole, thiophene, furan, or pyrrole; particularly preferred Z is thiazole, isothiazole, oxazole, isoxazole, pyrazole, imidazole, thiophene, furan, or pyrrole;

especially preferred Z is thiophene, furan, or pyrrole;

particularly preferred Z is selected from below groups A to G,

wherein

R 3 is halogen, CHO, CN, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

m is 0 or 1 ;

R 4 is halogen, CHO, CN, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

X is O, S, or NR 3A ; and

# denotes the point of attachment to the pyrimidine ring.

Preferred R 3 is halogen, CN, NO2, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkoxy, or C 3 -C 6 - cycloalkyl;

also preferred R 3 is halogen, CN, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy,

particularly preferred R 3 is halogen, CN, C 1 -C 6 -alkyl, or C 1 -C 6 -alkoxy;

especially preferred halogen, or CH3; also especially preferred R 3 is halogen;

more preferred R 3 is CI, Br, or I;

most preferred R 3 is CI or Br.

Preferred R 3A is H, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkylcarbonyl, C 3 -C 6 -alkenyl, C 3 -C 6 - haloalkenyl, C 3 -C 6 -alkenyl, C 3 -C 6 -haloalkenyl, or C 3 -C 6 -cycloalkyl;

also preferred R 3A is H, Ci-Cralkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkylcarbonyl;

particularly preferred R 3A is H, C 1 -C 6 -alkyl, or C 1 -C 6 -alkylcarbonyl;

especially preferred R 3A is H, or Ci-Cralkyl;

most preferred R 3A is H, or CH3.

Preferred R 4 is halogen, CN, Ci-Cralkyl, C 1 -C 6 -haloalkyl, or Ci-Cralkoxy;

particularly preferred R 4 is halogen, Ci-Crhaloalkyl, or C 1 -C 6 -alkyl;

especially preferred R 4 is halogen;

also especially preferred R 4 is C 1 -C 6 -haloalkyl, or Ci-Cralkyl;

more preferred R 4 is F, CI, CHF 2 , CF 3 , CH 3 , or C 2 H 5 ;

most preferred R 4 is F;

also most preferred R 4 is CH 3 ;

also most preferred R 4 is CI.

also most preferred R 4 is CF3.

Preferred m is 0, 1 , or 2;

more preferred m is 0 or 1 ;

most preferred m is 0.

also most preferred m is 1.

Also preferred are the pyrimidine compounds of formula (I), and their use as herbicide, wherein

R 1 is preferably Ci-Cralkyl, C 1 -C 6 -alkoxy, or C3-Crcycloalkyl, wherein the cycloalkyl substituent is unsubstituted;

particularly preferred R 1 is C 3 -C 6 -cycloalkyl, wherein the cycloalkyl substituent is unsubstituted; R 2 is preferably C2-Cralkenyl, C 3 -C 6 -cycloalkyl-Ci-Cralkylidenyl, 5- or 6-membered heteroaryl, C 1 -C 6 -hydroxyalkyl, or C 2 -C 6 -dihydroxyalkyl;

particularly preferred R 2 is C 2 -C 6 -alkenyl, 5- or 6-membered heteroaryl, or Ci-Crhydroxyalkyl; also particularly preferred R 2 is C 3 -C 6 -cycloalkyl-C 1 -C 6 -alkylidenyl, C2-Crdihydroxyalkyl or 5- or 6-membered heteroaryl; ,

more preferred R 2 is CH=CH-CH 3 , CH=C(CH 2 ) 3 , or CH=C(CH 2 ) 4 ;

also more preferred R 2 is 2-furyl, 3-furyl, 2-methyl-3-furyl, 3-methyl-2-furyl, 4-methyloxazol-5- yl, CHOH-CHOH-CeHs, or CHOH-CHOH-2-furyl;

most preferred R 2 is CH=CH-CH 3 , CH=C(CH 2 ) 3 , 2-furyl, 3-furyl, CHOH-CHOH-C 6 H 5 , CHOH- CHOH-2-furyl, or 4-methyl-5-oxazolyl.

wherein acyclic aliphatic groups of R 2 are unsubstituted or substituted by R d .

A is preferably CR 3 or NR 3A ;

particularly preferred A is CR 3 ;

also particularly preferred A is NR 3A ;

Z is preferably pyridine, pyrrole, furan, or thiophene;

particularly preferred Z is pyridine;

also particularly preferred Z is pyrrole, furan, or thiophene; more preferred Z is pyridine, furan, or thiophene;

most preferred Z is selected from groups A to G, as defined above;

specially preferred Z is A;

also specially preferred Z is C;

R 3 is preferably halogen, CN, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

particularly preferred R 3 is halogen or CH3;

R 3A is preferably H or C 1 -C 6 -alkyl;

particularly preferred R 3A is H or CH 3 ;

m is preferably 0 or 1 ;

R 4 is preferably halogen or CF3.

Also preferred are the pyrimidine compounds of formula (I), wherein

R 1 is C-C3H5;

R 2 is Ci-Ce-alkyl, C2-C 6 -alkenyl, C 3 -C 6 -cycloalkyl-Ci-Ce-alkyl, C 3 -C 6 -cycloalkenyl-Ci-Ce- alkyl, C 3 -C 6 -cycloalkyl-C 1 -C 6 -alkylidenyl, C 1 -C 6 -hydroxyalkyl, hydroxycarbonyl-C 1 -C 6 -alkyl, hydroxycarbonyl-C 1 -C 6 -haloalkyl, C 1 -C 6 -alkoxycarbonyl-C 1 -C 6 -alkyl, C 1 -C 6 -alkoxycarbonyl-Ci- C6-haloalkyl, or 5- membered heteroaryl;

wherein OH groups of R 2 are unsubstituted or substituted by R b ,

cyclic groups of R 2 are unsubstituted or substituted by R c , and

acyclic aliphatic groups of R 2 are unsubstituted or substituted by R d ;

R b is Ci-Ce-alkyl;

R c is Ci-Ce-alkyl or OH;

R d is phenyl or 5- or 6- membered heteroaryl;

wherein the substituent R d is unsubstituted or substituted by R e ;

R e is halogen, CN, N0 2 , C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, OH, C 1 -C 6 -alkoxy, C 1 -C 6 -haloalkoxy, Ci-Ce-alkylsulfonyl;

Z is A, E, G, or F;

X is S;

R 3 is CI, Br, F, I, CH 3 , or OCF 3 ;

m is 0 or 1 ;

R 4 is Br.

Also preferred are the pyrimidine compounds of formula (I), wherein

R 1 is C-C3H5;

R 2 is Ci-Ce-alkyl, C 2 -C 6 -alkenyl, C 3 -C 6 -cycloalkyl-Ci-Ce-alkyl, C 3 -C 6 -cycloalkenyl-Ci-Ce- alkyl, C 3 -C 6 -cycloalkyl-C 1 -C 6 -alkylidenyl, C 1 -C 6 -hydroxyalkyl, hydroxycarbonyl-C 1 -C 6 -alkyl, hydroxycarbonyl-C 1 -C 6 -haloalkyl, C 1 -C 6 -alkoxycarbonyl-C 1 -C 6 -alkyl, C 1 -C 6 -alkoxycarbonyl-Ci- C6-haloalkyl, or 5- membered heteroaryl;

wherein OH groups of R 2 are unsubstituted or substituted by R b ,

cyclic groups of R 2 are unsubstituted or substituted by R c , and

acyclic aliphatic groups of R 2 are unsubstituted or substituted by R d ;

R b is Ci-Ce-alkyl;

R c is Ci-Ce-alkyl or OH;

R d is phenyl or 5- or 6- membered heteroaryl;

wherein the substituent R d is unsubstituted or substituted by R e ; R e is halogen, CN, N0 2 , C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, OH, C 1 -C 6 -alkoxy, C 1 -C 6 -haloalkoxy, C 1 -C 6 -alkylsulfonyl;

Z is A or C;

R 3 is CI, Br, F, I, CH 3 , or OCF 3 ;

m is 0 or 1 ;

R 4 is halogen, preferably Br.

Also preferred are the pyrimidine compounds of formula (I), wherein

R 1 is c-C 3 H 5 ;

R2 is R2-9, R2-10 or R 2 -15, preferably R 2 -9;

Z is A or C;

R 3 is R 3 is halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkoxy, or C 1 -C 6 -haloalkoxy;

preferrably C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -haloalkoxy; more preferrably CI, Br, F, I, CH3, or OCF 3 ;

m is 0 or 1 ;

R 4 is F, Br, CI, CHF 2 , CH 3 , CF 3 , or C2H5.

Also preferred are the pyrimidine compounds of formula (1.1) (corresponds to pyrimidine compounds of formula (I) wherein R 2 is CH=CH-CH3), and their use as herbicide,

R

wherein the dotted line (----- ) is a single bond or a double bond;

R 1 is C 3 -C 6 -cycloalkyl, C 1 -C 6 -alkyl, or C 1 -C 6 -alkoxy;

A is CR 3 or NR 3A ;

R 3 is halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

R 3A is H or Ci-Ce-alkyl;

Z is pyridine, thiophene, furan, or pyrrol;

m is 0 or 1 ;

R 4 is F, CI, CHF 2 , CF 3 , CH 3 , or C2H5.

Also preferred are the pyrimidine compounds of formula (I.2) (corresponds to pyrimidine compounds of formula (I) wherein R 2 is CH=C(CH2) 3 ), and their use as herbicide,

wherein the dotted line (----- ) is a single bond or a double bond;

R 1 is C 3 -C6-cycloalkyl, C 1 -C 6 -alkyl, or C 1 -C 6 -alkoxy;

A is CR 3 ;

R 3 is halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

Z is pyridine, thiophene, furan, or pyrrol;

m is 0 or 1 ; R 4 is F, CI, CHF 2 , CH 3 , CF 3 , or C 2 H 5 .

Also preferred are the pyrimidine compounds of formula (1.3) (corresponds to pyrimidine compounds of formula (I) wherein R 2 is CH=C(CH2)4), and their use as herbicide,

wherein the dotted line (----- ) is single bond or double bond;

R 1 is C 3 -C 6 -cycloalkyl, C 1 -C 6 -alkyl, or C 1 -C 6 -alkoxy;

A is CR 3 ;

R 3 is halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

Z is pyridine, thiophene, furan, or pyrrol;

m is 0 or 1 ;

R 4 is F, CI, CHF 2 , CH 3 , CF 3 , or C 2 H 5 .

Also preferred are the pyrimidine compounds of formula (I.4) (corresponds to pyrimidine compounds of formula (I) wherein R 2 is 2-furyl), and their use as herbicide,

wherein the dotted line (----- ) is a single bond or a double bond;

R 1 is C 3 -C 6 -cycloalkyl, C 1 -C 6 -alkyl, or C 1 -C 6 -alkoxy;

A is CR 3 ;

R 3 is halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

Z is pyridine, thiophene, furan, or pyrrol;

m is 0 or 1 ;

R 4 is F, CI, CHF 2 , CH 3 , CF 3 , or C 2 H 5 .

Also preferred are the pyrimidine compounds of formula (1.5) (corresponds to pyrimidine compounds of formula (I) wherein R 2 is 3-furyl), and their use as herbicide,

wherein the dotted line (----- ) is a single bond or a double bond;

R 1 is C 3 -C6-cycloalkyl, C 1 -C 6 -alkyl, or C 1 -C 6 -alkoxy;

A is CR 3 ;

R 3 is halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

Z is pyridine, thiophene, furan, or pyrrol;

m is 0 or 1 ; R 4 is F, CI, CHF 2 , CH 3 , CF 3 , or C 2 H 5 .

Also preferred are the pyrimidine compounds of formula (1.6) (corresponds to pyrimidine compounds of formula (I) wherein R 2 is 3-methyl-2-furyl), and their use as herbicide,

R

wherein the dotted line (----- ) is a single bond or a double bond;

R 1 is C 3 -C 6 -cycloalkyl, C 1 -C 6 -alkyl, or C 1 -C 6 -alkoxy;

A is CR 3 ;

R 3 is halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

Z is pyridine, thiophene, furan, or pyrrol;

m is 0 or 1 ;

R 4 is F, CI, CHF 2 , CH 3 , CF 3 , or C 2 H 5 .

Also preferred are the pyrimidine compounds of formula (1.7) (corresponds to pyrimidine compounds of formula (I) wherein R 2 is 2-methyl-3-furyl), and their use as herbicide,

wherein the dotted line (----- ) is a single bond or a double bond;

R 1 is C 3 -C 6 -cycloalkyl, C 1 -C 6 -alkyl, or C 1 -C 6 -alkoxy;

A is CR 3 ;

R 3 is halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

Z is pyridine, thiophene, furan, or pyrrol;

m is 0 or 1 ;

R 4 is F, CI, CHF 2 , CH 3 , CF 3 , or C 2 H 5 .

Also preferred are the pyrimidine compounds of formula (1.8) (corresponds to pyrimidine compounds of formula (I) wherein R 2 is CHOH-CHOH-C6H5), and their use as herbicide,

HO

wherein the dotted line (----- ) is a single bond or a double bond;

R 1 is C 3 -C6-cycloalkyl, C 1 -C 6 -alkyl, or C 1 -C 6 -alkoxy;

A is CR 3 ;

R 3 is halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

Z is pyridine, thiophene, furan, or pyrrol;

m is 0 or 1 ; R 4 is F, CI, CHF 2 , CH 3 , CF 3 , or C 2 H 5 .

Also preferred are the pyrimidine compounds of formula (1.9) (corresponds to pyrimidine compounds of formula (I) wherein R 2 is CHOH-CHOH-2-furyl), and their use as herbicide,

wherein the dotted line (----- ) is a single bond or a double bond;

R 1 is C 3 -C 6 -cycloalkyl, C 1 -C 6 -alkyl, or C 1 -C 6 -alkoxy;

A is CR 3 ;

R 3 is halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

Z is pyridine, thiophene, furan, or pyrrol;

m is 0 or 1 ;

R 4 is F, CI, CHF 2 , CH 3 , CF 3 , or C 2 H 5 .

Also preferred are the pyrimidine compounds of formula (1.10) (corresponds to pyrimidine compounds of formula (I) wherein R 2 is 4-methyl-5-oxazolyl), and their use as herbicide,

wherein the dotted line (----- ) is a single bond or a double bond;

R 1 is C 3 -C 6 -cycloalkyl, C 1 -C 6 -alkyl, or C 1 -C 6 -alkoxy;

A is CR 3 ;

R 3 is halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

Z is pyridine, thiophene, furan, or pyrrol;

m is 0 or 1 ;

R 4 is F, CI, CHF 2 , CH 3 , CF 3 , or C 2 H 5

Also preferred are the pyrimidine compounds of formula (1.11) (corresponds to pyrimidine compounds of formula (I) wherein R 2 is R 2 -9), and their use as herbicide,

Y

wherein the dotted line (----- ) is a single bond or a double bond;

X and Y independently are selected from H, CH 3 , C 2 H5, n-propyl, iso-propyl, iso-butyl, n-butyl 2-butyl, t-butyl, OH, OCH 3 , SCH 3 , S(0)CH 3 , S(0) 2 CH 3 , CN, F, CI, Br, I, CH 2 CF 3 , CF 2 CF 3 , CF 2 CH 3 , CF 3 , CF 2 H, OCF 2 H, and OCF 3 ;

R 1 is C 3 -C6-cycloalkyl, C 1 -C 6 -alkyl, or C 1 -C 6 -alkoxy; preferably c-C 3 H 5 ; A is CR 3 ;

R 3 is halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

Z is pyridine, thiophene, furan, or pyrrol;

m is 0 or 1 ;

R 4 is F, Br, CI, CHF 2 , CH 3 , CF 3 , or C 2 H 5 ; preferably F, CI, CHF 2 , CH 3 , CF 3 , or C 2 H 5 ; also preferably Br.

Also preferred are the pyrimidine compounds of formula (1.1 1. A) (corresponds to pyrimidine compounds of formula (I), wherein wherein R 2 is R 2 -9 and Z is A) and their use as herbicide,

Y

wherein

X and Y independently are selected from H, CH 3 , C 2 H5, n-propyl, iso-propyl, iso-butyl, n-butyl, 2-butyl, t-butyl, OH, OCH 3 , SCH 3 , S(0)CH 3 , S(0) 2 CH 3 , CN, F, CI, Br, I, CH 2 CF 3 , CF 2 CF 3 , CF 2 CH 3 , CF 3 , CF 2 H, OCF 2 H, and OCF 3 ;

R 1 is C 3 -C6-cycloalkyl, C 1 -C 6 -alkyl, or C 1 -C 6 -alkoxy; preferably c-C 3 H5;

R 3 is halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

m is 0 or 1 ;

R 4 is F, Br, CI, CHF 2 , CH 3 , CF 3 , or C 2 H 5 .

Also preferred are the pyrimidine compounds of formula (1.1 1.C) (corresponds to pyrimidine compounds of formula (I), wherein wherein R 2 is R 2 -9 and Z is C) and their use as herbicide,

Y

wherein

X and Y independently are selected from H, CH 3 , C 2 H5, n-propyl, iso-propyl, iso-butyl, n-butyl, 2-butyl, t-butyl, OH, OCH 3 , SCH 3 , S(0)CH 3 , S(0) 2 CH 3 , CN, F, CI, Br, I, CH 2 CF 3 , CF 2 CF 3 , CF 2 CH 3 , CF 3 , CF 2 H, OCF 2 H, and OCF 3 ;

R 1 is C 3 -C6-cycloalkyl, C 1 -C 6 -alkyl, or C 1 -C 6 -alkoxy; preferably c-C 3 H 5 ;

R 3 is halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, or C 1 -C 6 -alkoxy;

m is 0 or 1 ;

R 4 is F, Br, CI, CHF 2 , CH 3 , CF 3 , or C 2 H 5 .

Particular preference is given to the pyrimidine compounds of formula I.A to I.G (corresponds to pyrimidine compounds of formula (I)), and their use as herbicide, wherein X is O, NR 3A , or S.

Preferred compounds of formula I, and their use as herbicide, are the compounds of the formulae I .A to I.G wherein

R 1 is C 2 H 5 , C-C3H5, C-C4H7, or OCH3;

R 2 is CH=CH-CH 3 , CH=C(CH 2 ) 3 , CH=C(CH 2 )4, 2-furyl, 3-furyl, 4-methyl-2-fury, 2-methyl-3-furyl CHOH-CHOH-CeHs, CHOH-CHOH-2-furyl or 4-methyl-5-oxazolyl;

R 3 is CH 3 , OCH3, CI, Br, CHF 2 , F, or I;

X is O, S, or NR 3A ;

m is 0 or 1 ;

R 4 is F or CF 3 .

Each of the groups mentioned for a substituent in the tables is furthermore per se,

independently of the combination in which it is mentioned, a particularly preferred aspect of the substituent in question.

According to particularly preferred embodiment of the compound of formula I, and their use as herbicide, compounds of the invention are the compounds of the formulae l-A to l-G that are compiled in the Tables 1 to 26, wherein the meaning for the combination of variables R 1 , R 2 , and R 3 for each individual compound of tables 1 to 26 corresponds to each line of Table A. The term "formula" used in below tables 1 to 26 denotes "compounds of formula".

The specific number for each single compound is deductible as follows:

Compound 1.1 .1-3 e.g. comprises the compound of formula 1.1 from Table 1 and line I-3 from Table A;

According to another particularly preferred embodiment of the compounds of formula I and their use as herbicide, compounds of the invention are the compounds of formulae I.A or I.C, wherein

R 1 is C2H5, C-C3H5, C-C4H7, or OCH3;

R 2 is selected from R 2 -9.1 to R 2 -9.676 from Table R 2 -9, R 2 -10.1 to R 2 -10.676 from Table R 2 - 10, and R 2 -15.1 to R 2 -15.676 from Table R 2 -15;

R 3 is CH 3 , OCH3, CI, Br, CHF 2 , F, or I;

m is 0 or 1 ;

R 4 is F.

According to another particularly preferred embodiment of the compounds of formula I and their use as herbicide, compounds of the invention are the compounds of formulae I.A that are compiled in tables 27 to 2054, wherein the meaning for the combination of variables R 1 , R 3 , m, and R 4 for each individual compound of tables 27 to 2054 corresponds to each line of Table A1 . Each of the groups mentioned for a substituent in the tables is furthermore per se,

independently of the combination in which it is mentioned, a particularly preferred aspect of the substituent in question.

The term "formula" used in below tables 27 to 2054 denotes "compounds of formula".

Table 27. Compounds of formula I.A, wherein R 2 is R 2 -9.17(=formula 1.27).

Table 28. Compounds of formula I.A, wherein R 2 is R 2 -9.18(=formula 1.28).

Table 29. Compounds of formula I.A, wherein R 2 is R 2 -9.19(=formula 1.29).

Table 30. Compounds of formula I. A, wherein R 2 is R 2 -9.20(=formula 1.30).

Table 31. Compounds of formula I.A, wherein R 2 is R 2 -9.21 (=formula 1.31 ).

Table 32. Compounds of formula I. A, wherein R 2 is R 2 -9.22(=formula 1.32).

Table 33. Compounds of formula I. A, wherein R 2 is R 2 -9.23(=formula 1.33). Tab e 34. Compounds wherein R 2 s R 2 -9.24 =formu .34).

Tab e 35. Compounds wherein R 2 s R 2 -9.25 =formu .35).

Tab e 36. Compounds wherein R 2 s R 2 -9.26 =formu .36).

Tab e 37. Compounds wherein R 2 s R 2 -9.27 =formu .37).

Tab e 38. Compounds wherein R 2 s R 2 -9.28 =formu .38).

Tab e 39. Compounds wherein R 2 s R 2 -9.29 =formu .39).

Tab e 40. Compounds wherein R 2 s R 2 -9.30 =formu .40).

Tab e 41. Compounds wherein R 2 s R 2 -9.31 =formu .41).

Tab e 42. Compounds wherein R 2 s R 2 -9.32 =formu .42).

Tab e 43. Compounds wherein R 2 s R 2 -9.33 =formu .43).

Tab e 44. Compounds wherein R 2 s R 2 -9.34 =formu .44).

Tab e 45. Compounds wherein R 2 s R 2 -9.35 =formu .45).

Tab e 46. Compounds wherein R 2 s R 2 -9.36 =formu .46).

Tab e 47. Compounds wherein R 2 s R 2 -9.37 =formu .47).

Tab e 48. Compounds wherein R 2 s R 2 -9.38 =formu .48).

Tab e 49. Compounds wherein R 2 s R 2 -9.39 =formu .49).

Tab e 50. Compounds wherein R 2 s R 2 -9.40 =formu .50).

Tab e 51. Compounds wherein R 2 s R 2 -9.41 =formu .51).

Tab e 52. Compounds wherein R 2 s R 2 -9.42 =formu .52).

Tab e 53. Compounds wherein R 2 s R 2 -9.43 =formu .53).

Tab e 54. Compounds wherein R 2 s R 2 -9.44 =formu .54).

Tab e 55. Compounds wherein R 2 s R 2 -9.45 =formu .55).

Tab e 56. Compounds wherein R 2 s R 2 -9.46 =formu .56).

Tab e 57. Compounds wherein R 2 s R 2 -9.47 =formu .57).

Tab e 58. Compounds wherein R 2 s R 2 -9.48 =formu .58).

Tab e 59. Compounds wherein R 2 s R 2 -9.49 =formu .59).

Tab e 60. Compounds wherein R 2 s R 2 -9.50 =formu .60).

Tab e 61. Compounds wherein R 2 s R 2 -9.51 =formu .61).

Tab e 62. Compounds wherein R 2 s R 2 -9.52 =formu .62).

Tab e 63. Compounds wherein R 2 s R 2 -9.53 =formu .63).

Tab e 64. Compounds wherein R 2 s R 2 -9.54 =formu .64).

Tab e 65. Compounds wherein R 2 s R 2 -9.55 =formu .65).

Tab e 66. Compounds wherein R 2 s R 2 -9.56 =formu .66).

Tab e 67. Compounds wherein R 2 s R 2 -9.57 =formu .67).

Tab e 68. Compounds wherein R 2 s R 2 -9.58 =formu .68).

Tab e 69. Compounds wherein R 2 s R 2 -9.59 =formu .69).

Tab e 70. Compounds wherein R 2 s R 2 -9.60 =formu .70).

Tab e 71. Compounds wherein R 2 s R 2 -9.61 =formu .71).

Tab e 72. Compounds wherein R 2 s R 2 -9.62 =formu .72).

Tab e 73. Compounds wherein R 2 s R 2 -9.63 =formu .73).

Tab e 74. Compounds wherein R 2 s R 2 -9.64 =formu .74).

Tab e 75. Compounds wherein R 2 s R 2 -9.65 =formu .75).

Tab e 76. Compounds wherein R 2 s R 2 -9.66 =formu .76).

Tab e 77. Compounds wherein R 2 s R 2 -9.67 =formu .77). Table 78. Compounds of formu a I .A, wherein R2 is R2-9.68(= formula 1.78).

Table 79. Compounds of formu a I .A, wherein R2 is R2-9.69(= formula 1 .79).

Table 80. Compounds of formu a I .A, wherein R2 is R2-9.70(= formula 1 .80).

Table 81. Compounds of formu a I .A, wherein R2 is R2-9.71 (= formula 1 .81 ).

Table 82. Compounds of formu a I .A, wherein R2 is R2-9.72(= formula 1 .82).

Table 83. Compounds of formu a I .A, wherein R2 is R2-9.73(= formula 1 .83).

Table 84. Compounds of formu a I .A, wherein R2 is R2-9.74(= formula 1 .84).

Table 85. Compounds of formu a I .A, wherein R2 is R2-9.75(= formula 1 .85).

Table 86. Compounds of formu a I .A, wherein R2 is R2-9.76(= formula 1 .86).

Table 87. Compounds of formu a I .A, wherein R2 is R2-9.77(= formula 1 .87).

Table 88. Compounds of formu a I .A, wherein R2 is R2-9.78(= formula 1 .88).

Table 89. Compounds of formu a I .A, wherein R2 is R2-9.79(= formula 1 .89).

Table 90. Compounds of formu a I .A, wherein R2 is R2-9.80(= formula 1 .90).

Table 91. Compounds of formu a I .A, wherein R2 is R2-9.81 (= formula 1 .91 ).

Table 92. Compounds of formu a I .A, wherein R2 is R2-9.82(= formula 1 .92).

Table 93. Compounds of formu a I .A, wherein R2 is R2-9.83(= formula 1 .93).

Table 94. Compounds of formu a I .A, wherein R2 is R2-9.84(= formula 1 .94).

Table 95. Compounds of formu a I .A, wherein R2 is R2-9.85(= formula 1 .95).

Table 96. Compounds of formu a I .A, wherein R2 is R2-9.86(= formula 1 .96).

Table 97. Compounds of formu a I .A, wherein R2 is R2-9.87(= formula 1 .97).

Table 98. Compounds of formu a I .A, wherein R2 is R2-9.88(= formula 1 .98).

Table 99. Compounds of formu a I .A, wherein R2 is R2-9.89(= formula 1 .99).

Table 100. Compounds of formu a I .A, wherein R2 is R2-9.90(= formula 1 .100).

Table 101 . Compounds of formu a I .A, wherein R2 is R2-9.91 (= formula 1 .101 ).

Table 102. Compounds of formu a I .A, wherein R2 is R2-9.92(= formula 1 .102).

Table 103. Compounds of formu a I .A, wherein R2 is R2-9.93(= formula 1 .103).

Table 104. Compounds of formu a I .A, wherein R2 is R2-9.94(= formula 1 .104).

Table 105. Compounds of formu a I .A, wherein R2 is R2-9.95(= formula 1 .105).

Table 106. Compounds of formu a I .A, wherein R2 is R2-9.96(= formula 1 .106).

Table 107. Compounds of formu a I .A, wherein R2 is R2-9.97(= formula 1 .107).

Table 108. Compounds of formu a I .A, wherein R2 is R2-9.98(= formula 1 .108).

Table 109. Compounds of formu a I .A, wherein R2 is R2-9.99(= formula 1 .109).

Table 1 10. Compounds of formu a I .A, wherein R2 is R2-9.100( =formula 1 .1 10).

Table 1 1 1 . Compounds of formu a I .A, wherein R2 is R2-9.101 ( =formula 1 .1 1 1 ).

Table 1 12. Compounds of formu a I .A, wherein R2 is R2-9.102( =formula 1 .1 12).

Table 1 13. Compounds of formu a I .A, wherein R2 is R2-9.103( =formula 1 .1 13).

Table 1 14. Compounds of formu a I .A, wherein R2 is R2-9.104( =formula 1 .1 14).

Table 1 15. Compounds of formu a I .A, wherein R2 is R2-9.105( =formula 1 .1 15).

Table 1 16. Compounds of formu a I .A, wherein R2 is R2-9.106( =formula 1 .1 16).

Table 1 17. Compounds of formu a I .A, wherein R2 is R2-9.107( =formula 1 .1 17).

Table 1 18. Compounds of formu a I .A, wherein R2 is R2-9.108( =formula 1 .1 18).

Table 1 19. Compounds of formu a I .A, wherein R2 is R2-9.109( =formula 1 .1 19).

Table 120. Compounds of formu a I .A, wherein R2 is R2-9.1 10( =formula 1 .120).

Table 121 . Compounds of formu a I .A, wherein R2 is R2-9.1 1 1 ( =formula 1 .121 ). Table 122. Compounds of formu a I .A, wherein R2 is R2-9.1 12I = Formu a 1 .122).

Table 123. Compounds of formu a I .A, wherein R2 is R2-9.1 13I = Formu a 1 .123).

Table 124. Compounds of formu a I .A, wherein R2 is R2-9.1 14I = Formu a 1 .124).

Table 125. Compounds of formu a I .A, wherein R2 is R2-9.1 15I = Formu a 1 .125).

Table 126. Compounds of formu a I .A, wherein R2 is R2-9.1 16I = Formu a 1 .126).

Table 127. Compounds of formu a I .A, wherein R2 is R2-9.1 17I = Formu a 1 .127).

Table 128. Compounds of formu a I .A, wherein R2 is R2-9.1 18I = Formu a 1 .128).

Table 129. Compounds of formu a I .A, wherein R2 is R2-9.1 19I = Formu a 1 .129).

Table 130. Compounds of formu a I .A, wherein R2 is R2-9.120I = Formu a 1 .130).

Table 131 . Compounds of formu a I .A, wherein R2 is R2-9.121 I = Formu a 1 .131 ).

Table 132. Compounds of formu a I .A, wherein R2 is R2-9.122I = Formu a 1 .132).

Table 133. Compounds of formu a I .A, wherein R2 is R2-9.123I = Formu a 1 .133).

Table 134. Compounds of formu a I .A, wherein R2 is R2-9.124I = Formu a 1 .134).

Table 135. Compounds of formu a I .A, wherein R2 is R2-9.125I = Formu a 1 .135).

Table 136. Compounds of formu a I .A, wherein R2 is R2-9.126I = Formu a 1 .136).

Table 137. Compounds of formu a I .A, wherein R2 is R2-9.127I = Formu a 1 .137).

Table 138. Compounds of formu a I .A, wherein R2 is R2-9.128I = Formu a 1 .138).

Table 139. Compounds of formu a I .A, wherein R2 is R2-9.129I = Formu a 1 .139).

Table 140. Compounds of formu a I .A, wherein R2 is R2-9.130I = Formu a 1 .140).

Table 141 . Compounds of formu a I .A, wherein R2 is R2-9.131 I = Formu a 1 .141 ).

Table 142. Compounds of formu a I .A, wherein R2 is R2-9.132I = Formu a 1 .142).

Table 143. Compounds of formu a I .A, wherein R2 is R2-9.133I = Formu a 1 .143).

Table 144. Compounds of formu a I .A, wherein R2 is R2-9.134I = Formu a 1 .144).

Table 145. Compounds of formu a I .A, wherein R2 is R2-9.135I = Formu a 1 .145).

Table 146. Compounds of formu a I .A, wherein R2 is R2-9.136I = Formu a 1 .146).

Table 147. Compounds of formu a I .A, wherein R2 is R2-9.137I = Formu a 1 .147).

Table 148. Compounds of formu a I .A, wherein R2 is R2-9.138I = Formu a 1 .148).

Table 149. Compounds of formu a I .A, wherein R2 is R2-9.139I = Formu a 1 .149).

Table 150. Compounds of formu a I .A, wherein R2 is R2-9.140I = Formu a 1 .150).

Table 151 . Compounds of formu a I .A, wherein R2 is R2-9.141 I = Formu a 1 .151 ).

Table 152. Compounds of formu a I .A, wherein R2 is R2-9.142I = Formu a 1 .152).

Table 153. Compounds of formu a I .A, wherein R2 is R2-9.143I = Formu a 1 .153).

Table 154. Compounds of formu a I .A, wherein R2 is R2-9.144I = Formu a 1 .154).

Table 155. Compounds of formu a I .A, wherein R2 is R2-9.145I = Formu a 1 .155).

Table 156. Compounds of formu a I .A, wherein R2 is R2-9.146I = Formu a 1 .156).

Table 157. Compounds of formu a I .A, wherein R2 is R2-9.147I = Formu a 1 .157).

Table 158. Compounds of formu a I .A, wherein R2 is R2-9.148I = Formu a 1 .158).

Table 159. Compounds of formu a I .A, wherein R2 is R2-9.149I = Formu a 1 .159).

Table 160. Compounds of formu a I .A, wherein R2 is R2-9.150I = Formu a 1 .160).

Table 161 . Compounds of formu a I .A, wherein R2 is R2-9.151 I = Formu a 1 .161 ).

Table 162. Compounds of formu a I .A, wherein R2 is R2-9.152I = Formu a 1 .162).

Table 163. Compounds of formu a I .A, wherein R2 is R2-9.153I = Formu a 1 .163).

Table 164. Compounds of formu a I .A, wherein R2 is R2-9.154I = Formu a 1 .164).

Table 165. Compounds of formu a I .A, wherein R2 is R2-9.155I = Formu a 1 .165). Table 166. Compounds of formu a I .A, wherein R2 is R2-9.156I = Formu a ' .166).

Table 167. Compounds of formu a I .A, wherein R2 is R2-9.157I = Formu a ' .167).

Table 168. Compounds of formu a I .A, wherein R2 is R2-9.158I = Formu a ' .168).

Table 169. Compounds of formu a I .A, wherein R2 is R2-9.159I = Formu a ' .169).

Table 170. Compounds of formu a I .A, wherein R2 is R2-9.160I = Formu a ' .170).

Table 171 . Compounds of formu a I .A, wherein R2 is R2-9.161 I = Formu a ' .171 ).

Table 172. Compounds of formu a I .A, wherein R2 is R2-9.162I = Formu a ' .172).

Table 173. Compounds of formu a I .A, wherein R2 is R2-9.163I = Formu a ' .173).

Table 174. Compounds of formu a I .A, wherein R2 is R2-9.164I = Formu a ' .174).

Table 175. Compounds of formu a I .A, wherein R2 is R2-9.165I = Formu a ' .175).

Table 176. Compounds of formu a I .A, wherein R2 is R2-9.166I = Formu a ' .176).

Table 177. Compounds of formu a I .A, wherein R2 is R2-9.167I = Formu a ' .177).

Table 178. Compounds of formu a I .A, wherein R2 is R2-9.168I = Formu a ' .178).

Table 179. Compounds of formu a I .A, wherein R2 is R2-9.169I = Formu a ' .179).

Table 180. Compounds of formu a I .A, wherein R2 is R2-9.170I = Formu a ' .180).

Table 181 . Compounds of formu a I .A, wherein R2 is R2-9.171 I = Formu a ' .181 ).

Table 182. Compounds of formu a I .A, wherein R2 is R2-9.172I = Formu a ' .182).

Table 183. Compounds of formu a I .A, wherein R2 is R2-9.173I = Formu a ' .183).

Table 184. Compounds of formu a I .A, wherein R2 is R2-9.174I = Formu a ' .184).

Table 185. Compounds of formu a I .A, wherein R2 is R2-9.175I = Formu a ' .185).

Table 186. Compounds of formu a I .A, wherein R2 is R2-9.176I = Formu a ' .186).

Table 187. Compounds of formu a I .A, wherein R2 is R2-9.177I = Formu a ' .187).

Table 188. Compounds of formu a I .A, wherein R2 is R2-9.178I = Formu a ' .188).

Table 189. Compounds of formu a I .A, wherein R2 is R2-9.179I = Formu a ' .189).

Table 190. Compounds of formu a I .A, wherein R2 is R2-9.180I = Formu a ' .190).

Table 191 . Compounds of formu a I .A, wherein R2 is R2-9.181 I = Formu a ' .191 ).

Table 192. Compounds of formu a I .A, wherein R2 is R2-9.182I = Formu a ' .192).

Table 193. Compounds of formu a I .A, wherein R2 is R2-9.183I = Formu a ' .193).

Table 194. Compounds of formu a I .A, wherein R2 is R2-9.184I = Formu a ' .194).

Table 195. Compounds of formu a I .A, wherein R2 is R2-9.185I = Formu a ' .195).

Table 196. Compounds of formu a I .A, wherein R2 is R2-9.186I = Formu a ' .196).

Table 197. Compounds of formu a I .A, wherein R2 is R2-9.187I = Formu a ' .197).

Table 198. Compounds of formu a I .A, wherein R2 is R2-9.188I = Formu a ' .198).

Table 199. Compounds of formu a I .A, wherein R2 is R2-9.189I = Formu a ' .199).

Table 200. Compounds of formu a I .A, wherein R2 is R2-9.190I = Formu a ' .200).

Table 201 . Compounds of formu a I .A, wherein R2 is R2-9.191 I = Formu a ' .201 ).

Table 202. Compounds of formu a I .A, wherein R2 is R2-9.192I = Formu a ' .202).

Table 203. Compounds of formu a I .A, wherein R2 is R2-9.193I = Formu a ' .203).

Table 204. Compounds of formu a I .A, wherein R2 is R2-9.194I = Formu a ' .204).

Table 205. Compounds of formu a I .A, wherein R2 is R2-9.195I = Formu a ' .205).

Table 206. Compounds of formu a I .A, wherein R2 is R2-9.196I = Formu a ' .206).

Table 207. Compounds of formu a I .A, wherein R2 is R2-9.197I = Formu a ' .207).

Table 208. Compounds of formu a I .A, wherein R2 is R2-9.198I = Formu a ' .208).

Table 209. Compounds of formu a I .A, wherein R2 is R2-9.199I = Formu a ' .209). Table 210. Compounds of formu a I .A, wherein R2 is R2- -9.200I =formu a 1.210)

Table 211. Compounds of formu a I .A, wherein R2 is R2- 9.2011 =formu a 1.211)

Table 212. Compounds of formu a I .A, wherein R2 is R2- 9.2021 =formu a 1.212)

Table 213. Compounds of formu a I .A, wherein R2 is R2- 9.2031 =formu a 1.213)

Table 214. Compounds of formu a I .A, wherein R2 is R2- 9.2041 =formu a 1.214)

Table 215. Compounds of formu a I .A, wherein R2 is R2- 9.2051 =formu a 1.215)

Table 216. Compounds of formu a I .A, wherein R2 is R2- 9.2061 =formu a 1.216)

Table 217. Compounds of formu a I .A, wherein R2 is R2- 9.2071 =formu a 1.217)

Table 218. Compounds of formu a I .A, wherein R2 is R2- 9.2081 =formu a 1.218)

Table 219. Compounds of formu a I .A, wherein R2 is R2- 9.2091 =formu a 1.219)

Table 220. Compounds of formu a I .A, wherein R2 is R2- 9.2101 =formu a 1.220)

Table 221. Compounds of formu a I .A, wherein R2 is R2- 9.2111 =formu a 1.221)

Table 222. Compounds of formu a I .A, wherein R2 is R2- 9.2121 =formu a 1.222)

Table 223. Compounds of formu a I .A, wherein R2 is R2- 9.2131 =formu a 1.223)

Table 224. Compounds of formu a I .A, wherein R2 is R2- 9.2141 =formu a 1.224)

Table 225. Compounds of formu a I .A, wherein R2 is R2- 9.2151 =formu a 1.225)

Table 226. Compounds of formu a I .A, wherein R2 is R2- 9.2161 =formu a 1.226)

Table 227. Compounds of formu a I .A, wherein R2 is R2- 9.2171 =formu a 1.227)

Table 228. Compounds of formu a I .A, wherein R2 is R2- 9.2181 =formu a 1.228)

Table 229. Compounds of formu a I .A, wherein R2 is R2- 9.2191 =formu a 1.229)

Table 230. Compounds of formu a I .A, wherein R2 is R2- 9.2201 =formu a 1.230)

Table 231. Compounds of formu a I .A, wherein R2 is R2- 9.2211 =formu a 1.231)

Table 232. Compounds of formu a I .A, wherein R2 is R2- 9.2221 =formu a 1.232)

Table 233. Compounds of formu a I .A, wherein R2 is R2- 9.2231 =formu a 1.233)

Table 234. Compounds of formu a I .A, wherein R2 is R2- 9.2241 =formu a 1.234)

Table 235. Compounds of formu a I .A, wherein R2 is R2- 9.2251 =formu a 1.235)

Table 236. Compounds of formu a I .A, wherein R2 is R2- 9.2261 =formu a 1.236)

Table 237. Compounds of formu a I .A, wherein R2 is R2- 9.2271 =formu a 1.237)

Table 238. Compounds of formu a I .A, wherein R2 is R2- 9.2281 =formu a 1.238)

Table 239. Compounds of formu a I .A, wherein R2 is R2- 9.2291 =formu a 1.239)

Table 240. Compounds of formu a I .A, wherein R2 is R2- 9.2301 =formu a 1.240)

Table 241. Compounds of formu a I .A, wherein R2 is R2- 9.2311 =formu a 1.241)

Table 242. Compounds of formu a I .A, wherein R2 is R2- 9.2321 =formu a 1.242)

Table 243. Compounds of formu a I .A, wherein R2 is R2- 9.2331 =formu a 1.243)

Table 244. Compounds of formu a I .A, wherein R2 is R2- 9.2341 =formu a 1.244)

Table 245. Compounds of formu a I .A, wherein R2 is R2- 9.2351 =formu a 1.245)

Table 246. Compounds of formu a I .A, wherein R2 is R2- 9.2361 =formu a 1.246)

Table 247. Compounds of formu a I .A, wherein R2 is R2- 9.2371 =formu a 1.247)

Table 248. Compounds of formu a I .A, wherein R2 is R2- 9.2381 =formu a 1.248)

Table 249. Compounds of formu a I .A, wherein R2 is R2- 9.2391 =formu a 1.249)

Table 250. Compounds of formu a I .A, wherein R2 is R2- 9.2401 =formu a 1.250)

Table 251. Compounds of formu a I .A, wherein R2 is R2- 9.2411 =formu a 1.251)

Table 252. Compounds of formu a I .A, wherein R2 is R2- 9.2421 =formu a 1.252)

Table 253. Compounds of formu a I .A, wherein R2 is R2- 9.243 (=formula 1.253) Table 254. Compounds of formu a I .A, wherein R2 is R2- -9.244I =formula ' 1 .254).

Table 255. Compounds of formu a I .A, wherein R2 is R2- -9.245I =formula ' 1 .255).

Table 256. Compounds of formu a I .A, wherein R2 is R2- -9.246I =formula ' 1 .256).

Table 257. Compounds of formu a I .A, wherein R2 is R2- -9.247I =formula ' 1 .257).

Table 258. Compounds of formu a I .A, wherein R2 is R2- -9.248I =formula ' 1 .258).

Table 259. Compounds of formu a I .A, wherein R2 is R2- -9.249I =formula ' 1 .259).

Table 260. Compounds of formu a I .A, wherein R2 is R2- -9.250I =formula ' 1 .260).

Table 261 . Compounds of formu a I .A, wherein R2 is R2- 9.2511 =formula ' 1 .261 ).

Table 262. Compounds of formu a I .A, wherein R2 is R2- 9.2521 =formula ' 1 .262).

Table 263. Compounds of formu a I .A, wherein R2 is R2- 9.2531 =formula ' 1 .263).

Table 264. Compounds of formu a I .A, wherein R2 is R2- 9.2541 =formula ' 1 .264).

Table 265. Compounds of formu a I .A, wherein R2 is R2- 9.2551 =formula ' 1 .265).

Table 266. Compounds of formu a I .A, wherein R2 is R2- 9.2561 =formula ' 1 .266).

Table 267. Compounds of formu a I .A, wherein R2 is R2- 9.2571 =formula ' 1 .267).

Table 268. Compounds of formu a I .A, wherein R2 is R2- 9.2581 =formula ' 1 .268).

Table 269. Compounds of formu a I .A, wherein R2 is R2- 9.2591 =formula ' 1 .269).

Table 270. Compounds of formu a I .A, wherein R2 is R2- 9.2601 =formula ' 1 .270).

Table 271 . Compounds of formu a I .A, wherein R2 is R2- 9.2611 =formula ' 1 .271 ).

Table 272. Compounds of formu a I .A, wherein R2 is R2- 9.2621 =formula ' 1 .272).

Table 273. Compounds of formu a I .A, wherein R2 is R2- 9.2631 =formula ' 1 .273).

Table 274. Compounds of formu a I .A, wherein R2 is R2- 9.2641 =formula ' 1 .274).

Table 275. Compounds of formu a I .A, wherein R2 is R2- 9.265 (=formula 1.275)

Table 276. Compounds of formu a I .A, wherein R2 is R2- 9.266 (=formula 1.276)

Table 277. Compounds of formu a I .A, wherein R2 is R2- 9.2671 =formula ' 1 .277).

Table 278. Compounds of formu a I .A, wherein R2 is R2- 9.2681 =formula ' 1 .278).

Table 279. Compounds of formu a I .A, wherein R2 is R2- 9.2691 =formula ' 1 .279).

Table 280. Compounds of formu a I .A, wherein R2 is R2- 9.270 (=formula 1.280)

Table 281 . Compounds of formu a I .A, wherein R2 is R2- 9.2711 =formula ' 1 .281 ).

Table 282. Compounds of formu a I .A, wherein R2 is R2- 9.2721 =formula ' 1 .282).

Table 283. Compounds of formu a I .A, wherein R2 is R2- 9.273 (=formula 1.283)

Table 284. Compounds of formu a I .A, wherein R2 is R2- 9.274 (=formula 1.284)

Table 285. Compounds of formu a I .A, wherein R2 is R2- 9.275 (=formula 1.285)

Table 286. Compounds of formu a I .A, wherein R2 is R2- 9.276 (=formula 1.286)

Table 287. Compounds of formu a I .A, wherein R2 is R2- 9.2771 =formula ' 1 .287).

Table 288. Compounds of formu a I .A, wherein R2 is R2- 9.2781 =formula ' 1 .288).

Table 289. Compounds of formu a I .A, wherein R2 is R2- 9.2791 =formula ' 1 .289).

Table 290. Compounds of formu a I .A, wherein R2 is R2- 9.2801 =formula ' 1 .290).

Table 291 . Compounds of formu a I .A, wherein R2 is R2- 9.2811 =formula ' 1 .291 ).

Table 292. Compounds of formu a I .A, wherein R2 is R2- 9.2821 =formula ' 1 .292).

Table 293. Compounds of formu a I .A, wherein R2 is R2- 9.2831 =formula ' 1 .293).

Table 294. Compounds of formu a I .A, wherein R2 is R2- 9.2841 =formula ' 1 .294).

Table 295. Compounds of formu a I .A, wherein R2 is R2- 9.2851 =formula ' 1 .295).

Table 296. Compounds of formu a I .A, wherein R2 is R2- 9.2861 =formula ' 1 .296).

Table 297. Compounds of formu a I .A, wherein R2 is R2- 9.2871 =formula ' 1 .297). Table 298. Compounds of formu a I .A, wherein R2 is R2- -9.288I =formu a 1.298)

Table 299. Compounds of formu a I .A, wherein R2 is R2- -9.289I =formu a 1.299)

Table 300. Compounds of formu a I .A, wherein R2 is R2- -9.290I =formu a 1.300)

Table 301. Compounds of formu a I .A, wherein R2 is R2- 9.2911 =formu a 1.301)

Table 302. Compounds of formu a I .A, wherein R2 is R2- 9.2921 =formu a 1.302)

Table 303. Compounds of formu a I .A, wherein R2 is R2- 9.2931 =formu a 1.303)

Table 304. Compounds of formu a I .A, wherein R2 is R2- 9.2941 =formu a 1.304)

Table 305. Compounds of formu a I .A, wherein R2 is R2- 9.2951 =formu a 1.305)

Table 306. Compounds of formu a I .A, wherein R2 is R2- 9.2961 =formu a 1.306)

Table 307. Compounds of formu a I .A, wherein R2 is R2- 9.2971 =formu a 1.307)

Table 308. Compounds of formu a I .A, wherein R2 is R2- 9.2981 =formu a 1.308)

Table 309. Compounds of formu a I .A, wherein R2 is R2- 9.2991 =formu a 1.309)

Table 310. Compounds of formu a I .A, wherein R2 is R2- 9.300 (=formula 1.310)

Table 311. Compounds of formu a I .A, wherein R2 is R2- 9.3011 =formu a 1.311)

Table 312. Compounds of formu a I .A, wherein R2 is R2- 9.3021 =formu a 1.312)

Table 313. Compounds of formu a I .A, wherein R2 is R2- 9.3031 =formu a 1.313)

Table 314. Compounds of formu a I .A, wherein R2 is R2- 9.3041 =formu a 1.314)

Table 315. Compounds of formu a I .A, wherein R2 is R2- 9.3051 =formu a 1.315)

Table 316. Compounds of formu a I .A, wherein R2 is R2- 9.3061 =formu a 1.316)

Table 317. Compounds of formu a I .A, wherein R2 is R2- 9.3071 =formu a 1.317)

Table 318. Compounds of formu a I .A, wherein R2 is R2- 9.3081 =formu a 1.318)

Table 319. Compounds of formu a I .A, wherein R2 is R2- 9.3091 =formu a 1.319)

Table 320. Compounds of formu a I .A, wherein R2 is R2- 9.3101 =formu a 1.320)

Table 321. Compounds of formu a I .A, wherein R2 is R2- 9.3111 =formu a 1.321)

Table 322. Compounds of formu a I .A, wherein R2 is R2- 9.3121 =formu a 1.322)

Table 323. Compounds of formu a I .A, wherein R2 is R2- 9.3131 =formu a 1.323)

Table 324. Compounds of formu a I .A, wherein R2 is R2- 9.3141 =formu a 1.324)

Table 325. Compounds of formu a I .A, wherein R2 is R2- 9.3151 =formu a 1.325)

Table 326. Compounds of formu a I .A, wherein R2 is R2- 9.3161 =formu a 1.326)

Table 327. Compounds of formu a I .A, wherein R2 is R2- 9.3171 =formu a 1.327)

Table 328. Compounds of formu a I .A, wherein R2 is R2- 9.3181 =formu a 1.328)

Table 329. Compounds of formu a I .A, wherein R2 is R2- 9.3191 =formu a 1.329)

Table 330. Compounds of formu a I .A, wherein R2 is R2- 9.3201 =formu a 1.330)

Table 331. Compounds of formu a I .A, wherein R2 is R2- 9.3211 =formu a 1.331)

Table 332. Compounds of formu a I .A, wherein R2 is R2- 9.3221 =formu a 1.332)

Table 333. Compounds of formu a I .A, wherein R2 is R2- 9.3231 =formu a 1.333)

Table 334. Compounds of formu a I .A, wherein R2 is R2- 9.3241 =formu a 1.334)

Table 335. Compounds of formu a I .A, wherein R2 is R2- 9.3251 =formu a 1.335)

Table 336. Compounds of formu a I .A, wherein R2 is R2- 9.3261 =formu a 1.336)

Table 337. Compounds of formu a I .A, wherein R2 is R2- 9.3271 =formu a 1.337)

Table 338. Compounds of formu a I .A, wherein R2 is R2- 9.3281 =formu a 1.338)

Table 339. Compounds of formu a I .A, wherein R2 is R2- 9.3291 =formu a 1.339)

Table 340. Compounds of formu a I .A, wherein R2 is R2- 9.3301 =formu a 1.340)

Table 341. Compounds of formu a I .A, wherein R2 is R2- 9.3311 =formu a 1.341) Table 342. Compounds of formula .A, wherein R 2 s R 2 -9.332( formula 1 .342) .

Table 343. Compounds of formula wherein R 2 s R 2 -9.333( formula 1 .343) .

Table 344. Compounds of formula wherein R 2 s R 2 -9.334( formula 1 .344) .

Table 345. Compounds of formula wherein R 2 s R 2 -9.335( formula 1 .345) .

Table 346. Compounds of formula wherein R 2 s R 2 -9.336( formula 1 .346) .

Table 347. Compounds of formula wherein R 2 s R 2 -9.334( formula 1 .347) .

Table 348. Compounds of formula wherein R 2 s R 2 -9.338( formula 1 .348) .

Table 349. Compounds of formula wherein R 2 s R 2 -9.339( formula 1 .349) .

Table 350. Compounds of formula wherein R 2 s R 2 -9.340( formula 1 .350) .

Table 351 . Compounds of formula wherein R 2 s R 2 -9.341 ( formula 1 .351 ) .

Table 352. Compounds of formula I. A, wherein R 2 is R 2 -9.342( =formula 1 .352) .

Table 353. Compounds of formula wherein R 2 s R 2 -9.343( formula 1 .353) .

Table 354. Compounds of formula wherein R 2 s R 2 -9.344( formula 1 .354) .

Table 355. Compounds of formula wherein R 2 s R 2 -9.345( formula 1 .355) .

Table 356. Compounds of formula wherein R 2 s R 2 -9.346( formula 1 .356) .

Table 357. Compounds of formula wherein R 2 s R 2 -9.347( formula 1 .357) .

Table 358. Compounds of formula wherein R 2 s R 2 -9.348( formula 1 .358) .

Table 359. Compounds of formula wherein R 2 s R 2 -9.349( formula 1 .359) .

Table 360. Compounds of formula wherein R 2 s R 2 -9.350( formula 1 .360) .

Table 361 . Compounds of formula wherein R 2 s R 2 -9.351 ( formula 1 .361 ) .

Table 362. Compounds of formula I. A, wherein R 2 is R 2 -9.352( =formula 1 .362) .

Table 363. Compounds of formula wherein R 2 s R 2 -9.353( formula 1 .363) .

Table 364. Compounds of formula wherein R 2 s R 2 -9.354( formula 1 .364) .

Table 365. Compounds of formula wherein R 2 s R 2 -9.355( formula 1 .365) .

Table 366. Compounds of formula wherein R 2 s R 2 -9.356( formula 1 .366) .

Table 367. Compounds of formula wherein R 2 s R 2 -9.357( formula 1 .367) .

Table 368. Compounds of formula wherein R 2 s R 2 -9.358( formula 1 .368) .

Table 369. Compounds of formula wherein R 2 s R 2 -9.359( formula 1 .369) .

Table 370. Compounds of formula wherein R 2 s R 2 -9.360( formula 1 .370) .

Table 371 . Compounds of formula wherein R 2 s R 2 -9.361 ( formula 1 .371 ) .

Table 372. Compounds of formula I. A, wherein R 2 is R 2 -9.362( =formula 1 .372) .

Table 373. Compounds of formula wherein R 2 s R 2 -9.363( formula 1 .373) .

Table 374. Compounds of formula wherein R 2 s R 2 -9.364( formula 1 .374) .

Table 375. Compounds of formula wherein R 2 s R 2 -9.365( formula 1 .375) .

Table 376. Compounds of formula wherein R 2 s R 2 -9.366( formula 1 .376) .

Table 377. Compounds of formula wherein R 2 s R 2 -9.367( formula 1 .377) .

Table 378. Compounds of formula wherein R 2 s R 2 -9.368( formula 1 .378) .

Table 379. Compounds of formula wherein R 2 s R 2 -9.369( formula 1 .379) .

Table 380. Compounds of formula wherein R 2 s R 2 -9.370( formula 1 .380) .

Table 381 . Compounds of formula wherein R 2 s R 2 -9.371 ( formula 1 .381 ) .

Table 382. Compounds of formula wherein R 2 s R 2 -9.372( formula 1 .382) .

Table 383. Compounds of formula wherein R 2 s R 2 -9.373( formula 1 .383) .

Table 384. Compounds of formula wherein R 2 s R 2 -9.374( formula 1 .384) .

Table 385. Compounds of formula wherein R 2 s R 2 -9.375( formula 1 .385) . Table 386. Compounds of formula I .A, wherein R 2 is R 2 -9.376I =formula 1 .386).

Table 387. Compounds of formula I .A, wherein R 2 is R 2 -9.377I =formula 1 .387).

Table 388. Compounds of formula I .A, wherein R 2 is R 2 -9.378I =formula 1 .388).

Table 389. Compounds of formula I .A, wherein R 2 is R 2 -9.379I =formula 1 .389).

Table 390. Compounds of formula I .A, wherein R 2 is R 2 -9.380I =formula 1 .390).

Table 391 . Compounds of formula I .A, wherein R 2 is R 2 -9.381 I =formula 1 .391 ).

Table 392. Compounds of formula I .A, wherein R 2 is R 2 -9.382I =formula 1 .392).

Table 393. Compounds of formula I .A, wherein R 2 is R 2 -9.383I =formula 1 .393).

Table 394. Compounds of formula I .A, wherein R 2 is R 2 -9.384I =formula 1 .394).

Table 395. Compounds of formula I .A, wherein R 2 is R 2 -9.385I =formula 1 .395).

Table 396. Compounds of formula I .A, wherein R 2 is R 2 -9.386I =formula 1 .396).

Table 397. Compounds of formula I .A, wherein R 2 is R 2 -9.387I =formula 1 .397).

Table 398. Compounds of formula I .A, wherein R 2 is R 2 -9.388I =formula 1 .398).

Table 399. Compounds of formula I .A, wherein R 2 is R 2 -9.389I =formula 1 .399).

Table 400. Compounds of formula I .A, wherein R 2 is R 2 -9.390I =formula 1 .400).

Table 401 . Compounds of formula I .A, wherein R 2 is R 2 -9.391 I =formula 1 .401 ).

Table 402. Compounds of formula LA, wherein R 2 is R 2 -9.392(=formula 1 .402).

Table 403. Compounds of formula I .A, wherein R 2 is R 2 -9.393I =formula 1 .403).

Table 404. Compounds of formula I .A, wherein R 2 is R 2 -9.394I =formula 1 .404).

Table 405. Compounds of formula I .A, wherein R 2 is R 2 -9.395I =formula 1 .405).

Table 406. Compounds of formula I .A, wherein R 2 is R 2 -9.396I =formula 1 .406).

Table 407. Compounds of formula I .A, wherein R 2 is R 2 -9.397I =formula 1 .407).

Table 408. Compounds of formula I .A, wherein R 2 is R 2 -9.398I =formula 1 .408).

Table 409. Compounds of formula I .A, wherein R 2 is R 2 -9.399I =formula 1 .409).

Table 410. Compounds of formula I .A, wherein R 2 is R 2 -9.400I =formula 1 .410).

Table 41 1 . Compounds of formula I .A, wherein R 2 is R 2 -9.401 I =formula 1 .41 1 ).

Table 412. Compounds of formula I .A, wherein R 2 is R 2 -9.402I =formula 1 .412).

Table 413. Compounds of formula I .A, wherein R 2 is R 2 -9.403I =formula 1 .413).

Table 414. Compounds of formula I .A, wherein R 2 is R 2 -9.404I =formula 1 .414).

Table 415. Compounds of formula I .A, wherein R 2 is R 2 -9.405I =formula 1 .415).

Table 416. Compounds of formula I .A, wherein R 2 is R 2 -9.406I =formula 1 .416).

Table 417. Compounds of formula I .A, wherein R 2 is R 2 -9.407I =formula 1 .417).

Table 418. Compounds of formula I .A, wherein R 2 is R 2 -9.408I =formula 1 .418).

Table 419. Compounds of formula I .A, wherein R 2 is R 2 -9.409I =formula 1 .419).

Table 420. Compounds of formula I .A, wherein R 2 is R 2 -9.410I =formula 1 .420).

Table 421 . Compounds of formula I .A, wherein R 2 is R 2 -9.41 1 I =formula 1 .421 ).

Table 422. Compounds of formula I .A, wherein R 2 is R 2 -9.412I =formula 1 .422).

Table 423. Compounds of formula I .A, wherein R 2 is R 2 -9.413I =formula 1 .423).

Table 424. Compounds of formula I .A, wherein R 2 is R 2 -9.414I =formula 1 .424).

Table 425. Compounds of formula I .A, wherein R 2 is R 2 -9.415I =formula 1 .425).

Table 426. Compounds of formula I .A, wherein R 2 is R 2 -9.416I =formula 1 .426).

Table 427. Compounds of formula I .A, wherein R 2 is R 2 -9.417I =formula 1 .427).

Table 428. Compounds of formula I .A, wherein R 2 is R 2 -9.418I =formula 1 .428).

Table 429. Compounds of formula I .A, wherein R 2 is R 2 -9.419I =formula 1 .429). Table 430. Compounds of formu a wherein R 2 is R 2 -9.420 =formu 1 .430) .

Table 431 . Compounds of formu a wherein R 2 is R 2 -9.421 =formu 1 .431 ) .

Table 432. Compounds of formula LA, wherein R 2 is R 2 -9.422(=formula 1 .432) .

Table 433. Compounds of formu a wherein R 2 s R 2 -9.423 ormu 1 .433) .

Table 434. Compounds of formu a wherein R 2 s R 2 -9.424 : ormu 1 .434) .

Table 435. Compounds of formu a wherein R 2 s R 2 -9.425 : ormu 1 .435) .

Table 436. Compounds of formu a wherein R 2 s R 2 -9.426 : ormu 1 .436) .

Table 437. Compounds of formu a wherein R 2 s R 2 -9.427 : ormu 1 .437) .

Table 438. Compounds of formu a wherein R 2 s R 2 -9.428 : ormu 1 .438) .

Table 439. Compounds of formu a wherein R 2 s R 2 -9.429 : ormu 1 .439) .

Table 440. Compounds of formu a wherein R 2 s R 2 -9.430 : ormu 1 .440) .

Table 441 . Compounds of formu a wherein R 2 s R 2 -9.431 : ormu 1 .441 ) .

Table 442. Compounds of formu a wherein R 2 s R 2 -9.432 : ormu 1 .442) .

Table 443. Compounds of formu a wherein R 2 s R 2 -9.433 : ormu 1 .443) .

Table 444. Compounds of formu a wherein R 2 s R 2 -9.434 : ormu 1 .444) .

Table 445. Compounds of formu a wherein R 2 s R 2 -9.435 : ormu 1 .445) .

Table 446. Compounds of formu a wherein R 2 s R 2 -9.436 : ormu 1 .446) .

Table 447. Compounds of formu a wherein R 2 s R 2 -9.437 : ormu 1 .447) .

Table 448. Compounds of formu a wherein R 2 s R 2 -9.438 : ormu 1 .448) .

Table 449. Compounds of formu a wherein R 2 s R 2 -9.439 : ormu 1 .449) .

Table 450. Compounds of formu a wherein R 2 s R 2 -9.440 : ormu 1 .450) .

Table 451 . Compounds of formu a wherein R 2 s R 2 -9.441 : ormu 1 .451 ) .

Table 452. Compounds of formu a wherein R 2 s R 2 -9.442 : ormu 1 .452) .

Table 453. Compounds of formu a wherein R 2 s R 2 -9.443 : ormu 1 .453) .

Table 454. Compounds of formu a wherein R 2 s R 2 -9.444 : ormu 1 .454) .

Table 455. Compounds of formu a wherein R 2 s R 2 -9.445 : ormu 1 .455) .

Table 456. Compounds of formu a wherein R 2 s R 2 -9.446 : ormu 1 .456) .

Table 457. Compounds of formu a wherein R 2 s R 2 -9.447 : ormu 1 .457) .

Table 458. Compounds of formu a wherein R 2 s R 2 -9.448 : ormu 1 .458) .

Table 459. Compounds of formu a wherein R 2 s R 2 -9.449 : ormu 1 .459) .

Table 460. Compounds of formu a wherein R 2 s R 2 -9.450 : ormu 1 .460) .

Table 461 . Compounds of formu a wherein R 2 s R 2 -9.451 : ormu 1 .461 ) .

Table 462. Compounds of formu a wherein R 2 s R 2 -9.452 : ormu 1 .462) .

Table 463. Compounds of formu a wherein R 2 s R 2 -9.453 : ormu 1 .463) .

Table 464. Compounds of formu a wherein R 2 s R 2 -9.454 : ormu 1 .464) .

Table 465. Compounds of formu a wherein R 2 s R 2 -9.455 : ormu 1 .465) .

Table 466. Compounds of formu a wherein R 2 s R 2 -9.456 : ormu 1 .466) .

Table 467. Compounds of formu a wherein R 2 s R 2 -9.457 : ormu 1 .467) .

Table 468. Compounds of formu a wherein R 2 s R 2 -9.458 : ormu 1 .468) .

Table 469. Compounds of formu a wherein R 2 s R 2 -9.459 : ormu 1 .469) .

Table 470. Compounds of formu a wherein R 2 s R 2 -9.460 : ormu 1 .470) .

Table 471 . Compounds of formu a wherein R 2 s R 2 -9.461 : ormu 1 .471 ) .

Table 472. Compounds of formu a wherein R 2 s R 2 -9.462 : ormu 1 .472) .

Table 473. Compounds of formu a wherein R 2 s R 2 -9.463 : ormu 1 .473) . Table 474. Compounds of formu a I .A, wherein R2 is R2- -9.464I =formu a 1 .474)

Table 475. Compounds of formu a I .A, wherein R2 is R2- -9.465I =formu a 1 .475)

Table 476. Compounds of formu a I .A, wherein R2 is R2- -9.466I =formu a 1 .476)

Table 477. Compounds of formu a I .A, wherein R2 is R2- -9.467I =formu a 1 .477)

Table 478. Compounds of formu a I .A, wherein R2 is R2- -9.468I =formu a 1 .478)

Table 479. Compounds of formu a I .A, wherein R2 is R2- -9.469I =formu a 1 .479)

Table 480. Compounds of formu a I .A, wherein R2 is R2- -9.470I =formu a 1 .480)

Table 481 . Compounds of formu a I .A, wherein R2 is R2- 9.4711 =formu a 1 .481 )

Table 482. Compounds of formu a I .A, wherein R2 is R2- 9.4721 =formu a 1 .482)

Table 483. Compounds of formu a I .A, wherein R2 is R2- 9.4731 =formu a 1 .483)

Table 484. Compounds of formu a I .A, wherein R2 is R2- 9.4741 =formu a 1 .484)

Table 485. Compounds of formu a I .A, wherein R2 is R2- 9.4751 =formu a 1 .485)

Table 486. Compounds of formu a I .A, wherein R2 is R2- 9.4761 =formu a 1 .486)

Table 487. Compounds of formu a I .A, wherein R2 is R2- 9.4771 =formu a 1 .487)

Table 488. Compounds of formu a I .A, wherein R2 is R2- 9.4781 =formu a 1 .488)

Table 489. Compounds of formu a I .A, wherein R2 is R2- 9.4791 =formu a 1 .489)

Table 490. Compounds of formu a I .A, wherein R2 is R2- 9.4801 =formu a 1 .490)

Table 491 . Compounds of formu a I .A, wherein R2 is R2- 9.4811 =formu a 1 .491 )

Table 492. Compounds of formu a I .A, wherein R2 is R2- 9.4821 =formu a 1 .492)

Table 493. Compounds of formu a I .A, wherein R2 is R2- 9.4831 =formu a 1 .493)

Table 494. Compounds of formu a I .A, wherein R2 is R2- 9.4841 =formu a 1 .494)

Table 495. Compounds of formu a I .A, wherein R2 is R2- 9.4851 =formu a 1 .495)

Table 496. Compounds of formu a I .A, wherein R2 is R2- 9.4861 =formu a 1 .496)

Table 497. Compounds of formu a I .A, wherein R2 is R2- 9.4871 =formu a 1 .497)

Table 498. Compounds of formu a I .A, wherein R2 is R2- 9.4881 =formu a 1 .498)

Table 499. Compounds of formu a I .A, wherein R2 is R2- 9.4891 =formu a 1 .499)

Table 500. Compounds of formu a I .A, wherein R2 is R2- 9.4901 =formu a 1 .500)

Table 501 . Compounds of formu a I .A, wherein R2 is R2- 9.4911 =formu a 1 .501 )

Table 502. Compounds of formu a I .A, wherein R2 is R2- 9.492 (=formula 1.502)

Table 503. Compounds of formu a I .A, wherein R2 is R2- 9.4931 =formu a 1 .503)

Table 504. Compounds of formu a I .A, wherein R2 is R2- 9.4941 =formu a 1 .504)

Table 505. Compounds of formu a I .A, wherein R2 is R2- 9.4951 =formu a 1 .505)

Table 506. Compounds of formu a I .A, wherein R2 is R2- 9.4961 =formu a 1 .506)

Table 507. Compounds of formu a I .A, wherein R2 is R2- 9.4971 =formu a 1 .507)

Table 508. Compounds of formu a I .A, wherein R2 is R2- 9.4981 =formu a 1 .508)

Table 509. Compounds of formu a I .A, wherein R2 is R2- 9.4991 =formu a 1 .509)

Table 510. Compounds of formu a I .A, wherein R2 is R2- 9.5001 =formu a 1 .510)

Table 51 1 . Compounds of formu a I .A, wherein R2 is R2- 9.5011 =formu a 1 .51 1 )

Table 512. Compounds of formu a I .A, wherein R2 is R2- 9.5021 =formu a 1 .512)

Table 513. Compounds of formu a I .A, wherein R2 is R2- 9.5031 =formu a 1 .513)

Table 514. Compounds of formu a I .A, wherein R2 is R2- 9.5041 =formu a 1 .514)

Table 515. Compounds of formu a I .A, wherein R2 is R2- 9.5051 =formu a 1 .515)

Table 516. Compounds of formu a I .A, wherein R2 is R2- 9.5061 =formu a 1 .516)

Table 517. Compounds of formu a I .A, wherein R2 is R2- 9.5071 =formu a 1 .517) Table 518. Compounds of formu a I .A, wherein R2 is R2- -9.508I =formula 1.518).

Table 519. Compounds of formu a I .A, wherein R2 is R2- -9.509I =formula 1.519).

Table 520. Compounds of formu a I .A, wherein R2 is R2- 9.5101 =formula 1.520).

Table 521. Compounds of formu a I .A, wherein R2 is R2- 9.5111 =formula 1.521).

Table 522. Compounds of formu a I .A, wherein R2 is R2- 9.512 (=formula 1.522)

Table 523. Compounds of formu a I .A, wherein R2 is R2- 9.513 (=formula 1.523)

Table 524. Compounds of formu a I .A, wherein R2 is R2- 9.5141 =formula 1.524).

Table 525. Compounds of formu a I .A, wherein R2 is R2- 9.5151 =formula 1.525).

Table 526. Compounds of formu a I .A, wherein R2 is R2- 9.5161 =formula 1.526).

Table 527. Compounds of formu a I .A, wherein R2 is R2- 9.5171 =formula 1.527).

Table 528. Compounds of formu a I .A, wherein R2 is R2- 9.5181 =formula 1.528).

Table 529. Compounds of formu a I .A, wherein R2 is R2- 9.5191 =formula 1.529).

Table 530. Compounds of formu a I .A, wherein R2 is R2- 9.5201 =formula 1.530).

Table 531. Compounds of formu a I .A, wherein R2 is R2- 9.5211 =formula 1.531).

Table 532. Compounds of formu a I .A, wherein R2 is R2- 9.5221 =formula 1.532).

Table 533. Compounds of formu a I .A, wherein R2 is R2- 9.5231 =formula 1.533).

Table 534. Compounds of formu a I .A, wherein R2 is R2- 9.5241 =formula 1.534).

Table 535. Compounds of formu a I .A, wherein R2 is R2- 9.5251 =formula 1.535).

Table 536. Compounds of formu a I .A, wherein R2 is R2- 9.5261 =formula 1.536).

Table 537. Compounds of formu a I .A, wherein R2 is R2- 9.5271 =formula 1.537).

Table 538. Compounds of formu a I .A, wherein R2 is R2- 9.5281 =formula 1.538).

Table 539. Compounds of formu a I .A, wherein R2 is R2- 9.5291 =formula 1.539).

Table 540. Compounds of formu a I .A, wherein R2 is R2- 9.5301 =formula 1.540).

Table 541. Compounds of formu a I .A, wherein R2 is R2- 9.5311 =formula 1.541).

Table 542. Compounds of formu a I .A, wherein R2 is R2- 9.5321 =formula 1.542).

Table 543. Compounds of formu a I .A, wherein R2 is R2- 9.5331 =formula 1.543).

Table 544. Compounds of formu a I .A, wherein R2 is R2- 9.5341 =formula 1.544).

Table 545. Compounds of formu a I .A, wherein R2 is R2- 9.5351 =formula 1.545).

Table 546. Compounds of formu a I .A, wherein R2 is R2- 9.5361 =formula 1.546).

Table 547. Compounds of formu a I .A, wherein R2 is R2- 9.5371 =formula 1.547).

Table 548. Compounds of formu a I .A, wherein R2 is R2- 9.5381 =formula 1.548).

Table 549. Compounds of formu a I .A, wherein R2 is R2- 9.5391 =formula 1.549).

Table 550. Compounds of formu a I .A, wherein R2 is R2- 9.5401 =formula 1.550).

Table 551. Compounds of formu a I .A, wherein R2 is R2- 9.5411 =formula 1.551).

Table 552. Compounds of formu a I .A, wherein R2 is R2- 9.5421 =formula 1.552).

Table 553. Compounds of formu a I .A, wherein R2 is R2- 9.5431 =formula 1.553).

Table 554. Compounds of formu a I .A, wherein R2 is R2- 9.5441 =formula 1.554).

Table 555. Compounds of formu a I .A, wherein R2 is R2- 9.5451 =formula 1.555).

Table 556. Compounds of formu a I .A, wherein R2 is R2- 9.5461 =formula 1.556).

Table 557. Compounds of formu a I .A, wherein R2 is R2- 9.5471 =formula 1.557).

Table 558. Compounds of formu a I .A, wherein R2 is R2- 9.5481 =formula 1.558).

Table 559. Compounds of formu a I .A, wherein R2 is R2- 9.5491 =formula 1.559).

Table 560. Compounds of formu a I .A, wherein R2 is R2- 9.5501 =formula 1.560).

Table 561. Compounds of formu a I .A, wherein R2 is R2- 9.5511 =formula 1.561). Table 562. Compounds of formu a I .A, wherein R2 is R2- -9.552I =formu a 1 .562).

Table 563. Compounds of formu a I .A, wherein R2 is R2- -9.553I =formu a 1 .563).

Table 564. Compounds of formu a I .A, wherein R2 is R2- -9.554I =formu a 1 .564).

Table 565. Compounds of formu a I .A, wherein R2 is R2- -9.555I =formu a 1 .565).

Table 566. Compounds of formu a I .A, wherein R2 is R2- -9.556I =formu a 1 .566).

Table 567. Compounds of formu a I .A, wherein R2 is R2- -9.557I =formu a 1 .567).

Table 568. Compounds of formu a I .A, wherein R2 is R2- -9.558I =formu a 1 .568).

Table 569. Compounds of formu a I .A, wherein R2 is R2- -9.559I =formu a 1 .569).

Table 570. Compounds of formu a I .A, wherein R2 is R2- 9.560 (=formula 1 .570)

Table 571 . Compounds of formu a I .A, wherein R2 is R2- 9.5611 =formu a 1 .571 ).

Table 572. Compounds of formu a I .A, wherein R2 is R2- 9.5621 =formu a 1 .572).

Table 573. Compounds of formu a I .A, wherein R2 is R2- 9.5631 =formu a 1 .573).

Table 574. Compounds of formu a I .A, wherein R2 is R2- 9.5641 =formu a 1 .574).

Table 575. Compounds of formu a I .A, wherein R2 is R2- 9.5651 =formu a 1 .575).

Table 576. Compounds of formu a I .A, wherein R2 is R2- 9.5661 =formu a 1 .576).

Table 577. Compounds of formu a I .A, wherein R2 is R2- 9.5671 =formu a 1 .577).

Table 578. Compounds of formu a I .A, wherein R2 is R2- 9.5681 =formu a 1 .578).

Table 579. Compounds of formu a I .A, wherein R2 is R2- 9.5691 =formu a 1 .579).

Table 580. Compounds of formu a I .A, wherein R2 is R2- 9.5701 =formu a 1 .580).

Table 581 . Compounds of formu a I .A, wherein R2 is R2- 9.5711 =formu a 1 .581 ).

Table 582. Compounds of formu a I .A, wherein R2 is R2- 9.5721 =formu a 1 .582).

Table 583. Compounds of formu a I .A, wherein R2 is R2- 9.5731 =formu a 1 .583).

Table 584. Compounds of formu a I .A, wherein R2 is R2- 9.5741 =formu a 1 .584).

Table 585. Compounds of formu a I .A, wherein R2 is R2- 9.5751 =formu a 1 .585).

Table 586. Compounds of formu a I .A, wherein R2 is R2- 9.5761 =formu a 1 .586).

Table 587. Compounds of formu a I .A, wherein R2 is R2- 9.5771 =formu a 1 .587).

Table 588. Compounds of formu a I .A, wherein R2 is R2- 9.5781 =formu a 1 .588).

Table 589. Compounds of formu a I .A, wherein R2 is R2- 9.5791 =formu a 1 .589).

Table 590. Compounds of formu a I .A, wherein R2 is R2- 9.5801 =formu a 1 .590).

Table 591 . Compounds of formu a I .A, wherein R2 is R2- 9.5811 =formu a 1 .591 ).

Table 592. Compounds of formu a I .A, wherein R2 is R2- 9.5821 =formu a 1 .592).

Table 593. Compounds of formu a I .A, wherein R2 is R2- 9.5831 =formu a 1 .593).

Table 594. Compounds of formu a I .A, wherein R2 is R2- 9.5841 =formu a 1 .594).

Table 595. Compounds of formu a I .A, wherein R2 is R2- 9.5851 =formu a 1 .595).

Table 596. Compounds of formu a I .A, wherein R2 is R2- 9.5861 =formu a 1 .596).

Table 597. Compounds of formu a I .A, wherein R2 is R2- 9.5871 =formu a 1 .597).

Table 598. Compounds of formu a I .A, wherein R2 is R2- 9.5881 =formu a 1 .598).

Table 599. Compounds of formu a I .A, wherein R2 is R2- 9.5891 =formu a 1 .599).

Table 600. Compounds of formu a I .A, wherein R2 is R2- 9.5901 =formu a 1 .600).

Table 601 . Compounds of formu a I .A, wherein R2 is R2- 9.5911 =formu a 1 .601 ).

Table 602. Compounds of formu a I .A, wherein R2 is R2- 9.5921 =formu a 1 .602).

Table 603. Compounds of formu a I .A, wherein R2 is R2- 9.5931 =formu a 1 .603).

Table 604. Compounds of formu a I .A, wherein R2 is R2- 9.5941 =formu a 1 .604).

Table 605. Compounds of formu a I .A, wherein R2 is R2- 9.5951 =formu a 1 .605). Table 606. Compounds of formu a I .A, wherein R2 is R2-9.596I Formu a 1 .606)

Table 607. Compounds of formu a I .A, wherein R2 is R2-9.597I = Formu a 1 .607)

Table 608. Compounds of formu a I .A, wherein R2 is R2-9.598I = Formu a 1 .608)

Table 609. Compounds of formu a I .A, wherein R2 is R2-9.599I = Formu a 1 .609)

Table 610. Compounds of formu a I .A, wherein R2 is R2-9.600I = Formu a 1 .610)

Table 61 1 . Compounds of formu a I .A, wherein R2 is R2-9.601 I = Formu a 1 .61 1 )

Table 612. Compounds of formu a I .A, wherein R2 is R2-9.602I = Formu a 1 .612)

Table 613. Compounds of formu a I .A, wherein R2 is R2-9.603I = Formu a 1 .613)

Table 614. Compounds of formu a I .A, wherein R2 is R2-9.604I = Formu a 1 .614)

Table 615. Compounds of formu a I .A, wherein R2 is R2-9.605I = Formu a 1 .615)

Table 616. Compounds of formu a I .A, wherein R2 is R2-9.606I = Formu a 1 .616)

Table 617. Compounds of formu a I .A, wherein R2 is R2-9.607I = Formu a 1 .617)

Table 618. Compounds of formu a I .A, wherein R2 is R2-9.608I = Formu a 1 .618)

Table 619. Compounds of formu a I .A, wherein R2 is R2-9.609I = Formu a 1 .619)

Table 620. Compounds of formu a I .A, wherein R2 is R2-9.610I = Formu a 1 .620)

Table 621 . Compounds of formu a I .A, wherein R2 is R2-9.61 1 I = Formu a 1 .621 )

Table 622. Compounds of formu a I .A, wherein R2 is R2-9.612I = Formu a 1 .622)

Table 623. Compounds of formu a I .A, wherein R2 is R2-9.613I = Formu a 1 .623)

Table 624. Compounds of formu a I .A, wherein R2 is R2-9.614I = Formu a 1 .624)

Table 625. Compounds of formu a I .A, wherein R2 is R2-9.615I = Formu a 1 .625)

Table 626. Compounds of formu a I .A, wherein R2 is R2-9.616I = Formu a 1 .626)

Table 627. Compounds of formu a I .A, wherein R2 is R2-9.617I = Formu a 1 .627)

Table 628. Compounds of formu a I .A, wherein R2 is R2-9.618I = Formu a 1 .628)

Table 629. Compounds of formu a I .A, wherein R2 is R2-9.619I = Formu a 1 .629)

Table 630. Compounds of formu a I .A, wherein R2 is R2-9.620I = Formu a 1 .630)

Table 631 . Compounds of formu a I .A, wherein R2 is R2-9.621 I = Formu a 1 .631 )

Table 632. Compounds of formu a I .A, wherein R2 is R2-9.622I = Formu a 1 .632)

Table 633. Compounds of formu a I .A, wherein R2 is R2-9.623I = Formu a 1 .633)

Table 634. Compounds of formu a I .A, wherein R2 is R2-9.624I = Formu a 1 .634)

Table 635. Compounds of formu a I .A, wherein R2 is R2-9.625I = Formu a 1 .635)

Table 636. Compounds of formu a I .A, wherein R2 is R2-9.626I = Formu a 1 .636)

Table 637. Compounds of formu a I .A, wherein R2 is R2-9.627I = Formu a 1 .637)

Table 638. Compounds of formu a I .A, wherein R2 is R2-9.628I = Formu a 1 .638)

Table 639. Compounds of formu a I .A, wherein R2 is R2-9.629I = Formu a 1 .639)

Table 640. Compounds of formu a I .A, wherein R2 is R2-9.630I = Formu a 1 .640)

Table 641 . Compounds of formu a I .A, wherein R2 is R2-9.631 I = Formu a 1 .641 )

Table 642. Compounds of formu a I .A, wherein R2 is R2-9.632I = Formu a 1 .642)

Table 643. Compounds of formu a I .A, wherein R2 is R2-9.633I = Formu a 1 .643)

Table 644. Compounds of formu a I .A, wherein R2 is R2-9.634I = Formu a 1 .644)

Table 645. Compounds of formu a I .A, wherein R2 is R2-9.635I = Formu a 1 .645)

Table 646. Compounds of formu a I .A, wherein R2 is R2-9.636I = Formu a 1 .646)

Table 647. Compounds of formu a I .A, wherein R2 is R2-9.637I = Formu a 1 .647)

Table 648. Compounds of formu a I .A, wherein R2 is R2-9.638I = Formu a 1 .648)

Table 649. Compounds of formu a I .A, wherein R2 is R2-9.639I = Formu a 1 .649) Table 650. Compounds of formu a I .A, wherein R2 is R2-9.640(=formula 1.650).

Table 651. Compounds of formu a I .A, wherein R2 is R2-9.641 (=formula 1.651).

Table 652. Compounds of formu a I .A, wherein R2 is R2-9.642(=formula 1.652).

Table 653. Compounds of formu a I .A, wherein R2 is R2-9.643(=formula 1.653).

Table 654. Compounds of formu a I .A, wherein R2 is R2-9.644(=formula 1.654).

Table 655. Compounds of formu a I .A, wherein R2 is R2-9.645(=formula 1.655).

Table 656. Compounds of formu a I .A, wherein R2 is R2-9.646(=formula 1.656).

Table 657. Compounds of formu a I .A, wherein R2 is R2-9.647(=formula 1.657).

Table 658. Compounds of formu a I .A, wherein R2 is R2-9.648(=formula 1.658).

Table 659. Compounds of formu a I .A, wherein R2 is R2-9.649(=formula 1.659).

Table 660. Compounds of formu a I .A, wherein R2 is R2-9.650(=formula 1.660).

Table 661. Compounds of formu a I .A, wherein R2 is R2-9.651 (=formula 1.661).

Table 662. Compounds of formu a I .A, wherein R2 is R2-9.652(=formula 1.662).

Table 663. Compounds of formu a I .A, wherein R2 is R2-9.653(=formula 1.663).

Table 664. Compounds of formu a I .A, wherein R2 is R2-9.654(=formula 1.664).

Table 665. Compounds of formu a I .A, wherein R2 is R2-9.655(=formula 1.665).

Table 666. Compounds of formu a I .A, wherein R2 is R2-9.656(=formula 1.666).

Table 667. Compounds of formu a I .A, wherein R2 is R2-9.657(=formula 1.667).

Table 668. Compounds of formu a I .A, wherein R2 is R2-9.658(=formula 1.668).

Table 669. Compounds of formu a I .A, wherein R2 is R2-9.659(=formula 1.669).

Table 670. Compounds of formu a I .A, wherein R2 is R2-9.660(=formula 1.670).

Table 671. Compounds of formu a I .A, wherein R2 is R2-9.661 (=formula 1.671).

Table 672. Compounds of formu a I .A, wherein R2 is R2-9.662(=formula 1.672).

Table 673. Compounds of formu a I .A, wherein R2 is R2-9.663(=formula 1.673).

Table 674. Compounds of formu a I .A, wherein R2 is R2-9.664(=formula 1.674).

Table 675. Compounds of formu a I .A, wherein R2 is R2-9.665(=formula 1.675).

Table 676. Compounds of formu a I .A, wherein R2 is R2-9.666(=formula 1.676).

Table 677. Compounds of formu a I .A, wherein R2 is R2-9.667(=formula 1.677).

Table 678. Compounds of formu a I .A, wherein R2 is R2-9.668(=formula 1.678).

Table 679. Compounds of formu a I .A, wherein R2 is R2-9.669(=formula 1.679).

Table 680. Compounds of formu a I .A, wherein R2 is R2-9.670(=formula 1.680).

Table 681. Compounds of formu a I .A, wherein R2 is R2-9.671 (=formula 1.681).

Table 682. Compounds of formu a I .A, wherein R2 is R2-9.672(=formula 1.682).

Table 683. Compounds of formu a I .A, wherein R2 is R2-9.673(=formula 1.683).

Table 684. Compounds of formu a I .A, wherein R2 is R2-9.674(=formula 1.684).

Table 685. Compounds of formu a I .A, wherein R2 is R2-9.675(=formula 1.685).

Table 686. Compounds of formu a I .A, wherein R2 is R2-9.676(=formula 1.686).

Table 687. Compounds of formu a I .A, wherein R2 is R2-10.1(=formula 1.687).

Table 688. Compounds of formu a I .A, wherein R2 is R2-10.2(=formula 1.688).

Table 689. Compounds of formu a I .A, wherein R2 is R2-10.3(=formula 1.689).

Table 690. Compounds of formu a I .A, wherein R2 is R2_io.4(=formula 1.690).

Table 691. Compounds of formu a I .A, wherein R2 is R2-10.5(=formula 1.691).

Table 692. Compounds of formu a I .A, wherein R2 is R2-10.6(=formula 1.692).

Table 693. Compounds of formu a I .A, wherein R2 is R2-10.7(=formula 1.693). Table 694. Compounds of formu a I .A, wherein R2 is R2 0.8(=formula 1.694).

Table 695. Compounds of formu a I .A, wherein R2 is R2 0.9(=formula 1.695).

Table 696. Compounds of formu a I .A, wherein R2 is R2 0.101 Formu a 1 .696)

Table 697. Compounds of formu a I .A, wherein R2 is R2 0.1 11 = Formu a 1 .697)

Table 698. Compounds of formu a I .A, wherein R2 is R2 0.121 = Formu a 1 .698)

Table 699. Compounds of formu a I .A, wherein R2 is R2 0.131 = Formu a 1 .699)

Table 700. Compounds of formu a I .A, wherein R2 is R2 0.141 = Formu a 1 .700)

Table 701 . Compounds of formu a I .A, wherein R2 is R2 0.151 = Formu a 1 .701 )

Table 702. Compounds of formu a I .A, wherein R2 is R2 0.161 = Formu a 1 .702)

Table 703. Compounds of formu a I .A, wherein R2 is R2 0.171 = Formu a 1 .703)

Table 704. Compounds of formu a I .A, wherein R2 is R2 0.181 = Formu a 1 .704)

Table 705. Compounds of formu a I .A, wherein R2 is R2 0.191 = Formu a 1 .705)

Table 706. Compounds of formu a I .A, wherein R2 is R2 0.201 = Formu a 1 .706)

Table 707. Compounds of formu a I .A, wherein R2 is R2 0.211 = Formu a 1 .707)

Table 708. Compounds of formu a I .A, wherein R2 is R2 0.221 = Formu a 1 .708)

Table 709. Compounds of formu a I .A, wherein R2 is R2 0.231 = Formu a 1 .709)

Table 710. Compounds of formu a I .A, wherein R2 is R2 0.241 = Formu a 1 .710)

Table 71 1 . Compounds of formu a I .A, wherein R2 is R2 0.251 = Formu a 1 .71 1 )

Table 712. Compounds of formu a I .A, wherein R2 is R2 0.261 = Formu a 1 .712)

Table 713. Compounds of formu a I .A, wherein R2 is R2 0.271 = Formu a 1 .713)

Table 714. Compounds of formu a I .A, wherein R2 is R2 0.281 = Formu a 1 .714)

Table 715. Compounds of formu a I .A, wherein R2 is R2 0.291 = Formu a 1 .715)

Table 716. Compounds of formu a I .A, wherein R2 is R2 0.301 = Formu a 1 .716)

Table 717. Compounds of formu a I .A, wherein R2 is R2 0.311 = Formu a 1 .717)

Table 718. Compounds of formu a I .A, wherein R2 is R2 0.321 = Formu a 1 .718)

Table 719. Compounds of formu a I .A, wherein R2 is R2 0.331 = Formu a 1 .719)

Table 720. Compounds of formu a I .A, wherein R2 is R2 0.341 = Formu a 1 .720)

Table 721 . Compounds of formu a I .A, wherein R2 is R2 0.351 = Formu a 1 .721 )

Table 722. Compounds of formu a I .A, wherein R2 is R2 0.361 = Formu a 1 .722)

Table 723. Compounds of formu a I .A, wherein R2 is R2 0.371 = Formu a 1 .723)

Table 724. Compounds of formu a I .A, wherein R2 is R2 0.381 = Formu a 1 .724)

Table 725. Compounds of formu a I .A, wherein R2 is R2 0.391 = Formu a 1 .725)

Table 726. Compounds of formu a I .A, wherein R2 is R2 0.401 = Formu a 1 .726)

Table 727. Compounds of formu a I .A, wherein R2 is R2 0.411 = Formu a 1 .727)

Table 728. Compounds of formu a I .A, wherein R2 is R2 0.421 = Formu a 1 .728)

Table 729. Compounds of formu a I .A, wherein R2 is R2 0.431 = Formu a 1 .729)

Table 730. Compounds of formu a I .A, wherein R2 is R2 0.441 = Formu a 1 .730)

Table 731 . Compounds of formu a I .A, wherein R2 is R2 0.451 = Formu a 1 .731 )

Table 732. Compounds of formu a I .A, wherein R2 is R2 0.461 = Formu a 1 .732)

Table 733. Compounds of formu a I .A, wherein R2 is R2 0.471 = Formu a 1 .733)

Table 734. Compounds of formu a I .A, wherein R2 is R2 0.481 = Formu a 1 .734)

Table 735. Compounds of formu a I .A, wherein R2 is R2 0.491 = Formu a 1 .735)

Table 736. Compounds of formu a I .A, wherein R2 is R2 0.501 = Formu a 1 .736)

Table 737. Compounds of formu a I .A, wherein R2 is R2 0.511 = Formu a 1 .737) Table 738. Compounds of formu a ■A, wherein R2 is R2-- 0.52| = Formu a 1 .738).

Table 739. Compounds of formu a ■A, wherein R2 is R2-- 0.53I = Formu a 1 .739).

Table 740. Compounds of formu a ■A, wherein R2 is R2-- 0.54| = Formu a 1 .740).

Table 741 . Compounds of formu a ■A, wherein R2 is R2-- 0.55I = Formu a 1 .741 ).

Table 742. Compounds of formu a ■A, wherein R2 is R2-- 0.56I = Formu a 1 .742).

Table 743. Compounds of formu a ■A, wherein R2 is R2-- 0.57| = Formu a 1 .743).

Table 744. Compounds of formu a ■A, wherein R2 is R2-- 0.58I = Formu a 1 .744).

Table 745. Compounds of formu a ■A, wherein R2 is R2-- 0.59I = Formu a 1 .745).

Table 746. Compounds of formu a ■A, wherein R2 is R2-- 0.60I = Formu a 1 .746).

Table 747. Compounds of formu a ■A, wherein R2 is R2-- 0.611 = Formu a 1 .747).

Table 748. Compounds of formu a ■A, wherein R2 is R2-- 0.621 = Formu a 1 .748).

Table 749. Compounds of formu a ■A, wherein R2 is R2-- 0.631 = Formu a 1 .749).

Table 750. Compounds of formu a ■A, wherein R2 is R2-- 0.641 = Formu a 1 .750).

Table 751 . Compounds of formu a ■A, wherein R2 is R2-- 0.651 = Formu a 1 .751 ).

Table 752. Compounds of formu a ■A, wherein R2 is R2-- 0.661 = Formu a 1 .752).

Table 753. Compounds of formu a ■A, wherein R2 is R2-- 0.671 = Formu a 1 .753).

Table 754. Compounds of formu a ■A, wherein R2 is R2-- 0.681 = Formu a 1 .754).

Table 755. Compounds of formu a ■A, wherein R2 is R2-- 0.691 = Formu a 1 .755).

Table 756. Compounds of formu a ■A, wherein R2 is R2-- 0.701 = Formu a 1 .756).

Table 757. Compounds of formu a ■A, wherein R2 is R2-- 0.711 = Formu a 1 .757).

Table 758. Compounds of formu a ■A, wherein R2 is R2-- 0.721 = Formu a 1 .758).

Table 759. Compounds of formu a ■A, wherein R2 is R2-- 0.731 = Formu a 1 .759).

Table 760. Compounds of formu a ■A, wherein R2 is R2-- 0.741 = Formu a 1 .760).

Table 761 . Compounds of formu a ■A, wherein R2 is R2-- 0.751 = Formu a 1 .761 ).

Table 762. Compounds of formu a ■A, wherein R2 is R2-- 0.761 = Formu a 1 .762).

Table 763. Compounds of formu a ■A, wherein R2 is R2-- 0.771 = Formu a 1 .763).

Table 764. Compounds of formu a ■A, wherein R2 is R2-- 0.781 = Formu a 1 .764).

Table 765. Compounds of formu a ■A, wherein R2 is R2-- 0.791 = Formu a 1 .765).

Table 766. Compounds of formu a ■A, wherein R2 is R2-- 0.801 = Formu a 1 .766).

Table 767. Compounds of formu a ■A, wherein R2 is R2-- 0.811 = Formu a 1 .767).

Table 768. Compounds of formu a ■A, wherein R2 is R2-- 0.821 = Formu a 1 .768).

Table 769. Compounds of formu a ■A, wherein R2 is R2-- 0.831 = Formu a 1 .769).

Table 770. Compounds of formu a ■A, wherein R2 is R2-- 0.841 = Formu a 1 .770).

Table 771 . Compounds of formu a ■A, wherein R2 is R2-- 0.851 = Formu a 1 .771 ).

Table 772. Compounds of formu a ■A, wherein R2 is R2-- 0.861 = Formu a 1 .772).

Table 773. Compounds of formu a ■A, wherein R2 is R2-- 0.871 = Formu a 1 .773).

Table 774. Compounds of formu a ■A, wherein R2 is R2-- 0.881 = Formu a 1 .774).

Table 775. Compounds of formu a ■A, wherein R2 is R2-- 0.891 = Formu a 1 .775).

Table 776. Compounds of formu a ■A, wherein R2 is R2-- 0.901 = Formu a 1 .776).

Table 777. Compounds of formu a ■A, wherein R2 is R2-- 0.911 = Formu a 1 .777).

Table 778. Compounds of formu a ■A, wherein R2 is R2-- 0.921 = Formu a 1 .778).

Table 779. Compounds of formu a ■A, wherein R2 is R2-- 0.931 = Formu a 1 .779).

Table 780. Compounds of formu a ■A, wherein R2 is R2-- 0.941 = Formu a 1 .780).

Table 781 . Compounds of formu a ■A, wherein R2 is R2-- 0.951 = Formu a 1 .781 ). Table 782. Compounds of formu a I .A, wherein R2 is R2-- 0.96(=formula 1.782).

Table 783. Compounds of formu a I .A, wherein R2 is R2-- 0.97(=formula 1.783).

Table 784. Compounds of formu a I .A, wherein R2 is R2-- 0.98(=formula 1.784).

Table 785. Compounds of formu a I .A, wherein R2 is R2-- 0.99(=formula 1.785).

Table 786. Compounds of formu a I .A, wherein R2 is R2-- 0.100( =formula 1.786).

Table 787. Compounds of formu a I .A, wherein R2 is R2-- 0.101( =formula 1.787).

Table 788. Compounds of formu a I .A, wherein R2 is R2-- 0.102( =formula 1.788).

Table 789. Compounds of formu a I .A, wherein R2 is R2-- 0.103( =formula 1.789).

Table 790. Compounds of formu a I .A, wherein R2 is R2-- 0.104( =formula 1.790).

Table 791. Compounds of formu a I .A, wherein R2 is R2-- 0.105( =formula 1.791).

Table 792. Compounds of formu a I .A, wherein R2 is R2-- 0.106( =formula 1.792).

Table 793. Compounds of formu a I .A, wherein R2 is R2-- 0.107( =formula 1.793).

Table 794. Compounds of formu a I .A, wherein R2 is R2-- 0.108( =formula 1.794).

Table 795. Compounds of formu a I .A, wherein R2 is R2-- 0.109( =formula 1.795).

Table 796. Compounds of formu a I .A, wherein R2 is R2-- 0.110( =formula 1.796).

Table 797. Compounds of formu a I .A, wherein R2 is R2-- 0.111< =formula 1.797).

Table 798. Compounds of formu a I .A, wherein R2 is R2-- 0.112( =formula 1.798).

Table 799. Compounds of formu a I .A, wherein R2 is R2-- 0.113( =formula 1.799).

Table 800. Compounds of formu a I .A, wherein R2 is R2-- 0.114( =formula 1.800).

Table 801. Compounds of formu a I .A, wherein R2 is R2-- 0.115( =formula 1.801).

Table 802. Compounds of formu a I .A, wherein R2 is R2-- 0.116( =formula 1.802).

Table 803. Compounds of formu a I .A, wherein R2 is R2-- 0.117( =formula 1.803).

Table 804. Compounds of formu a I .A, wherein R2 is R2-- 0.118( =formula 1.804).

Table 805. Compounds of formu a I .A, wherein R2 is R2-- 0.119( =formula 1.805).

Table 806. Compounds of formu a I .A, wherein R2 is R2-- 0.120( =formula 1.806).

Table 807. Compounds of formu a I .A, wherein R2 is R2-- 0.121( =formula 1.807).

Table 808. Compounds of formu a I .A, wherein R2 is R2-- 0.122( =formula 1.808).

Table 809. Compounds of formu a I .A, wherein R2 is R2-- 0.123( =formula 1.809).

Table 810. Compounds of formu a I .A, wherein R2 is R2-- 0.124( =formula 1.810).

Table 811. Compounds of formu a I .A, wherein R2 is R2-- 0.125( =formula 1.811).

Table 812. Compounds of formu a I .A, wherein R2 is R2-- 0.126( =formula 1.812).

Table 813. Compounds of formu a I .A, wherein R2 is R2-- 0.127( =formula 1.813).

Table 814. Compounds of formu a I .A, wherein R2 is R2-- 0.128( =formula 1.814).

Table 815. Compounds of formu a I .A, wherein R2 is R2-- 0.129( =formula 1.815).

Table 816. Compounds of formu a I .A, wherein R2 is R2-- 0.130( =formula 1.816).

Table 817. Compounds of formu a I .A, wherein R2 is R2-- 0.131( =formula 1.817).

Table 818. Compounds of formu a I .A, wherein R2 is R2-- 0.132( =formula 1.818).

Table 819. Compounds of formu a I .A, wherein R2 is R2-- 0.133( =formula 1.819).

Table 820. Compounds of formu a I .A, wherein R2 is R2-- 0.134( =formula 1.820).

Table 821. Compounds of formu a I .A, wherein R2 is R2-- 0.135( =formula 1.821).

Table 822. Compounds of formu a I .A, wherein R2 is R2-- 0.136( =formula 1.822).

Table 823. Compounds of formu a I .A, wherein R2 is R2-- 0.137( =formula 1.823).

Table 824. Compounds of formu a I .A, wherein R2 is R2-- 0.138( =formula 1.824).

Table 825. Compounds of formu a I .A, wherein R2 is R2-- 0.139( =formula 1.825). Table 826. Compounds of formu a I .A, wherein R2 is R2-- 0.140( = Formu a 1.826).

Table 827. Compounds of formu a I .A, wherein R2 is R2-- 0.141 ( = Formu a 1.827).

Table 828. Compounds of formu a I .A, wherein R2 is R2-- 0.142( = Formu a 1.828).

Table 829. Compounds of formu a I .A, wherein R2 is R2-- 0.143( = Formu a 1.829).

Table 830. Compounds of formu a I .A, wherein R2 is R2-- 0.144( = Formu a 1.830).

Table 831 . Compounds of formu a I .A, wherein R2 is R2-- 0.145( = Formu a 1.831 ).

Table 832. Compounds of formu a I .A, wherein R2 is R2-- 0.146( = Formu a 1.832).

Table 833. Compounds of formu a I .A, wherein R2 is R2-- 0.147( = Formu a 1.833).

Table 834. Compounds of formu a I .A, wherein R2 is R2-- 0.148( = Formu a 1.834).

Table 835. Compounds of formu a I .A, wherein R2 is R2-- 0.149( = Formu a 1.835).

Table 836. Compounds of formu a I .A, wherein R2 is R2-- 0.150( = Formu a 1.836).

Table 837. Compounds of formu a I .A, wherein R2 is R2-- 0.151 ( = Formu a 1.837).

Table 838. Compounds of formu a I .A, wherein R2 is R2-- 0.152( = Formu a 1.838).

Table 839. Compounds of formu a I .A, wherein R2 is R2-- 0.153( = Formu a 1.839).

Table 840. Compounds of formu a I .A, wherein R2 is R2-- 0.154( = Formu a 1.840).

Table 841 . Compounds of formu a I .A, wherein R2 is R2-- 0.155( = Formu a 1.841 ).

Table 842. Compounds of formu a I .A, wherein R2 is R2-- 0.156( = Formu a 1.842).

Table 843. Compounds of formu a I .A, wherein R2 is R2-- 0.157( = Formu a 1.843).

Table 844. Compounds of formu a I .A, wherein R2 is R2-- 0.158( = Formu a 1.844).

Table 845. Compounds of formu a I .A, wherein R2 is R2-- 0.159( = Formu a 1.845).

Table 846. Compounds of formu a I .A, wherein R2 is R2-- 0.160( = Formu a 1.846).

Table 847. Compounds of formu a I .A, wherein R2 is R2-- 0.161 ( = Formu a 1.847).

Table 848. Compounds of formu a I .A, wherein R2 is R2-- 0.162( = Formu a 1.848).

Table 849. Compounds of formu a I .A, wherein R2 is R2-- 0.163( = Formu a 1.849).

Table 850. Compounds of formu a I .A, wherein R2 is R2-- 0.164( = Formu a 1.850).

Table 851 . Compounds of formu a I .A, wherein R2 is R2-- 0.165( = Formu a 1.851 ).

Table 852. Compounds of formu a I .A, wherein R2 is R2-- 0.166( = Formu a 1.852).

Table 853. Compounds of formu a I .A, wherein R2 is R2-- 0.167( = Formu a 1.853).

Table 854. Compounds of formu a I .A, wherein R2 is R2-- 0.168( = Formu a 1.854).

Table 855. Compounds of formu a I .A, wherein R2 is R2-- 0.169( = Formu a 1.855).

Table 856. Compounds of formu a I .A, wherein R2 is R2-- 0.170( = Formu a 1.856).

Table 857. Compounds of formu a I .A, wherein R2 is R2-- 0.171 ( = Formu a 1.857).

Table 858. Compounds of formu a I .A, wherein R2 is R2-- 0.172( = Formu a 1.858).

Table 859. Compounds of formu a I .A, wherein R2 is R2-- 0.173( = Formu a 1.859).

Table 860. Compounds of formu a I .A, wherein R2 is R2-- 0.174( = Formu a 1.860).

Table 861 . Compounds of formu a I .A, wherein R2 is R2-- 0.175( = Formu a 1.861 ).

Table 862. Compounds of formu a I .A, wherein R2 is R2-- 0.176( = Formu a 1.862).

Table 863. Compounds of formu a I .A, wherein R2 is R2-- 0.177( = Formu a 1.863).

Table 864. Compounds of formu a I .A, wherein R2 is R2-- 0.178( = Formu a 1.864).

Table 865. Compounds of formu a I .A, wherein R2 is R2-- 0.179( = Formu a 1.865).

Table 866. Compounds of formu a I .A, wherein R2 is R2-- 0.180( = Formu a 1.866).

Table 867. Compounds of formu a I .A, wherein R2 is R2-- 0.181 ( = Formu a 1.867).

Table 868. Compounds of formu a I .A, wherein R2 is R2-- 0.182( = Formu a 1.868).

Table 869. Compounds of formu a I .A, wherein R2 is R2-- 0.183( = Formu a 1.869). Table 870. Compounds of formu a I .A, wherein R2 is R2-- 0.184( = Formu a 1.870).

Table 871 . Compounds of formu a I .A, wherein R2 is R2-- 0.185( = Formu a 1.871 ).

Table 872. Compounds of formu a I .A, wherein R2 is R2-- 0.186( = Formu a 1.872).

Table 873. Compounds of formu a I .A, wherein R2 is R2-- 0.187( = Formu a 1.873).

Table 874. Compounds of formu a I .A, wherein R2 is R2-- 0.188( = Formu a 1.874).

Table 875. Compounds of formu a I .A, wherein R2 is R2-- 0.189( = Formu a 1.875).

Table 876. Compounds of formu a I .A, wherein R2 is R2-- 0.190( = Formu a 1.876).

Table 877. Compounds of formu a I .A, wherein R2 is R2-- 0.191 ( = Formu a 1.877).

Table 878. Compounds of formu a I .A, wherein R2 is R2-- 0.192( = Formu a 1.878).

Table 879. Compounds of formu a I .A, wherein R2 is R2-- 0.193( = Formu a 1.879).

Table 880. Compounds of formu a I .A, wherein R2 is R2-- 0.194( = Formu a 1.880).

Table 881 . Compounds of formu a I .A, wherein R2 is R2-- 0.195( = Formu a 1.881 ).

Table 882. Compounds of formu a I .A, wherein R2 is R2-- 0.196( = Formu a 1.882).

Table 883. Compounds of formu a I .A, wherein R2 is R2-- 0.197( = Formu a 1.883).

Table 884. Compounds of formu a I .A, wherein R2 is R2-- 0.198( = Formu a 1.884).

Table 885. Compounds of formu a I .A, wherein R2 is R2-- 0.199( = Formu a 1.885).

Table 886. Compounds of formu a I .A, wherein R2 is R2-- 0.200( = Formu a 1.886).

Table 887. Compounds of formu a I .A, wherein R2 is R2-- 0.201 ( = Formu a 1.887).

Table 888. Compounds of formu a I .A, wherein R2 is R2-- 0.202( = Formu a 1.888).

Table 889. Compounds of formu a I .A, wherein R2 is R2-- 0.203( = Formu a 1.889).

Table 890. Compounds of formu a I .A, wherein R2 is R2-- 0.204( = Formu a 1.890).

Table 891 . Compounds of formu a I .A, wherein R2 is R2-- 0.205( = Formu a 1.891 ).

Table 892. Compounds of formu a I .A, wherein R2 is R2-- 0.206( = Formu a 1.892).

Table 893. Compounds of formu a I .A, wherein R2 is R2-- 0.207( = Formu a 1.893).

Table 894. Compounds of formu a I .A, wherein R2 is R2-- 0.208( = Formu a 1.894).

Table 895. Compounds of formu a I .A, wherein R2 is R2-- 0.209( = Formu a 1.895).

Table 896. Compounds of formu a I .A, wherein R2 is R2-- 0.210( = Formu a 1.896).

Table 897. Compounds of formu a I .A, wherein R2 is R2-- 0.21 1 ( = Formu a 1.897).

Table 898. Compounds of formu a I .A, wherein R2 is R2-- 0.212( = Formu a 1.898).

Table 899. Compounds of formu a I .A, wherein R2 is R2-- 0.213( = Formu a 1.899).

Table 900. Compounds of formu a I .A, wherein R2 is R2-- 0.214( = Formu a 1.900).

Table 901 . Compounds of formu a I .A, wherein R2 is R2-- 0.215( = Formu a 1.901 ).

Table 902. Compounds of formu a I .A, wherein R2 is R2-- 0.216( = Formu a 1.902).

Table 903. Compounds of formu a I .A, wherein R2 is R2-- 0.217( = Formu a 1.903).

Table 904. Compounds of formu a I .A, wherein R2 is R2-- 0.218( = Formu a 1.904).

Table 905. Compounds of formu a I .A, wherein R2 is R2-- 0.219( = Formu a 1.905).

Table 906. Compounds of formu a I .A, wherein R2 is R2-- 0.220( = Formu a 1.906).

Table 907. Compounds of formu a I .A, wherein R2 is R2-- 0.221 ( = Formu a 1.907).

Table 908. Compounds of formu a I .A, wherein R2 is R2-- 0.222( = Formu a 1.908).

Table 909. Compounds of formu a I .A, wherein R2 is R2-- 0.223( = Formu a 1.909).

Table 910. Compounds of formu a I .A, wherein R2 is R2-- 0.224( = Formu a 1.910).

Table 91 1 . Compounds of formu a I .A, wherein R2 is R2-- 0.225( = Formu a 1.91 1 ).

Table 912. Compounds of formu a I .A, wherein R2 is R2-- 0.226( = Formu a 1.912).

Table 913. Compounds of formu a I .A, wherein R2 is R2-- 0.227( = Formu a 1.913). Table 914. Compounds of formu a I .A, wherein R2 is R2-- 0.228( Formu a 1.914).

Table 915. Compounds of formu a I .A, wherein R2 is R2-- 0.229( = Formu a 1.915).

Table 916. Compounds of formu a I .A, wherein R2 is R2-- 0.230( = Formu a 1.916).

Table 917. Compounds of formu a I .A, wherein R2 is R2-- 0.231 ( = Formu a 1.917).

Table 918. Compounds of formu a I .A, wherein R2 is R2-- 0.232( = Formu a 1.918).

Table 919. Compounds of formu a I .A, wherein R2 is R2-- 0.233( = Formu a 1.919).

Table 920. Compounds of formu a I .A, wherein R2 is R2-- 0.234( = Formu a 1.920).

Table 921 . Compounds of formu a I .A, wherein R2 is R2-- 0.235( = Formu a 1.921 ).

Table 922. Compounds of formu a I .A, wherein R2 is R2-- 0.236( = Formu a 1.922).

Table 923. Compounds of formu a I .A, wherein R2 is R2-- 0.237( = Formu a 1.923).

Table 924. Compounds of formu a I .A, wherein R2 is R2-- 0.238( = Formu a 1.924).

Table 925. Compounds of formu a I .A, wherein R2 is R2-- 0.239( = Formu a 1.925).

Table 926. Compounds of formu a I .A, wherein R2 is R2-- 0.240( = Formu a 1.926).

Table 927. Compounds of formu a I .A, wherein R2 is R2-- 0.241 ( = Formu a 1.927).

Table 928. Compounds of formu a I .A, wherein R2 is R2-- 0.242( = Formu a 1.928).

Table 929. Compounds of formu a I .A, wherein R2 is R2-- 0.243( = Formu a 1.929).

Table 930. Compounds of formu a I .A, wherein R2 is R2-- 0.244( = Formu a 1.930).

Table 931 . Compounds of formu a I .A, wherein R2 is R2-- 0.245( = Formu a 1.931 ).

Table 932. Compounds of formu a I .A, wherein R2 is R2-- 0.246( = Formu a 1.932).

Table 933. Compounds of formu a I .A, wherein R2 is R2-- 0.247( = Formu a 1.933).

Table 934. Compounds of formu a I .A, wherein R2 is R2-- 0.248( = Formu a 1.934).

Table 935. Compounds of formu a I .A, wherein R2 is R2-- 0.249( = Formu a 1.935).

Table 936. Compounds of formu a I .A, wherein R2 is R2-- 0.250( = Formu a 1.936).

Table 937. Compounds of formu a I .A, wherein R2 is R2-- 0.251 ( = Formu a 1.937).

Table 938. Compounds of formu a I .A, wherein R2 is R2-- 0.252( = Formu a 1.938).

Table 939. Compounds of formu a I .A, wherein R2 is R2-- 0.253( = Formu a 1.939).

Table 940. Compounds of formu a I .A, wherein R2 is R2-- 0.254( = Formu a 1.940).

Table 941 . Compounds of formu a I .A, wherein R2 is R2-- 0.255( = Formu a 1.941 ).

Table 942. Compounds of formu a I .A, wherein R2 is R2-- 0.256( = Formu a 1.942).

Table 943. Compounds of formu a I .A, wherein R2 is R2-- 0.257( = Formu a 1.943).

Table 944. Compounds of formu a I .A, wherein R2 is R2-- 0.258( = Formu a 1.944).

Table 945. Compounds of formu a I .A, wherein R2 is R2-- 0.259( = Formu a 1.945).

Table 946. Compounds of formu a I .A, wherein R2 is R2-- 0.260( = Formu a 1.946).

Table 947. Compounds of formu a I .A, wherein R2 is R2-- 0.261 ( = Formu a 1.947).

Table 948. Compounds of formu a I .A, wherein R2 is R2-- 0.262( = Formu a 1.948).

Table 949. Compounds of formu a I .A, wherein R2 is R2-- 0.263( = Formu a 1.949).

Table 950. Compounds of formu a I .A, wherein R2 is R2-- 0.264( = Formu a 1.950).

Table 951 . Compounds of formu a I .A, wherein R2 is R2-- 0.265( = Formu a 1.951 ).

Table 952. Compounds of formu a I .A, wherein R2 is R2-- 0.266( = Formu a 1.952).

Table 953. Compounds of formu a I .A, wherein R2 is R2-- 0.267( = Formu a 1.953).

Table 954. Compounds of formu a I .A, wherein R2 is R2-- 0.268( = Formu a 1.954).

Table 955. Compounds of formu a I .A, wherein R2 is R2-- 0.269( = Formu a 1.955).

Table 956. Compounds of formu a I .A, wherein R2 is R2-- 0.270( = Formu a 1.956).

Table 957. Compounds of formu a I .A, wherein R2 is R2-- 0.271 ( = Formu a 1.957). Table 958. Compounds of formu a I .A, wherein R2 is R2-- 0.272( Formu a 1.958).

Table 959. Compounds of formu a I .A, wherein R2 is R2-- 0.273( = Formu a 1.959).

Table 960. Compounds of formu a I .A, wherein R2 is R2-- 0.274( = Formu a 1.960).

Table 961 . Compounds of formu a I .A, wherein R2 is R2-- 0.275( = Formu a 1.961 ).

Table 962. Compounds of formu a I .A, wherein R2 is R2-- 0.276( = Formu a 1.962).

Table 963. Compounds of formu a I .A, wherein R2 is R2-- 0.277( = Formu a 1.963).

Table 964. Compounds of formu a I .A, wherein R2 is R2-- 0.278( = Formu a 1.964).

Table 965. Compounds of formu a I .A, wherein R2 is R2-- 0.279( = Formu a 1.965).

Table 966. Compounds of formu a I .A, wherein R2 is R2-- 0.280( = Formu a 1.966).

Table 967. Compounds of formu a I .A, wherein R2 is R2-- 0.281 ( = Formu a 1.967).

Table 968. Compounds of formu a I .A, wherein R2 is R2-- 0.282( = Formu a 1.968).

Table 969. Compounds of formu a I .A, wherein R2 is R2-- 0.283( = Formu a 1.969).

Table 970. Compounds of formu a I .A, wherein R2 is R2-- 0.284( = Formu a 1.970).

Table 971 . Compounds of formu a I .A, wherein R2 is R2-- 0.285( = Formu a 1.971 ).

Table 972. Compounds of formu a I .A, wherein R2 is R2-- 0.286( = Formu a 1.972).

Table 973. Compounds of formu a I .A, wherein R2 is R2-- 0.287( = Formu a 1.973).

Table 974. Compounds of formu a I .A, wherein R2 is R2-- 0.288( = Formu a 1.974).

Table 975. Compounds of formu a I .A, wherein R2 is R2-- 0.289( = Formu a 1.975).

Table 976. Compounds of formu a I .A, wherein R2 is R2-- 0.290( = Formu a 1.976).

Table 977. Compounds of formu a I .A, wherein R2 is R2-- 0.291 ( = Formu a 1.977).

Table 978. Compounds of formu a I .A, wherein R2 is R2-- 0.292( = Formu a 1.978).

Table 979. Compounds of formu a I .A, wherein R2 is R2-- 0.293( = Formu a 1.979).

Table 980. Compounds of formu a I .A, wherein R2 is R2-- 0.294( = Formu a 1.980).

Table 981 . Compounds of formu a I .A, wherein R2 is R2-- 0.295( = Formu a 1.981 ).

Table 982. Compounds of formu a I .A, wherein R2 is R2-- 0.296( = Formu a 1.982).

Table 983. Compounds of formu a I .A, wherein R2 is R2-- 0.297( = Formu a 1.983).

Table 984. Compounds of formu a I .A, wherein R2 is R2-- 0.298( = Formu a 1.984).

Table 985. Compounds of formu a I .A, wherein R2 is R2-- 0.299( = Formu a 1.985).

Table 986. Compounds of formu a I .A, wherein R2 is R2-- 0.300( = Formu a 1.986).

Table 987. Compounds of formu a I .A, wherein R2 is R2-- 0.301 ( = Formu a 1.987).

Table 988. Compounds of formu a I .A, wherein R2 is R2-- 0.302( = Formu a 1.988).

Table 989. Compounds of formu a I .A, wherein R2 is R2-- 0.303( = Formu a 1.989).

Table 990. Compounds of formu a I .A, wherein R2 is R2-- 0.304( = Formu a 1.990).

Table 991 . Compounds of formu a I .A, wherein R2 is R2-- 0.305( = Formu a 1.991 ).

Table 992. Compounds of formu a I .A, wherein R2 is R2-- 0.306( = Formu a 1.992).

Table 993. Compounds of formu a I .A, wherein R2 is R2-- 0.307( = Formu a 1.993).

Table 994. Compounds of formu a I .A, wherein R2 is R2-- 0.308( = Formu a 1.994).

Table 995. Compounds of formu a I .A, wherein R2 is R2-- 0.309( = Formu a 1.995).

Table 996. Compounds of formu a I .A, wherein R2 is R2-- 0.310( = Formu a 1.996).

Table 997. Compounds of formu a I .A, wherein R2 is R2-- 0.31 1 ( = Formu a 1.997).

Table 998. Compounds of formu a I .A, wherein R2 is R2-- 0.312( = Formu a 1.998).

Table 999. Compounds of formu a I .A, wherein R2 is R2-- 0.313( = Formu a 1.999).

Table 1000. Compounds of formu a I .A, wherein R2 is R2-- 0.314( = Formu a 1.1000)

Table 1001. Compounds of formu a I .A, wherein R2 is R2-- 0.315( = Formu a 1.1001 ) Table 1002. Compounds of formu a I .A, wherein R2 is R2-- 0.316( Formu a 1.1002)

Table 1003. Compounds of formu a I .A, wherein R2 is R2-- 0.317( = Formu a 1 .1003)

Table 1004. Compounds of formu a I .A, wherein R2 is R2-- 0.318( = Formu a 1 .1004)

Table 1005. Compounds of formu a I .A, wherein R2 is R2-- 0.319( = Formu a 1 .1005)

Table 1006. Compounds of formu a I .A, wherein R2 is R2-- 0.320( = Formu a 1 .1006)

Table 1007. Compounds of formu a I .A, wherein R2 is R2-- 0.321 ( = Formu a 1 .1007)

Table 1008. Compounds of formu a I .A, wherein R2 is R2-- 0.322( = Formu a 1 .1008)

Table 1009. Compounds of formu a I .A, wherein R2 is R2-- 0.323( = Formu a 1 .1009)

Table 1010. Compounds of formu a I .A, wherein R2 is R2-- 0.324( = Formu a 1 .1010)

Table 101 1. Compounds of formu a I .A, wherein R2 is R2-- 0.325( = Formu a 1 .101 1 )

Table 1012. Compounds of formu a I .A, wherein R2 is R2-- 0.326( = Formu a 1 .1012)

Table 1013. Compounds of formu a I .A, wherein R2 is R2-- 0.327( = Formu a 1 .1013)

Table 1014. Compounds of formu a I .A, wherein R2 is R2-- 0.328( = Formu a 1 .1014)

Table 1015. Compounds of formu a I .A, wherein R2 is R2-- 0.329( = Formu a 1 .1015)

Table 1016. Compounds of formu a I .A, wherein R2 is R2-- 0.330( = Formu a 1 .1016)

Table 1017. Compounds of formu a I .A, wherein R2 is R2-- 0.331 ( = Formu a 1 .1017)

Table 1018. Compounds of formu a I .A, wherein R2 is R2-- 0.332( = Formu a 1 .1018)

Table 1019. Compounds of formu a I .A, wherein R2 is R2-- 0.333( = Formu a 1 .1019)

Table 1020. Compounds of formu a I .A, wherein R2 is R2-- 0.334( = Formu a 1 .1020)

Table 1021. Compounds of formu a I .A, wherein R2 is R2-- 0.335( = Formu a 1 .1021 )

Table 1022. Compounds of formu a I .A, wherein R2 is R2-- 0.336( = Formu a 1 .1022)

Table 1023. Compounds of formu a I .A, wherein R2 is R2-- 0.334( = Formu a 1 .1023)

Table 1024. Compounds of formu a I .A, wherein R2 is R2-- 0.338( = Formu a 1 .1024)

Table 1025. Compounds of formu a I .A, wherein R2 is R2-- 0.339( = Formu a 1 .1025)

Table 1026. Compounds of formu a I .A, wherein R2 is R2-- 0.340( = Formu a 1 .1026)

Table 1027. Compounds of formu a I .A, wherein R2 is R2-- 0.341 ( = Formu a 1 .1027)

Table 1028. Compounds of formu a I .A, wherein R2 is R2-- 0.342( = Formu a 1 .1028)

Table 1029. Compounds of formu a I .A, wherein R2 is R2-- 0.343( = Formu a 1 .1029)

Table 1030. Compounds of formu a I .A, wherein R2 is R2-- 0.344( = Formu a 1 .1030)

Table 1031. Compounds of formu a I .A, wherein R2 is R2-- 0.345( = Formu a 1 .1031 )

Table 1032. Compounds of formu a I .A, wherein R2 is R2-- 0.346( = Formu a 1 .1032)

Table 1033. Compounds of formu a I .A, wherein R2 is R2-- 0.347( = Formu a 1 .1033)

Table 1034. Compounds of formu a I .A, wherein R2 is R2-- 0.348( = Formu a 1 .1034)

Table 1035. Compounds of formu a I .A, wherein R2 is R2-- 0.349( = Formu a 1 .1035)

Table 1036. Compounds of formu a I .A, wherein R2 is R2-- 0.350( = Formu a 1 .1036)

Table 1037. Compounds of formu a I .A, wherein R2 is R2-- 0.351 ( = Formu a 1 .1037)

Table 1038. Compounds of formu a I .A, wherein R2 is R2-- 0.352( = Formu a 1 .1038)

Table 1039. Compounds of formu a I .A, wherein R2 is R2-- 0.353( = Formu a 1 .1039)

Table 1040. Compounds of formu a I .A, wherein R2 is R2-- 0.354( = Formu a 1 .1040)

Table 1041. Compounds of formu a I .A, wherein R2 is R2-- 0.355( = Formu a 1 .1041 )

Table 1042. Compounds of formu a I .A, wherein R2 is R2-- 0.356( = Formu a 1 .1042)

Table 1043. Compounds of formu a I .A, wherein R2 is R2-- 0.357( = Formu a 1 .1043)

Table 1044. Compounds of formu a I .A, wherein R2 is R2-- 0.358( = Formu a 1 .1044)

Table 1045. Compounds of formu a I .A, wherein R2 is R2-- 0.359( = Formu a 1 .1045) Table 1046. Compounds of formu a I .A, wherein R2 is R2-- 0.360( = Formu a 1 .1046).

Table 1047. Compounds of formu a I .A, wherein R2 is R2-- 0.361 ( = Formu a 1 .1047).

Table 1048. Compounds of formu a I .A, wherein R2 is R2-- 0.362( = Formu a 1 .1048).

Table 1049. Compounds of formu a I .A, wherein R2 is R2-- 0.363( = Formu a 1 .1049).

Table 1050. Compounds of formu a I .A, wherein R2 is R2-- 0.364( = Formu a 1 .1050).

Table 1051. Compounds of formu a I .A, wherein R2 is R2-- 0.365( = Formu a 1 .1051 ).

Table 1052. Compounds of formu a I .A, wherein R2 is R2-- 0.366( = Formu a 1 .1052).

Table 1053. Compounds of formu a I .A, wherein R2 is R2-- 0.367( = Formu a 1 .1053).

Table 1054. Compounds of formu a I .A, wherein R2 is R2-- 0.368( = Formu a 1 .1054).

Table 1055. Compounds of formu a I .A, wherein R2 is R2-- 0.369( = Formu a 1 .1055).

Table 1056. Compounds of formu a I .A, wherein R2 is R2-- 0.370( = Formu a 1 .1056).

Table 1057. Compounds of formu a I .A, wherein R2 is R2-- 0.371 ( = Formu a 1 .1057).

Table 1058. Compounds of formu a I .A, wherein R2 is R2-- 0.372( = Formu a 1 .1058).

Table 1059. Compounds of formu a I .A, wherein R2 is R2-- 0.373( = Formu a 1 .1059).

Table 1060. Compounds of formu a I .A, wherein R2 is R2-- 0.374( = Formu a 1 .1060).

Table 1061. Compounds of formu a I .A, wherein R2 is R2-- 0.375( = Formu a 1 .1061 ).

Table 1062. Compounds of formu a I .A, wherein R2 is R2-- 0.376( = Formu a 1 .1062).

Table 1063. Compounds of formu a I .A, wherein R2 is R2-- 0.377( = Formu a 1 .1063).

Table 1064. Compounds of formu a I .A, wherein R2 is R2-- 0.378( = Formu a 1 .1064).

Table 1065. Compounds of formu a I .A, wherein R2 is R2-- 0.379( = Formu a 1 .1065).

Table 1066. Compounds of formu a I .A, wherein R2 is R2-- 0.380( = Formu a 1 .1066).

Table 1067. Compounds of formu a I .A, wherein R2 is R2-- 0.381 ( = Formu a 1 .1067).

Table 1068. Compounds of formu a I .A, wherein R2 is R2-- 0.382( = Formu a 1 .1068).

Table 1069. Compounds of formu a I .A, wherein R2 is R2-- 0.383( = Formu a 1 .1069).

Table 1070. Compounds of formu a I .A, wherein R2 is R2-- 0.384( = Formu a 1 .1070).

Table 1071. Compounds of formu a I .A, wherein R2 is R2-- 0.385( = Formu a 1 .1071 ).

Table 1072. Compounds of formu a I .A, wherein R2 is R2-- 0.386( = Formu a 1 .1072).

Table 1073. Compounds of formu a I .A, wherein R2 is R2-- 0.387( = Formu a 1 .1073).

Table 1074. Compounds of formu a I .A, wherein R2 is R2-- 0.388( = Formu a 1 .1074).

Table 1075. Compounds of formu a I .A, wherein R2 is R2-- 0.389( = Formu a 1 .1075).

Table 1076. Compounds of formu a I .A, wherein R2 is R2-- 0.390( = Formu a 1 .7076).

Table 1077. Compounds of formu a I .A, wherein R2 is R2-- 0.391 ( = Formu a 1 .1077).

Table 1078. Compounds of formu a I .A, wherein R2 is R2-- 0.392( = Formu a 1 .1078).

Table 1079. Compounds of formu a I .A, wherein R2 is R2-- 0.393( = Formu a 1 .1079).

Table 1080. Compounds of formu a I .A, wherein R2 is R2-- 0.394( = Formu a 1 .1080).

Table 1081. Compounds of formu a I .A, wherein R2 is R2-- 0.395( = Formu a 1 .1081 ).

Table 1082. Compounds of formu a I .A, wherein R2 is R2-- 0.396( = Formu a 1 .1082).

Table 1083. Compounds of formu a I .A, wherein R2 is R2-- 0.397( = Formu a 1 .1083).

Table 1084. Compounds of formu a I .A, wherein R2 is R2-- 0.398( = Formu a 1 .1084).

Table 1085. Compounds of formu a I .A, wherein R2 is R2-- 0.399( = Formu a 1 .1085).

Table 1086. Compounds of formu a I .A, wherein R2 is R2-- 0.400( = Formu a 1 .1086).

Table 1087. Compounds of formu a I .A, wherein R2 is R2-- 0.401 ( = Formu a 1 .1087).

Table 1088. Compounds of formu a I .A, wherein R2 is R2-- 0.402( = Formu a 1 .1088).

Table 1089. Compounds of formu a I .A, wherein R2 is R2-- 0.403( = Formu a 1 .1089). Table 1090. Compounds of formu a I .A, wherein R2 is R2-- 0.404( = Formu a 1.1090).

Table 1091. Compounds of formu a I .A, wherein R2 is R2-- 0.405( = Formu a 1 .1091).

Table 1092. Compounds of formu a I .A, wherein R2 is R2-- 0.406( = Formu a 1 .1092).

Table 1093. Compounds of formu a I .A, wherein R2 is R2-- 0.407( = Formu a 1 .1093).

Table 1094. Compounds of formu a I .A, wherein R2 is R2-- 0.408( = Formu a 1 .1094).

Table 1095. Compounds of formu a I .A, wherein R2 is R2-- 0.409( = Formu a 1 .1095).

Table 1096. Compounds of formu a I .A, wherein R2 is R2-- 0.410( = Formu a 1 .1096).

Table 1097. Compounds of formu a I .A, wherein R2 is R2-- 0.411( = Formu a 1 .1097).

Table 1098. Compounds of formu a I .A, wherein R2 is R2-- 0.412( = Formu a 1 .1098).

Table 1099. Compounds of formu a I .A, wherein R2 is R2-- 0.413( = Formu a 1 .1099).

Table 1100. Compounds of formu a I .A, wherein R2 is R2-- 0.414( = Formu a 1 .1100).

Table 1101. Compounds of formu a I .A, wherein R2 is R2-- 0.415( = Formu a 1 .1101).

Table 1102. Compounds of formu a I .A, wherein R2 is R2-- 0.416( = Formu a 1 .1102).

Table 1103. Compounds of formu a I .A, wherein R2 is R2-- 0.417( = Formu a 1 .1103).

Table 1104. Compounds of formu a I .A, wherein R2 is R2-- 0.418( = Formu a 1 .1104).

Table 1105. Compounds of formu a I .A, wherein R2 is R2-- 0.419( = Formu a 1 .1105).

Table 1106. Compounds of formu a I .A, wherein R2 is R2-- 0.420( = Formu a 1 .1106).

Table 1107. Compounds of formu a I .A, wherein R2 is R2-- 0.421 ( = Formu a 1 .1107).

Table 1108. Compounds of formu a I .A, wherein R2 is R2-- 0.422( = Formu a 1 .1108).

Table 1109. Compounds of formu a I .A, wherein R2 is R2-- 0.423( = Formu a 1 .1109).

Table 1110. Compounds of formu a I .A, wherein R2 is R2-- 0.424( = Formu a 1 .1110).

Table 1111. Compounds of formu a I .A, wherein R2 is R2-- 0.425( = Formu a 1 .1111).

Table 1112. Compounds of formu a I .A, wherein R2 is R2-- 0.426( = Formu a 1 .1112).

Table 1113. Compounds of formu a I .A, wherein R2 is R2-- 0.427( = Formu a 1 .1113).

Table 1114. Compounds of formu a I .A, wherein R2 is R2-- 0.428( = Formu a 1 .1114).

Table 1115. Compounds of formu a I .A, wherein R2 is R2-- 0.429( = Formu a 1 .1115).

Table 1116. Compounds of formu a I .A, wherein R2 is R2-- 0.430( = Formu a 1 .1116).

Table 1117. Compounds of formu a I .A, wherein R2 is R2-- 0.431 ( = Formu a 1 .1117).

Table 1118. Compounds of formu a I .A, wherein R2 is R2-- 0.432( = Formu a 1 .1118).

Table 1119. Compounds of formu a I .A, wherein R2 is R2-- 0.433( = Formu a 1 .1119).

Table 1120. Compounds of formu a I .A, wherein R2 is R2-- 0.434( = Formu a 1 .1120).

Table 1121. Compounds of formu a I .A, wherein R2 is R2-- 0.435( = Formu a 1 .1121).

Table 1122. Compounds of formu a I .A, wherein R2 is R2-- 0.436( = Formu a 1 .1122).

Table 1123. Compounds of formu a I .A, wherein R2 is R2-- 0.437( = Formu a 1 .1123).

Table 1124. Compounds of formu a I .A, wherein R2 is R2-- 0.438( = Formu a 1 .1124).

Table 1125. Compounds of formu a I .A, wherein R2 is R2-- 0.439( = Formu a 1 .1125).

Table 1126. Compounds of formu a I .A, wherein R2 is R2-- 0.440( = Formu a 1 .1126).

Table 1127. Compounds of formu a I .A, wherein R2 is R2-- 0.441 ( = Formu a 1 .1127).

Table 1128. Compounds of formu a I .A, wherein R2 is R2-- 0.442( = Formu a 1 .1128).

Table 1129. Compounds of formu a I .A, wherein R2 is R2-- 0.443( = Formu a 1 .1129).

Table 1130. Compounds of formu a I .A, wherein R2 is R2-- 0.444( = Formu a 1 .1130).

Table 1131. Compounds of formu a I .A, wherein R2 is R2-- 0.445( = Formu a 1 .1131).

Table 1132. Compounds of formu a I .A, wherein R2 is R2-- 0.446( = Formu a 1 .1132).

Table 1133. Compounds of formu a I .A, wherein R2 is R2-- 0.447( = Formu a 1 .1133). Table 1134. Compounds of formu a I .A, wherein R2 is R2-- 0.448( = Formu a 1.1134).

Table 1135. Compounds of formu a I .A, wherein R2 is R2-- 0.449( = Formu a 1 .1135).

Table 1136. Compounds of formu a I .A, wherein R2 is R2-- 0.450( = Formu a 1 .1136).

Table 1137. Compounds of formu a I .A, wherein R2 is R2-- 0.451 ( = Formu a 1 .1137).

Table 1138. Compounds of formu a I .A, wherein R2 is R2-- 0.452( = Formu a 1 .1138).

Table 1139. Compounds of formu a I .A, wherein R2 is R2-- 0.453( = Formu a 1 .1139).

Table 1140. Compounds of formu a I .A, wherein R2 is R2-- 0.454( = Formu a 1 .1140).

Table 1141. Compounds of formu a I .A, wherein R2 is R2-- 0.455( = Formu a 1 .1141).

Table 1142. Compounds of formu a I .A, wherein R2 is R2-- 0.456( = Formu a 1 .1142).

Table 1143. Compounds of formu a I .A, wherein R2 is R2-- 0.457( = Formu a 1 .1143).

Table 1144. Compounds of formu a I .A, wherein R2 is R2-- 0.458( = Formu a 1 .1144).

Table 1145. Compounds of formu a I .A, wherein R2 is R2-- 0.459( = Formu a 1 .1145).

Table 1146. Compounds of formu a I .A, wherein R2 is R2-- 0.460( = Formu a 1 .1146).

Table 1147. Compounds of formu a I .A, wherein R2 is R2-- 0.461 ( = Formu a 1 .1147).

Table 1148. Compounds of formu a I .A, wherein R2 is R2-- 0.462( = Formu a 1 .1148).

Table 1149. Compounds of formu a I .A, wherein R2 is R2-- 0.463( = Formu a 1 .1149).

Table 1150. Compounds of formu a I .A, wherein R2 is R2-- 0.464( = Formu a 1 .1150).

Table 1151. Compounds of formu a I .A, wherein R2 is R2-- 0.465( = Formu a 1 .1151).

Table 1152. Compounds of formu a I .A, wherein R2 is R2-- 0.466( = Formu a 1 .1152).

Table 1153. Compounds of formu a I .A, wherein R2 is R2-- 0.467( = Formu a 1 .1153).

Table 1154. Compounds of formu a I .A, wherein R2 is R2-- 0.468( = Formu a 1 .1154).

Table 1155. Compounds of formu a I .A, wherein R2 is R2-- 0.469( = Formu a 1 .1154).

Table 1156. Compounds of formu a I .A, wherein R2 is R2-- 0.470( = Formu a 1 .1156).

Table 1157. Compounds of formu a I .A, wherein R2 is R2-- 0.471 ( = Formu a 1 .1157).

Table 1158. Compounds of formu a I .A, wherein R2 is R2-- 0.472( = Formu a 1 .1158).

Table 1159. Compounds of formu a I .A, wherein R2 is R2-- 0.473( = Formu a 1 .1159).

Table 1160. Compounds of formu a I .A, wherein R2 is R2-- 0.474( = Formu a 1 .1160).

Table 1161. Compounds of formu a I .A, wherein R2 is R2-- 0.475( = Formu a 1 .1161).

Table 1162. Compounds of formu a I .A, wherein R2 is R2-- 0.476( = Formu a 1 .1162).

Table 1163. Compounds of formu a I .A, wherein R2 is R2-- 0.477( = Formu a 1 .1163).

Table 1164. Compounds of formu a I .A, wherein R2 is R2-- 0.478( = Formu a 1 .1164).

Table 1165. Compounds of formu a I .A, wherein R2 is R2-- 0.479( = Formu a 1 .1165).

Table 1166. Compounds of formu a I .A, wherein R2 is R2-- 0.480( = Formu a 1 .1166).

Table 1167. Compounds of formu a I .A, wherein R2 is R2-- 0.481 ( = Formu a 1 .1167).

Table 1168. Compounds of formu a I .A, wherein R2 is R2-- 0.482( = Formu a 1 .1168).

Table 1169. Compounds of formu a I .A, wherein R2 is R2-- 0.483( = Formu a 1 .1169).

Table 1170. Compounds of formu a I .A, wherein R2 is R2-- 0.484( = Formu a 1 .1170).

Table 1171. Compounds of formu a I .A, wherein R2 is R2-- 0.485( = Formu a 1 .1171).

Table 1172. Compounds of formu a I .A, wherein R2 is R2-- 0.486( = Formu a 1 .1172).

Table 1173. Compounds of formu a I .A, wherein R2 is R2-- 0.487( = Formu a 1 .1173).

Table 1174. Compounds of formu a I .A, wherein R2 is R2-- 0.488( = Formu a 1 .1174).

Table 1175. Compounds of formu a I .A, wherein R2 is R2-- 0.489( = Formu a 1 .1175).

Table 1176. Compounds of formu a I .A, wherein R2 is R2-- 0.490( = Formu a 1 .1176).

Table 1177. Compounds of formu a I .A, wherein R2 is R2-- 0.491 ( = Formu a 1 .1177). Table 1 178. Compounds of formu a I .A, wherein R2 is R2-- 0.492( Formu a 1.1 178)

Table 1 179. Compounds of formu a I .A, wherein R2 is R2-- 0.493( = Formu a 1 .1 179)

Table 1 180. Compounds of formu a I .A, wherein R2 is R2-- 0.494( = Formu a 1 .1 180)

Table 1 181. Compounds of formu a I .A, wherein R2 is R2-- 0.495( = Formu a 1 .1 181 )

Table 1 182. Compounds of formu a I .A, wherein R2 is R2-- 0.496( = Formu a 1 .1 182)

Table 1 183. Compounds of formu a I .A, wherein R2 is R2-- 0.497( = Formu a 1 .1 183)

Table 1 184. Compounds of formu a I .A, wherein R2 is R2-- 0.498( = Formu a 1 .1 184)

Table 1 185. Compounds of formu a I .A, wherein R2 is R2-- 0.499( = Formu a 1 .1 185)

Table 1 186. Compounds of formu a I .A, wherein R2 is R2-- 0.500( = Formu a 1 .1 186)

Table 1 187. Compounds of formu a I .A, wherein R2 is R2-- 0.501 ( = Formu a 1 .1 187)

Table 1 188. Compounds of formu a I .A, wherein R2 is R2-- 0.502( = Formu a 1 .1 188)

Table 1 189. Compounds of formu a I .A, wherein R2 is R2-- 0.503( = Formu a 1 .1 189)

Table 1 190. Compounds of formu a I .A, wherein R2 is R2-- 0.504( = Formu a 1 .1 190)

Table 1 191. Compounds of formu a I .A, wherein R2 is R2-- 0.505( = Formu a 1 .1 191 )

Table 1 192. Compounds of formu a I .A, wherein R2 is R2-- 0.506( = Formu a 1 .1 192)

Table 1 193. Compounds of formu a I .A, wherein R2 is R2-- 0.507( = Formu a 1 .1 193)

Table 1 194. Compounds of formu a I .A, wherein R2 is R2-- 0.508( = Formu a 1 .1 194)

Table 1 195. Compounds of formu a I .A, wherein R2 is R2-- 0.509( = Formu a 1 .1 195)

Table 1 196. Compounds of formu a I .A, wherein R2 is R2-- 0.510( = Formu a 1 .1 196)

Table 1 197. Compounds of formu a I .A, wherein R2 is R2-- 0.51 1 ( = Formu a 1 .1 197)

Table 1 198. Compounds of formu a I .A, wherein R2 is R2-- 0.512( = Formu a 1 .1 198)

Table 1 199. Compounds of formu a I .A, wherein R2 is R2-- 0.513( = Formu a 1 .1 199)

Table 1200. Compounds of formu a I .A, wherein R2 is R2-- 0.514( = Formu a 1 .1200)

Table 1201. Compounds of formu a I .A, wherein R2 is R2-- 0.515( = Formu a 1 .1201 )

Table 1202. Compounds of formu a I .A, wherein R2 is R2-- 0.516( = Formu a 1 .1202)

Table 1203. Compounds of formu a I .A, wherein R2 is R2-- 0.517( = Formu a 1 .1203)

Table 1204. Compounds of formu a I .A, wherein R2 is R2-- 0.518( = Formu a 1 .1204)

Table 1205. Compounds of formu a I .A, wherein R2 is R2-- 0.519( = Formu a 1 .1205)

Table 1206. Compounds of formu a I .A, wherein R2 is R2-- 0.520( = Formu a 1 .1206)

Table 1207. Compounds of formu a I .A, wherein R2 is R2-- 0.521 ( = Formu a 1 .1207)

Table 1208. Compounds of formu a I .A, wherein R2 is R2-- 0.522( = Formu a 1 .1208)

Table 1209. Compounds of formu a I .A, wherein R2 is R2-- 0.523( = Formu a 1 .1209)

Table 1210. Compounds of formu a I .A, wherein R2 is R2-- 0.524( = Formu a 1 .1210)

Table 121 1. Compounds of formu a I .A, wherein R2 is R2-- 0.525( = Formu a 1 .121 1 )

Table 1212. Compounds of formu a I .A, wherein R2 is R2-- 0.526( = Formu a 1 .1212)

Table 1213. Compounds of formu a I .A, wherein R2 is R2-- 0.527( = Formu a 1 .1213)

Table 1214. Compounds of formu a I .A, wherein R2 is R2-- 0.528( = Formu a 1 .1212)

Table 1215. Compounds of formu a I .A, wherein R2 is R2-- 0.529( = Formu a 1 .1215)

Table 1216. Compounds of formu a I .A, wherein R2 is R2-- 0.530( = Formu a 1 .1216)

Table 1217. Compounds of formu a I .A, wherein R2 is R2-- 0.531 ( = Formu a 1 .1217)

Table 1218. Compounds of formu a I .A, wherein R2 is R2-- 0.532( = Formu a 1 .1218)

Table 1219. Compounds of formu a I .A, wherein R2 is R2-- 0.533( = Formu a 1 .1219)

Table 1220. Compounds of formu a I .A, wherein R2 is R2-- 0.534( = Formu a 1 .1220)

Table 1221. Compounds of formu a I .A, wherein R2 is R2-- 0.535( = Formu a 1 .1221 ) Table 1222. Compounds of formu a I .A, wherein R2 is R2-- 0.536( = Formu a 1.1222).

Table 1223. Compounds of formu a I .A, wherein R2 is R2-- 0.537( = Formu a 1 .1223).

Table 1224. Compounds of formu a I .A, wherein R2 is R2-- 0.538( = Formu a 1 .1224).

Table 1225. Compounds of formu a I .A, wherein R2 is R2-- 0.539( = Formu a 1 .1225).

Table 1226. Compounds of formu a I .A, wherein R2 is R2-- 0.540( = Formu a 1 .1226).

Table 1227. Compounds of formu a I .A, wherein R2 is R2-- 0.541 ( = Formu a 1 .1227).

Table 1228. Compounds of formu a I .A, wherein R2 is R2-- 0.542( = Formu a 1 .1228).

Table 1229. Compounds of formu a I .A, wherein R2 is R2-- 0.543( = Formu a 1 .1229).

Table 1230. Compounds of formu a I .A, wherein R2 is R2-- 0.544( = Formu a 1 .1230).

Table 1231. Compounds of formu a I .A, wherein R2 is R2-- 0.545( = Formu a 1 .1231 ).

Table 1232. Compounds of formu a I .A, wherein R2 is R2-- 0.546( = Formu a 1 .1232).

Table 1233. Compounds of formu a I .A, wherein R2 is R2-- 0.547( = Formu a 1 .1233).

Table 1234. Compounds of formu a I .A, wherein R2 is R2-- 0.548( = Formu a 1 .1234).

Table 1235. Compounds of formu a I .A, wherein R2 is R2-- 0.549( = Formu a 1 .1235).

Table 1236. Compounds of formu a I .A, wherein R2 is R2-- 0.550( = Formu a 1 .1236).

Table 1237. Compounds of formu a I .A, wherein R2 is R2-- 0.551 ( = Formu a 1 .1237).

Table 1238. Compounds of formu a I .A, wherein R2 is R2-- 0.552( = Formu a 1 .1238).

Table 1239. Compounds of formu a I .A, wherein R2 is R2-- 0.553( = Formu a 1 .1239).

Table 1240. Compounds of formu a I .A, wherein R2 is R2-- 0.554( = Formu a 1 .1240).

Table 1241. Compounds of formu a I .A, wherein R2 is R2-- 0.555( = Formu a 1 .1241 ).

Table 1242. Compounds of formu a I .A, wherein R2 is R2-- 0.556( = Formu a 1 .1242).

Table 1243. Compounds of formu a I .A, wherein R2 is R2-- 0.557( = Formu a 1 .1243).

Table 1244. Compounds of formu a I .A, wherein R2 is R2-- 0.558( = Formu a 1 .1244).

Table 1245. Compounds of formu a I .A, wherein R2 is R2-- 0.559( = Formu a 1 .1245).

Table 1246. Compounds of formu a I .A, wherein R2 is R2-- 0.560( = Formu a 1 .1246).

Table 1247. Compounds of formu a I .A, wherein R2 is R2-- 0.561 ( = Formu a 1 .1247).

Table 1248. Compounds of formu a I .A, wherein R2 is R2-- 0.562( = Formu a 1 .1248).

Table 1249. Compounds of formu a I .A, wherein R2 is R2-- 0.563( = Formu a 1 .1249).

Table 1250. Compounds of formu a I .A, wherein R2 is R2-- 0.564( = Formu a 1 .1350).

Table 1251. Compounds of formu a I .A, wherein R2 is R2-- 0.565( = Formu a 1 .1251 ).

Table 1252. Compounds of formu a I .A, wherein R2 is R2-- 0.566( = Formu a 1 .1252).

Table 1253. Compounds of formu a I .A, wherein R2 is R2-- 0.567( = Formu a 1 .1253).

Table 1254. Compounds of formu a I .A, wherein R2 is R2-- 0.568( = Formu a 1 .1254).

Table 1255. Compounds of formu a I .A, wherein R2 is R2-- 0.569( = Formu a 1 .1255).

Table 1256. Compounds of formu a I .A, wherein R2 is R2-- 0.570( = Formu a 1 .1256).

Table 1257. Compounds of formu a I .A, wherein R2 is R2-- 0.571 ( = Formu a 1 .1257).

Table 1258. Compounds of formu a I .A, wherein R2 is R2-- 0.572( = Formu a 1 .1258).

Table 1259. Compounds of formu a I .A, wherein R2 is R2-- 0.573( = Formu a 1 .1259).

Table 1260. Compounds of formu a I .A, wherein R2 is R2-- 0.574( = Formu a 1 .1260).

Table 1261. Compounds of formu a I .A, wherein R2 is R2-- 0.575( = Formu a 1 .1261 ).

Table 1262. Compounds of formu a I .A, wherein R2 is R2-- 0.576( = Formu a 1 .1262).

Table 1263. Compounds of formu a I .A, wherein R2 is R2-- 0.577( = Formu a 1 .1263).

Table 1264. Compounds of formu a I .A, wherein R2 is R2-- 0.578( = Formu a 1 .1264).

Table 1265. Compounds of formu a I .A, wherein R2 is R2-- 0.579( = Formu a 1 .1265). Table 1266. Compounds of formu a I .A, wherein R2 is R2-- 0.580( = Formu a 1.1266).

Table 1267. Compounds of formu a I .A, wherein R2 is R2-- 0.581 ( = Formu a 1 .1267).

Table 1268. Compounds of formu a I .A, wherein R2 is R2-- 0.582( = Formu a 1 .1268).

Table 1269. Compounds of formu a I .A, wherein R2 is R2-- 0.583( = Formu a 1 .1269).

Table 1270. Compounds of formu a I .A, wherein R2 is R2-- 0.584( = Formu a 1 .1270).

Table 1271. Compounds of formu a I .A, wherein R2 is R2-- 0.585( = Formu a 1 .1271).

Table 1272. Compounds of formu a I .A, wherein R2 is R2-- 0.586( = Formu a 1 .1272).

Table 1273. Compounds of formu a I .A, wherein R2 is R2-- 0.587( = Formu a 1 .1273).

Table 1274. Compounds of formu a I .A, wherein R2 is R2-- 0.588( = Formu a 1 .1274).

Table 1275. Compounds of formu a I .A, wherein R2 is R2-- 0.589( = Formu a 1 .1275).

Table 1276. Compounds of formu a I .A, wherein R2 is R2-- 0.590( = Formu a 1 .1276).

Table 1277. Compounds of formu a I .A, wherein R2 is R2-- 0.591 ( = Formu a 1 .1277).

Table 1278. Compounds of formu a I .A, wherein R2 is R2-- 0.592( = Formu a 1 .1278).

Table 1279. Compounds of formu a I .A, wherein R2 is R2-- 0.593( = Formu a 1 .1279).

Table 1280. Compounds of formu a I .A, wherein R2 is R2-- 0.594( = Formu a 1 .1280).

Table 1281. Compounds of formu a I .A, wherein R2 is R2-- 0.595( = Formu a 1 .1281).

Table 1282. Compounds of formu a I .A, wherein R2 is R2-- 0.596( = Formu a 1 .1282).

Table 1283. Compounds of formu a I .A, wherein R2 is R2-- 0.597( = Formu a 1 .1283).

Table 1284. Compounds of formu a I .A, wherein R2 is R2-- 0.598( = Formu a 1 .1284).

Table 1285. Compounds of formu a I .A, wherein R2 is R2-- 0.599( = Formu a 1 .1285).

Table 1286. Compounds of formu a I .A, wherein R2 is R2-- 0.600( = Formu a 1 .1286).

Table 1287. Compounds of formu a I .A, wherein R2 is R2-- 0.601 ( = Formu a 1 .1287).

Table 1288. Compounds of formu a I .A, wherein R2 is R2-- 0.602( = Formu a 1 .1288).

Table 1289. Compounds of formu a I .A, wherein R2 is R2-- 0.603( = Formu a 1 .1289).

Table 1290. Compounds of formu a I .A, wherein R2 is R2-- 0.604( = Formu a 1 .1290).

Table 1291. Compounds of formu a I .A, wherein R2 is R2-- 0.605( = Formu a 1 .1291).

Table 1292. Compounds of formu a I .A, wherein R2 is R2-- 0.606( = Formu a 1 .1292).

Table 1293. Compounds of formu a I .A, wherein R2 is R2-- 0.607( = Formu a 1 .1293).

Table 1294. Compounds of formu a I .A, wherein R2 is R2-- 0.608( = Formu a 1 .1294).

Table 1295. Compounds of formu a I .A, wherein R2 is R2-- 0.609( = Formu a 1 .1295).

Table 1296. Compounds of formu a I .A, wherein R2 is R2-- 0.610( = Formu a 1 .1296).

Table 1297. Compounds of formu a I .A, wherein R2 is R2-- 0.611( = Formu a 1 .1297).

Table 1298. Compounds of formu a I .A, wherein R2 is R2-- 0.612( = Formu a 1 .1298).

Table 1299. Compounds of formu a I .A, wherein R2 is R2-- 0.613( = Formu a 1 .1299).

Table 1300. Compounds of formu a I .A, wherein R2 is R2-- 0.614( = Formu a 1 .1300).

Table 1301. Compounds of formu a I .A, wherein R2 is R2-- 0.615( = Formu a 1 .1301).

Table 1302. Compounds of formu a I .A, wherein R2 is R2-- 0.616( = Formu a 1 .1302).

Table 1303. Compounds of formu a I .A, wherein R2 is R2-- 0.617( = Formu a 1 .1303).

Table 1304. Compounds of formu a I .A, wherein R2 is R2-- 0.618( = Formu a 1 .1304).

Table 1305. Compounds of formu a I .A, wherein R2 is R2-- 0.619( = Formu a 1 .1305).

Table 1306. Compounds of formu a I .A, wherein R2 is R2-- 0.620( = Formu a 1 .1306).

Table 1307. Compounds of formu a I .A, wherein R2 is R2-- 0.621 ( = Formu a 1 .1307).

Table 1308. Compounds of formu a I .A, wherein R2 is R2-- 0.622( = Formu a 1 .1308).

Table 1309. Compounds of formu a I .A, wherein R2 is R2-- 0.623( = Formu a 1 .1309). Table 1310. Compounds of formu a I .A, wherein R2 is R2-- 0.624( Formu a 1.1310)

Table 131 1. Compounds of formu a I .A, wherein R2 is R2-- 0.625( = Formu a 1 .131 1 )

Table 1312. Compounds of formu a I .A, wherein R2 is R2-- 0.626( = Formu a 1 .1312)

Table 1313. Compounds of formu a I .A, wherein R2 is R2-- 0.627( = Formu a 1 .1313)

Table 1314. Compounds of formu a I .A, wherein R2 is R2-- 0.628( = Formu a 1 .1314)

Table 1315. Compounds of formu a I .A, wherein R2 is R2-- 0.629( = Formu a 1 .1315)

Table 1316. Compounds of formu a I .A, wherein R2 is R2-- 0.630( = Formu a 1 .1316)

Table 1317. Compounds of formu a I .A, wherein R2 is R2-- 0.631 ( = Formu a 1 .1317)

Table 1318. Compounds of formu a I .A, wherein R2 is R2-- 0.632( = Formu a 1 .1318)

Table 1319. Compounds of formu a I .A, wherein R2 is R2-- 0.633( = Formu a 1 .1319)

Table 1320. Compounds of formu a I .A, wherein R2 is R2-- 0.634( = Formu a 1 .1320)

Table 1321. Compounds of formu a I .A, wherein R2 is R2-- 0.635( = Formu a 1 .1321 )

Table 1322. Compounds of formu a I .A, wherein R2 is R2-- 0.636( = Formu a 1 .1322)

Table 1323. Compounds of formu a I .A, wherein R2 is R2-- 0.637( = Formu a 1 .1323)

Table 1324. Compounds of formu a I .A, wherein R2 is R2-- 0.638( = Formu a 1 .1324)

Table 1325. Compounds of formu a I .A, wherein R2 is R2-- 0.639( = Formu a 1 .1325)

Table 1326. Compounds of formu a I .A, wherein R2 is R2-- 0.640( = Formu a 1 .1326)

Table 1327. Compounds of formu a I .A, wherein R2 is R2-- 0.641 ( = Formu a 1 .1327)

Table 1328. Compounds of formu a I .A, wherein R2 is R2-- 0.642( = Formu a 1 .1328)

Table 1329. Compounds of formu a I .A, wherein R2 is R2-- 0.643( = Formu a 1 .1329)

Table 1330. Compounds of formu a I .A, wherein R2 is R2-- 0.644( = Formu a 1 .1330)

Table 1331. Compounds of formu a I .A, wherein R2 is R2-- 0.645( = Formu a 1 .1331 )

Table 1332. Compounds of formu a I .A, wherein R2 is R2-- 0.646( = Formu a 1 .1332)

Table 1333. Compounds of formu a I .A, wherein R2 is R2-- 0.647( = Formu a 1 .1333)

Table 1334. Compounds of formu a I .A, wherein R2 is R2-- 0.648( = Formu a 1 .1334)

Table 1335. Compounds of formu a I .A, wherein R2 is R2-- 0.649( = Formu a 1 .1335)

Table 1336. Compounds of formu a I .A, wherein R2 is R2-- 0.650( = Formu a 1 .1336)

Table 1337. Compounds of formu a I .A, wherein R2 is R2-- 0.651 ( = Formu a 1 .1337)

Table 1338. Compounds of formu a I .A, wherein R2 is R2-- 0.652( = Formu a 1 .1338)

Table 1339. Compounds of formu a I .A, wherein R2 is R2-- 0.653( = Formu a 1 .1339)

Table 1340. Compounds of formu a I .A, wherein R2 is R2-- 0.654( = Formu a 1 .1340)

Table 1341. Compounds of formu a I .A, wherein R2 is R2-- 0.655( = Formu a 1 .1341 )

Table 1342. Compounds of formu a I .A, wherein R2 is R2-- 0.656( = Formu a 1 .1342)

Table 1343. Compounds of formu a I .A, wherein R2 is R2-- 0.657( = Formu a 1 .1343)

Table 1344. Compounds of formu a I .A, wherein R2 is R2-- 0.658( = Formu a 1 .1344)

Table 1345. Compounds of formu a I .A, wherein R2 is R2-- 0.659( = Formu a 1 .1345)

Table 1346. Compounds of formu a I .A, wherein R2 is R2-- 0.660( = Formu a 1 .1346)

Table 1347. Compounds of formu a I .A, wherein R2 is R2-- 0.661 ( = Formu a 1 .1347)

Table 1348. Compounds of formu a I .A, wherein R2 is R2-- 0.662( = Formu a 1 .1348)

Table 1349. Compounds of formu a I .A, wherein R2 is R2-- 0.663( = Formu a 1 .1349)

Table 1350. Compounds of formu a I .A, wherein R2 is R2-- 0.664( = Formu a 1 .1350)

Table 1351. Compounds of formu a I .A, wherein R2 is R2-- 0.665( = Formu a 1 .1351 )

Table 1352. Compounds of formu a I .A, wherein R2 is R2-- 0.666( = Formu a 1 .1352)

Table 1353. Compounds of formu a I .A, wherein R2 is R2-- 0.667( = Formu a 1 .1353) Table 1354. Compounds of formu a I .A, wherein R2 is R2 0.668(=formula 1.1354).

Table 1355. Compounds of formu a I .A, wherein R2 is R2 0.669(=formula 1.1355).

Table 1356. Compounds of formu a I .A, wherein R2 is R2 0.670(=formula 1.1356).

Table 1357. Compounds of formu a I .A, wherein R2 is R2 0.671 (=formula 1.1357).

Table 1358. Compounds of formu a I .A, wherein R2 is R2 0.672(=formula 1.1358).

Table 1359. Compounds of formu a I .A, wherein R2 is R2 0.673(=formula 1.1359).

Table 1360. Compounds of formu a I .A, wherein R2 is R2 0.674(=formula 1.1360).

Table 1361. Compounds of formu a I .A, wherein R2 is R2 0.675(=formula 1.1361).

Table 1362. Compounds of formu a I .A, wherein R2 is R2 0.676(=formula 1.1362).

Table 1363. Compounds of formu a I .A, wherein R2 is R2 5.1(=formula 1.1363).

Table 1364. Compounds of formu a I .A, wherein R2 is R2 5.2(=formula 1.1364).

Table 1365. Compounds of formu a I .A, wherein R2 is R2 5.3(=formula 1.1365).

Table 1366. Compounds of formu a I .A, wherein R2 is R2 5.4(=formula 1.1366).

Table 1367. Compounds of formu a I .A, wherein R2 is R2 5.5(=formula 1.1367).

Table 1368. Compounds of formu a I .A, wherein R2 is R2 5.6(=formula 1.1368).

Table 1369. Compounds of formu a I .A, wherein R2 is R2 5.7(=formula 1.1369).

Table 1370. Compounds of formu a I .A, wherein R2 is R2 5.8(=formula 1.1370).

Table 1371. Compounds of formu a I .A, wherein R2 is R2 5.9(=formula 1.1371).

Table 1372. Compounds of formu a I .A, wherein R2 is R2 5.10(=formula 1.1372).

Table 1373. Compounds of formu a I .A, wherein R2 is R2 5.11 (=formula 1.1373).

Table 1374. Compounds of formu a I .A, wherein R2 is R2 5.12(=formula 1.1374).

Table 1375. Compounds of formu a I .A, wherein R2 is R2 5.13(=formula 1.1375).

Table 1376. Compounds of formu a I .A, wherein R2 is R2 5.14(=formula 1.1376).

Table 1377. Compounds of formu a I .A, wherein R2 is R2 5.15(=formula 1.1377).

Table 1378. Compounds of formu a I .A, wherein R2 is R2 5.16(=formula 1.1378).

Table 1379. Compounds of formu a I .A, wherein R2 is R2 5.17(=formula 1.1379).

Table 1380. Compounds of formu a I .A, wherein R2 is R2 5.18(=formula 1.1380).

Table 1381. Compounds of formu a I .A, wherein R2 is R2 5.19(=formula 1.1381).

Table 1382. Compounds of formu a I .A, wherein R2 is R2 5.20(=formula 1.1382).

Table 1383. Compounds of formu a I .A, wherein R2 is R2 5.21 (=formula 1.1383).

Table 1384. Compounds of formu a I .A, wherein R2 is R2 5.22(=formula 1.1384).

Table 1385. Compounds of formu a I .A, wherein R2 is R2 5.23(=formula 1.1385).

Table 1386. Compounds of formu a I .A, wherein R2 is R2 5.24(=formula 1.1386).

Table 1387. Compounds of formu a I .A, wherein R2 is R2 5.25(=formula 1.1387).

Table 1388. Compounds of formu a I .A, wherein R2 is R2 5.26(=formula 1.1388).

Table 1389. Compounds of formu a I .A, wherein R2 is R2 5.27(=formula 1.1389).

Table 1390. Compounds of formu a I .A, wherein R2 is R2 5.28(=formula 1.1390).

Table 1391. Compounds of formu a I .A, wherein R2 is R2 5.29(=formula 1.1391).

Table 1392. Compounds of formu a I .A, wherein R2 is R2 5.30(=formula 1.1392).

Table 1393. Compounds of formu a I .A, wherein R2 is R2 5.31 (=formula 1.1393).

Table 1394. Compounds of formu a I .A, wherein R2 is R2 5.32(=formula 1.1394).

Table 1395. Compounds of formu a I .A, wherein R2 is R2 5.33(=formula 1.1395).

Table 1396. Compounds of formu a I .A, wherein R2 is R2 5.34(=formula 1.1396).

Table 1397. Compounds of formu a I .A, wherein R2 is R2 5.35(=formula 1.1397). Table 1398. Compounds of formu a I .A, wherein R2 is R2-- 5.36I Formu a 1 .1398).

Table 1399. Compounds of formu a I .A, wherein R2 is R2-- 5.37| = Formu a 1 .1399).

Table 1400. Compounds of formu a I .A, wherein R2 is R2-- 5.38I = Formu a 1 .1400).

Table 1401. Compounds of formu a I .A, wherein R2 is R2-- 5.39I = Formu a 1 .1401 ).

Table 1402. Compounds of formu a I .A, wherein R2 is R2-- 5.40I = Formu a 1 . 1402)

Table 1403. Compounds of formu a I .A, wherein R2 is R2-- 5.411 = Formu a 1 . 1403)

Table 1404. Compounds of formu a I .A, wherein R2 is R2-- 5.421 = Formu a 1 . 1404)

Table 1405. Compounds of formu a I .A, wherein R2 is R2-- 5.431 = Formu a 1 . 1405)

Table 1406. Compounds of formu a I .A, wherein R2 is R2-- 5.441 = Formu a 1 . 1406)

Table 1407. Compounds of formu a I .A, wherein R2 is R2-- 5.451 = Formu a 1 . 1407)

Table 1408. Compounds of formu a I .A, wherein R2 is R2-- 5.461 = Formu a 1 .1408).

Table 1409. Compounds of formu a I .A, wherein R2 is R2-- 5.471 = Formu a 1 .1409).

Table 1410. Compounds of formu a I .A, wherein R2 is R2-- 5.481 = Formu a 1 .1410).

Table 141 1. Compounds of formu a I .A, wherein R2 is R2-- 5.491 = Formu a 1 .141 1 ).

Table 1412. Compounds of formu a I .A, wherein R2 is R2-- 5.501 = Formu a 1 .1412).

Table 1413. Compounds of formu a I .A, wherein R2 is R2-- 5.511 = Formu a 1 .1413).

Table 1414. Compounds of formu a I .A, wherein R2 is R2-- 5.521 = Formu a 1 .1414).

Table 1415. Compounds of formu a I .A, wherein R2 is R2-- 5.531 = Formu a 1 .1415).

Table 1416. Compounds of formu a I .A, wherein R2 is R2-- 5.541 = Formu a 1 .1416).

Table 1417. Compounds of formu a I .A, wherein R2 is R2-- 5.551 = Formu a 1 .1417).

Table 1418. Compounds of formu a I .A, wherein R2 is R2-- 5.561 = Formu a 1 .1418).

Table 1419. Compounds of formu a I .A, wherein R2 is R2-- 5.571 = Formu a 1 .1419).

Table 1420. Compounds of formu a I .A, wherein R2 is R2-- 5.581 = Formu a 1 .1420).

Table 1421. Compounds of formu a I .A, wherein R2 is R2-- 5.591 = Formu a 1 .1421 ).

Table 1422. Compounds of formu a I .A, wherein R2 is R2-- 5.601 = Formu a 1 .1422).

Table 1423. Compounds of formu a I .A, wherein R2 is R2-- 5.611 = Formu a 1 .1423).

Table 1424. Compounds of formu a I .A, wherein R2 is R2-- 5.621 = Formu a 1 .1424).

Table 1425. Compounds of formu a I .A, wherein R2 is R2-- 5.631 = Formu a 1 .1425).

Table 1426. Compounds of formu a I .A, wherein R2 is R2-- 5.641 = Formu a 1 .1426).

Table 1427. Compounds of formu a I .A, wherein R2 is R2-- 5.651 = Formu a 1 .1427).

Table 1428. Compounds of formu a I .A, wherein R2 is R2-- 5.661 = Formu a 1 .1428).

Table 1429. Compounds of formu a I .A, wherein R2 is R2-- 5.671 = Formu a 1 .1429).

Table 1430. Compounds of formu a I .A, wherein R2 is R2-- 5.681 = Formu a 1 .1430).

Table 1431. Compounds of formu a I .A, wherein R2 is R2-- 5.691 = Formu a 1 .1431 ).

Table 1432. Compounds of formu a I .A, wherein R2 is R2-- 5.701 = Formu a 1 .1432).

Table 1433. Compounds of formu a I .A, wherein R2 is R2-- 5.711 = Formu a 1 .1433).

Table 1434. Compounds of formu a I .A, wherein R2 is R2-- 5.721 = Formu a 1 .1434).

Table 1435. Compounds of formu a I .A, wherein R2 is R2-- 5.731 = Formu a 1 .1435).

Table 1436. Compounds of formu a I .A, wherein R2 is R2-- 5.741 = Formu a 1 .1436).

Table 1437. Compounds of formu a I .A, wherein R2 is R2-- 5.751 = Formu a 1 .1437).

Table 1438. Compounds of formu a I .A, wherein R2 is R2-- 5.761 = Formu a 1 .1438).

Table 1439. Compounds of formu a I .A, wherein R2 is R2-- 5.771 = Formu a 1 .1439).

Table 1440. Compounds of formu a I .A, wherein R2 is R2-- 5.781 = Formu a 1 .1440).

Table 1441. Compounds of formu a I .A, wherein R2 is R2-- 5.791 = Formu a 1 .1441 ). Table 1442. Compounds of formu a I .A, wherein R2 is R2 5.80(=formula 1.1442).

Table 1443. Compounds of formu a I .A, wherein R2 is R2 5.81 (=formula 1. 1443).

Table 1444. Compounds of formu a I .A, wherein R2 is R2 5.82(=formula 1. 1444).

Table 1445. Compounds of formu a I .A, wherein R2 is R2 5.83(=formula 1. 1445).

Table 1446. Compounds of formu a I .A, wherein R2 is R2 5.84(=formula 1. 1446).

Table 1447. Compounds of formu a I .A, wherein R2 is R2 5.85(=formula 1. 1447).

Table 1448. Compounds of formu a I .A, wherein R2 is R2 5.86(=formula 1. 1448).

Table 1449. Compounds of formu a I .A, wherein R2 is R2 5.87(=formula 1. 1449).

Table 1450. Compounds of formu a I .A, wherein R2 is R2 5.88(=formula 1. 1450).

Table 1451. Compounds of formu a I .A, wherein R2 is R2 5.89(=formula 1. 1451).

Table 1452. Compounds of formu a I .A, wherein R2 is R2 5.90(=formula 1. 1452).

Table 1453. Compounds of formu a I .A, wherein R2 is R2 5.91 (=formula 1. 1453).

Table 1454. Compounds of formu a I .A, wherein R2 is R2 5.92(=formula 1. 1454).

Table 1455. Compounds of formu a I .A, wherein R2 is R2 5.93(=formula 1. 1455).

Table 1456. Compounds of formu a I .A, wherein R2 is R2 5.94(=formula 1. 1456).

Table 1457. Compounds of formu a I .A, wherein R2 is R2 5.95(=formula 1. 1457).

Table 1458. Compounds of formu a I .A, wherein R2 is R2 5.96(=formula 1. 1458).

Table 1459. Compounds of formu a I .A, wherein R2 is R2 5.97(=formula 1. 1459).

Table 1460. Compounds of formu a I .A, wherein R2 is R2 5.98(=formula 1. 1460).

Table 1461. Compounds of formu a I .A, wherein R2 is R2 5.99(=formula 1. 1461).

Table 1462. Compounds of formu a I .A, wherein R2 is R2 5.100(=formula ' 1.1462).

Table 1463. Compounds of formu a I .A, wherein R2 is R2 5.101(=formula ' 1.1463).

Table 1464. Compounds of formu a I .A, wherein R2 is R2 5.102(=formula ' 1.1464).

Table 1465. Compounds of formu a I .A, wherein R2 is R2 5.103(=formula ' 1.1465).

Table 1466. Compounds of formu a I .A, wherein R2 is R2 5.104(=formula ' 1.1466).

Table 1467. Compounds of formu a I .A, wherein R2 is R2 5.105(=formula ' 1.1467).

Table 1468. Compounds of formu a I .A, wherein R2 is R2 5.106(=formula ' 1.1468).

Table 1469. Compounds of formu a I .A, wherein R2 is R2 5.107(=formula ' 1.1469).

Table 1470. Compounds of formu a I .A, wherein R2 is R2 5.108(=formula ' 1.1470).

Table 1471. Compounds of formu a I .A, wherein R2 is R2 5.109(=formula ' 1.1471).

Table 1472. Compounds of formu a I .A, wherein R2 is R2 5.110(=formula ' 1.1472).

Table 1473. Compounds of formu a I .A, wherein R2 is R2 5.111(=formula ' 1.1473).

Table 1474. Compounds of formu a I .A, wherein R2 is R2 5.112(=formula ' 1.1475).

Table 1475. Compounds of formu a I .A, wherein R2 is R2 5.113(=formula ' 1.1475).

Table 1476. Compounds of formu a I .A, wherein R2 is R2 5.114(=formula ' 1.1476).

Table 1477. Compounds of formu a I .A, wherein R2 is R2 5.115(=formula ' 1.1477).

Table 1478. Compounds of formu a I .A, wherein R2 is R2 5.116(=formula ' 1.1478).

Table 1479. Compounds of formu a I .A, wherein R2 is R2 5.117(=formula ' 1.1479).

Table 1480. Compounds of formu a I .A, wherein R2 is R2 5.118(=formula ' 1.1480).

Table 1481. Compounds of formu a I .A, wherein R2 is R2 5.119(=formula ' 1.1481).

Table 1482. Compounds of formu a I .A, wherein R2 is R2 5.120(=formula ' 1.1482).

Table 1483. Compounds of formu a I .A, wherein R2 is R2 5.121 (=formula ' 1.1483).

Table 1484. Compounds of formu a I .A, wherein R2 is R2 5.122(=formula ' 1.1484).

Table 1485. Compounds of formu a I .A, wherein R2 is R2 5.123(=formula ' 1.1485). Table 1486. Compounds of formu a I .A, wherein R2 is R2-- 5.124( Formu a 1.1486)

Table 1487. Compounds of formu a I .A, wherein R2 is R2-- 5.125( = Formu a 1 .1487)

Table 1488. Compounds of formu a I .A, wherein R2 is R2-- 5.126( = Formu a 1 .1488)

Table 1489. Compounds of formu a I .A, wherein R2 is R2-- 5.127( = Formu a 1 .1489)

Table 1490. Compounds of formu a I .A, wherein R2 is R2-- 5.128( = Formu a 1 .1490)

Table 1491. Compounds of formu a I .A, wherein R2 is R2-- 5.129( = Formu a 1 .1491 )

Table 1492. Compounds of formu a I .A, wherein R2 is R2-- 5.130( = Formu a 1 .1492)

Table 1493. Compounds of formu a I .A, wherein R2 is R2-- 5.131 ( = Formu a 1 .1493)

Table 1494. Compounds of formu a I .A, wherein R2 is R2-- 5.132( = Formu a 1 .1494)

Table 1495. Compounds of formu a I .A, wherein R2 is R2-- 5.133( = Formu a 1 .1495)

Table 1496. Compounds of formu a I .A, wherein R2 is R2-- 5.134( = Formu a 1 .1496)

Table 1497. Compounds of formu a I .A, wherein R2 is R2-- 5.135( = Formu a 1 .1497)

Table 1498. Compounds of formu a I .A, wherein R2 is R2-- 5.136( = Formu a 1 .1498)

Table 1499. Compounds of formu a I .A, wherein R2 is R2-- 5.137( = Formu a 1 .1499)

Table 1500. Compounds of formu a I .A, wherein R2 is R2-- 5.138( = Formu a 1 .1500)

Table 1501. Compounds of formu a I .A, wherein R2 is R2-- 5.139( = Formu a 1 .1501 )

Table 1502. Compounds of formu a I .A, wherein R2 is R2-- 5.140( = Formu a 1 .1502)

Table 1503. Compounds of formu a I .A, wherein R2 is R2-- 5.141 ( = Formu a 1 .1503)

Table 1504. Compounds of formu a I .A, wherein R2 is R2-- 5.142( = Formu a 1 .1504)

Table 1505. Compounds of formu a I .A, wherein R2 is R2-- 5.143( = Formu a 1 .1505)

Table 1506. Compounds of formu a I .A, wherein R2 is R2-- 5.144( = Formu a 1 .1506)

Table 1507. Compounds of formu a I .A, wherein R2 is R2-- 5.145( = Formu a 1 .1507)

Table 1508. Compounds of formu a I .A, wherein R2 is R2-- 5.146( = Formu a 1 .1508)

Table 1509. Compounds of formu a I .A, wherein R2 is R2-- 5.147( = Formu a 1 .1509)

Table 1510. Compounds of formu a I .A, wherein R2 is R2-- 5.148( = Formu a 1 .1510)

Table 151 1. Compounds of formu a I .A, wherein R2 is R2-- 5.149( = Formu a 1 .151 1 )

Table 1512. Compounds of formu a I .A, wherein R2 is R2-- 5.150( = Formu a 1 .1512)

Table 1513. Compounds of formu a I .A, wherein R2 is R2-- 5.151 ( = Formu a 1 .1513)

Table 1514. Compounds of formu a I .A, wherein R2 is R2-- 5.152( = Formu a 1 .1514)

Table 1515. Compounds of formu a I .A, wherein R2 is R2-- 5.153( = Formu a 1 .1515)

Table 1516. Compounds of formu a I .A, wherein R2 is R2-- 5.154( = Formu a 1 .1516)

Table 1517. Compounds of formu a I .A, wherein R2 is R2-- 5.155( = Formu a 1 .1517)

Table 1518. Compounds of formu a I .A, wherein R2 is R2-- 5.156( = Formu a 1 .1518)

Table 1519. Compounds of formu a I .A, wherein R2 is R2-- 5.157( = Formu a 1 .1519)

Table 1520. Compounds of formu a I .A, wherein R2 is R2-- 5.158( = Formu a 1 .1520)

Table 1521. Compounds of formu a I .A, wherein R2 is R2-- 5.159( = Formu a 1 .1521 )

Table 1522. Compounds of formu a I .A, wherein R2 is R2-- 5.160( = Formu a 1 .1522)

Table 1523. Compounds of formu a I .A, wherein R2 is R2-- 5.161 ( = Formu a 1 .1523)

Table 1524. Compounds of formu a I .A, wherein R2 is R2-- 5.162( = Formu a 1 .1524)

Table 1525. Compounds of formu a I .A, wherein R2 is R2-- 5.163( = Formu a 1 .1525)

Table 1526. Compounds of formu a I .A, wherein R2 is R2-- 5.164( = Formu a 1 .1526)

Table 1527. Compounds of formu a I .A, wherein R2 is R2-- 5.165( = Formu a 1 .1527)

Table 1528. Compounds of formu a I .A, wherein R2 is R2-- 5.166( = Formu a 1 .1528)

Table 1529. Compounds of formu a I .A, wherein R2 is R2-- 5.167( = Formu a 1 .1529) Table 1530. Compounds of formu a I .A, wherein R2 is R2-- 5.168( = Formu a 1.1530).

Table 1531. Compounds of formu a I .A, wherein R2 is R2-- 5.169( = Formu a 1 .1531 ).

Table 1532. Compounds of formu a I .A, wherein R2 is R2-- 5.170( = Formu a 1 .1532).

Table 1533. Compounds of formu a I .A, wherein R2 is R2-- 5.171 ( = Formu a 1 .1533).

Table 1534. Compounds of formu a I .A, wherein R2 is R2-- 5.172( = Formu a 1 .1534).

Table 1535. Compounds of formu a I .A, wherein R2 is R2-- 5.173( = Formu a 1 .1535).

Table 1536. Compounds of formu a I .A, wherein R2 is R2-- 5.174( = Formu a 1 .1536).

Table 1537. Compounds of formu a I .A, wherein R2 is R2-- 5.175( = Formu a 1 .1537).

Table 1538. Compounds of formu a I .A, wherein R2 is R2-- 5.176( = Formu a 1 .1538).

Table 1539. Compounds of formu a I .A, wherein R2 is R2-- 5.177( = Formu a 1 .1539).

Table 1540. Compounds of formu a I .A, wherein R2 is R2-- 5.178( = Formu a 1 .1540).

Table 1541. Compounds of formu a I .A, wherein R2 is R2-- 5.179( = Formu a 1 .1541 ).

Table 1542. Compounds of formu a I .A, wherein R2 is R2-- 5.180( = Formu a 1 .1542).

Table 1543. Compounds of formu a I .A, wherein R2 is R2-- 5.181 ( = Formu a 1 .1543).

Table 1544. Compounds of formu a I .A, wherein R2 is R2-- 5.182( = Formu a 1 .1544).

Table 1545. Compounds of formu a I .A, wherein R2 is R2-- 5.183( = Formu a 1 .1545).

Table 1546. Compounds of formu a I .A, wherein R2 is R2-- 5.184( = Formu a 1 .1546).

Table 1547. Compounds of formu a I .A, wherein R2 is R2-- 5.185( = Formu a 1 .1547).

Table 1548. Compounds of formu a I .A, wherein R2 is R2-- 5.186( = Formu a 1 .1548).

Table 1549. Compounds of formu a I .A, wherein R2 is R2-- 5.187( = Formu a 1 .1549).

Table 1550. Compounds of formu a I .A, wherein R2 is R2-- 5.188( = Formu a 1 .1550).

Table 1551. Compounds of formu a I .A, wherein R2 is R2-- 5.189( = Formu a 1 .1551 ).

Table 1552. Compounds of formu a I .A, wherein R2 is R2-- 5.190( = Formu a 1 .1552).

Table 1553. Compounds of formu a I .A, wherein R2 is R2-- 5.191 ( = Formu a 1 .1553).

Table 1554. Compounds of formu a I .A, wherein R2 is R2-- 5.192( = Formu a 1 .1554).

Table 1555. Compounds of formu a I .A, wherein R2 is R2-- 5.193( = Formu a 1 .1555).

Table 1556. Compounds of formu a I .A, wherein R2 is R2-- 5.194( = Formu a 1 .1556).

Table 1557. Compounds of formu a I .A, wherein R2 is R2-- 5.195( = Formu a 1 .1557).

Table 1558. Compounds of formu a I .A, wherein R2 is R2-- 5.196( = Formu a 1 .1558).

Table 1559. Compounds of formu a I .A, wherein R2 is R2-- 5.197( = Formu a 1 .1559).

Table 1560. Compounds of formu a I .A, wherein R2 is R2-- 5.198( = Formu a 1 .1560).

Table 1561. Compounds of formu a I .A, wherein R2 is R2-- 5.199( = Formu a 1 .1561 ).

Table 1562. Compounds of formu a I .A, wherein R2 is R2-- 5.200( = Formu a 1 .1562).

Table 1563. Compounds of formu a I .A, wherein R2 is R2-- 5.201 ( = Formu a 1 .1563).

Table 1564. Compounds of formu a I .A, wherein R2 is R2-- 5.202( = Formu a 1 .1564).

Table 1565. Compounds of formu a I .A, wherein R2 is R2-- 5.203( = Formu a 1 .1565).

Table 1566. Compounds of formu a I .A, wherein R2 is R2-- 5.204( = Formu a 1 .1566).

Table 1567. Compounds of formu a I .A, wherein R2 is R2-- 5.205( = Formu a 1 .1567).

Table 1568. Compounds of formu a I .A, wherein R2 is R2-- 5.206( = Formu a 1 .1568).

Table 1569. Compounds of formu a I .A, wherein R2 is R2-- 5.207( = Formu a 1 .1569).

Table 1570. Compounds of formu a I .A, wherein R2 is R2-- 5.208( = Formu a 1 .1570).

Table 1571. Compounds of formu a I .A, wherein R2 is R2-- 5.209( = Formu a 1 .1571 ).

Table 1572. Compounds of formu a I .A, wherein R2 is R2-- 5.210( = Formu a 1 .1572).

Table 1573. Compounds of formu a I .A, wherein R2 is R2-- 5.21 1 ( = Formu a 1 .1573). Table 1574. Compounds of formu a I .A, wherein R2 is R2-- 5.212( Formu a 1.1574)

Table 1575. Compounds of formu a I .A, wherein R2 is R2-- 5.213( = Formu a 1 .1575)

Table 1576. Compounds of formu a I .A, wherein R2 is R2-- 5.214( = Formu a 1 .1576)

Table 1577. Compounds of formu a I .A, wherein R2 is R2-- 5.215( = Formu a 1 .1577)

Table 1578. Compounds of formu a I .A, wherein R2 is R2-- 5.216( = Formu a 1 .1578)

Table 1579. Compounds of formu a I .A, wherein R2 is R2-- 5.217( = Formu a 1 .1579)

Table 1580. Compounds of formu a I .A, wherein R2 is R2-- 5.218( = Formu a 1 .1580)

Table 1581. Compounds of formu a I .A, wherein R2 is R2-- 5.219( = Formu a 1 .1581 )

Table 1582. Compounds of formu a I .A, wherein R2 is R2-- 5.220( = Formu a 1 .1582)

Table 1583. Compounds of formu a I .A, wherein R2 is R2-- 5.221 ( = Formu a 1 .1583)

Table 1584. Compounds of formu a I .A, wherein R2 is R2-- 5.222( = Formu a 1 .1584)

Table 1585. Compounds of formu a I .A, wherein R2 is R2-- 5.223( = Formu a 1 .1585)

Table 1586. Compounds of formu a I .A, wherein R2 is R2-- 5.224( = Formu a 1 .1586)

Table 1587. Compounds of formu a I .A, wherein R2 is R2-- 5.225( = Formu a 1 .1587)

Table 1588. Compounds of formu a I .A, wherein R2 is R2-- 5.226( = Formu a 1 .1588)

Table 1589. Compounds of formu a I .A, wherein R2 is R2-- 5.227( = Formu a 1 .1589)

Table 1590. Compounds of formu a I .A, wherein R2 is R2-- 5.228( = Formu a 1 .1590)

Table 1591. Compounds of formu a I .A, wherein R2 is R2-- 5.229( = Formu a 1 .1591 )

Table 1592. Compounds of formu a I .A, wherein R2 is R2-- 5.230( = Formu a 1 .1592)

Table 1593. Compounds of formu a I .A, wherein R2 is R2-- 5.231 ( = Formu a 1 .1593)

Table 1594. Compounds of formu a I .A, wherein R2 is R2-- 5.232( = Formu a 1 .1594)

Table 1595. Compounds of formu a I .A, wherein R2 is R2-- 5.233( = Formu a 1 .1595)

Table 1596. Compounds of formu a I .A, wherein R2 is R2-- 5.234( = Formu a 1 .1596)

Table 1597. Compounds of formu a I .A, wherein R2 is R2-- 5.235( = Formu a 1 .1597)

Table 1598. Compounds of formu a I .A, wherein R2 is R2-- 5.236( = Formu a 1 .1598)

Table 1599. Compounds of formu a I .A, wherein R2 is R2-- 5.237( = Formu a 1 .1599)

Table 1600. Compounds of formu a I .A, wherein R2 is R2-- 5.238( = Formu a 1 .1600)

Table 1601. Compounds of formu a I .A, wherein R2 is R2-- 5.239( = Formu a 1 .1601 )

Table 1602. Compounds of formu a I .A, wherein R2 is R2-- 5.240( = Formu a 1 .1602)

Table 1603. Compounds of formu a I .A, wherein R2 is R2-- 5.241 ( = Formu a 1 .1603)

Table 1604. Compounds of formu a I .A, wherein R2 is R2-- 5.242( = Formu a 1 .1604)

Table 1605. Compounds of formu a I .A, wherein R2 is R2-- 5.243( = Formu a 1 .1605)

Table 1606. Compounds of formu a I .A, wherein R2 is R2-- 5.244( = Formu a 1 .1606)

Table 1607. Compounds of formu a I .A, wherein R2 is R2-- 5.245( = Formu a 1 .1607)

Table 1608. Compounds of formu a I .A, wherein R2 is R2-- 5.246( = Formu a 1 .1608)

Table 1609. Compounds of formu a I .A, wherein R2 is R2-- 5.247( = Formu a 1 .1609)

Table 1610. Compounds of formu a I .A, wherein R2 is R2-- 5.248( = Formu a 1 .1610)

Table 161 1. Compounds of formu a I .A, wherein R2 is R2-- 5.249( = Formu a 1 .161 1 )

Table 1612. Compounds of formu a I .A, wherein R2 is R2-- 5.250( = Formu a 1 .1612)

Table 1613. Compounds of formu a I .A, wherein R2 is R2-- 5.251 ( = Formu a 1 .1613)

Table 1614. Compounds of formu a I .A, wherein R2 is R2-- 5.252( = Formu a 1 .1614)

Table 1615. Compounds of formu a I .A, wherein R2 is R2-- 5.253( = Formu a 1 .1615)

Table 1616. Compounds of formu a I .A, wherein R2 is R2-- 5.254( = Formu a 1 .1616)

Table 1617. Compounds of formu a I .A, wherein R2 is R2-- 5.255( = Formu a 1 .1617) Table 1618. Compounds of formu a I .A, wherein R2 is R2-- 5.256( = Formu a 1.1618).

Table 1619. Compounds of formu a I .A, wherein R2 is R2-- 5.257( = Formu a 1 .1619).

Table 1620. Compounds of formu a I .A, wherein R2 is R2-- 5.258( = Formu a 1 .1620).

Table 1621. Compounds of formu a I .A, wherein R2 is R2-- 5.259( = Formu a 1 .1621 ).

Table 1622. Compounds of formu a I .A, wherein R2 is R2-- 5.260( = Formu a 1 .1622).

Table 1623. Compounds of formu a I .A, wherein R2 is R2-- 5.261 ( = Formu a 1 .1623).

Table 1624. Compounds of formu a I .A, wherein R2 is R2-- 5.262( = Formu a 1 .1624).

Table 1625. Compounds of formu a I .A, wherein R2 is R2-- 5.263( = Formu a 1 .1625).

Table 1626. Compounds of formu a I .A, wherein R2 is R2-- 5.264( = Formu a 1 .1626).

Table 1627. Compounds of formu a I .A, wherein R2 is R2-- 5.265( = Formu a 1 .1627).

Table 1628. Compounds of formu a I .A, wherein R2 is R2-- 5.266( = Formu a 1 .1628).

Table 1629. Compounds of formu a I .A, wherein R2 is R2-- 5.267( = Formu a 1 .1629).

Table 1630. Compounds of formu a I .A, wherein R2 is R2-- 5.268( = Formu a 1 .1630).

Table 1631. Compounds of formu a I .A, wherein R2 is R2-- 5.269( = Formu a 1 .1631 ).

Table 1632. Compounds of formu a I .A, wherein R2 is R2-- 5.270( = Formu a 1 .1632).

Table 1633. Compounds of formu a I .A, wherein R2 is R2-- 5.271 ( = Formu a 1 .1633).

Table 1634. Compounds of formu a I .A, wherein R2 is R2-- 5.272( = Formu a 1 .1634).

Table 1635. Compounds of formu a I .A, wherein R2 is R2-- 5.273( = Formu a 1 .1635).

Table 1636. Compounds of formu a I .A, wherein R2 is R2-- 5.274( = Formu a 1 .1636).

Table 1637. Compounds of formu a I .A, wherein R2 is R2-- 5.275( = Formu a 1 .1637).

Table 1638. Compounds of formu a I .A, wherein R2 is R2-- 5.276( = Formu a 1 .1638).

Table 1639. Compounds of formu a I .A, wherein R2 is R2-- 5.277( = Formu a 1 .1639).

Table 1640. Compounds of formu a I .A, wherein R2 is R2-- 5.278( = Formu a 1 .1640).

Table 1641. Compounds of formu a I .A, wherein R2 is R2-- 5.279( = Formu a 1 .1641 ).

Table 1642. Compounds of formu a I .A, wherein R2 is R2-- 5.280( = Formu a 1 .1642).

Table 1643. Compounds of formu a I .A, wherein R2 is R2-- 5.281 ( = Formu a 1 .1643).

Table 1644. Compounds of formu a I .A, wherein R2 is R2-- 5.282( = Formu a 1 .1644).

Table 1645. Compounds of formu a I .A, wherein R2 is R2-- 5.283( = Formu a 1 .1645).

Table 1646. Compounds of formu a I .A, wherein R2 is R2-- 5.284( = Formu a 1 .1646).

Table 1647. Compounds of formu a I .A, wherein R2 is R2-- 5.285( = Formu a 1 .1647).

Table 1648. Compounds of formu a I .A, wherein R2 is R2-- 5.286( = Formu a 1 .1648).

Table 1649. Compounds of formu a I .A, wherein R2 is R2-- 5.287( = Formu a 1 .1649).

Table 1650. Compounds of formu a I .A, wherein R2 is R2-- 5.288( = Formu a 1 .1650).

Table 1651. Compounds of formu a I .A, wherein R2 is R2-- 5.289( = Formu a 1 .1651 ).

Table 1652. Compounds of formu a I .A, wherein R2 is R2-- 5.290( = Formu a 1 .1652).

Table 1653. Compounds of formu a I .A, wherein R2 is R2-- 5.291 ( = Formu a 1 .1653).

Table 1654. Compounds of formu a I .A, wherein R2 is R2-- 5.292( = Formu a 1 .1654).

Table 1655. Compounds of formu a I .A, wherein R2 is R2-- 5.293( = Formu a 1 .1655).

Table 1656. Compounds of formu a I .A, wherein R2 is R2-- 5.294( = Formu a 1 .1656).

Table 1657. Compounds of formu a I .A, wherein R2 is R2-- 5.295( = Formu a 1 .1657).

Table 1658. Compounds of formu a I .A, wherein R2 is R2-- 5.296( = Formu a 1 .1658).

Table 1659. Compounds of formu a I .A, wherein R2 is R2-- 5.297( = Formu a 1 .1659).

Table 1660. Compounds of formu a I .A, wherein R2 is R2-- 5.298( = Formu a 1 .1660).

Table 1661. Compounds of formu a I .A, wherein R2 is R2-- 5.299( = Formu a 1 .1661 ). Table 1662. Compounds of formu a I .A, wherein R2 is R2-- 5.300( = Formu a 1.1662).

Table 1663. Compounds of formu a I .A, wherein R2 is R2-- 5.301 ( = Formu a 1 .1663).

Table 1664. Compounds of formu a I .A, wherein R2 is R2-- 5.302( = Formu a 1 .1664).

Table 1665. Compounds of formu a I .A, wherein R2 is R2-- 5.303( = Formu a 1 .1665).

Table 1666. Compounds of formu a I .A, wherein R2 is R2-- 5.304( = Formu a 1 .1666).

Table 1667. Compounds of formu a I .A, wherein R2 is R2-- 5.305( = Formu a 1 .1667).

Table 1668. Compounds of formu a I .A, wherein R2 is R2-- 5.306( = Formu a 1 .1668).

Table 1669. Compounds of formu a I .A, wherein R2 is R2-- 5.307( = Formu a 1 .1669).

Table 1670. Compounds of formu a I .A, wherein R2 is R2-- 5.308( = Formu a 1 .1670).

Table 1671. Compounds of formu a I .A, wherein R2 is R2-- 5.309( = Formu a 1 .1671 ).

Table 1672. Compounds of formu a I .A, wherein R2 is R2-- 5.310( = Formu a 1 .1672).

Table 1673. Compounds of formu a I .A, wherein R2 is R2-- 5.31 1 ( = Formu a 1 .1673).

Table 1674. Compounds of formu a I .A, wherein R2 is R2-- 5.312( = Formu a 1 .1674).

Table 1675. Compounds of formu a I .A, wherein R2 is R2-- 5.313( = Formu a 1 .1675).

Table 1676. Compounds of formu a I .A, wherein R2 is R2-- 5.314( = Formu a 1 .1676).

Table 1677. Compounds of formu a I .A, wherein R2 is R2-- 5.315( = Formu a 1 .1676).

Table 1678. Compounds of formu a I .A, wherein R2 is R2-- 5.316( = Formu a 1 .1678).

Table 1679. Compounds of formu a I .A, wherein R2 is R2-- 5.317( = Formu a 1 .1679).

Table 1680. Compounds of formu a I .A, wherein R2 is R2-- 5.318( = Formu a 1 .1680).

Table 1681. Compounds of formu a I .A, wherein R2 is R2-- 5.319( = Formu a 1 .1681 ).

Table 1682. Compounds of formu a I .A, wherein R2 is R2-- 5.320( = Formu a 1 .1682).

Table 1683. Compounds of formu a I .A, wherein R2 is R2-- 5.321 ( = Formu a 1 .1683).

Table 1684. Compounds of formu a I .A, wherein R2 is R2-- 5.322( = Formu a 1 .1684).

Table 1685. Compounds of formu a I .A, wherein R2 is R2-- 5.323( = Formu a 1 .1685).

Table 1686. Compounds of formu a I .A, wherein R2 is R2-- 5.324( = Formu a 1 .1686).

Table 1687. Compounds of formu a I .A, wherein R2 is R2-- 5.325( = Formu a 1 .1687).

Table 1688. Compounds of formu a I .A, wherein R2 is R2-- 5.326( = Formu a 1 .1688).

Table 1689. Compounds of formu a I .A, wherein R2 is R2-- 5.327( = Formu a 1 .1689).

Table 1690. Compounds of formu a I .A, wherein R2 is R2-- 5.328( = Formu a 1 .1690).

Table 1691. Compounds of formu a I .A, wherein R2 is R2-- 5.329( = Formu a 1 .1691 ).

Table 1692. Compounds of formu a I .A, wherein R2 is R2-- 5.330( = Formu a 1 .1692).

Table 1693. Compounds of formu a I .A, wherein R2 is R2-- 5.331 ( = Formu a 1 .1693).

Table 1694. Compounds of formu a I .A, wherein R2 is R2-- 5.332( = Formu a 1 .1694).

Table 1695. Compounds of formu a I .A, wherein R2 is R2-- 5.333( = Formu a 1 .1695).

Table 1696. Compounds of formu a I .A, wherein R2 is R2-- 5.334( = Formu a 1 .1696).

Table 1697. Compounds of formu a I .A, wherein R2 is R2-- 5.335( = Formu a 1 .1697).

Table 1698. Compounds of formu a I .A, wherein R2 is R2-- 5.336( = Formu a 1 .1698).

Table 1699. Compounds of formu a I .A, wherein R2 is R2-- 5.334( = Formu a 1 .1699).

Table 1700. Compounds of formu a I .A, wherein R2 is R2-- 5.338( = Formu a 1 .1700).

Table 1701. Compounds of formu a I .A, wherein R2 is R2-- 5.339( = Formu a 1 .1701 ).

Table 1702. Compounds of formu a I .A, wherein R2 is R2-- 5.340( = Formu a 1 .1702).

Table 1703. Compounds of formu a I .A, wherein R2 is R2-- 5.341 ( = Formu a 1 .1703).

Table 1704. Compounds of formu a I .A, wherein R2 is R2-- 5.342( = Formu a 1 .1704).

Table 1705. Compounds of formu a I .A, wherein R2 is R2-- 5.343( = Formu a 1 .1705). Table 1706. Compounds of formu a I .A, wherein R2 is R2-- 5.344( Formu a 1.1706)

Table 1707. Compounds of formu a I .A, wherein R2 is R2-- 5.345( = Formu a 1 .1707)

Table 1708. Compounds of formu a I .A, wherein R2 is R2-- 5.346( = Formu a 1 .1708)

Table 1709. Compounds of formu a I .A, wherein R2 is R2-- 5.347( = Formu a 1 .1709)

Table 1710. Compounds of formu a I .A, wherein R2 is R2-- 5.348( = Formu a 1 .1710)

Table 171 1. Compounds of formu a I .A, wherein R2 is R2-- 5.349( = Formu a 1 .171 1 )

Table 1712. Compounds of formu a I .A, wherein R2 is R2-- 5.350( = Formu a 1 .1712)

Table 1713. Compounds of formu a I .A, wherein R2 is R2-- 5.351 ( = Formu a 1 .1713)

Table 1714. Compounds of formu a I .A, wherein R2 is R2-- 5.352( = Formu a 1 .1714)

Table 1715. Compounds of formu a I .A, wherein R2 is R2-- 5.353( = Formu a 1 .1715)

Table 1716. Compounds of formu a I .A, wherein R2 is R2-- 5.354( = Formu a 1 .1716)

Table 1717. Compounds of formu a I .A, wherein R2 is R2-- 5.355( = Formu a 1 .1717)

Table 1718. Compounds of formu a I .A, wherein R2 is R2-- 5.356( = Formu a 1 .1718)

Table 1719. Compounds of formu a I .A, wherein R2 is R2-- 5.357( = Formu a 1 .1719)

Table 1720. Compounds of formu a I .A, wherein R2 is R2-- 5.358( = Formu a 1 .1720)

Table 1721. Compounds of formu a I .A, wherein R2 is R2-- 5.359( = Formu a 1 .1721 )

Table 1722. Compounds of formu a I .A, wherein R2 is R2-- 5.360( = Formu a 1 .1722)

Table 1723. Compounds of formu a I .A, wherein R2 is R2-- 5.361 ( = Formu a 1 .1723)

Table 1724. Compounds of formu a I .A, wherein R2 is R2-- 5.362( = Formu a 1 .1724)

Table 1725. Compounds of formu a I .A, wherein R2 is R2-- 5.363( = Formu a 1 .1725)

Table 1726. Compounds of formu a I .A, wherein R2 is R2-- 5.364( = Formu a 1 .1726)

Table 1727. Compounds of formu a I .A, wherein R2 is R2-- 5.365( = Formu a 1 .1727)

Table 1728. Compounds of formu a I .A, wherein R2 is R2-- 5.366( = Formu a 1 .1728)

Table 1729. Compounds of formu a I .A, wherein R2 is R2-- 5.367( = Formu a 1 .1729)

Table 1730. Compounds of formu a I .A, wherein R2 is R2-- 5.368( = Formu a 1 .1730)

Table 1731. Compounds of formu a I .A, wherein R2 is R2-- 5.369( = Formu a 1 .1731 )

Table 1732. Compounds of formu a I .A, wherein R2 is R2-- 5.370( = Formu a 1 .1732)

Table 1733. Compounds of formu a I .A, wherein R2 is R2-- 5.371 ( = Formu a 1 .1733)

Table 1734. Compounds of formu a I .A, wherein R2 is R2-- 5.372( = Formu a 1 .1734)

Table 1735. Compounds of formu a I .A, wherein R2 is R2-- 5.373( = Formu a 1 .1735)

Table 1736. Compounds of formu a I .A, wherein R2 is R2-- 5.374( = Formu a 1 .1736)

Table 1737. Compounds of formu a I .A, wherein R2 is R2-- 5.375( = Formu a 1 .1737)

Table 1738. Compounds of formu a I .A, wherein R2 is R2-- 5.376( = Formu a 1 .1738)

Table 1739. Compounds of formu a I .A, wherein R2 is R2-- 5.377( = Formu a 1 .1739)

Table 1740. Compounds of formu a I .A, wherein R2 is R2-- 5.378( = Formu a 1 .1740)

Table 1741. Compounds of formu a I .A, wherein R2 is R2-- 5.379( = Formu a 1 .1741 )

Table 1742. Compounds of formu a I .A, wherein R2 is R2-- 5.380( = Formu a 1 .1742)

Table 1743. Compounds of formu a I .A, wherein R2 is R2-- 5.381 ( = Formu a 1 .1743)

Table 1744. Compounds of formu a I .A, wherein R2 is R2-- 5.382( = Formu a 1 .1744)

Table 1745. Compounds of formu a I .A, wherein R2 is R2-- 5.383( = Formu a 1 .1745)

Table 1746. Compounds of formu a I .A, wherein R2 is R2-- 5.384( = Formu a 1 .1746)

Table 1747. Compounds of formu a I .A, wherein R2 is R2-- 5.385( = Formu a 1 .1747)

Table 1748. Compounds of formu a I .A, wherein R2 is R2-- 5.386( = Formu a 1 .1748)

Table 1749. Compounds of formu a I .A, wherein R2 is R2-- 5.387( = Formu a 1 .1749) Table 1750. Compounds of formu a I .A, wherein R2 is R2-- 5.388( = Formu a 1.1750).

Table 1751. Compounds of formu a I .A, wherein R2 is R2-- 5.389( = Formu a 1 .1751 ).

Table 1752. Compounds of formu a I .A, wherein R2 is R2-- 5.390( = Formu a 1 .1752).

Table 1753. Compounds of formu a I .A, wherein R2 is R2-- 5.391 ( = Formu a 1 .1753).

Table 1754. Compounds of formu a I .A, wherein R2 is R2-- 5.392( = Formu a 1 .1754).

Table 1755. Compounds of formu a I .A, wherein R2 is R2-- 5.393( = Formu a 1 .1755).

Table 1756. Compounds of formu a I .A, wherein R2 is R2-- 5.394( = Formu a 1 .1756).

Table 1757. Compounds of formu a I .A, wherein R2 is R2-- 5.395( = Formu a 1 .1757).

Table 1758. Compounds of formu a I .A, wherein R2 is R2-- 5.396( = Formu a 1 .1758).

Table 1759. Compounds of formu a I .A, wherein R2 is R2-- 5.397( = Formu a 1 .1759).

Table 1760. Compounds of formu a I .A, wherein R2 is R2-- 5.398( = Formu a 1 .1760).

Table 1761. Compounds of formu a I .A, wherein R2 is R2-- 5.399( = Formu a 1 .1761 ).

Table 1762. Compounds of formu a I .A, wherein R2 is R2-- 5.400( = Formu a 1 .1762).

Table 1763. Compounds of formu a I .A, wherein R2 is R2-- 5.401 ( = Formu a 1 .1763).

Table 1764. Compounds of formu a I .A, wherein R2 is R2-- 5.402( = Formu a 1 .1764).

Table 1765. Compounds of formu a I .A, wherein R2 is R2-- 5.403( = Formu a 1 .1765).

Table 1766. Compounds of formu a I .A, wherein R2 is R2-- 5.404( = Formu a 1 .1766).

Table 1767. Compounds of formu a I .A, wherein R2 is R2-- 5.405( = Formu a 1 .1767).

Table 1768. Compounds of formu a I .A, wherein R2 is R2-- 5.406( = Formu a 1 .1768).

Table 1769. Compounds of formu a I .A, wherein R2 is R2-- 5.407( = Formu a 1 .1769).

Table 1770. Compounds of formu a I .A, wherein R2 is R2-- 5.408( = Formu a 1 .1770).

Table 1771. Compounds of formu a I .A, wherein R2 is R2-- 5.409( = Formu a 1 .1771 ).

Table 1772. Compounds of formu a I .A, wherein R2 is R2-- 5.410( = Formu a 1 .1772).

Table 1773. Compounds of formu a I .A, wherein R2 is R2-- 5.41 1 ( = Formu a 1 .1773).

Table 1774. Compounds of formu a I .A, wherein R2 is R2-- 5.412( = Formu a 1 .1774).

Table 1775. Compounds of formu a I .A, wherein R2 is R2-- 5.413( = Formu a 1 .1775).

Table 1776. Compounds of formu a I .A, wherein R2 is R2-- 5.414( = Formu a 1 .1776).

Table 1777. Compounds of formu a I .A, wherein R2 is R2-- 5.415( = Formu a 1 .1777).

Table 1778. Compounds of formu a I .A, wherein R2 is R2-- 5.416( = Formu a 1 .1778).

Table 1779. Compounds of formu a I .A, wherein R2 is R2-- 5.417( = Formu a 1 .1779).

Table 1780. Compounds of formu a I .A, wherein R2 is R2-- 5.418( = Formu a 1 .1780).

Table 1781. Compounds of formu a I .A, wherein R2 is R2-- 5.419( = Formu a 1 .1781 ).

Table 1782. Compounds of formu a I .A, wherein R2 is R2-- 5.420( = Formu a 1 .1782).

Table 1783. Compounds of formu a I .A, wherein R2 is R2-- 5.421 ( = Formu a 1 .1783).

Table 1784. Compounds of formu a I .A, wherein R2 is R2-- 5.422( = Formu a 1 .1784).

Table 1785. Compounds of formu a I .A, wherein R2 is R2-- 5.423( = Formu a 1 .1785).

Table 1786. Compounds of formu a I .A, wherein R2 is R2-- 5.424( = Formu a 1 .1786).

Table 1787. Compounds of formu a I .A, wherein R2 is R2-- 5.425( = Formu a 1 .1787).

Table 1788. Compounds of formu a I .A, wherein R2 is R2-- 5.426( = Formu a 1 .1788).

Table 1789. Compounds of formu a I .A, wherein R2 is R2-- 5.427( = Formu a 1 .1789).

Table 1790. Compounds of formu a I .A, wherein R2 is R2-- 5.428( = Formu a 1 .1790).

Table 1791. Compounds of formu a I .A, wherein R2 is R2-- 5.429( = Formu a 1 .1791 ).

Table 1792. Compounds of formu a I .A, wherein R2 is R2-- 5.430( = Formu a 1 .1792).

Table 1793. Compounds of formu a I .A, wherein R2 is R2-- 5.431 ( = Formu a 1 .1793). Table 1794. Compounds of formu a I .A, wherein R2 is R2-- 5.432( Formu a 1.1794

Table 1795. Compounds of formu a I .A, wherein R2 is R2-- 5.433( = Formu a 1 .1795

Table 1796. Compounds of formu a I .A, wherein R2 is R2-- 5.434( = Formu a 1 .1796

Table 1797. Compounds of formu a I .A, wherein R2 is R2-- 5.435( = Formu a 1 .1797

Table 1798. Compounds of formu a I .A, wherein R2 is R2-- 5.436( = Formu a 1 .1798

Table 1799. Compounds of formu a I .A, wherein R2 is R2-- 5.437( = Formu a 1 .1799

Table 1800. Compounds of formu a I .A, wherein R2 is R2-- 5.438( = Formu a 1 .1800

Table 1801. Compounds of formu a I .A, wherein R2 is R2-- 5.439( = Formu a 1 .1801

Table 1802. Compounds of formu a I .A, wherein R2 is R2-- 5.440( = Formu a 1 .1802

Table 1803. Compounds of formu a I .A, wherein R2 is R2-- 5.441 ( = Formu a 1 .1803

Table 1804. Compounds of formu a I .A, wherein R2 is R2-- 5.442( = Formu a 1 .1804

Table 1805. Compounds of formu a I .A, wherein R2 is R2-- 5.443( = Formu a 1 .1805

Table 1806. Compounds of formu a I .A, wherein R2 is R2-- 5.444( = Formu a 1 .1806

Table 1807. Compounds of formu a I .A, wherein R2 is R2-- 5.445( = Formu a 1 .1807

Table 1808. Compounds of formu a I .A, wherein R2 is R2-- 5.446( = Formu a 1 .1808

Table 1809. Compounds of formu a I .A, wherein R2 is R2-- 5.447( = Formu a 1 .1809

Table 1810. Compounds of formu a I .A, wherein R2 is R2-- 5.448( = Formu a 1 .1810

Table 181 1. Compounds of formu a I .A, wherein R2 is R2-- 5.449( = Formu a 1 .181 1

Table 1812. Compounds of formu a I .A, wherein R2 is R2-- 5.450( = Formu a 1 .1812

Table 1813. Compounds of formu a I .A, wherein R2 is R2-- 5.451 ( = Formu a 1 .1813

Table 1814. Compounds of formu a I .A, wherein R2 is R2-- 5.452( = Formu a 1 .1814

Table 1815. Compounds of formu a I .A, wherein R2 is R2-- 5.453( = Formu a 1 .1815

Table 1816. Compounds of formu a I .A, wherein R2 is R2-- 5.454( = Formu a 1 .1816

Table 1817. Compounds of formu a I .A, wherein R2 is R2-- 5.455( = Formu a 1 .1817

Table 1818. Compounds of formu a I .A, wherein R2 is R2-- 5.456( = Formu a 1 .1818

Table 1819. Compounds of formu a I .A, wherein R2 is R2-- 5.457( = Formu a 1 .1819

Table 1820. Compounds of formu a I .A, wherein R2 is R2-- 5.458( = Formu a 1 .1820

Table 1821. Compounds of formu a I .A, wherein R2 is R2-- 5.459( = Formu a 1 .1821

Table 1822. Compounds of formu a I .A, wherein R2 is R2-- 5.460( = Formu a 1 .1822

Table 1823. Compounds of formu a I .A, wherein R2 is R2-- 5.461 ( = Formu a 1 .1823

Table 1824. Compounds of formu a I .A, wherein R2 is R2-- 5.462( = Formu a 1 .1824

Table 1825. Compounds of formu a I .A, wherein R2 is R2-- 5.463( = Formu a 1 .1825

Table 1826. Compounds of formu a I .A, wherein R2 is R2-- 5.464( = Formu a 1 .1826

Table 1827. Compounds of formu a I .A, wherein R2 is R2-- 5.465( = Formu a 1 .1827

Table 1828. Compounds of formu a I .A, wherein R2 is R2-- 5.466( = Formu a 1 .1828

Table 1829. Compounds of formu a I .A, wherein R2 is R2-- 5.467( = Formu a 1 .1829

Table 1830. Compounds of formu a I .A, wherein R2 is R2-- 5.468( = Formu a 1 .1830

Table 1831. Compounds of formu a I .A, wherein R2 is R2-- 5.469( = Formu a 1 .1831

Table 1832. Compounds of formu a I .A, wherein R2 is R2-- 5.470( = Formu a 1 .1832

Table 1833. Compounds of formu a I .A, wherein R2 is R2-- 5.471 ( = Formu a 1 .1833

Table 1834. Compounds of formu a I .A, wherein R2 is R2-- 5.472( = Formu a 1 .1834

Table 1835. Compounds of formu a I .A, wherein R2 is R2-- 5.473( = Formu a 1 .1835

Table 1836. Compounds of formu a I .A, wherein R2 is R2-- 5.474( = Formu a 1 .1836

Table 1837. Compounds of formu a I .A, wherein R2 is R2-- 5.475( = Formu a 1 .1837 Table 1838. Compounds of formu a I .A, wherein R2 is R2-- 5.476( = Formu a 1.1838).

Table 1839. Compounds of formu a I .A, wherein R2 is R2-- 5.477( = Formu a 1 .1839).

Table 1840. Compounds of formu a I .A, wherein R2 is R2-- 5.478( = Formu a 1 .1840).

Table 1841. Compounds of formu a I .A, wherein R2 is R2-- 5.479( = Formu a 1 .1841 ).

Table 1842. Compounds of formu a I .A, wherein R2 is R2-- 5.480( = Formu a 1 .1842).

Table 1843. Compounds of formu a I .A, wherein R2 is R2-- 5.481 ( = Formu a 1 .1843).

Table 1844. Compounds of formu a I .A, wherein R2 is R2-- 5.482( = Formu a 1 .1844).

Table 1845. Compounds of formu a I .A, wherein R2 is R2-- 5.483( = Formu a 1 .1845).

Table 1846. Compounds of formu a I .A, wherein R2 is R2-- 5.484( = Formu a 1 .1846).

Table 1847. Compounds of formu a I .A, wherein R2 is R2-- 5.485( = Formu a 1 .1847).

Table 1848. Compounds of formu a I .A, wherein R2 is R2-- 5.486( = Formu a 1 .1848).

Table 1849. Compounds of formu a I .A, wherein R2 is R2-- 5.487( = Formu a 1 .1849).

Table 1850. Compounds of formu a I .A, wherein R2 is R2-- 5.488( = Formu a 1 .1850).

Table 1851. Compounds of formu a I .A, wherein R2 is R2-- 5.489( = Formu a 1 .1851 ).

Table 1852. Compounds of formu a I .A, wherein R2 is R2-- 5.490( = Formu a 1 .1852).

Table 1853. Compounds of formu a I .A, wherein R2 is R2-- 5.491 ( = Formu a 1 .1853).

Table 1854. Compounds of formu a I .A, wherein R2 is R2-- 5.492( = Formu a 1 .1854).

Table 1855. Compounds of formu a I .A, wherein R2 is R2-- 5.493( = Formu a 1 .1855).

Table 1856. Compounds of formu a I .A, wherein R2 is R2-- 5.494( = Formu a 1 .1856).

Table 1857. Compounds of formu a I .A, wherein R2 is R2-- 5.495( = Formu a 1 .1857).

Table 1858. Compounds of formu a I .A, wherein R2 is R2-- 5.496( = Formu a 1 .1858).

Table 1859. Compounds of formu a I .A, wherein R2 is R2-- 5.497( = Formu a 1 .1859).

Table 1860. Compounds of formu a I .A, wherein R2 is R2-- 5.498( = Formu a 1 .1860).

Table 1861. Compounds of formu a I .A, wherein R2 is R2-- 5.499( = Formu a 1 .1861 ).

Table 1862. Compounds of formu a I .A, wherein R2 is R2-- 5.500( = Formu a 1 .1862).

Table 1863. Compounds of formu a I .A, wherein R2 is R2-- 5.501 ( = Formu a 1 .1863).

Table 1864. Compounds of formu a I .A, wherein R2 is R2-- 5.502( = Formu a 1 .1864).

Table 1865. Compounds of formu a I .A, wherein R2 is R2-- 5.503( = Formu a 1 .1865).

Table 1866. Compounds of formu a I .A, wherein R2 is R2-- 5.504( = Formu a 1 .1866).

Table 1867. Compounds of formu a I .A, wherein R2 is R2-- 5.505( = Formu a 1 .1867).

Table 1868. Compounds of formu a I .A, wherein R2 is R2-- 5.506( = Formu a 1 .1868).

Table 1869. Compounds of formu a I .A, wherein R2 is R2-- 5.507( = Formu a 1 .1869).

Table 1870. Compounds of formu a I .A, wherein R2 is R2-- 5.508( = Formu a 1 .1870).

Table 1871. Compounds of formu a I .A, wherein R2 is R2-- 5.509( = Formu a 1 .1871 ).

Table 1872. Compounds of formu a I .A, wherein R2 is R2-- 5.510( = Formu a 1 .1872).

Table 1873. Compounds of formu a I .A, wherein R2 is R2-- 5.51 1 ( = Formu a 1 .1873).

Table 1874. Compounds of formu a I .A, wherein R2 is R2-- 5.512( = Formu a 1 .1874).

Table 1875. Compounds of formu a I .A, wherein R2 is R2-- 5.513( = Formu a 1 .1875).

Table 1876. Compounds of formu a I .A, wherein R2 is R2-- 5.514( = Formu a 1 .1876).

Table 1877. Compounds of formu a I .A, wherein R2 is R2-- 5.515( = Formu a 1 .1877).

Table 1878. Compounds of formu a I .A, wherein R2 is R2-- 5.516( = Formu a 1 .1878).

Table 1879. Compounds of formu a I .A, wherein R2 is R2-- 5.517( = Formu a 1 .1879).

Table 1880. Compounds of formu a I .A, wherein R2 is R2-- 5.518( = Formu a 1 .1880).

Table 1881. Compounds of formu a I .A, wherein R2 is R2-- 5.519( = Formu a 1 .1881 ). Table 1882. Compounds of formu a I .A, wherein R2 is R2-- 5.520( Formu a 1.1882)

Table 1883. Compounds of formu a I .A, wherein R2 is R2-- 5.521 ( = Formu a 1 .1883)

Table 1884. Compounds of formu a I .A, wherein R2 is R2-- 5.522( = Formu a 1 .1884)

Table 1885. Compounds of formu a I .A, wherein R2 is R2-- 5.523( = Formu a 1 .1885)

Table 1886. Compounds of formu a I .A, wherein R2 is R2-- 5.524( = Formu a 1 .1886)

Table 1887. Compounds of formu a I .A, wherein R2 is R2-- 5.525( = Formu a 1 .1887)

Table 1888. Compounds of formu a I .A, wherein R2 is R2-- 5.526( = Formu a 1 .1888)

Table 1889. Compounds of formu a I .A, wherein R2 is R2-- 5.527( = Formu a 1 .1889)

Table 1890. Compounds of formu a I .A, wherein R2 is R2-- 5.528( = Formu a 1 .1890)

Table 1891. Compounds of formu a I .A, wherein R2 is R2-- 5.529( = Formu a 1 .1891 )

Table 1892. Compounds of formu a I .A, wherein R2 is R2-- 5.530( = Formu a 1 .1892)

Table 1893. Compounds of formu a I .A, wherein R2 is R2-- 5.531 ( = Formu a 1 .1893)

Table 1894. Compounds of formu a I .A, wherein R2 is R2-- 5.532( = Formu a 1 .1894)

Table 1895. Compounds of formu a I .A, wherein R2 is R2-- 5.533( = Formu a 1 .1895)

Table 1896. Compounds of formu a I .A, wherein R2 is R2-- 5.534( = Formu a 1 .1896)

Table 1897. Compounds of formu a I .A, wherein R2 is R2-- 5.535( = Formu a 1 .1897)

Table 1898. Compounds of formu a I .A, wherein R2 is R2-- 5.536( = Formu a 1 .1898)

Table 1899. Compounds of formu a I .A, wherein R2 is R2-- 5.537( = Formu a 1 .1899)

Table 1900. Compounds of formu a I .A, wherein R2 is R2-- 5.538( = Formu a 1 .1900)

Table 1901. Compounds of formu a I .A, wherein R2 is R2-- 5.539( = Formu a 1 .1901 )

Table 1902. Compounds of formu a I .A, wherein R2 is R2-- 5.540( = Formu a 1 .1902)

Table 1903. Compounds of formu a I .A, wherein R2 is R2-- 5.541 ( = Formu a 1 .1903)

Table 1904. Compounds of formu a I .A, wherein R2 is R2-- 5.542( = Formu a 1 .1904)

Table 1905. Compounds of formu a I .A, wherein R2 is R2-- 5.543( = Formu a 1 .1905)

Table 1906. Compounds of formu a I .A, wherein R2 is R2-- 5.544( = Formu a 1 .1906)

Table 1907. Compounds of formu a I .A, wherein R2 is R2-- 5.545( = Formu a 1 .1907)

Table 1908. Compounds of formu a I .A, wherein R2 is R2-- 5.546( = Formu a 1 .1908)

Table 1909. Compounds of formu a I .A, wherein R2 is R2-- 5.547( = Formu a 1 .1909)

Table 1910. Compounds of formu a I .A, wherein R2 is R2-- 5.548( = Formu a 1 .1910)

Table 191 1. Compounds of formu a I .A, wherein R2 is R2-- 5.549( = Formu a 1 .191 1 )

Table 1912. Compounds of formu a I .A, wherein R2 is R2-- 5.550( = Formu a 1 .1912)

Table 1913. Compounds of formu a I .A, wherein R2 is R2-- 5.551 ( = Formu a 1 .1913)

Table 1914. Compounds of formu a I .A, wherein R2 is R2-- 5.552( = Formu a 1 .1914)

Table 1915. Compounds of formu a I .A, wherein R2 is R2-- 5.553( = Formu a 1 .1915)

Table 1916. Compounds of formu a I .A, wherein R2 is R2-- 5.554( = Formu a 1 .1916)

Table 1917. Compounds of formu a I .A, wherein R2 is R2-- 5.555( = Formu a 1 .1917)

Table 1918. Compounds of formu a I .A, wherein R2 is R2-- 5.556( = Formu a 1 .1918)

Table 1919. Compounds of formu a I .A, wherein R2 is R2-- 5.557( = Formu a 1 .1919)

Table 1920. Compounds of formu a I .A, wherein R2 is R2-- 5.558( = Formu a 1 .1920)

Table 1921. Compounds of formu a I .A, wherein R2 is R2-- 5.559( = Formu a 1 .1921 )

Table 1922. Compounds of formu a I .A, wherein R2 is R2-- 5.560( = Formu a 1 .1922)

Table 1923. Compounds of formu a I .A, wherein R2 is R2-- 5.561 ( = Formu a 1 .1923)

Table 1924. Compounds of formu a I .A, wherein R2 is R2-- 5.562( = Formu a 1 .1924)

Table 1925. Compounds of formu a I .A, wherein R2 is R2-- 5.563( = Formu a 1 .1925) Table 1926. Compounds of formu a I .A, wherein R2 is R2-- 5.564( = Formu a 1.1926).

Table 1927. Compounds of formu a I .A, wherein R2 is R2-- 5.565( = Formu a 1 .1927).

Table 1928. Compounds of formu a I .A, wherein R2 is R2-- 5.566( = Formu a 1 .1928).

Table 1929. Compounds of formu a I .A, wherein R2 is R2-- 5.567( = Formu a 1 .1929).

Table 1930. Compounds of formu a I .A, wherein R2 is R2-- 5.568( = Formu a 1 .1930).

Table 1931. Compounds of formu a I .A, wherein R2 is R2-- 5.569( = Formu a 1 .1931).

Table 1932. Compounds of formu a I .A, wherein R2 is R2-- 5.570( = Formu a 1 .1932).

Table 1933. Compounds of formu a I .A, wherein R2 is R2-- 5.571 ( = Formu a 1 .1933).

Table 1934. Compounds of formu a I .A, wherein R2 is R2-- 5.572( = Formu a 1 .1934).

Table 1935. Compounds of formu a I .A, wherein R2 is R2-- 5.573( = Formu a 1 .1935).

Table 1936. Compounds of formu a I .A, wherein R2 is R2-- 5.574( = Formu a 1 .1936).

Table 1937. Compounds of formu a I .A, wherein R2 is R2-- 5.575( = Formu a 1 .1937).

Table 1938. Compounds of formu a I .A, wherein R2 is R2-- 5.576( = Formu a 1 .1938).

Table 1939. Compounds of formu a I .A, wherein R2 is R2-- 5.577( = Formu a 1 .1939).

Table 1940. Compounds of formu a I .A, wherein R2 is R2-- 5.578( = Formu a 1 .1940).

Table 1941. Compounds of formu a I .A, wherein R2 is R2-- 5.579( = Formu a 1 .1941).

Table 1942. Compounds of formu a I .A, wherein R2 is R2-- 5.580( = Formu a 1 .1942).

Table 1943. Compounds of formu a I .A, wherein R2 is R2-- 5.581 ( = Formu a 1 .1943).

Table 1944. Compounds of formu a I .A, wherein R2 is R2-- 5.582( = Formu a 1 .1944).

Table 1945. Compounds of formu a I .A, wherein R2 is R2-- 5.583( = Formu a 1 .1945).

Table 1946. Compounds of formu a I .A, wherein R2 is R2-- 5.584( = Formu a 1 .1946).

Table 1947. Compounds of formu a I .A, wherein R2 is R2-- 5.585( = Formu a 1 .1947).

Table 1948. Compounds of formu a I .A, wherein R2 is R2-- 5.586( = Formu a 1 .1948).

Table 1949. Compounds of formu a I .A, wherein R2 is R2-- 5.587( = Formu a 1 .1949).

Table 1950. Compounds of formu a I .A, wherein R2 is R2-- 5.588( = Formu a 1 .1950).

Table 1951. Compounds of formu a I .A, wherein R2 is R2-- 5.589( = Formu a 1 .1951).

Table 1952. Compounds of formu a I .A, wherein R2 is R2-- 5.590( = Formu a 1 .1952).

Table 1953. Compounds of formu a I .A, wherein R2 is R2-- 5.591 ( = Formu a 1 .1953).

Table 1954. Compounds of formu a I .A, wherein R2 is R2-- 5.592( = Formu a 1 .1954).

Table 1955. Compounds of formu a I .A, wherein R2 is R2-- 5.593( = Formu a 1 .1955).

Table 1956. Compounds of formu a I .A, wherein R2 is R2-- 5.594( = Formu a 1 .1956).

Table 1957. Compounds of formu a I .A, wherein R2 is R2-- 5.595( = Formu a 1 .1957).

Table 1958. Compounds of formu a I .A, wherein R2 is R2-- 5.596( = Formu a 1 .1958).

Table 1959. Compounds of formu a I .A, wherein R2 is R2-- 5.597( = Formu a 1 .1959).

Table 1960. Compounds of formu a I .A, wherein R2 is R2-- 5.598( = Formu a 1 .1960).

Table 1961. Compounds of formu a I .A, wherein R2 is R2-- 5.599( = Formu a 1 .1961).

Table 1962. Compounds of formu a I .A, wherein R2 is R2-- 5.600( = Formu a 1 .1962).

Table 1963. Compounds of formu a I .A, wherein R2 is R2-- 5.601 ( = Formu a 1 .1963).

Table 1964. Compounds of formu a I .A, wherein R2 is R2-- 5.602( = Formu a 1 .1964).

Table 1965. Compounds of formu a I .A, wherein R2 is R2-- 5.603( = Formu a 1 .1965).

Table 1966. Compounds of formu a I .A, wherein R2 is R2-- 5.604( = Formu a 1 .1966).

Table 1967. Compounds of formu a I .A, wherein R2 is R2-- 5.605( = Formu a 1 .1967).

Table 1968. Compounds of formu a I .A, wherein R2 is R2-- 5.606( = Formu a 1 .1968).

Table 1969. Compounds of formu a I .A, wherein R2 is R2-- 5.607( = Formu a 1 .1969). Table 1970. Compounds of formu a I .A, wherein R2 is R2-- 5.608( = Formu a ' 1.1970).

Table 1971. Compounds of formu a I .A, wherein R2 is R2-- 5.609( = Formu a ' 1.1971).

Table 1972. Compounds of formu a I .A, wherein R2 is R2-- 5.610( = Formu a ' 1.1972).

Table 1973. Compounds of formu a I .A, wherein R2 is R2-- 5.611( = Formu a ' 1.1973).

Table 1974. Compounds of formu a I .A, wherein R2 is R2-- 5.612( = Formu a ' 1.1974).

Table 1975. Compounds of formu a I .A, wherein R2 is R2-- 5.613( = Formu a ' 1.1975).

Table 1976. Compounds of formu a I .A, wherein R2 is R2-- 5.614( = Formu a ' 1.1976).

Table 1977. Compounds of formu a I .A, wherein R2 is R2-- 5.615( = Formu a ' 1.1977).

Table 1978. Compounds of formu a I .A, wherein R2 is R2-- 5.616( = Formu a ' 1.1978).

Table 1979. Compounds of formu a I .A, wherein R2 is R2-- 5.617( = Formu a ' 1.1979).

Table 1980. Compounds of formu a I .A, wherein R2 is R2-- 5.618( = Formu a ' 1.1980).

Table 1981. Compounds of formu a I .A, wherein R2 is R2-- 5.619( = Formu a ' 1.1981).

Table 1982. Compounds of formu a I .A, wherein R2 is R2-- 5.620( = Formu a ' 1.1982).

Table 1983. Compounds of formu a I .A, wherein R2 is R2-- 5.621 ( = Formu a ' 1.1983).

Table 1984. Compounds of formu a I .A, wherein R2 is R2-- 5.622( = Formu a ' 1.1984).

Table 1985. Compounds of formu a I .A, wherein R2 is R2-- 5.623( = Formu a ' 1.1985).

Table 1986. Compounds of formu a I .A, wherein R2 is R2-- 5.624( = Formu a ' 1.1986).

Table 1987. Compounds of formu a I .A, wherein R2 is R2-- 5.625( = Formu a ' 1.1987).

Table 1988. Compounds of formu a I .A, wherein R2 is R2-- 5.626( = Formu a ' 1.1988).

Table 1989. Compounds of formu a I .A, wherein R2 is R2-- 5.627( = Formu a ' 1.1989).

Table 1990. Compounds of formu a I .A, wherein R2 is R2-- 5.628( = Formu a ' 1.1990).

Table 1991. Compounds of formu a I .A, wherein R2 is R2-- 5.629( = Formu a ' 1.1991).

Table 1992. Compounds of formu a I .A, wherein R2 is R2-- 5.630( = Formu a ' 1.1992).

Table 1993. Compounds of formu a I .A, wherein R2 is R2-- 5.631 ( = Formu a ' 1.1993).

Table 1994. Compounds of formu a I .A, wherein R2 is R2-- 5.632( = Formu a ' 1.1994).

Table 1995. Compounds of formu a I .A, wherein R2 is R2-- 5.633( = Formu a ' 1.1995).

Table 1996. Compounds of formu a I .A, wherein R2 is R2-- 5.634( = Formu a ' 1.1996).

Table 1997. Compounds of formu a I .A, wherein R2 is R2-- 5.635( = Formu a ' 1.1997).

Table 1998. Compounds of formu a I .A, wherein R2 is R2-- 5.636( = Formu a ' 1.1998).

Table 1999. Compounds of formu a I .A, wherein R2 is R2-- 5.637( = Formu a ' 1.1999).

Table 2000. Compounds of formu a I .A, wherein R2 is R2-- 5.638( = Formu a ' 1.2000).

Table 2001. Compounds of formu a I .A, wherein R2 is R2-- 5.639( = Formu a ' 1.2001).

Table 2002. Compounds of formu a I .A, wherein R2 is R2-- 5.640( = Formu a ' 1.2002).

Table 2003. Compounds of formu a I .A, wherein R2 is R2-- 5.641 ( = Formu a ' 1.2003).

Table 2004. Compounds of formu a I .A, wherein R2 is R2-- 5.642( = Formu a ' 1.2004).

Table 2005. Compounds of formu a I .A, wherein R2 is R2-- 5.643( = Formu a ' 1.2005).

Table 2006. Compounds of formu a I .A, wherein R2 is R2-- 5.644( = Formu a ' 1.2006).

Table 2007. Compounds of formu a I .A, wherein R2 is R2-- 5.645( = Formu a ' 1.2007).

Table 2008. Compounds of formu a I .A, wherein R2 is R2-- 5.646( = Formu a ' 1.2008).

Table 2009. Compounds of formu a I .A, wherein R2 is R2-- 5.647( = Formu a ' 1.2009).

Table 2010. Compounds of formu a I .A, wherein R2 is R2-- 5.648( = Formu a ' 1.2010).

Table 2011. Compounds of formu a I .A, wherein R2 is R2-- 5.649( = Formu a ' 1.2011).

Table 2012. Compounds of formu a I .A, wherein R2 is R2-- 5.650( = Formu a ' 1.2012).

Table 2013. Compounds of formu a I .A, wherein R2 is R2-- 5.651 ( = Formu a ' 1.2013). Table 2014. Compounds of formu a I .A, wherein R2 is R2-15.652(=formula 1.2014).

Table 2015. Compounds of formu a I .A, wherein R2 is R2-15.653(=formula 1.2015).

Table 2016. Compounds of formu a I .A, wherein R2 is R2-15.654(=formula 1.2016).

Table 2017. Compounds of formu a I .A, wherein R2 is R2-15.655(=formula 1.2017).

Table 2018. Compounds of formu a I .A, wherein R2 is R2-15.656(=formula 1.2018).

Table 2019. Compounds of formu a I .A, wherein R2 is R2-15.657(=formula 1.2019).

Table 2020. Compounds of formu a I .A, wherein R2 is R2-15.658(=formula 1.2020).

Table 2021. Compounds of formu a I .A, wherein R2 is R2-15.659(=formula 1.2021).

Table 2022. Compounds of formu a I .A, wherein R2 is R2-15.660(=formula 1.2022).

Table 2023. Compounds of formu a I .A, wherein R2 is R2-15.661 (=formula 1.2023).

Table 2024. Compounds of formu a I .A, wherein R2 is R2-15.662(=formula 1.2024).

Table 2025. Compounds of formu a I .A, wherein R2 is R2-15.663(=formula 1.2025).

Table 2026. Compounds of formu a I .A, wherein R2 is R2-15.664(=formula 1.2026).

Table 2027. Compounds of formu a I .A, wherein R2 is R2-15.665(=formula 1.2027).

Table 2028. Compounds of formu a I .A, wherein R2 is R2-15.666(=formula 1.2028).

Table 2029. Compounds of formu a I .A, wherein R2 is R2-15.667(=formula 1.2029).

Table 2030. Compounds of formu a I .A, wherein R2 is R2-15.668(=formula 1.2030).

Table 2031. Compounds of formu a I .A, wherein R2 is R2-15.669(=formula 1.2031).

Table 2032. Compounds of formu a I .A, wherein R2 is R2-15.670(=formula 1.2032).

Table 2033. Compounds of formu a I .A, wherein R2 is R2-15.671 (=formula 1.2033).

Table 2034. Compounds of formu a I .A, wherein R2 is R2-15.672(=formula 1.2034).

Table 2035. Compounds of formu a I .A, wherein R2 is R2-15.673(=formula 1.2035).

Table 2036. Compounds of formu a I .A, wherein R2 is R2-15.674(=formula 1.2036).

Table 2037. Compounds of formu a I .A, wherein R2 is R2-15.675(=formula 1.2037).

Table 2038. Compounds of formu a I .A, wherein R2 is R2-15.676(=formula 1.2038).

Table 2039. Compounds of formu a I .A, wherein R2 is R2-9.1 (=formula 1.2039).

Table 2040. Compounds of formu a I .A, wherein R2 is R2-9.2(=formula 1.2040).

Table 2041. Compounds of formu a I .A, wherein R2 is R2-9.3(=formula 1.2041).

Table 2042. Compounds of formu a I .A, wherein R2 is R2-9.4(=formula 1.2042).

Table 2043. Compounds of formu a I .A, wherein R2 is R2-9.5(=formula 1.2043).

Table 2044. Compounds of formu a I .A, wherein R2 is R2-9.6(=formula 1.2044).

Table 2045. Compounds of formu a I .A, wherein R2 is R2-9.7(=formula 1.2045).

Table 2046. Compounds of formu a I .A, wherein R2 is R2-9.8(=formula 1.2046).

Table 2047. Compounds of formu a I .A, wherein R2 is R2-9.9(=formula 1.2047).

Table 2048. Compounds of formu a I .A, wherein R2 is R2-9.10(=formula 1.2048).

Table 2049. Compounds of formu a I .A, wherein R2 is R2-9.11(=formula 1.2049).

Table 2050. Compounds of formu a I .A, wherein R2 is R2-9.12(=formula 1.2050).

Table 2051. Compounds of formu a I .A, wherein R2 is R2-9.13(=formula 1.2051).

Table 2052. Compounds of formu a I .A, wherein R2 is R2-9.14(=formula 1.2052).

Table 2053. Compounds of formu a I .A, wherein R2 is R2-9.15(=formula 1.2053).

Table 2054. Compounds of formu a I .A, wherein R2 is R2-9.16(=formula 1.2054).

TableAI :

The specific number for each single compound is deductible as follows:

Compound 1.27.1-317 e.g. comprises the compound of formula 1.27 from Table 27 and line I- 317 from Table A1 ;

According to another particularly preferred embodiment of the compounds of formula I and their use as herbicide, compounds of the invention are the compounds of formulae I that are compiled in tables 2055 to 4082, wherein the meaning for the combination of variables R 1 , R 3 , m, and R 4 for each individual compound of tables 2055 to 4082 corresponds to each line of Table A2. Each of the groups mentioned for a substituent in the tables is furthermore per se, independently of the combination in which it is mentioned, a particularly preferred aspect of the substituent in question. The term "formula" used in below tables 2055 to 4082 denotes

"compounds of formula".

Table 2055. Compounds of formu a I.C, wherein R2 is R2-9.17I Formu a 1 .2055).

Table 2056. Compounds of formu a I.C, wherein R2 is R2-9.18I = Formu a 1 .2056).

Table 2057. Compounds of formu a I.C, wherein R2 is R2-9.19I = Formu a 1 .2057).

Table 2058. Compounds of formu a I.C, wherein R2 is R2-9.20I = Formu a 1 . 2058)

Table 2059. Compounds of formu a I.C, wherein R2 is R2-9.21 I = Formu a 1 . 2059)

Table 2060. Compounds of formu a I.C, wherein R2 is R2-9.22I = Formu a 1 . 2060)

Table 2061. Compounds of formu a I.C, wherein R2 is R2-9.23I = Formu a 1 . 2061 )

Table 2062. Compounds of formu a I.C, wherein R2 is R2-9.24I = Formu a 1 . 2062)

Table 2063. Compounds of formu a I.C, wherein R2 is R2-9.25I = Formu a 1 . 2063)

Table 2064. Compounds of formu a I.C, wherein R2 is R2-9.26I = Formu a 1 . 2064)

Table 2065. Compounds of formu a I.C, wherein R2 is R2-9.27I = Formu a 1 . 2065)

Table 2066. Compounds of formu a I.C, wherein R2 is R2-9.28I = Formu a 1 . 2066)

Table 2067. Compounds of formu a I.C, wherein R2 is R2-9.29I = Formu a 1 . 2067)

Table 2068. Compounds of formu a I.C, wherein R2 is R2-9.30I = Formu a 1 . 2068)

Table 2069. Compounds of formu a I.C, wherein R2 is R2-9.31 I = Formu a 1 . 2069)

Table 2070. Compounds of formu a I.C, wherein R2 is R2-9.32I = Formu a 1 . 2070)

Table 2071. Compounds of formu a I.C, wherein R2 is R2-9.33I = Formu a 1 . 2071 )

Table 2072. Compounds of formu a I.C, wherein R2 is R2-9.34I = Formu a 1 . 2072)

Table 2073. Compounds of formu a I.C, wherein R2 is R2-9.35I = Formu a 1 . 2073)

Table 2074. Compounds of formu a I.C, wherein R2 is R2-9.36I = Formu a 1 . 2074)

Table 2075. Compounds of formu a I.C, wherein R2 is R2-9.37I = Formu a 1 . 2075)

Table 2076. Compounds of formu a I.C, wherein R2 is R2-9.38I = Formu a 1 . 2076)

Table 2077. Compounds of formu a I.C, wherein R2 is R2-9.39I = Formu a 1 . 2077)

Table 2078. Compounds of formu a I.C, wherein R2 is R2-9.40I = Formu a 1 . 2078)

Table 2079. Compounds of formu a I.C, wherein R2 is R2-9.41 I = Formu a 1 . 2079)

Table 2080. Compounds of formu a I.C, wherein R2 is R2-9.42I = Formu a 1 .2080).

Table 2081. Compounds of formu a I.C, wherein R2 is R2-9.43I = Formu a 1 .2081 ).

Table 2082. Compounds of formu a I.C, wherein R2 is R2-9.44I = Formu a 1 .2082).

Table 2083. Compounds of formu a I.C, wherein R2 is R2-9.45I = Formu a 1 .2083).

Table 2084. Compounds of formu a I.C, wherein R2 is R2-9.46I = Formu a 1 .2084).

Table 2085. Compounds of formu a I.C, wherein R2 is R2-9.47I = Formu a 1 .2085).

Table 2086. Compounds of formu a I.C, wherein R2 is R2-9.48I = Formu a 1 .2086).

Table 2087. Compounds of formu a I.C, wherein R2 is R2-9.49I = Formu a 1 .2087).

Table 2088. Compounds of formu a I.C, wherein R2 is R2-9.50I = Formu a 1 .2088).

Table 2089. Compounds of formu a I.C, wherein R2 is R2-9.51 I = Formu a 1 .2089).

Table 2090. Compounds of formu a I.C, wherein R2 is R2-9.52I = Formu a 1 .2090).

Table 2091. Compounds of formu a I.C, wherein R2 is R2-9.53I = Formu a 1 .2091 ).

Table 2092. Compounds of formu a I.C, wherein R2 is R2-9.54I = Formu a 1 .2092).

Table 2093. Compounds of formu a I.C, wherein R2 is R2-9.55I = Formu a 1 .2093).

Table 2094. Compounds of formu a I.C, wherein R2 is R2-9.56I = Formu a 1 .2094).

Table 2095. Compounds of formu a I.C, wherein R2 is R2-9.57I = Formu a 1 .2095). Table 2096. Compounds of formu a I.C, wherein R2 is R2-9.58I Formula 1 .2096).

Table 2097. Compounds of formu a I.C, wherein R2 is R2-9.59I = Formula 1 .2097).

Table 2098. Compounds of formu a I.C, wherein R2 is R2-9.60I = Formula 1 .2098).

Table 2099. Compounds of formu a I.C, wherein R2 is R2-9.61 I = Formula 1 .2099).

Table 2' 100. Compounds of formu a I.C, wherein R2 is R2-9.62I = Formula 1 .2100).

Table 2' 101. Compounds of formu a I.C, wherein R2 is R2-9.63I = Formula 1 . 2101 ).

Table 2' 102. Compounds of formu a I.C, wherein R2 is R2-9.64I = Formula 1 . 2102).

Table 2' 103. Compounds of formu a I.C, wherein R2 is R2-9.65I = Formula 1 . 2103).

Table 2' 104. Compounds of formu a I.C, wherein R2 is R2-9.66I = Formula 1 . 2104).

Table 2' 105. Compounds of formu a I.C, wherein R2 is R2-9.67I = Formula 1 . 2105).

Table 2' 106. Compounds of formu a I.C, wherein R2 is R2-9.68I = Formula 1 . 2106).

Table 2' 107. Compounds of formu a I.C, wherein R2 is R2-9.69I = Formula 1 . 2107).

Table 2' 108. Compounds of formu a I.C, wherein R2 is R2-9.70I = Formula 1 . 2108).

Table 2' 109. Compounds of formu a I.C, wherein R2 is R2-9.71 I = Formula 1 . 2109).

Table 2' 1 10. Compounds of formu a I.C, wherein R2 is R2-9.72I = Formula 1 . 21 10).

Table 2' 1 1 1. Compounds of formu a I.C, wherein R2 is R2-9.73I = Formula 1 . 21 1 1 ).

Table 2' 1 12. Compounds of formu a I.C, wherein R2 is R2-9.74I = Formula 1 . 21 12).

Table 2' 1 13. Compounds of formu a I.C, wherein R2 is R2-9.75I = Formula 1 . 21 13).

Table 2' 1 14. Compounds of formu a I.C, wherein R2 is R2-9.76I = Formula 1 . 21 14).

Table 2' 1 15. Compounds of formu a I.C, wherein R2 is R2-9.77I = Formula 1 . 21 15).

Table 2' 1 16. Compounds of formu a I.C, wherein R2 is R2-9.78I = Formula 1 . 21 16).

Table 2' 1 17. Compounds of formu a I.C, wherein R2 is R2-9.79I = Formula 1 . 21 17).

Table 2' 1 18. Compounds of formu a I.C, wherein R2 is R2-9.80I = Formula 1 .21 18).

Table 2' 1 19. Compounds of formu a I.C, wherein R2 is R2-9.81 I = Formula 1 .21 19).

Table 2' I20. Compounds of formu a I.C, wherein R2 is R2-9.82I = Formula 1 .2120).

Table 2' 121. Compounds of formu a I.C, wherein R2 is R2-9.83I = Formula 1 .2121 ).

Table 2' 122. Compounds of formu a I.C, wherein R2 is R2-9.84I = Formula 1 .2122).

Table 2' I23. Compounds of formu a I.C, wherein R2 is R2-9.85I = Formula 1 .2123).

Table 2' 124. Compounds of formu a I.C, wherein R2 is R2-9.86I = Formula 1 .2124).

Table 2' I25. Compounds of formu a I.C, wherein R2 is R2-9.87I = Formula 1 .2125).

Table 2' I26. Compounds of formu a I.C, wherein R2 is R2-9.88I = Formula 1 .2126).

Table 2' I27. Compounds of formu a I.C, wherein R2 is R2-9.89I = Formula 1 .2127).

Table 2' I28. Compounds of formu a I.C, wherein R2 is R2-9.90I = Formula 1 .2128).

Table 2' I29. Compounds of formu a I.C, wherein R2 is R2-9.91 I = Formula 1 .2129).

Table 2' 130. Compounds of formu a I.C, wherein R2 is R2-9.92I = Formula 1 .2130).

Table 2' 131. Compounds of formu a I.C, wherein R2 is R2-9.93I = Formula 1 .2131 ).

Table 2' 132. Compounds of formu a I.C, wherein R2 is R2-9.94I = Formula 1 .2132).

Table 2' 133. Compounds of formu a I.C, wherein R2 is R2-9.95I = Formula 1 .2133).

Table 2' 134. Compounds of formu a I.C, wherein R2 is R2-9.96I = Formula 1 .2134).

Table 2' 135. Compounds of formu a I.C, wherein R2 is R2-9.97I = Formula 1 .2135).

Table 2' 136. Compounds of formu a I.C, wherein R2 is R2-9.98I = Formula 1 .2136).

Table 2' 137. Compounds of formu a I.C, wherein R2 is R2-9.99I = Formula 1 .2137).

Table 2' 138. Compounds of formu a I.C, wherein R2 is R2-9.100(=formula 1.2138).

Table 2' 139. Compounds of formu a I.C, wherein R2 is R2-9.101 (=formula 1.2139). Tab e 2140. Compounds of ormu a I.C, wherein R2 is R2-9. 02( = Formu a 1.2140).

Tab e 2141. Compounds of ormu a I.C, wherein R2 is R2-9. 03( = Formu a 1.2141 ).

Tab e 2142. Compounds of ormu a I.C, wherein R2 is R2-9. 04( = Formu a 1.2142).

Tab e 2143. Compounds of ormu a I.C, wherein R2 is R2-9. 05( = Formu a 1.2143).

Tab e 2144. Compounds of ormu a I.C, wherein R2 is R2-9. 06( = Formu a 1.2144).

Tab Θ 2145. Compounds of ormu a I.C, wherein R2 is R2-9. 07( = Formu a 1.2145).

Tab Θ 2146. Compounds of ormu a I.C, wherein R2 is R2-9. 08( = Formu a 1.2146).

Tab Θ 2147. Compounds of ormu a I.C, wherein R2 is R2-9. 09( = Formu a 1.2147).

Tab Θ 2148. Compounds of ormu a I.C, wherein R2 is R2-9. 10( = Formu a 1.2148).

Tab Θ 2149. Compounds of ormu a I.C, wherein R2 is R2-9. 1 1 ( = Formu a 1.2149).

Tab Θ 2150. Compounds of ormu a I.C, wherein R2 is R2-9. 12( = Formu a 1.2150).

Tab Θ 2151. Compounds of ormu a I.C, wherein R2 is R2-9. 13( = Formu a 1.2151 ).

Tab Θ 2152. Compounds of ormu a I.C, wherein R2 is R2-9. 14( = Formu a 1.2152).

Tab Θ 2153. Compounds of ormu a I.C, wherein R2 is R2-9. 15( = Formu a 1.2153).

Tab Θ 2154. Compounds of ormu a I.C, wherein R2 is R2-9. 16( = Formu a 1.2154).

Tab Θ 2155. Compounds of ormu a I.C, wherein R2 is R2-9. 17( = Formu a 1.2155).

Tab Θ 2156. Compounds of ormu a I.C, wherein R2 is R2-9. 18( = Formu a 1.2156).

Tab Θ 2157. Compounds of ormu a I.C, wherein R2 is R2-9. 19( = Formu a 1.2157).

Tab Θ 2158. Compounds of ormu a I.C, wherein R2 is R2-9. 20( = Formu a 1.2158).

Tab Θ 2159. Compounds of ormu a I.C, wherein R2 is R2-9. 21 ( = Formu a 1.2159).

Tab Θ 2160. Compounds of ormu a I.C, wherein R2 is R2-9. 22( = Formu a 1.2160).

Tab Θ 2161. Compounds of ormu a I.C, wherein R2 is R2-9. 23( = Formu a 1.2161 ).

Tab Θ 2162. Compounds of ormu a I.C, wherein R2 is R2-9. 24( = Formu a 1.2162).

Tab Θ 2163. Compounds of ormu a I.C, wherein R2 is R2-9. 25( = Formu a 1.2163).

Tab Θ 2164. Compounds of ormu a I.C, wherein R2 is R2-9. 26( = Formu a 1.2164).

Tab Θ 2165. Compounds of ormu a I.C, wherein R2 is R2-9. 27( = Formu a 1.2165).

Tab Θ 2166. Compounds of ormu a I.C, wherein R2 is R2-9. 28( = Formu a 1.2166).

Tab Θ 2167. Compounds of ormu a I.C, wherein R2 is R2-9. 29( = Formu a 1.2167).

Tab Θ 2168. Compounds of ormu a I.C, wherein R2 is R2-9. 30( = Formu a 1.2168).

Tab Θ 2169. Compounds of ormu a I.C, wherein R2 is R2-9. 31 ( = Formu a 1.2169).

Tab Θ 2170. Compounds of ormu a I.C, wherein R2 is R2-9. 32( = Formu a 1.2170).

Tab Θ 2171. Compounds of ormu a I.C, wherein R2 is R2-9. 33( = Formu a 1.2171 ).

Tab Θ 2172. Compounds of ormu a I.C, wherein R2 is R2-9. 34( = Formu a 1.2172).

Tab Θ 2173. Compounds of ormu a I.C, wherein R2 is R2-9. 35( = Formu a 1.2173).

Tab Θ 2174. Compounds of ormu a I.C, wherein R2 is R2-9. 36( = Formu a 1.2174).

Tab Θ 2175. Compounds of ormu a I.C, wherein R2 is R2-9. 37( = Formu a 1.2175).

Tab Θ 2176. Compounds of ormu a I.C, wherein R2 is R2-9. 38( = Formu a 1.2176).

Tab Θ 2177. Compounds of ormu a I.C, wherein R2 is R2-9. 39( = Formu a 1.2177).

Tab Θ 2178. Compounds of ormu a I.C, wherein R2 is R2-9. 40( = Formu a 1.2178).

Tab Θ 2179. Compounds of ormu a I.C, wherein R2 is R2-9. 41 ( = Formu a 1.2179).

Tab Θ 2180. Compounds of ormu a I.C, wherein R2 is R2-9. 42( = Formu a 1.2180).

Tab Θ 2181. Compounds of ormu a I.C, wherein R2 is R2-9. 43( = Formu a 1.2181 ).

Tab Θ 2182. Compounds of ormu a I.C, wherein R2 is R2-9. 44( = Formu a 1.2182).

Tab Θ 2183. Compounds of ormu a I.C, wherein R2 is R2-9. 45( = Formu a 1.2183). Tab e 2184. Compounds of ormu a I.C, wherein R2 is R2-9. 46( Formu a 1.2184).

Tab e 2185. Compounds of ormu a I.C, wherein R2 is R2-9. 47( = Formu a 1.2185).

Tab e 2186. Compounds of ormu a I.C, wherein R2 is R2-9. 48( = Formu a 1.2186).

Tab e 2187. Compounds of ormu a I.C, wherein R2 is R2-9. 49( = Formu a 1.2187).

Tab e 2188. Compounds of ormu a I.C, wherein R2 is R2-9. 50( = Formu a 1.2188).

Tab e 2189. Compounds of ormu a I.C, wherein R2 is R2-9. 51 ( = Formu a 1.2189).

Tab e 2190. Compounds of ormu a I.C, wherein R2 is R2-9. 52( = Formu a 1.2190).

Tab e 2191. Compounds of ormu a I.C, wherein R2 is R2-9. 53( = Formu a 1.2191 ).

Tab Θ 2192. Compounds of ormu a I.C, wherein R2 is R2-9. 54( = Formu a 1.2192).

Tab e 2193. Compounds of ormu a I.C, wherein R2 is R2-9. 55( = Formu a 1.2193).

Tab Θ 2194. Compounds of ormu a I.C, wherein R2 is R2-9. 56( = Formu a 1.2194).

Tab Θ 2195. Compounds of ormu a I.C, wherein R2 is R2-9. 57( = Formu a 1.2195).

Tab Θ 2196. Compounds of ormu a I.C, wherein R2 is R2-9. 58( = Formu a 1.2196).

Tab Θ 2197. Compounds of ormu a I.C, wherein R2 is R2-9. 59( = Formu a 1.2197).

Tab Θ 2198. Compounds of ormu a I.C, wherein R2 is R2-9. 60( = Formu a 1.2198).

Tab Θ 2199. Compounds of ormu a I.C, wherein R2 is R2-9. 61 ( = Formu a 1.2199).

Tab e 2200. Compounds of ormu a I.C, wherein R2 is R2-9. 62( = Formu a 1.2200).

Tab e 2201. Compounds of ormu a I.C, wherein R2 is R2-9. 63( = Formu a 1.2201 ).

Tab e 2202. Compounds of ormu a I.C, wherein R2 is R2-9. 64( = Formu a 1.2202).

Tab e 2203. Compounds of ormu a I.C, wherein R2 is R2-9. 65( = Formu a 1.2203).

Tab e 2204. Compounds of ormu a I.C, wherein R2 is R2-9. 66( = Formu a 1.2204).

Tab e 2205. Compounds of ormu a I.C, wherein R2 is R2-9. 67( = Formu a 1.2205).

Tab e 2206. Compounds of ormu a I.C, wherein R2 is R2-9. 68( = Formu a 1.2206).

Tab e 2207. Compounds of ormu a I.C, wherein R2 is R2-9. 69( = Formu a 1.2207).

Tab e 2208. Compounds of ormu a I.C, wherein R2 is R2-9. 70( = Formu a 1.2208).

Tab e 2209. Compounds of ormu a I.C, wherein R2 is R2-9. 71 ( = Formu a 1.2209).

Tab e 2210. Compounds of ormu a I.C, wherein R2 is R2-9. 72( = Formu a 1.2210).

Tab e 2211. Compounds of ormu a I.C, wherein R2 is R2-9. 73( = Formu a 1.221 1 ).

Tab e 2212. Compounds of ormu a I.C, wherein R2 is R2-9. 74( = Formu a 1.2212).

Tab Θ 2213. Compounds of ormu a I.C, wherein R2 is R2-9. 75( = Formu a 1.2213).

Tab Θ 2214. Compounds of ormu a I.C, wherein R2 is R2-9. 76( = Formu a 1.2214).

Tab Θ 2215. Compounds of ormu a I.C, wherein R2 is R2-9. 77( = Formu a 1.2215).

Tab Θ 2216. Compounds of ormu a I.C, wherein R2 is R2-9. 78( = Formu a 1.2216).

Tab Θ 2217. Compounds of ormu a I.C, wherein R2 is R2-9. 79( = Formu a 1.2217).

Tab Θ 2218. Compounds of ormu a I.C, wherein R2 is R2-9. 80( = Formu a 1.2218).

Tab Θ 2219. Compounds of ormu a I.C, wherein R2 is R2-9. 81 ( = Formu a 1.2219).

Tab e 2220. Compounds of ormu a I.C, wherein R2 is R2-9. 82( = Formu a 1.2220).

Tab Θ 2221. Compounds of ormu a I.C, wherein R2 is R2-9. 83( = Formu a 1.2221 ).

Tab e 2222. Compounds of ormu a I.C, wherein R2 is R2-9. 84( = Formu a 1.2222).

Tab e 2223. Compounds of ormu a I.C, wherein R2 is R2-9. 85( = Formu a 1. 2223).

Tab e 2224. Compounds of ormu a I.C, wherein R2 is R2-9. 86( = Formu a 1. 2224).

Tab e 2225. Compounds of ormu a I.C, wherein R2 is R2-9. 87( = Formu a 1. 2225).

Tab e 2226. Compounds of ormu a I.C, wherein R2 is R2-9. 88( = Formu a 1.2226).

Tab e 2227. Compounds of ormu a I.C, wherein R2 is R2-9. 89( = Formu a 1.2227). Tab e 2228. Compounds o ormu a I.C, wherein R2 is R2-9.190( Formu a 1.2228).

Tab e 2229. Compounds o ormu a I.C, wherein R2 is R2-9.191( = Formu a 1.2229).

Tab e 2230. Compounds o ormu a I.C, wherein R2 is R2-9.192( = Formu a 1.2230).

Tab e 2231. Compounds o ormu a I.C, wherein R2 is R2-9.193( = Formu a 1.2231).

Tab e 2232. Compounds o ormu a I.C, wherein R2 is R2-9.194( = Formu a 1.2232).

Tab e 2233. Compounds o ormu a I.C, wherein R2 is R2-9.195( = Formu a 1.2233).

Tab e 2234. Compounds o ormu a I.C, wherein R2 is R2-9.196( = Formu a 1.2234).

Tab e 2235. Compounds o ormu a I.C, wherein R2 is R2-9.197( = Formu a 1.2235).

Tab e 2236. Compounds o ormu a I.C, wherein R2 is R2-9.198( = Formu a 1.2236).

Tab e 2237. Compounds o ormu a I.C, wherein R2 is R2-9.199( = Formu a 1.2237).

Tab e 2238. Compounds o ormu a I.C, wherein R2 is R2-9.200( = Formu a 1.2238).

Tab e 2239. Compounds o ormu a I.C, wherein R2 is R2-9.201< = Formu a 1.2239).

Tab e 2240. Compounds o ormu a I.C, wherein R2 is R2-9.202( = Formu a 1.2240).

Tab e 2241. Compounds o ormu a I.C, wherein R2 is R2-9.203( = Formu a 1.2241).

Tab e 2242. Compounds o ormu a I.C, wherein R2 is R2-9.204( = Formu a 1.2242).

Tab e 2243. Compounds o ormu a I.C, wherein R2 is R2-9.205( = Formu a 1.2243).

Tab e 2244. Compounds o ormu a I.C, wherein R2 is R2-9.206( = Formu a 1.2244).

Tab e 2245. Compounds o ormu a I.C, wherein R2 is R2-9.207( = Formu a 1.2245).

Tab e 2246. Compounds o ormu a I.C, wherein R2 is R2-9.208( = Formu a 1.2246).

Tab e 2247. Compounds o ormu a I.C, wherein R2 is R2-9.209( = Formu a 1.2247).

Tab e 2248. Compounds o ormu a I.C, wherein R2 is R2-9.210( = Formu a 1.2248).

Tab e 2249. Compounds o ormu a I.C, wherein R2 is R2-9.211< = Formu a 1.2249).

Tab e 2250. Compounds o ormu a I.C, wherein R2 is R2-9.212( = Formu a 1.2250).

Tab e 2251. Compounds o ormu a I.C, wherein R2 is R2-9.213( = Formu a 1.2251).

Tab e 2252. Compounds o ormu a I.C, wherein R2 is R2-9.214( = Formu a 1.2252).

Tab e 2253. Compounds o ormu a I.C, wherein R2 is R2-9.215( = Formu a 1.2253).

Tab e 2254. Compounds o ormu a I.C, wherein R2 is R2-9.216( = Formu a 1.2254).

Tab e 2255. Compounds o ormu a I.C, wherein R2 is R2-9.217( = Formu a 1.2255).

Tab e 2256. Compounds o ormu a I.C, wherein R2 is R2-9.218( = Formu a 1.2256).

Tab e 2257. Compounds o ormu a I.C, wherein R2 is R2-9.219( = Formu a 1.2257).

Tab e 2258. Compounds o ormu a I.C, wherein R2 is R2-9.220( = Formu a 1.2258).

Tab e 2259. Compounds o ormu a I.C, wherein R2 is R2-9.221< = Formu a 1.2259).

Tab e 2260. Compounds o ormu a I.C, wherein R2 is R2-9.222( = Formu a 1.2260).

Tab e 2261. Compounds o ormu a I.C, wherein R2 is R2-9.223( = Formu a 1.2261).

Tab e 2262. Compounds o ormu a I.C, wherein R2 is R2-9.224( = Formu a 1.2262).

Tab e 2263. Compounds o ormu a I.C, wherein R2 is R2-9.225( = Formu a 1.2263).

Tab e 2264. Compounds o ormu a I.C, wherein R2 is R2-9.226( = Formu a 1.2264).

Tab e 2265. Compounds o ormu a I.C, wherein R2 is R2-9.227( = Formu a 1.2265).

Tab e 2266. Compounds o ormu a I.C, wherein R2 is R2-9.228( = Formu a 1.2266).

Tab e 2267. Compounds o ormu a I.C, wherein R2 is R2-9.229( = Formu a 1.2267).

Tab e 2268. Compounds o ormu a I.C, wherein R2 is R2-9.230( = Formu a 1.2268).

Tab e 2269. Compounds o ormu a I.C, wherein R2 is R2-9.231< = Formu a 1.2269).

Tab e 2270. Compounds o ormu a I.C, wherein R2 is R2-9.232( = Formu a 1.2270).

Tab e 2271. Compounds o ormu a I.C, wherein R2 is R2-9.233( = Formu a 1.2271). Table 2272. Compounds of formu a I.C, wherein R2 is R2- 9.234( =formula 1.2272).

Table 2273. Compounds of formu a I.C, wherein R2 is R2- -9.235< =formula 1.2273).

Table 2274. Compounds of formu a I.C, wherein R2 is R2- -9.236< =formula 1.2274).

Table 2275. Compounds of formu a I.C, wherein R2 is R2- -9.237< =formula 1.2275).

Table 2276. Compounds of formu a I.C, wherein R2 is R2- -9.238< =formula 1.2276).

Table 2277. Compounds of formu a I.C, wherein R2 is R2- 9.239( =formula 1.2277).

Table 2278. Compounds of formu a I.C, wherein R2 is R2- 9.240( =formula 1.2278).

Table 2279. Compounds of formu a I.C, wherein R2 is R2- 9.241 ( =formula 1.2279).

Table 2280. Compounds of formu a I.C, wherein R2 is R2- 9.242( =formula 1.2280).

Table 2281. Compounds of formu a I.C, wherein R2 is R2- 9.243 (=formula 1.2281)

Table 2282. Compounds of formu a I.C, wherein R2 is R2- 9.244( =formula 1.2282).

Table 2283. Compounds of formu a I.C, wherein R2 is R2- 9.245( =formula 1.2283).

Table 2284. Compounds of formu a I.C, wherein R2 is R2- 9.246( =formula 1.2284).

Table 2285. Compounds of formu a I.C, wherein R2 is R2- 9.247( =formula 1.2285).

Table 2286. Compounds of formu a I.C, wherein R2 is R2- 9.248( =formula 1.2286).

Table 2287. Compounds of formu a I.C, wherein R2 is R2- 9.249( =formula 1.2287).

Table 2288. Compounds of formu a I.C, wherein R2 is R2- 9.250( =formula 1.2288).

Table 2289. Compounds of formu a I.C, wherein R2 is R2- 9.251 ( =formula 1.2289).

Table 2290. Compounds of formu a I.C, wherein R2 is R2- 9.252( =formula 1.2290).

Table 2291. Compounds of formu a I.C, wherein R2 is R2- 9.253( =formula 1.2291).

Table 2292. Compounds of formu a I.C, wherein R2 is R2- 9.254( =formula 1.2292).

Table 2293. Compounds of formu a I.C, wherein R2 is R2- 9.255( =formula 1.2293).

Table 2294. Compounds of formu a I.C, wherein R2 is R2- 9.256( =formula 1.2294).

Table 2295. Compounds of formu a I.C, wherein R2 is R2- 9.257( =formula 1.2295).

Table 2296. Compounds of formu a I.C, wherein R2 is R2- 9.258( =formula 1.2296).

Table 2297. Compounds of formu a I.C, wherein R2 is R2- 9.259( =formula 1.2297).

Table 2298. Compounds of formu a I.C, wherein R2 is R2- 9.260( =formula 1.2298).

Table 2299. Compounds of formu a I.C, wherein R2 is R2- 9.261 ( =formula 1.2299).

Table 2300. Compounds of formu a I.C, wherein R2 is R2- 9.262( =formula 1.2300).

Table 2301. Compounds of formu a I.C, wherein R2 is R2- 9.263( =formula 1.2301).

Table 2302. Compounds of formu a I.C, wherein R2 is R2- 9.264( =formula 1.2302).

Table 2303. Compounds of formu a I.C, wherein R2 is R2- 9.265 (=formula 1.2303)

Table 2304. Compounds of formu a I.C, wherein R2 is R2- 9.266 (=formula 1.2304)

Table 2305. Compounds of formu a I.C, wherein R2 is R2- 9.267( =formula 1.2305).

Table 2306. Compounds of formu a I.C, wherein R2 is R2- 9.268( =formula 1.2306).

Table 2307. Compounds of formu a I.C, wherein R2 is R2- 9.269( =formula 1.2307).

Table 2308. Compounds of formu a I.C, wherein R2 is R2- 9.270 (=formula 1.2308)

Table 2309. Compounds of formu a I.C, wherein R2 is R2- 9.271 ( =formula 1.2309).

Table 2310. Compounds of formu a I.C, wherein R2 is R2- 9.272( =formula 1.2310).

Table 2311. Compounds of formu a I.C, wherein R2 is R2- 9.273 (=formula 1.2311)

Table 2312. Compounds of formu a I.C, wherein R2 is R2- 9.274 (=formula 1.2312)

Table 2313. Compounds of formu a I.C, wherein R2 is R2- 9.275 (=formula 1.2313)

Table 2314. Compounds of formu a I.C, wherein R2 is R2- 9.276 (=formula 1.2314)

Table 2315. Compounds of formu a I.C, wherein R2 is R2- 9.277( =formula 1.2315). Table 2316. Compounds of formu a I.C, wherein R2 is R2- 9.278( =formu a 1.2316).

Table 2317. Compounds of formu a I.C, wherein R2 is R2- 9.279( =formu a 1.2317).

Table 2318. Compounds of formu a I.C, wherein R2 is R2- 9.280( =formu a 1.2318).

Table 2319. Compounds of formu a I.C, wherein R2 is R2- 9.281 ( =formu a 1.2319).

Table 2320. Compounds of formu a I.C, wherein R2 is R2- -9.282< =formu a 1.2320).

Table 2321. Compounds of formu a I.C, wherein R2 is R2- -9.283< =formu a 1.2321).

Table 2322. Compounds of formu a I.C, wherein R2 is R2- 9.284( =formu a 1.2322).

Table 2323. Compounds of formu a I.C, wherein R2 is R2- 9.285( =formu a 1.2323).

Table 2324. Compounds of formu a I.C, wherein R2 is R2- 9.286( =formu a 1.2324).

Table 2325. Compounds of formu a I.C, wherein R2 is R2- 9.287( =formu a 1.2325).

Table 2326. Compounds of formu a I.C, wherein R2 is R2- 9.288( =formu a 1.2326).

Table 2327. Compounds of formu a I.C, wherein R2 is R2- 9.289( =formu a 1.2327).

Table 2328. Compounds of formu a I.C, wherein R2 is R2- 9.290( =formu a 1.2328).

Table 2329. Compounds of formu a I.C, wherein R2 is R2- 9.291 ( =formu a 1.2329).

Table 2330. Compounds of formu a I.C, wherein R2 is R2- 9.292( =formu a 1.2330).

Table 2331. Compounds of formu a I.C, wherein R2 is R2- 9.293( =formu a 1.2331).

Table 2332. Compounds of formu a I.C, wherein R2 is R2- 9.294( =formu a 1.2332).

Table 2333. Compounds of formu a I.C, wherein R2 is R2- 9.295( =formu a 1.2333).

Table 2334. Compounds of formu a I.C, wherein R2 is R2- 9.296( =formu a 1.2334).

Table 2335. Compounds of formu a I.C, wherein R2 is R2- 9.297( =formu a 1.2335).

Table 2336. Compounds of formu a I.C, wherein R2 is R2- 9.298( =formu a 1.2336).

Table 2337. Compounds of formu a I.C, wherein R2 is R2- 9.299( =formu a 1.2337).

Table 2338. Compounds of formu a I.C, wherein R2 is R2- 9.300 (=formula 1.2338).

Table 2339. Compounds of formu a I.C, wherein R2 is R2- 9.301 ( =formu a 1.2339).

Table 2340. Compounds of formu a I.C, wherein R2 is R2- 9.302( =formu a 1.2340).

Table 2341. Compounds of formu a I.C, wherein R2 is R2- 9.303( =formu a 1.2341).

Table 2342. Compounds of formu a I.C, wherein R2 is R2- 9.304( =formu a 1.2342).

Table 2343. Compounds of formu a I.C, wherein R2 is R2- 9.305( =formu a 1.2343).

Table 2344. Compounds of formu a I.C, wherein R2 is R2- 9.306( =formu a 1.2344).

Table 2345. Compounds of formu a I.C, wherein R2 is R2- 9.307( =formu a 1.2345).

Table 2346. Compounds of formu a I.C, wherein R2 is R2- 9.308( =formu a 1.2346).

Table 2347. Compounds of formu a I.C, wherein R2 is R2- 9.309( =formu a 1.2347).

Table 2348. Compounds of formu a I.C, wherein R2 is R2- 9.310( =formu a 1.2348).

Table 2349. Compounds of formu a I.C, wherein R2 is R2- 9.311( =formu a 1.2349).

Table 2350. Compounds of formu a I.C, wherein R2 is R2- 9.312( =formu a 1.2350).

Table 2351. Compounds of formu a I.C, wherein R2 is R2- 9.313( =formu a 1.2351).

Table 2352. Compounds of formu a I.C, wherein R2 is R2- 9.314( =formu a 1.2352).

Table 2353. Compounds of formu a I.C, wherein R2 is R2- 9.315( =formu a 1.2353).

Table 2354. Compounds of formu a I.C, wherein R2 is R2- 9.316( =formu a 1.2354).

Table 2355. Compounds of formu a I.C, wherein R2 is R2- 9.317( =formu a 1.2355).

Table 2356. Compounds of formu a I.C, wherein R2 is R2- 9.318( =formu a 1.2356).

Table 2357. Compounds of formu a I.C, wherein R2 is R2- 9.319( =formu a 1.2357).

Table 2358. Compounds of formu a I.C, wherein R2 is R2- 9.320( =formu a 1.2358).

Table 2359. Compounds of formu a I.C, wherein R2 is R2- 9.321 ( =formu a 1.2359). Table 2360. Compounds of formula wherein R 2 s R 2 -9.322(: formula 1.2360) .

Table 2361. Compounds of formula wherein R 2 s R 2 -9.323( : formula 1.2361) .

Table 2362. Compounds of formula wherein R 2 s R 2 -9.324(: formula 1.2362) .

Table 2363. Compounds of formula wherein R 2 s R 2 -9.325( : formula 1.2363) . Table 2364. Compounds of formula wherein R 2 s R 2 -9.326( : formula 1.2364) .

Table 2365. Compounds of formula wherein R 2 s R 2 -9.327(: formula 1.2365) .

Table 2366. Compounds of formula wherein R 2 s R 2 -9.328( : formula 1.2366) .

Table 2367. Compounds of formula wherein R 2 s R 2 -9.329( : formula 1.2367) .

Table 2368. Compounds of formula wherein R 2 s R 2 -9.330( : formula 1.2368) . Table 2369. Compounds of formula wherein R 2 s R 2 -9.331( : formula 1.2369) .

Table 2370. Compounds of formula wherein R 2 s R 2 -9.332(: formula 1.2370) .

Table 2371. Compounds of formula wherein R 2 s R 2 -9.333( : formula 1.2371) .

Table 2372. Compounds of formula wherein R 2 s R 2 -9.334(: formula 1.2372) .

Table 2373. Compounds of formula wherein R 2 s R 2 -9.335( : formula 1.2373) . Table 2374. Compounds of formula wherein R 2 s R 2 -9.336( : formula 1.2374) .

Table 2375. Compounds of formula wherein R 2 s R 2 -9.334(: formula 1.2375) .

Table 2376. Compounds of formula wherein R 2 s R 2 -9.338( : formula 1.2376) .

Table 2377. Compounds of formula wherein R 2 s R 2 -9.339( : formula 1.2377) .

Table 2378. Compounds of formula wherein R 2 s R 2 -9.340( : formula 1.2378) . Table 2379. Compounds of formula wherein R 2 s R 2 -9.341(: formula 1.2379) .

Table 2380. Compounds of formula I.C, wherein R 2 is R 2 -9.342( ; =formula 1.2380) .

Table 2381. Compounds of formula wherein R 2 s R 2 -9.343( : formula 1.2381) .

Table 2382. Compounds of formula wherein R 2 s R 2 -9.344(: formula 1.2382) .

Table 2383. Compounds of formula wherein R 2 s R 2 -9.345( : formula 1.2383) . Table 2384. Compounds of formula wherein R 2 s R 2 -9.346( : formula 1.2384) .

Table 2385. Compounds of formula wherein R 2 s R 2 -9.347(: formula 1.2385) .

Table 2386. Compounds of formula wherein R 2 s R 2 -9.348( : formula 1.2386) .

Table 2387. Compounds of formula wherein R 2 s R 2 -9.349( : formula 1.2387) .

Table 2388. Compounds of formula wherein R 2 s R 2 -9.350( : formula 1.2388) . Table 2389. Compounds of formula wherein R 2 s R 2 -9.351( : formula 1.2389) .

Table 2390. Compounds of formula I.C, wherein R 2 is R 2 -9.352( ; =formula 1.2390) .

Table 2391. Compounds of formula .C, wherein R 2 is R 2 -9.353( ; formula 1.2391) .

Table 2392. Compounds of formula .C, wherein R 2 is R 2 -9.354( ; formula 1.2392) .

Table 2393. Compounds of formula .C, wherein R 2 is R 2 -9.355( ; formula 1.2393) . Table 2394. Compounds of formula .C, wherein R 2 is R 2 -9.356( ; formula 1.2394) .

Table 2395. Compounds of formula .C, wherein R 2 is R 2 -9.357( ; formula 1.2395) .

Table 2396. Compounds of formula .C, wherein R 2 is R 2 -9.358( ; formula 1.2396) .

Table 2397. Compounds of formula .C, wherein R 2 is R 2 -9.359( ; formula 1.2397) .

Table 2398. Compounds of formula .C, wherein R 2 is R 2 -9.360( ; formula 1.2398) . Table 2399. Compounds of formula .C, wherein R 2 is R 2 -9.361( ; formula 1.2399) .

Table 2400. Compounds of formula I.C, wherein R 2 is R 2 -9.362( ; =formula 1.2400) .

Table 2401. Compounds of formula .C, wherein R 2 is R 2 -9.363( formula 1.2401) .

Table 2402. Compounds of formula .C, wherein R 2 is R 2 -9.364( formula 1.2402) .

Table 2403. Compounds of formula .C, wherein R 2 is R 2 -9.365( formula 1.2403) . Table 2404. Compounds of formu a I.C, wherein R2 is R2- 9.366( =formu a 1.2404)

Table 2405. Compounds of formu a I.C, wherein R2 is R2- 9.367( =formu a 1.2405)

Table 2406. Compounds of formu a I.C, wherein R2 is R2- 9.368( =formu a 1.2406)

Table 2407. Compounds of formu a I.C, wherein R2 is R2- 9.369( =formu a 1.2407)

Table 2408. Compounds of formu a I.C, wherein R2 is R2- 9.370( =formu a 1.2408)

Table 2409. Compounds of formu a I.C, wherein R2 is R2- 9.371 ( =formu a 1.2409)

Table 2410. Compounds of formu a I.C, wherein R2 is R2- -9.372< =formu a 1.2410)

Table 2411. Compounds of formu a I.C, wherein R2 is R2- -9.373< =formu a 1.2411)

Table 2412. Compounds of formu a I.C, wherein R2 is R2- 9.374( =formu a 1.2412)

Table 2413. Compounds of formu a I.C, wherein R2 is R2- 9.375( =formu a 1.2413)

Table 2414. Compounds of formu a I.C, wherein R2 is R2- 9.376( =formu a 1.2414)

Table 2415. Compounds of formu a I.C, wherein R2 is R2- 9.377( =formu a 1.2415)

Table 2416. Compounds of formu a I.C, wherein R2 is R2- 9.378( =formu a 1.2416)

Table 2417. Compounds of formu a I.C, wherein R2 is R2- 9.379( =formu a 1.2417)

Table 2418. Compounds of formu a I.C, wherein R2 is R2- 9.380( =formu a 1.2418)

Table 2419. Compounds of formu a I.C, wherein R2 is R2- 9.381 ( =formu a 1.2419)

Table 2420. Compounds of formu a I.C, wherein R2 is R2- 9.382( =formu a 1.2420)

Table 2421. Compounds of formu a I.C, wherein R2 is R2- 9.383( =formu a 1.2421)

Table 2422. Compounds of formu a I.C, wherein R2 is R2- 9.384( =formu a 1.2422)

Table 2423. Compounds of formu a I.C, wherein R2 is R2- 9.385( =formu a 1.2423)

Table 2424. Compounds of formu a I.C, wherein R2 is R2- 9.386( =formu a 1.2424)

Table 2425. Compounds of formu a I.C, wherein R2 is R2- 9.387( =formu a 1.2425)

Table 2426. Compounds of formu a I.C, wherein R2 is R2- 9.388( =formu a 1.2426)

Table 2427. Compounds of formu a I.C, wherein R2 is R2- 9.389( =formu a 1.2427)

Table 2428. Compounds of formu a I.C, wherein R2 is R2- 9.390( =formu a 1.2428)

Table 2429. Compounds of formu a I.C, wherein R2 is R2- 9.391 ( =formu a 1.2429)

Table 2430. Compounds of formula I.C, wherein R2 is R2-9.392(=formula 1.2430

Table 2431. Compounds of formu a I.C, wherein R2 is R2- 9.393( =formu a 1.2431)

Table 2432. Compounds of formu a I.C, wherein R2 is R2- 9.394( =formu a 1.2432)

Table 2433. Compounds of formu a I.C, wherein R2 is R2- 9.395( =formu a 1.2433)

Table 2434. Compounds of formu a I.C, wherein R2 is R2- 9.396( =formu a 1.2434)

Table 2435. Compounds of formu a I.C, wherein R2 is R2- 9.397( =formu a 1.2435)

Table 2436. Compounds of formu a I.C, wherein R2 is R2- 9.398( =formu a 1.2436)

Table 2437. Compounds of formu a I.C, wherein R2 is R2- 9.399( =formu a 1.2437)

Table 2438. Compounds of formu a I.C, wherein R2 is R2- 9.400( =formu a 1.2438)

Table 2439. Compounds of formu a I.C, wherein R2 is R2- 9.401 ( =formu a 1.2439)

Table 2440. Compounds of formu a I.C, wherein R2 is R2- 9.402( =formu a 1.2440)

Table 2441. Compounds of formu a I.C, wherein R2 is R2- 9.403( =formu a 1.2441)

Table 2442. Compounds of formu a I.C, wherein R2 is R2- 9.404( =formu a 1.2442)

Table 2443. Compounds of formu a I.C, wherein R2 is R2- 9.405( =formu a 1.2443)

Table 2444. Compounds of formu a I.C, wherein R2 is R2- 9.406( =formu a 1.2444)

Table 2445. Compounds of formu a I.C, wherein R2 is R2- 9.407( =formu a 1.2445)

Table 2446. Compounds of formu a I.C, wherein R2 is R2- 9.408( =formu a 1.2446)

Table 2447. Compounds of formu a I.C, wherein R2 is R2- 9.409( =formu a 1.2447) Table 2448. Compounds of formu a wherein R 2 s R 2 -9.410 =formu 1.2448) .

Table 2449. Compounds of formu a wherein R 2 s R 2 -9.41 1 =formu 1.2449) .

Table 2450. Compounds of formu a wherein R 2 s R 2 -9.412 =formu 1.2450) .

Table 2451. Compounds of formu a wherein R 2 s R 2 -9.413 =formu 1.2451 ) .

Table 2452. Compounds of formu a wherein R 2 s R 2 -9.414 =formu 1.2452) .

Table 2453. Compounds of formu a wherein R 2 s R 2 -9.415 =formu 1.2453) .

Table 2454. Compounds of formu a wherein R 2 s R 2 -9.416 =formu 1.2454) .

Table 2455. Compounds of formu a wherein R 2 s R 2 -9.417 =formu 1.2455) .

Table 2456. Compounds of formu a wherein R 2 s R 2 -9.418 =formu 1.2456) .

Table 2457. Compounds of formu a wherein R 2 s R 2 -9.419 =formu 1.2457) .

Table 2458. Compounds of formu a wherein R 2 s R 2 -9.420 =formu 1.2458) .

Table 2459. Compounds of formu a wherein R 2 s R 2 -9.421 =formu 1.2459) .

Table 2460. Compounds of formula I.C, wherein R 2 is R 2 -9.422( -formula 1.2460) .

Table 2461. Compounds of formu a wherein R 2 s R 2 -9.423 =formu 1.2461 ) .

Table 2462. Compounds of formu a wherein R 2 s R 2 -9.424 =formu 1.2462) .

Table 2463. Compounds of formu a wherein R 2 s R 2 -9.425 =formu 1.2463) .

Table 2464. Compounds of formu a wherein R 2 s R 2 -9.426 =formu 1.2464) .

Table 2465. Compounds of formu a wherein R 2 s R 2 -9.427 =formu 1.2465) .

Table 2466. Compounds of formu a wherein R 2 s R 2 -9.428 =formu 1.2466) .

Table 2467. Compounds of formu a wherein R 2 s R 2 -9.429 =formu 1.2467) .

Table 2468. Compounds of formu a wherein R 2 s R 2 -9.430 =formu 1.2468) .

Table 2469. Compounds of formu a wherein R 2 s R 2 -9.431 =formu 1.2469) .

Table 2470. Compounds of formu a wherein R 2 s R 2 -9.432 =formu 1.2470) .

Table 2471. Compounds of formu a wherein R 2 s R 2 -9.433 =formu 1.2471 ) .

Table 2472. Compounds of formu a wherein R 2 s R 2 -9.434 =formu 1.2472) .

Table 2473. Compounds of formu a wherein R 2 s R 2 -9.435 =formu 1.2473) .

Table 2474. Compounds of formu a wherein R 2 s R 2 -9.436 =formu 1.2474) .

Table 2475. Compounds of formu a wherein R 2 s R 2 -9.437 =formu 1.2475) .

Table 2476. Compounds of formu a wherein R 2 s R 2 -9.438 =formu 1.2476) .

Table 2477. Compounds of formu a wherein R 2 s R 2 -9.439 =formu 1.2477) .

Table 2478. Compounds of formu a wherein R 2 s R 2 -9.440 =formu 1.2478) .

Table 2479. Compounds of formu a wherein R 2 s R 2 -9.441 =formu 1.2479) .

Table 2480. Compounds of formu a wherein R 2 s R 2 -9.442 =formu 1.2480) .

Table 2481. Compounds of formu a wherein R 2 s R 2 -9.443 =formu 1.2481 ) .

Table 2482. Compounds of formu a wherein R 2 s R 2 -9.444 =formu 1.2482) .

Table 2483. Compounds of formu a wherein R 2 s R 2 -9.445 =formu 1.2483) .

Table 2484. Compounds of formu a wherein R 2 s R 2 -9.446 =formu 1.2484) .

Table 2485. Compounds of formu a wherein R 2 s R 2 -9.447 =formu 1.2485) .

Table 2486. Compounds of formu a wherein R 2 s R 2 -9.448 =formu 1.2486) .

Table 2487. Compounds of formu a wherein R 2 s R 2 -9.449 =formu 1.2487) .

Table 2488. Compounds of formu a wherein R 2 s R 2 -9.450 =formu 1.2488) .

Table 2489. Compounds of formu a wherein R 2 s R 2 -9.451 =formu 1.2489) .

Table 2490. Compounds of formu a wherein R 2 s R 2 -9.452 =formu 1.2490) .

Table 2491. Compounds of formu a wherein R 2 s R 2 -9.453 =formu 1.2491 ) . Table 2492. Compounds of formu a I.C, wherein R2 is R2- 9.454( =formu a 1.2492)

Table 2493. Compounds of formu a I.C, wherein R2 is R2- 9.455( =formu a 1.2493)

Table 2494. Compounds of formu a I.C, wherein R2 is R2- 9.456( =formu a 1.2494)

Table 2495. Compounds of formu a I.C, wherein R2 is R2- 9.457( =formu a 1.2495)

Table 2496. Compounds of formu a I.C, wherein R2 is R2- 9.458( =formu a 1.2496)

Table 2497. Compounds of formu a I.C, wherein R2 is R2- 9.459( =formu a 1.2497)

Table 2498. Compounds of formu a I.C, wherein R2 is R2- 9.460( =formu a 1.2498)

Table 2499. Compounds of formu a I.C, wherein R2 is R2- 9.461 ( =formu a 1.2499)

Table 2500. Compounds of formu a I.C, wherein R2 is R2- 9.462( =formu a 1.2500)

Table 2501. Compounds of formu a I.C, wherein R2 is R2- 9.463( =formu a 1.2501)

Table 2502. Compounds of formu a I.C, wherein R2 is R2- 9.464( =formu a 1.2502)

Table 2503. Compounds of formu a I.C, wherein R2 is R2- 9.465( =formu a 1.2503)

Table 2504. Compounds of formu a I.C, wherein R2 is R2- 9.466( =formu a 1.2504)

Table 2505. Compounds of formu a I.C, wherein R2 is R2- 9.467( =formu a 1.2505)

Table 2506. Compounds of formu a I.C, wherein R2 is R2- 9.468( =formu a 1.2506)

Table 2507. Compounds of formu a I.C, wherein R2 is R2- 9.469( =formu a 1.2507)

Table 2508. Compounds of formu a I.C, wherein R2 is R2- 9.470( =formu a 1.2508)

Table 2509. Compounds of formu a I.C, wherein R2 is R2- 9.471 ( =formu a 1.2509)

Table 2510. Compounds of formu a I.C, wherein R2 is R2- 9.472( =formu a 1.2510)

Table 2511. Compounds of formu a I.C, wherein R2 is R2- 9.473( =formu a 1.2511)

Table 2512. Compounds of formu a I.C, wherein R2 is R2- 9.474( =formu a 1.2512)

Table 2513. Compounds of formu a I.C, wherein R2 is R2- 9.475( =formu a 1.2513)

Table 2514. Compounds of formu a I.C, wherein R2 is R2- 9.476( =formu a 1.2514)

Table 2515. Compounds of formu a I.C, wherein R2 is R2- 9.477( =formu a 1.2515)

Table 2516. Compounds of formu a I.C, wherein R2 is R2- 9.478( =formu a 1.2516)

Table 2517. Compounds of formu a I.C, wherein R2 is R2- 9.479( =formu a 1.2517)

Table 2518. Compounds of formu a I.C, wherein R2 is R2- 9.480( =formu a 1.2518)

Table 2519. Compounds of formu a I.C, wherein R2 is R2- 9.481 ( =formu a 1.2519)

Table 2520. Compounds of formu a I.C, wherein R2 is R2- 9.482( =formu a 1.2520)

Table 2521. Compounds of formu a I.C, wherein R2 is R2- 9.483( =formu a 1.2521)

Table 2522. Compounds of formu a I.C, wherein R2 is R2- 9.484( =formu a 1.2522)

Table 2523. Compounds of formu a I.C, wherein R2 is R2- 9.485( =formu a 1.2523)

Table 2524. Compounds of formu a I.C, wherein R2 is R2- 9.486( =formu a 1.2521)

Table 2525. Compounds of formu a I.C, wherein R2 is R2- 9.487( =formu a 1.2525)

Table 2526. Compounds of formu a I.C, wherein R2 is R2- 9.488( =formu a 1.2526)

Table 2527. Compounds of formu a I.C, wherein R2 is R2- 9.489( =formu a 1.2527)

Table 2528. Compounds of formu a I.C, wherein R2 is R2- 9.490( =formu a 1.2528)

Table 2529. Compounds of formu a I.C, wherein R2 is R2- 9.491 ( =formu a 1.2529)

Table 2530. Compounds of formu a I.C, wherein R2 is R2- 9.492 (=formula 1.2530)

Table 2531. Compounds of formu a I.C, wherein R2 is R2- 9.493( =formu a 1.2531)

Table 2532. Compounds of formu a I.C, wherein R2 is R2- 9.494( =formu a 1.2532)

Table 2533. Compounds of formu a I.C, wherein R2 is R2- 9.495( =formu a 1.2533)

Table 2534. Compounds of formu a I.C, wherein R2 is R2- 9.496( =formu a 1.2534)

Table 2535. Compounds of formu a I.C, wherein R2 is R2- 9.497( =formu a 1.2535) Table 2536. Compounds of formu a I.C, wherein R2 is R2- 9.498( =formula 1.2536).

Table 2537. Compounds of formu a I.C, wherein R2 is R2- 9.499( =formula 1.2537).

Table 2538. Compounds of formu a I.C, wherein R2 is R2- 9.500( =formula 1.2538).

Table 2539. Compounds of formu a I.C, wherein R2 is R2- 9.501 ( =formula 1.2539).

Table 2540. Compounds of formu a I.C, wherein R2 is R2- 9.502( =formula 1.2540).

Table 2541. Compounds of formu a I.C, wherein R2 is R2- 9.503( =formula 1.2541).

Table 2542. Compounds of formu a I.C, wherein R2 is R2- 9.504( =formula 1.2542).

Table 2543. Compounds of formu a I.C, wherein R2 is R2- 9.505( =formula 1.2543).

Table 2544. Compounds of formu a I.C, wherein R2 is R2- 9.506( =formula 1.2544).

Table 2545. Compounds of formu a I.C, wherein R2 is R2- 9.507( =formula 1.2545).

Table 2546. Compounds of formu a I.C, wherein R2 is R2- 9.508( =formula 1.2546).

Table 2547. Compounds of formu a I.C, wherein R2 is R2- 9.509( =formula 1.2547).

Table 2548. Compounds of formu a I.C, wherein R2 is R2- 9.510( =formula 1.2548).

Table 2549. Compounds of formu a I.C, wherein R2 is R2- 9.511( =formula 1.2549).

Table 2550. Compounds of formu a I.C, wherein R2 is R2- 9.512 (=formula 1.2550)

Table 2551. Compounds of formu a I.C, wherein R2 is R2- 9.513 (=formula 1.2551)

Table 2552. Compounds of formu a I.C, wherein R2 is R2- 9.514( =formula 1.2552).

Table 2553. Compounds of formu a I.C, wherein R2 is R2- 9.515( =formula 1.2553).

Table 2554. Compounds of formu a I.C, wherein R2 is R2- 9.516( =formula 1.2554).

Table 2555. Compounds of formu a I.C, wherein R2 is R2- 9.517( =formula 1.2555).

Table 2556. Compounds of formu a I.C, wherein R2 is R2- 9.518( =formula 1.2556).

Table 2557. Compounds of formu a I.C, wherein R2 is R2- 9.519( =formula 1.2557).

Table 2558. Compounds of formu a I.C, wherein R2 is R2- 9.520( =formula 1.2558).

Table 2559. Compounds of formu a I.C, wherein R2 is R2- 9.521 ( =formula 1.2559).

Table 2560. Compounds of formu a I.C, wherein R2 is R2- 9.522( =formula 1.2560).

Table 2561. Compounds of formu a I.C, wherein R2 is R2- 9.523( =formula 1.2561).

Table 2562. Compounds of formu a I.C, wherein R2 is R2- 9.524( =formula 1.2562).

Table 2563. Compounds of formu a I.C, wherein R2 is R2- 9.525( =formula 1.2563).

Table 2564. Compounds of formu a I.C, wherein R2 is R2- 9.526( =formula 1.2564).

Table 2565. Compounds of formu a I.C, wherein R2 is R2- 9.527( =formula 1.2565).

Table 2566. Compounds of formu a I.C, wherein R2 is R2- 9.528( =formula 1.2566).

Table 2567. Compounds of formu a I.C, wherein R2 is R2- 9.529( =formula 1.2567).

Table 2568. Compounds of formu a I.C, wherein R2 is R2- 9.530( =formula 1.2568).

Table 2569. Compounds of formu a I.C, wherein R2 is R2- 9.531 ( =formula 1.2569).

Table 2570. Compounds of formu a I.C, wherein R2 is R2- 9.532( =formula 1.2570).

Table 2571. Compounds of formu a I.C, wherein R2 is R2- 9.533( =formula 1.2571).

Table 2572. Compounds of formu a I.C, wherein R2 is R2- 9.534( =formula 1.2572).

Table 2573. Compounds of formu a I.C, wherein R2 is R2- 9.535( =formula 1.2573).

Table 2574. Compounds of formu a I.C, wherein R2 is R2- 9.536( =formula 1.2574).

Table 2575. Compounds of formu a I.C, wherein R2 is R2- 9.537( =formula 1.2575).

Table 2576. Compounds of formu a I.C, wherein R2 is R2- 9.538( =formula 1.2576).

Table 2577. Compounds of formu a I.C, wherein R2 is R2- 9.539( =formula 1.2577).

Table 2578. Compounds of formu a I.C, wherein R2 is R2- 9.540( =formula 1.2578).

Table 2579. Compounds of formu a I.C, wherein R2 is R2- 9.541 ( =formula 1.2579). Table 2580. Compounds of formu a I.C, wherein R2 is R2- 9.542( =formu a 1.2580).

Table 2581. Compounds of formu a I.C, wherein R2 is R2- 9.543( =formu a 1.2581).

Table 2582. Compounds of formu a I.C, wherein R2 is R2- 9.544( =formu a 1.2582).

Table 2583. Compounds of formu a I.C, wherein R2 is R2- 9.545( =formu a 1.2583).

Table 2584. Compounds of formu a I.C, wherein R2 is R2- 9.546( =formu a 1.2584).

Table 2585. Compounds of formu a I.C, wherein R2 is R2- 9.547( =formu a 1.2585).

Table 2586. Compounds of formu a I.C, wherein R2 is R2- 9.548( =formu a 1.2586).

Table 2587. Compounds of formu a I.C, wherein R2 is R2- 9.549( =formu a 1.2587).

Table 2588. Compounds of formu a I.C, wherein R2 is R2- 9.550( =formu a 1.2588).

Table 2589. Compounds of formu a I.C, wherein R2 is R2- 9.551 ( =formu a 1.2589).

Table 2590. Compounds of formu a I.C, wherein R2 is R2- 9.552( =formu a 1.2590).

Table 2591. Compounds of formu a I.C, wherein R2 is R2- 9.553( =formu a 1.2591).

Table 2592. Compounds of formu a I.C, wherein R2 is R2- 9.554( =formu a 1.2592).

Table 2593. Compounds of formu a I.C, wherein R2 is R2- 9.555( =formu a 1.2593).

Table 2594. Compounds of formu a I.C, wherein R2 is R2- 9.556( =formu a 1.2594).

Table 2595. Compounds of formu a I.C, wherein R2 is R2- 9.557( =formu a 1.2595).

Table 2596. Compounds of formu a I.C, wherein R2 is R2- 9.558( =formu a 1.2596).

Table 2597. Compounds of formu a I.C, wherein R2 is R2- 9.559( =formu a 1.2597).

Table 2598. Compounds of formu a I.C, wherein R2 is R2- 9.560 (=formula 1.2598)

Table 2599. Compounds of formu a I.C, wherein R2 is R2- 9.561 ( =formu a 1.2599).

Table 2600. Compounds of formu a I.C, wherein R2 is R2- 9.562( =formu a 1.2600).

Table 2601. Compounds of formu a I.C, wherein R2 is R2- 9.563( =formu a 1.2601).

Table 2602. Compounds of formu a I.C, wherein R2 is R2- 9.564( =formu a 1.2602).

Table 2603. Compounds of formu a I.C, wherein R2 is R2- 9.565( =formu a 1.2603).

Table 2604. Compounds of formu a I.C, wherein R2 is R2- 9.566( =formu a 1.2604).

Table 2605. Compounds of formu a I.C, wherein R2 is R2- 9.567( =formu a 1.2605).

Table 2606. Compounds of formu a I.C, wherein R2 is R2- 9.568( =formu a 1.2606).

Table 2607. Compounds of formu a I.C, wherein R2 is R2- 9.569( =formu a 1.2607).

Table 2608. Compounds of formu a I.C, wherein R2 is R2- 9.570( =formu a 1.2608).

Table 2609. Compounds of formu a I.C, wherein R2 is R2- 9.571 ( =formu a 1.2609).

Table 2610. Compounds of formu a I.C, wherein R2 is R2- 9.572( =formu a 1.2610).

Table 2611. Compounds of formu a I.C, wherein R2 is R2- 9.573( =formu a 1.2611).

Table 2612. Compounds of formu a I.C, wherein R2 is R2- 9.574( =formu a 1.2612).

Table 2613. Compounds of formu a I.C, wherein R2 is R2- 9.575( =formu a 1.2613).

Table 2614. Compounds of formu a I.C, wherein R2 is R2- 9.576( =formu a 1.2614).

Table 2615. Compounds of formu a I.C, wherein R2 is R2- 9.577( =formu a 1.2615).

Table 2616. Compounds of formu a I.C, wherein R2 is R2- 9.578( =formu a 1.2616).

Table 2617. Compounds of formu a I.C, wherein R2 is R2- 9.579( =formu a 1.2617).

Table 2618. Compounds of formu a I.C, wherein R2 is R2- 9.580( =formu a 1.2618).

Table 2619. Compounds of formu a I.C, wherein R2 is R2- 9.581 ( =formu a 1.2619).

Table 2620. Compounds of formu a I.C, wherein R2 is R2- 9.582( =formu a 1.2620).

Table 2621. Compounds of formu a I.C, wherein R2 is R2- 9.583( =formu a 1.2621).

Table 2622. Compounds of formu a I.C, wherein R2 is R2- 9.584( =formu a 1.2622).

Table 2623. Compounds of formu a I.C, wherein R2 is R2- 9.585( =formu a 1.2623). Tab e 2624. Compounds o ormu a I.C, wherein R2 is R2-9.586( Formu a 1.2624).

Tab e 2625. Compounds o ormu a I.C, wherein R2 is R2-9.587( = Formu a 1.2625).

Tab e 2626. Compounds o ormu a I.C, wherein R2 is R2-9.588( = Formu a 1.2626).

Tab e 2627. Compounds o ormu a I.C, wherein R2 is R2-9.589( = Formu a 1.2627).

Tab e 2628. Compounds o ormu a I.C, wherein R2 is R2-9.590( = Formu a 1.2628).

Tab e 2629. Compounds o ormu a I.C, wherein R2 is R2-9.591< = Formu a 1.2629).

Tab e 2630. Compounds o ormu a I.C, wherein R2 is R2-9.592( = Formu a 1.2630).

Tab e 2631. Compounds o ormu a I.C, wherein R2 is R2-9.593( = Formu a 1.2631).

Tab e 2632. Compounds o ormu a I.C, wherein R2 is R2-9.594( = Formu a 1.2632).

Tab e 2633. Compounds o ormu a I.C, wherein R2 is R2-9.595( = Formu a 1.2633).

Tab e 2634. Compounds o ormu a I.C, wherein R2 is R2-9.596( = Formu a 1.2634).

Tab e 2635. Compounds o ormu a I.C, wherein R2 is R2-9.597( = Formu a 1.2635).

Tab e 2636. Compounds o ormu a I.C, wherein R2 is R2-9.598( = Formu a 1.2636).

Tab e 2637. Compounds o ormu a I.C, wherein R2 is R2-9.599( = Formu a 1.2637).

Tab e 2638. Compounds o ormu a I.C, wherein R2 is R2-9.600( = Formu a 1.2638).

Tab e 2639. Compounds o ormu a I.C, wherein R2 is R2-9.601< = Formu a 1.2639).

Tab e 2640. Compounds o ormu a I.C, wherein R2 is R2-9.602( = Formu a 1.2640).

Tab e 2641. Compounds o ormu a I.C, wherein R2 is R2-9.603( = Formu a 1.2641).

Tab e 2642. Compounds o ormu a I.C, wherein R2 is R2-9.604( = Formu a 1.2642).

Tab e 2643. Compounds o ormu a I.C, wherein R2 is R2-9.605( = Formu a 1.2643).

Tab e 2644. Compounds o ormu a I.C, wherein R2 is R2-9.606( = Formu a 1.2644).

Tab e 2645. Compounds o ormu a I.C, wherein R2 is R2-9.607( = Formu a 1.2645).

Tab e 2646. Compounds o ormu a I.C, wherein R2 is R2-9.608( = Formu a 1.2646).

Tab e 2647. Compounds o ormu a I.C, wherein R2 is R2-9.609( = Formu a 1.2647).

Tab e 2648. Compounds o ormu a I.C, wherein R2 is R2-9.610( = Formu a 1.2648).

Tab e 2649. Compounds o ormu a I.C, wherein R2 is R2-9.611( = Formu a 1.2649).

Tab e 2650. Compounds o ormu a I.C, wherein R2 is R2-9.612( = Formu a 1.2650).

Tab e 2651. Compounds o ormu a I.C, wherein R2 is R2-9.613( = Formu a 1.2651).

Tab e 2652. Compounds o ormu a I.C, wherein R2 is R2-9.614( = Formu a 1.2652).

Tab e 2653. Compounds o ormu a I.C, wherein R2 is R2-9.615( = Formu a 1.2653).

Tab e 2654. Compounds o ormu a I.C, wherein R2 is R2-9.616( = Formu a 1.2654).

Tab e 2655. Compounds o ormu a I.C, wherein R2 is R2-9.617( = Formu a 1.2655).

Tab e 2656. Compounds o ormu a I.C, wherein R2 is R2-9.618( = Formu a 1.2656).

Tab e 2657. Compounds o ormu a I.C, wherein R2 is R2-9.619( = Formu a 1.2657).

Tab e 2658. Compounds o ormu a I.C, wherein R2 is R2-9.620( = Formu a 1.2658).

Tab e 2659. Compounds o ormu a I.C, wherein R2 is R2-9.621< = Formu a 1.2659).

Tab e 2660. Compounds o ormu a I.C, wherein R2 is R2-9.622( = Formu a 1.2660).

Tab e 2661. Compounds o ormu a I.C, wherein R2 is R2-9.623( = Formu a 1.2661).

Tab e 2662. Compounds o ormu a I.C, wherein R2 is R2-9.624( = Formu a 1.2662).

Tab e 2663. Compounds o ormu a I.C, wherein R2 is R2-9.625( = Formu a 1.2663).

Tab e 2664. Compounds o ormu a I.C, wherein R2 is R2-9.626( = Formu a 1.2664).

Tab e 2665. Compounds o ormu a I.C, wherein R2 is R2-9.627( = Formu a 1.2665).

Tab e 2666. Compounds o ormu a I.C, wherein R2 is R2-9.628( = Formu a 1.2666).

Tab e 2667. Compounds o ormu a I.C, wherein R2 is R2-9.629( = Formu a 1.2667). Tab e 2668. Compounds o ormu a I.C, wherein R2 is R2-9.630( Formu a 1.2668).

Tab e 2669. Compounds o ormu a I.C, wherein R2 is R2-9.631< = Formu a 1.2669).

Tab e 2670. Compounds o ormu a I.C, wherein R2 is R2-9.632( = Formu a 1.2670).

Tab e 2671. Compounds o ormu a I.C, wherein R2 is R2-9.633( = Formu a 1.2671).

Tab e 2672. Compounds o ormu a I.C, wherein R2 is R2-9.634( = Formu a 1.2672).

Tab e 2673. Compounds o ormu a I.C, wherein R2 is R2-9.635( = Formu a 1.2673).

Tab e 2674. Compounds o ormu a I.C, wherein R2 is R2-9.636( = Formu a 1.2674).

Tab e 2675. Compounds o ormu a I.C, wherein R2 is R2-9.637( = Formu a 1.2675).

Tab e 2676. Compounds o ormu a I.C, wherein R2 is R2-9.638( = Formu a 1.2676).

Tab e 2677. Compounds o ormu a I.C, wherein R2 is R2-9.639( = Formu a 1.2677).

Tab e 2678. Compounds o ormu a I.C, wherein R2 is R2-9.640( = Formu a 1.2678).

Tab e 2679. Compounds o ormu a I.C, wherein R2 is R2-9.641< = Formu a 1.2679).

Tab e 2680. Compounds o ormu a I.C, wherein R2 is R2-9.642( = Formu a 1.2680).

Tab e 2681. Compounds o ormu a I.C, wherein R2 is R2-9.643( = Formu a 1.2681).

Tab e 2682. Compounds o ormu a I.C, wherein R2 is R2-9.644( = Formu a 1.2682).

Tab e 2683. Compounds o ormu a I.C, wherein R2 is R2-9.645( = Formu a 1.2683).

Tab e 2684. Compounds o ormu a I.C, wherein R2 is R2-9.646( = Formu a 1.2684).

Tab e 2685. Compounds o ormu a I.C, wherein R2 is R2-9.647( = Formu a 1.2685).

Tab e 2686. Compounds o ormu a I.C, wherein R2 is R2-9.648( = Formu a 1.2686).

Tab e 2687. Compounds o ormu a I.C, wherein R2 is R2-9.649( = Formu a 1.2687).

Tab e 2688. Compounds o ormu a I.C, wherein R2 is R2-9.650( = Formu a 1.2688).

Tab e 2689. Compounds o ormu a I.C, wherein R2 is R2-9.651< = Formu a 1.2689).

Tab e 2690. Compounds o ormu a I.C, wherein R2 is R2-9.652( = Formu a 1.2690).

Tab e 2691. Compounds o ormu a I.C, wherein R2 is R2-9.653( = Formu a 1.2691).

Tab e 2692. Compounds o ormu a I.C, wherein R2 is R2-9.654( = Formu a 1.2692).

Tab e 2693. Compounds o ormu a I.C, wherein R2 is R2-9.655( = Formu a 1.2693).

Tab e 2694. Compounds o ormu a I.C, wherein R2 is R2-9.656( = Formu a 1.2694).

Tab e 2695. Compounds o ormu a I.C, wherein R2 is R2-9.657( = Formu a 1.2695).

Tab e 2696. Compounds o ormu a I.C, wherein R2 is R2-9.658( = Formu a 1.2696).

Tab e 2697. Compounds o ormu a I.C, wherein R2 is R2-9.659( = Formu a 1.2697).

Tab e 2698. Compounds o ormu a I.C, wherein R2 is R2-9.660( = Formu a 1.2698).

Tab e 2699. Compounds o ormu a I.C, wherein R2 is R2-9.661< = Formu a 1.2699).

Tab e 2700. Compounds o ormu a I.C, wherein R2 is R2-9.662( = Formu a 1.2700).

Tab e 2701. Compounds o ormu a I.C, wherein R2 is R2-9.663( = Formu a 1.2701).

Tab e 2702. Compounds o ormu a I.C, wherein R2 is R2-9.664( = Formu a 1.2702).

Tab e 2703. Compounds o ormu a I.C, wherein R2 is R2-9.665( = Formu a 1.2703).

Tab e 2704. Compounds o ormu a I.C, wherein R2 is R2-9.666( = Formu a 1.2704).

Tab e 2705. Compounds o ormu a I.C, wherein R2 is R2-9.667( = Formu a 1.2705).

Tab e 2706. Compounds o ormu a I.C, wherein R2 is R2-9.668( = Formu a 1.2706).

Tab e 2707. Compounds o ormu a I.C, wherein R2 is R2-9.669( = Formu a 1.2707).

Tab e 2708. Compounds o ormu a I.C, wherein R2 is R2-9.670( = Formu a 1.2708).

Tab e 2709. Compounds o ormu a I.C, wherein R2 is R2-9.671< = Formu a 1.2709).

Tab e 2710. Compounds o ormu a I.C, wherein R2 is R2-9.672( = Formu a 1.2710).

Tab e 2711. Compounds o ormu a I.C, wherein R2 is R2-9.673( = Formu a 1.2711). Table 2712. Compounds of formu a I.C, wherein R2 is R2J 3.674(=formula 1.2712).

Table 2713. Compounds of formu a I.C, wherein R2 is R2J 3.675(=formula 1.2713).

Table 2714. Compounds of formu a I.C, wherein R2 is R2J 3.676(=formula 1.2714).

Table 2715. Compounds of formu a I.C, wherein R2 is R2- 10.1 (= formula 1.2715).

Table 2716. Compounds of formu a I.C, wherein R2 is R2- 10.2(= formula 1.2716).

Table 2717. Compounds of formu a I.C, wherein R2 is R2- 10.3(= formula 1.2717).

Table 2718. Compounds of formu a I.C, wherein R2 is R2- 10.4(= formula 1.2718).

Table 2719. Compounds of formu a I.C, wherein R2 is R2- 10.5(= formula 1.2719).

Table 2720. Compounds of formu a I.C, wherein R2 is R2- 10.6(= formula 1.2720).

Table 2721. Compounds of formu a I.C, wherein R2 is R2- 10.7(= formula 1.2721).

Table 2722. Compounds of formu a I.C, wherein R2 is R2- 10.8(= formula 1.2722).

Table 2723. Compounds of formu a I.C, wherein R2 is R2- 10.9(= formula 1.2723).

Table 2724. Compounds of formu a I.C, wherein R2 is R2- 10.101 =formula 1.2724).

Table 2725. Compounds of formu a I.C, wherein R2 is R2- 10.111 =formula 1.2725).

Table 2726. Compounds of formu a I.C, wherein R2 is R2- 10.121 =formula 1.2726).

Table 2727. Compounds of formu a I.C, wherein R2 is R2- 10.131 =formula 1.2727).

Table 2728. Compounds of formu a I.C, wherein R2 is R2- 10.141 =formula 1.2728).

Table 2729. Compounds of formu a I.C, wherein R2 is R2- 10.151 =formula 1.2729).

Table 2730. Compounds of formu a I.C, wherein R2 is R2- 10.161 =formula 1.2730).

Table 2731. Compounds of formu a I.C, wherein R2 is R2- 10.171 =formula 1.2731).

Table 2732. Compounds of formu a I.C, wherein R2 is R2- 10.181 =formula 1.2732).

Table 2733. Compounds of formu a I.C, wherein R2 is R2- 10.191 =formula 1.2733).

Table 2734. Compounds of formu a I.C, wherein R2 is R2- 10.201 =formula 1.2734).

Table 2735. Compounds of formu a I.C, wherein R2 is R2- 10.211 =formula 1.2735).

Table 2736. Compounds of formu a I.C, wherein R2 is R2- 10.221 =formula 1.2736).

Table 2737. Compounds of formu a I.C, wherein R2 is R2- 10.231 =formula 1.2737).

Table 2738. Compounds of formu a I.C, wherein R2 is R2- 10.241 =formula 1.2738).

Table 2739. Compounds of formu a I.C, wherein R2 is R2- 10.251 =formula 1.2739).

Table 2740. Compounds of formu a I.C, wherein R2 is R2- 10.261 =formula 1.2740).

Table 2741. Compounds of formu a I.C, wherein R2 is R2- 10.271 =formula 1.2741).

Table 2742. Compounds of formu a I.C, wherein R2 is R2- 10.281 =formula 1.2742).

Table 2743. Compounds of formu a I.C, wherein R2 is R2- 10.291 =formula 1.2743).

Table 2744. Compounds of formu a I.C, wherein R2 is R2- 10.301 =formula 1.2744).

Table 2745. Compounds of formu a I.C, wherein R2 is R2- 10.311 =formula 1.2745).

Table 2746. Compounds of formu a I.C, wherein R2 is R2- 10.321 =formula 1.2746).

Table 2747. Compounds of formu a I.C, wherein R2 is R2- 10.331 =formula 1.2747).

Table 2748. Compounds of formu a I.C, wherein R2 is R2- 10.341 =formula 1.2748).

Table 2749. Compounds of formu a I.C, wherein R2 is R2- 10.351 =formula 1.2749).

Table 2750. Compounds of formu a I.C, wherein R2 is R2- 10.361 =formula 1.2750).

Table 2751. Compounds of formu a I.C, wherein R2 is R2- 10.371 =formula 1.2751).

Table 2752. Compounds of formu a I.C, wherein R2 is R2- 10.381 =formula 1.2752).

Table 2753. Compounds of formu a I.C, wherein R2 is R2- 10.391 =formula 1.2753).

Table 2754. Compounds of formu a I.C, wherein R2 is R2- 10.401 =formula 1.2754).

Table 2755. Compounds of formu a I.C, wherein R2 is R2- 10.411 =formula 1.2755). Tab e 2756. Compounds o ormu a I.C, wherein R2 is R2-- I 0.42( Formu a 1.2756).

Tab e 2757. Compounds o ormu a I.C, wherein R2 is R2-- I 0.43( = Formu a 1.2757).

Tab e 2758. Compounds o ormu a I.C, wherein R2 is R2-- I 0.44( = Formu a 1.2758).

Tab e 2759. Compounds o ormu a I.C, wherein R2 is R2-- I 0.45( = Formu a 1.2759).

Tab e 2760. Compounds o ormu a I.C, wherein R2 is R2-- I 0.46( = Formu a 1.2760).

Tab e 2761. Compounds o ormu a I.C, wherein R2 is R2-- I 0.47( = Formu a 1.2761 ).

Tab e 2762. Compounds o ormu a I.C, wherein R2 is R2-- I 0.48( = Formu a 1.2762).

Tab e 2763. Compounds o ormu a I.C, wherein R2 is R2-- I 0.49( = Formu a 1.2763).

Tab e 2764. Compounds o ormu a I.C, wherein R2 is R2-- I 0.50( = Formu a 1.2764).

Tab e 2765. Compounds o ormu a I.C, wherein R2 is R2-- I 0.51 ( = Formu a 1.2765).

Tab e 2766. Compounds o ormu a I.C, wherein R2 is R2-- I 0.52( = Formu a 1.2766).

Tab e 2767. Compounds o ormu a I.C, wherein R2 is R2-- I 0.53( = Formu a 1.2767).

Tab e 2768. Compounds o ormu a I.C, wherein R2 is R2-- I 0.54( = Formu a 1.2768).

Tab e 2769. Compounds o ormu a I.C, wherein R2 is R2-- I 0.55( = Formu a 1.2769).

Tab e 2770. Compounds o ormu a I.C, wherein R2 is R2-- I 0.56( = Formu a 1.2770).

Tab e 2771. Compounds o ormu a I.C, wherein R2 is R2-- I 0.57( = Formu a 1.2771 ).

Tab e 2772. Compounds o ormu a I.C, wherein R2 is R2-- I 0.58( = Formu a 1.2772).

Tab e 2773. Compounds o ormu a I.C, wherein R2 is R2-- I 0.59( = Formu a 1.2773).

Tab e 2774. Compounds o ormu a I.C, wherein R2 is R2-- I 0.60( = Formu a 1.2774).

Tab e 2775. Compounds o ormu a I.C, wherein R2 is R2-- I 0.61 ( = Formu a 1.2775).

Tab e 2776. Compounds o ormu a I.C, wherein R2 is R2-- I 0.62( = Formu a 1.2776).

Tab e 2777. Compounds o ormu a I.C, wherein R2 is R2-- I 0.63( = Formu a 1.2777).

Tab e 2778. Compounds o ormu a I.C, wherein R2 is R2-- I 0.64( = Formu a 1.2778).

Tab e 2779. Compounds o ormu a I.C, wherein R2 is R2-- I 0.65( = Formu a 1.2779).

Tab e 2780. Compounds o ormu a I.C, wherein R2 is R2-- I 0.66( = Formu a 1.2780).

Tab e 2781. Compounds o ormu a I.C, wherein R2 is R2-- I 0.67( = Formu a 1.2781 ).

Tab e 2782. Compounds o ormu a I.C, wherein R2 is R2-- I 0.68( = Formu a 1.2782).

Tab e 2783. Compounds o ormu a I.C, wherein R2 is R2-- I 0.69( = Formu a 1.2783).

Tab e 2784. Compounds o ormu a I.C, wherein R2 is R2-- I 0.70( = Formu a 1.2784).

Tab e 2785. Compounds o ormu a I.C, wherein R2 is R2-- I 0.71 ( = Formu a 1.2785).

Tab e 2786. Compounds o ormu a I.C, wherein R2 is R2-- I 0.72( = Formu a 1.2786).

Tab e 2787. Compounds o ormu a I.C, wherein R2 is R2-- I 0.73( = Formu a 1.2787).

Tab e 2788. Compounds o ormu a I.C, wherein R2 is R2-- I 0.74( = Formu a 1.2788).

Tab e 2789. Compounds o ormu a I.C, wherein R2 is R2-- I 0.75( = Formu a 1.2789).

Tab e 2790. Compounds o ormu a I.C, wherein R2 is R2-- I 0.76( = Formu a 1.2790).

Tab e 2791. Compounds o ormu a I.C, wherein R2 is R2-- I 0.77( = Formu a 1.2791 ).

Tab e 2792. Compounds o ormu a I.C, wherein R2 is R2-- I 0.78( = Formu a 1.2792).

Tab e 2793. Compounds o ormu a I.C, wherein R2 is R2-- I 0.79( = Formu a 1.2793).

Tab e 2794. Compounds o ormu a I.C, wherein R2 is R2-- I 0.80( = Formu a 1.2794).

Tab e 2795. Compounds o ormu a I.C, wherein R2 is R2-- I 0.81 ( = Formu a 1.2795).

Tab e 2796. Compounds o ormu a I.C, wherein R2 is R2-- I 0.82( = Formu a 1.2796).

Tab e 2797. Compounds o ormu a I.C, wherein R2 is R2-- I 0.83( = Formu a 1.2797).

Tab e 2798. Compounds o ormu a I.C, wherein R2 is R2-- I 0.84( = Formu a 1.2798).

Tab e 2799. Compounds o ormu a I.C, wherein R2 is R2-- I 0.85( = Formu a 1.2799). Table 2800. Compounds of formu a I.C, wherein R2 is R2 0.86(= formula 1.2800).

Table 2801. Compounds of formu a I.C, wherein R2 is R2 0.87(= formula 1 .2801).

Table 2802. Compounds of formu a I.C, wherein R2 is R2 0.88(= formula 1 .2802).

Table 2803. Compounds of formu a I.C, wherein R2 is R2 0.89(= formula 1 .2803).

Table 2804. Compounds of formu a I.C, wherein R2 is R2 0.90(= formula 1 .2804).

Table 2805. Compounds of formu a I.C, wherein R2 is R2 0.91(= formula 1 .2805).

Table 2806. Compounds of formu a I.C, wherein R2 is R2 0.92(= formula 1 .2806).

Table 2807. Compounds of formu a I.C, wherein R2 is R2 0.93(= formula 1 .2807).

Table 2808. Compounds of formu a I.C, wherein R2 is R2 0.94(= formula 1 .2808).

Table 2809. Compounds of formu a I.C, wherein R2 is R2 0.95(= formula 1 .2809).

Table 2810. Compounds of formu a I.C, wherein R2 is R2 0.96(= formula 1 .2810).

Table 2811. Compounds of formu a I.C, wherein R2 is R2 0.97(= formula 1 .2811).

Table 2812. Compounds of formu a I.C, wherein R2 is R2 0.98(= formula 1 .2812).

Table 2813. Compounds of formu a I.C, wherein R2 is R2 0.99(= formula 1 .2813).

Table 2814. Compounds of formu a I.C, wherein R2 is R2 0.100 [=formula 1.2814).

Table 2815. Compounds of formu a I.C, wherein R2 is R2 0.101 [=formula 1.2815).

Table 2816. Compounds of formu a I.C, wherein R2 is R2 0.102 [=formula 1.2816).

Table 2817. Compounds of formu a I.C, wherein R2 is R2 0.103 [=formula 1.2817).

Table 2818. Compounds of formu a I.C, wherein R2 is R2 0.104 [=formula 1.2818).

Table 2819. Compounds of formu a I.C, wherein R2 is R2 0.105 [=formula 1.2819).

Table 2820. Compounds of formu a I.C, wherein R2 is R2 0.106 [=formula 1.2820).

Table 2821. Compounds of formu a I.C, wherein R2 is R2 0.107 [=formula 1.2821).

Table 2822. Compounds of formu a I.C, wherein R2 is R2 0.108 [=formula 1.2822).

Table 2823. Compounds of formu a I.C, wherein R2 is R2 0.109 [=formula 1.2823).

Table 2824. Compounds of formu a I.C, wherein R2 is R2 0.110 [=formula 1.2824).

Table 2825. Compounds of formu a I.C, wherein R2 is R2 0.111 [=formula 1.2825).

Table 2826. Compounds of formu a I.C, wherein R2 is R2 0.112 [=formula 1.2826).

Table 2827. Compounds of formu a I.C, wherein R2 is R2 0.113 [=formula 1.2827).

Table 2828. Compounds of formu a I.C, wherein R2 is R2 0.114 [=formula 1.2828).

Table 2829. Compounds of formu a I.C, wherein R2 is R2 0.115 [=formula 1.2829).

Table 2830. Compounds of formu a I.C, wherein R2 is R2 0.116 [=formula 1.2830).

Table 2831. Compounds of formu a I.C, wherein R2 is R2 0.117 [=formula 1.2831).

Table 2832. Compounds of formu a I.C, wherein R2 is R2 0.118 [=formula 1.2832).

Table 2833. Compounds of formu a I.C, wherein R2 is R2 0.119 [=formula 1.2833).

Table 2834. Compounds of formu a I.C, wherein R2 is R2 0.120 [=formula 1.2834).

Table 2835. Compounds of formu a I.C, wherein R2 is R2 0.121 [=formula 1.2835).

Table 2836. Compounds of formu a I.C, wherein R2 is R2 0.122 [=formula 1.2836).

Table 2837. Compounds of formu a I.C, wherein R2 is R2 0.123 [=formula 1.2837).

Table 2838. Compounds of formu a I.C, wherein R2 is R2 0.124 [=formula 1.2838).

Table 2839. Compounds of formu a I.C, wherein R2 is R2 0.125 [=formula 1.2839).

Table 2840. Compounds of formu a I.C, wherein R2 is R2 0.126 [=formula 1.2840).

Table 2841. Compounds of formu a I.C, wherein R2 is R2 0.127 [=formula 1.2841).

Table 2842. Compounds of formu a I.C, wherein R2 is R2 0.128 [=formula 1.2842).

Table 2843. Compounds of formu a I.C, wherein R2 is R2 0.129 [=formula 1.2843). Table 2844. Compounds of formu a I.C, wherein R2 is R2-- 10.1301 = Formu a 1 .2844).

Table 2845. Compounds of formu a I.C, wherein R2 is R2-- 10.1311 = Formu a 1 .2845).

Table 2846. Compounds of formu a I.C, wherein R2 is R2-- 10.1321 = Formu a 1 .2846).

Table 2847. Compounds of formu a I.C, wherein R2 is R2-- 10.1331 = Formu a 1 .2847).

Table 2848. Compounds of formu a I.C, wherein R2 is R2-- 10.1341 = Formu a 1 .2848).

Table 2849. Compounds of formu a I.C, wherein R2 is R2-- 10.1351 = Formu a 1 .2849).

Table 2850. Compounds of formu a I.C, wherein R2 is R2-- 10.1361 = Formu a 1 .2850).

Table 2851. Compounds of formu a I.C, wherein R2 is R2-- 10.1371 = Formu a 1 .2851 ).

Table 2852. Compounds of formu a I.C, wherein R2 is R2-- 10.1381 = Formu a 1 .2852).

Table 2853. Compounds of formu a I.C, wherein R2 is R2-- 10.1391 = Formu a 1 .2853).

Table 2854. Compounds of formu a I.C, wherein R2 is R2-- 10.1401 = Formu a 1 .2854).

Table 2855. Compounds of formu a I.C, wherein R2 is R2-- 10.1411 = Formu a 1 .2855).

Table 2856. Compounds of formu a I.C, wherein R2 is R2-- 10.1421 = Formu a 1 .2856).

Table 2857. Compounds of formu a I.C, wherein R2 is R2-- 10.1431 = Formu a 1 .2857).

Table 2858. Compounds of formu a I.C, wherein R2 is R2-- 10.1441 = Formu a 1 .2858).

Table 2859. Compounds of formu a I.C, wherein R2 is R2-- 10.1451 = Formu a 1 .2859).

Table 2860. Compounds of formu a I.C, wherein R2 is R2-- 10.1461 = Formu a 1 .2860).

Table 2861. Compounds of formu a I.C, wherein R2 is R2-- 10.1471 = Formu a 1 .2861 ).

Table 2862. Compounds of formu a I.C, wherein R2 is R2-- 10.1481 = Formu a 1 .2862).

Table 2863. Compounds of formu a I.C, wherein R2 is R2-- 10.1491 = Formu a 1 .2863).

Table 2864. Compounds of formu a I.C, wherein R2 is R2-- 10.1501 = Formu a 1 .2864).

Table 2865. Compounds of formu a I.C, wherein R2 is R2-- 10.1511 = Formu a 1 .2865).

Table 2866. Compounds of formu a I.C, wherein R2 is R2-- 10.1521 = Formu a 1 .2866).

Table 2867. Compounds of formu a I.C, wherein R2 is R2-- 10.1531 = Formu a 1 .2867).

Table 2868. Compounds of formu a I.C, wherein R2 is R2-- 10.1541 = Formu a 1 .2868).

Table 2869. Compounds of formu a I.C, wherein R2 is R2-- 10.1551 = Formu a 1 .2869).

Table 2870. Compounds of formu a I.C, wherein R2 is R2-- 10.1561 = Formu a 1 .2870).

Table 2871. Compounds of formu a I.C, wherein R2 is R2-- 10.1571 = Formu a 1 .2871 ).

Table 2872. Compounds of formu a I.C, wherein R2 is R2-- 10.1581 = Formu a 1 .2872).

Table 2873. Compounds of formu a I.C, wherein R2 is R2-- 10.1591 = Formu a 1 .2873).

Table 2874. Compounds of formu a I.C, wherein R2 is R2-- 10.1601 = Formu a 1 .2874).

Table 2875. Compounds of formu a I.C, wherein R2 is R2-- 10.1611 = Formu a 1 .2875).

Table 2876. Compounds of formu a I.C, wherein R2 is R2-- 10.1621 = Formu a 1 .2876).

Table 2877. Compounds of formu a I.C, wherein R2 is R2-- 10.1631 = Formu a 1 .2877).

Table 2878. Compounds of formu a I.C, wherein R2 is R2-- 10.1641 = Formu a 1 .2878).

Table 2879. Compounds of formu a I.C, wherein R2 is R2-- 10.1651 = Formu a 1 .2879).

Table 2880. Compounds of formu a I.C, wherein R2 is R2-- 10.1661 = Formu a 1 .2880).

Table 2881. Compounds of formu a I.C, wherein R2 is R2-- 10.1671 = Formu a 1 .2881 ).

Table 2882. Compounds of formu a I.C, wherein R2 is R2-- 10.1681 = Formu a 1 .2882).

Table 2883. Compounds of formu a I.C, wherein R2 is R2-- 10.1691 = Formu a 1 .2883).

Table 2884. Compounds of formu a I.C, wherein R2 is R2-- 10.1701 = Formu a 1 .2884).

Table 2885. Compounds of formu a I.C, wherein R2 is R2-- 10.1711 = Formu a 1 .2885).

Table 2886. Compounds of formu a I.C, wherein R2 is R2-- 10.1721 = Formu a 1 .2886).

Table 2887. Compounds of formu a I.C, wherein R2 is R2-- 10.1731 = Formu a 1 .2887). Table 2888. Compounds of formu a I.C, wherein R2 is R2-- 10.1741 = Formu a 1 .2888).

Table 2889. Compounds of formu a I.C, wherein R2 is R2-- 10.1751 = Formu a 1 .2889).

Table 2890. Compounds of formu a I.C, wherein R2 is R2-- 10.1761 = Formu a 1 .2890).

Table 2891. Compounds of formu a I.C, wherein R2 is R2-- 10.1771 = Formu a 1 .2891 ).

Table 2892. Compounds of formu a I.C, wherein R2 is R2-- 10.1781 = Formu a 1 .2892).

Table 2893. Compounds of formu a I.C, wherein R2 is R2-- 10.1791 = Formu a 1 .2893).

Table 2894. Compounds of formu a I.C, wherein R2 is R2-- 10.1801 = Formu a 1 .2894).

Table 2895. Compounds of formu a I.C, wherein R2 is R2-- 10.1811 = Formu a 1 .2895).

Table 2896. Compounds of formu a I.C, wherein R2 is R2-- 10.1821 = Formu a 1 .2896).

Table 2897. Compounds of formu a I.C, wherein R2 is R2-- 10.1831 = Formu a 1 .2897).

Table 2898. Compounds of formu a I.C, wherein R2 is R2-- 10.1841 = Formu a 1 .2898).

Table 2899. Compounds of formu a I.C, wherein R2 is R2-- 10.1851 = Formu a 1 .2899).

Table 2900. Compounds of formu a I.C, wherein R2 is R2-- 10.1861 = Formu a 1 .2900).

Table 2901. Compounds of formu a I.C, wherein R2 is R2-- 10.1871 = Formu a 1 .2901 ).

Table 2902. Compounds of formu a I.C, wherein R2 is R2-- 10.1881 = Formu a 1 .2902).

Table 2903. Compounds of formu a I.C, wherein R2 is R2-- 10.1891 = Formu a 1 .2903).

Table 2904. Compounds of formu a I.C, wherein R2 is R2-- 10.1901 = Formu a 1 .2904).

Table 2905. Compounds of formu a I.C, wherein R2 is R2-- 10.1911 = Formu a 1 .2905).

Table 2906. Compounds of formu a I.C, wherein R2 is R2-- 10.1921 = Formu a 1 .2906).

Table 2907. Compounds of formu a I.C, wherein R2 is R2-- 10.1931 = Formu a 1 .2907).

Table 2908. Compounds of formu a I.C, wherein R2 is R2-- 10.1941 = Formu a 1 .2908).

Table 2909. Compounds of formu a I.C, wherein R2 is R2-- 10.1951 = Formu a 1 .2909).

Table 2910. Compounds of formu a I.C, wherein R2 is R2-- 10.1961 = Formu a 1 .2910).

Table 291 1. Compounds of formu a I.C, wherein R2 is R2-- 10.1971 = Formu a 1 .291 1 ).

Table 2912. Compounds of formu a I.C, wherein R2 is R2-- 10.1981 = Formu a 1 .2912).

Table 2913. Compounds of formu a I.C, wherein R2 is R2-- 10.1991 = Formu a 1 .2913).

Table 2914. Compounds of formu a I.C, wherein R2 is R2-- 10.2001 = Formu a 1 .2914).

Table 2915. Compounds of formu a I.C, wherein R2 is R2-- 10.2011 = Formu a 1 .2915).

Table 2916. Compounds of formu a I.C, wherein R2 is R2-- 10.2021 = Formu a 1 .2916).

Table 2917. Compounds of formu a I.C, wherein R2 is R2-- 10.2031 = Formu a 1 .2917).

Table 2918. Compounds of formu a I.C, wherein R2 is R2-- 10.2041 = Formu a 1 .2918).

Table 2919. Compounds of formu a I.C, wherein R2 is R2-- 10.2051 = Formu a 1 .2919).

Table 2920. Compounds of formu a I.C, wherein R2 is R2-- 10.2061 = Formu a 1 .2920).

Table 2921. Compounds of formu a I.C, wherein R2 is R2-- 10.2071 = Formu a 1 .2921 ).

Table 2922. Compounds of formu a I.C, wherein R2 is R2-- 10.2081 = Formu a 1 .2922).

Table 2923. Compounds of formu a I.C, wherein R2 is R2-- 10.2091 = Formu a 1 .2923).

Table 2924. Compounds of formu a I.C, wherein R2 is R2-- 10.2101 = Formu a 1 .2924).

Table 2925. Compounds of formu a I.C, wherein R2 is R2-- 10.21 11 = Formu a 1 .2925).

Table 2926. Compounds of formu a I.C, wherein R2 is R2-- 10.2121 = Formu a 1 .2926).

Table 2927. Compounds of formu a I.C, wherein R2 is R2-- 10.2131 = Formu a 1 .2927).

Table 2928. Compounds of formu a I.C, wherein R2 is R2-- 10.2141 = Formu a 1 .2928).

Table 2929. Compounds of formu a I.C, wherein R2 is R2-- 10.2151 = Formu a 1 .2929).

Table 2930. Compounds of formu a I.C, wherein R2 is R2-- 10.2161 = Formu a 1 .2930).

Table 2931. Compounds of formu a I.C, wherein R2 is R2-- 10.2171 = Formu a 1 .2931 ). Table 2932. Compounds of formu a I.C, wherein R2 is R2-- 10.2181 = Formu a 1 .2932).

Table 2933. Compounds of formu a I.C, wherein R2 is R2-- 10.2191 = Formu a 1 .2933).

Table 2934. Compounds of formu a I.C, wherein R2 is R2-- 10.2201 = Formu a 1 .2934).

Table 2935. Compounds of formu a I.C, wherein R2 is R2-- 10.2211 = Formu a 1 .2935).

Table 2936. Compounds of formu a I.C, wherein R2 is R2-- 10.2221 = Formu a 1 .2936).

Table 2937. Compounds of formu a I.C, wherein R2 is R2-- 10.2231 = Formu a 1 .2937).

Table 2938. Compounds of formu a I.C, wherein R2 is R2-- 10.2241 = Formu a 1 .2938).

Table 2939. Compounds of formu a I.C, wherein R2 is R2-- 10.2251 = Formu a 1 .2939).

Table 2940. Compounds of formu a I.C, wherein R2 is R2-- 10.2261 = Formu a 1 .2940).

Table 2941. Compounds of formu a I.C, wherein R2 is R2-- 10.2271 = Formu a 1 .2941 ).

Table 2942. Compounds of formu a I.C, wherein R2 is R2-- 10.2281 = Formu a 1 .2942).

Table 2943. Compounds of formu a I.C, wherein R2 is R2-- 10.2291 = Formu a 1 .2943).

Table 2944. Compounds of formu a I.C, wherein R2 is R2-- 10.2301 = Formu a 1 .2944).

Table 2945. Compounds of formu a I.C, wherein R2 is R2-- 10.2311 = Formu a 1 .2945).

Table 2946. Compounds of formu a I.C, wherein R2 is R2-- 10.2321 = Formu a 1 .2946).

Table 2947. Compounds of formu a I.C, wherein R2 is R2-- 10.2331 = Formu a 1 .2947).

Table 2948. Compounds of formu a I.C, wherein R2 is R2-- 10.2341 = Formu a 1 .2948).

Table 2949. Compounds of formu a I.C, wherein R2 is R2-- 10.2351 = Formu a 1 .2949).

Table 2950. Compounds of formu a I.C, wherein R2 is R2-- 10.2361 = Formu a 1 .2950).

Table 2951. Compounds of formu a I.C, wherein R2 is R2-- 10.2371 = Formu a 1 .2951 ).

Table 2952. Compounds of formu a I.C, wherein R2 is R2-- 10.2381 = Formu a 1 .2952).

Table 2953. Compounds of formu a I.C, wherein R2 is R2-- 10.2391 = Formu a 1 .2953).

Table 2954. Compounds of formu a I.C, wherein R2 is R2-- 10.2401 = Formu a 1 .2954).

Table 2955. Compounds of formu a I.C, wherein R2 is R2-- 10.2411 = Formu a 1 .2955).

Table 2956. Compounds of formu a I.C, wherein R2 is R2-- 10.2421 = Formu a 1 .2956).

Table 2957. Compounds of formu a I.C, wherein R2 is R2-- 10.2431 = Formu a 1 .2957).

Table 2958. Compounds of formu a I.C, wherein R2 is R2-- 10.2441 = Formu a 1 .2958).

Table 2959. Compounds of formu a I.C, wherein R2 is R2-- 10.2451 = Formu a 1 .2959).

Table 2960. Compounds of formu a I.C, wherein R2 is R2-- 10.2461 = Formu a 1 .2960).

Table 2961. Compounds of formu a I.C, wherein R2 is R2-- 10.2471 = Formu a 1 .2961 ).

Table 2962. Compounds of formu a I.C, wherein R2 is R2-- 10.2481 = Formu a 1 .2962).

Table 2963. Compounds of formu a I.C, wherein R2 is R2-- 10.2491 = Formu a 1 .2963).

Table 2964. Compounds of formu a I.C, wherein R2 is R2-- 10.2501 = Formu a 1 .2964).

Table 2965. Compounds of formu a I.C, wherein R2 is R2-- 10.2511 = Formu a 1 .2965).

Table 2966. Compounds of formu a I.C, wherein R2 is R2-- 10.2521 = Formu a 1 .2966).

Table 2967. Compounds of formu a I.C, wherein R2 is R2-- 10.2531 = Formu a 1 .2967).

Table 2968. Compounds of formu a I.C, wherein R2 is R2-- 10.2541 = Formu a 1 .2968).

Table 2969. Compounds of formu a I.C, wherein R2 is R2-- 10.2551 = Formu a 1 .2969).

Table 2970. Compounds of formu a I.C, wherein R2 is R2-- 10.2561 = Formu a 1 .2970).

Table 2971. Compounds of formu a I.C, wherein R2 is R2-- 10.2571 = Formu a 1 .2971 ).

Table 2972. Compounds of formu a I.C, wherein R2 is R2-- 10.2581 = Formu a 1 .2972).

Table 2973. Compounds of formu a I.C, wherein R2 is R2-- 10.2591 = Formu a 1 .2973).

Table 2974. Compounds of formu a I.C, wherein R2 is R2-- 10.2601 = Formu a 1 .2974).

Table 2975. Compounds of formu a I.C, wherein R2 is R2-- 10.2611 = Formu a 1 .2975). Table 2976. Compounds of formu a I.C, wherein R2 is R2-- I 0.262I = Formu a 1 .2976).

Table 2977. Compounds of formu a I.C, wherein R2 is R2-- I 0.263I = Formu a 1 .2977).

Table 2978. Compounds of formu a I.C, wherein R2 is R2-- I 0.264I = Formu a 1 .2978).

Table 2979. Compounds of formu a I.C, wherein R2 is R2-- I 0.265I = Formu a 1 .2979).

Table 2980. Compounds of formu a I.C, wherein R2 is R2-- I 0.266I = Formu a 1 .2980).

Table 2981. Compounds of formu a I.C, wherein R2 is R2-- I 0.267I = Formu a 1 .2981 ).

Table 2982. Compounds of formu a I.C, wherein R2 is R2-- I 0.268I = Formu a 1 .2982).

Table 2983. Compounds of formu a I.C, wherein R2 is R2-- I 0.269I = Formu a 1 .2983).

Table 2984. Compounds of formu a I.C, wherein R2 is R2-- I 0.270I = Formu a 1 .2984).

Table 2985. Compounds of formu a I.C, wherein R2 is R2-- 10.2711 = Formu a 1 .2985).

Table 2986. Compounds of formu a I.C, wherein R2 is R2-- 10.2721 = Formu a 1 .2986).

Table 2987. Compounds of formu a I.C, wherein R2 is R2-- 10.2731 = Formu a 1 .2987).

Table 2988. Compounds of formu a I.C, wherein R2 is R2-- 10.2741 = Formu a 1 .2988).

Table 2989. Compounds of formu a I.C, wherein R2 is R2-- 10.2751 = Formu a 1 .2989).

Table 2990. Compounds of formu a I.C, wherein R2 is R2-- 10.2761 = Formu a 1 .2990).

Table 2991. Compounds of formu a I.C, wherein R2 is R2-- 10.2771 = Formu a 1 .2991 ).

Table 2992. Compounds of formu a I.C, wherein R2 is R2-- 10.2781 = Formu a 1 .2992).

Table 2993. Compounds of formu a I.C, wherein R2 is R2-- 10.2791 = Formu a 1 .2993.

Table 2994. Compounds of formu a I.C, wherein R2 is R2-- 10.2801 = Formu a 1 .2994).

Table 2995. Compounds of formu a I.C, wherein R2 is R2-- 10.2811 = Formu a 1 .2995).

Table 2996. Compounds of formu a I.C, wherein R2 is R2-- 10.2821 = Formu a 1 .2996).

Table 2997. Compounds of formu a I.C, wherein R2 is R2-- 10.2831 = Formu a 1 .2997).

Table 2998. Compounds of formu a I.C, wherein R2 is R2-- 10.2841 = Formu a 1 .2998).

Table 2999. Compounds of formu a I.C, wherein R2 is R2-- 10.2851 = Formu a 1 .2999).

Table 3000. Compounds of formu a I.C, wherein R2 is R2-- 10.2861 = Formu a 1 .3000).

Table 3001. Compounds of formu a I.C, wherein R2 is R2-- 10.2871 = Formu a 1 .3001 ).

Table 3002. Compounds of formu a I.C, wherein R2 is R2-- 10.2881 = Formu a 1 .3002).

Table 3003. Compounds of formu a I.C, wherein R2 is R2-- 10.2891 = Formu a 1 .3003).

Table 3004. Compounds of formu a I.C, wherein R2 is R2-- 10.2901 = Formu a 1 .3004).

Table 3005. Compounds of formu a I.C, wherein R2 is R2-- 10.2911 = Formu a 1 .3005).

Table 3006. Compounds of formu a I.C, wherein R2 is R2-- 10.2921 = Formu a 1 .3006).

Table 3007. Compounds of formu a I.C, wherein R2 is R2-- 10.2931 = Formu a 1 .3007).

Table 3008. Compounds of formu a I.C, wherein R2 is R2-- 10.2941 = Formu a 1 .3008).

Table 3009. Compounds of formu a I.C, wherein R2 is R2-- 10.2951 = Formu a 1 .3009).

Table 3010. Compounds of formu a I.C, wherein R2 is R2-- 10.2961 = Formu a 1 .3010).

Table 301 1. Compounds of formu a I.C, wherein R2 is R2-- 10.2971 = Formu a 1 .301 1 ).

Table 3012. Compounds of formu a I.C, wherein R2 is R2-- 10.2981 = Formu a 1 .3012).

Table 3013. Compounds of formu a I.C, wherein R2 is R2-- 10.2991 = Formu a 1 .3013).

Table 3014. Compounds of formu a I.C, wherein R2 is R2-- 10.3001 = Formu a 1 .3014).

Table 3015. Compounds of formu a I.C, wherein R2 is R2-- 10.3011 = Formu a 1 .3015).

Table 3016. Compounds of formu a I.C, wherein R2 is R2-- 10.3021 = Formu a 1 .3016).

Table 3017. Compounds of formu a I.C, wherein R2 is R2-- 10.3031 = Formu a 1 .3017).

Table 3018. Compounds of formu a I.C, wherein R2 is R2-- 10.3041 = Formu a 1 .3018).

Table 3019. Compounds of formu a I.C, wherein R2 is R2-- 10.3051 = Formu a 1 .3019). Table 3020. Compounds of formu a I.C, wherein R2 is R2-- I0.306I = Formu a 1.3020).

Table 3021. Compounds of formu a I.C, wherein R2 is R2-- I0.307I = Formu a 1.3021).

Table 3022. Compounds of formu a I.C, wherein R2 is R2-- I0.308I = Formu a 1.3022).

Table 3023. Compounds of formu a I.C, wherein R2 is R2-- I0.309I = Formu a 1.3023).

Table 3024. Compounds of formu a I.C, wherein R2 is R2-- 10.3101 = Formu a 1.3024).

Table 3025. Compounds of formu a I.C, wherein R2 is R2-- 10.3111 = Formu a 1.3025).

Table 3026. Compounds of formu a I.C, wherein R2 is R2-- 10.3121 = Formu a 1.3026).

Table 3027. Compounds of formu a I.C, wherein R2 is R2-- 10.3131 = Formu a 1.3027).

Table 3028. Compounds of formu a I.C, wherein R2 is R2-- 10.3141 = Formu a 1.3028).

Table 3029. Compounds of formu a I.C, wherein R2 is R2-- 10.3151 = Formu a 1.3029).

Table 3030. Compounds of formu a I.C, wherein R2 is R2-- 10.3161 = Formu a 1.3030).

Table 3031. Compounds of formu a I.C, wherein R2 is R2-- 10.3171 = Formu a 1.3031).

Table 3032. Compounds of formu a I.C, wherein R2 is R2-- 10.3181 = Formu a 1.3032).

Table 3033. Compounds of formu a I.C, wherein R2 is R2-- 10.3191 = Formu a 1.3033).

Table 3034. Compounds of formu a I.C, wherein R2 is R2-- 10.3201 = Formu a 1.3034).

Table 3035. Compounds of formu a I.C, wherein R2 is R2-- 10.3211 = Formu a 1.3035).

Table 3036. Compounds of formu a I.C, wherein R2 is R2-- 10.3221 = Formu a 1.3036).

Table 3037. Compounds of formu a I.C, wherein R2 is R2-- 10.3231 = Formu a 1.3037).

Table 3038. Compounds of formu a I.C, wherein R2 is R2-- 10.3241 = Formu a 1.3038).

Table 3039. Compounds of formu a I.C, wherein R2 is R2-- 10.3251 = Formu a 1.3039).

Table 3040. Compounds of formu a I.C, wherein R2 is R2-- 10.3261 = Formu a 1.3040).

Table 3041. Compounds of formu a I.C, wherein R2 is R2-- 10.3271 = Formu a 1.3041).

Table 3042. Compounds of formu a I.C, wherein R2 is R2-- 10.3281 = Formu a 1.3042).

Table 3043. Compounds of formu a I.C, wherein R2 is R2-- 10.3291 = Formu a 1.3043).

Table 3044. Compounds of formu a I.C, wherein R2 is R2-- 10.3301 = Formu a 1.3044).

Table 3045. Compounds of formu a I.C, wherein R2 is R2-- 10.3311 = Formu a 1.3045).

Table 3046. Compounds of formu a I.C, wherein R2 is R2-- 10.3321 = Formu a 1.3046).

Table 3047. Compounds of formu a I.C, wherein R2 is R2-- 10.3331 = Formu a 1.3047).

Table 3048. Compounds of formu a I.C, wherein R2 is R2-- 10.3341 = Formu a 1.3048).

Table 3049. Compounds of formu a I.C, wherein R2 is R2-- 10.3351 = Formu a 1.3049).

Table 3050. Compounds of formu a I.C, wherein R2 is R2-- 10.3361 = Formu a 1.3050).

Table 3051. Compounds of formu a I.C, wherein R2 is R2-- 10.3341 = Formu a 1.3051).

Table 3052. Compounds of formu a I.C, wherein R2 is R2-- 10.3381 = Formu a 1.3052).

Table 3053. Compounds of formu a I.C, wherein R2 is R2-- 10.3391 = Formu a 1.3053).

Table 3054. Compounds of formu a I.C, wherein R2 is R2-- 10.3401 = Formu a 1.3054).

Table 3055. Compounds of formu a I.C, wherein R2 is R2-- 10.3411 = Formu a 1.3055).

Table 3056. Compounds of formu a I.C, wherein R2 is R2-- 10.3421 = Formu a 1.3056).

Table 3057. Compounds of formu a I.C, wherein R2 is R2-- 10.3431 = Formu a 1.3057).

Table 3058. Compounds of formu a I.C, wherein R2 is R2-- 10.3441 = Formu a 1.3058).

Table 3059. Compounds of formu a I.C, wherein R2 is R2-- 10.3451 = Formu a 1.3059).

Table 3060. Compounds of formu a I.C, wherein R2 is R2-- 10.3461 = Formu a 1.3060).

Table 3061. Compounds of formu a I.C, wherein R2 is R2-- 10.3471 = Formu a 1.3061).

Table 3062. Compounds of formu a I.C, wherein R2 is R2-- 10.3481 = Formu a 1.3062).

Table 3063. Compounds of formu a I.C, wherein R2 is R2-- 10.3491 = Formu a 1.3063). Table 3064. Compounds of formu a I.C, wherein R2 is R2-- I 0.350I = Formu a 1 .3064).

Table 3065. Compounds of formu a I.C, wherein R2 is R2-- 10.3511 = Formu a 1 .3065).

Table 3066. Compounds of formu a I.C, wherein R2 is R2-- 10.3521 = Formu a 1 .3066).

Table 3067. Compounds of formu a I.C, wherein R2 is R2-- 10.3531 = Formu a 1 .3067).

Table 3068. Compounds of formu a I.C, wherein R2 is R2-- 10.3541 = Formu a 1 .3068).

Table 3069. Compounds of formu a I.C, wherein R2 is R2-- 10.3551 = Formu a 1 .3069).

Table 3070. Compounds of formu a I.C, wherein R2 is R2-- 10.3561 = Formu a 1 .3070).

Table 3071. Compounds of formu a I.C, wherein R2 is R2-- 10.3571 = Formu a 1 .3071 ).

Table 3072. Compounds of formu a I.C, wherein R2 is R2-- 10.3581 = Formu a 1 .3072).

Table 3073. Compounds of formu a I.C, wherein R2 is R2-- 10.3591 = Formu a 1 .3073).

Table 3074. Compounds of formu a I.C, wherein R2 is R2-- 10.3601 = Formu a 1 .3074).

Table 3075. Compounds of formu a I.C, wherein R2 is R2-- 10.3611 = Formu a 1 .3075).

Table 3076. Compounds of formu a I.C, wherein R2 is R2-- 10.3621 = Formu a 1 .3076).

Table 3077. Compounds of formu a I.C, wherein R2 is R2-- 10.3631 = Formu a 1 .3077).

Table 3078. Compounds of formu a I.C, wherein R2 is R2-- 10.3641 = Formu a 1 .3078).

Table 3079. Compounds of formu a I.C, wherein R2 is R2-- 10.3651 = Formu a 1 .3079).

Table 3080. Compounds of formu a I.C, wherein R2 is R2-- 10.3661 = Formu a 1 .3080).

Table 3081. Compounds of formu a I.C, wherein R2 is R2-- 10.3671 = Formu a 1 .3081 ).

Table 3082. Compounds of formu a I.C, wherein R2 is R2-- 10.3681 = Formu a 1 .3082).

Table 3083. Compounds of formu a I.C, wherein R2 is R2-- 10.3691 = Formu a 1 .3083).

Table 3084. Compounds of formu a I.C, wherein R2 is R2-- 10.3701 = Formu a 1 .3084).

Table 3085. Compounds of formu a I.C, wherein R2 is R2-- 10.3711 = Formu a 1 .3085).

Table 3086. Compounds of formu a I.C, wherein R2 is R2-- 10.3721 = Formu a 1 .3086).

Table 3087. Compounds of formu a I.C, wherein R2 is R2-- 10.3731 = Formu a 1 .3087).

Table 3088. Compounds of formu a I.C, wherein R2 is R2-- 10.3741 = Formu a 1 .3088).

Table 3089. Compounds of formu a I.C, wherein R2 is R2-- 10.3751 = Formu a 1 .3089).

Table 3090. Compounds of formu a I.C, wherein R2 is R2-- 10.3761 = Formu a 1 .3090).

Table 3091. Compounds of formu a I.C, wherein R2 is R2-- 10.3771 = Formu a 1 .3091 ).

Table 3092. Compounds of formu a I.C, wherein R2 is R2-- 10.3781 = Formu a 1 .3092).

Table 3093. Compounds of formu a I.C, wherein R2 is R2-- 10.3791 = Formu a 1 .3093).

Table 3094. Compounds of formu a I.C, wherein R2 is R2-- 10.3801 = Formu a 1 .3094).

Table 3095. Compounds of formu a I.C, wherein R2 is R2-- 10.3811 = Formu a 1 .3095).

Table 3096. Compounds of formu a I.C, wherein R2 is R2-- 10.3821 = Formu a 1 .3096).

Table 3097. Compounds of formu a I.C, wherein R2 is R2-- 10.3831 = Formu a 1 .3097).

Table 3098. Compounds of formu a I.C, wherein R2 is R2-- 10.3841 = Formu a 1 .3098).

Table 3099. Compounds of formu a I.C, wherein R2 is R2-- 10.3851 = Formu a 1 .3099).

Table 3100. Compounds of formu a I.C, wherein R2 is R2-- 10.3861 = Formu a 1 .3100).

Table 3101. Compounds of formu a I.C, wherein R2 is R2-- 10.3871 = Formu a 1 .3101 ).

Table 3102. Compounds of formu a I.C, wherein R2 is R2-- 10.3881 = Formu a 1 .3102).

Table 3103. Compounds of formu a I.C, wherein R2 is R2-- 10.3891 = Formu a 1 .3103).

Table 3104. Compounds of formu a I.C, wherein R2 is R2-- 10.3901 = Formu a 1 .3104).

Table 3105. Compounds of formu a I.C, wherein R2 is R2-- 10.3911 = Formu a 1 .3105).

Table 3106. Compounds of formu a I.C, wherein R2 is R2-- 10.3921 = Formu a 1 .3106).

Table 3107. Compounds of formu a I.C, wherein R2 is R2-- 10.3931 = Formu a 1 .3107). Tab e3108. Compounds o ormu a I.C, wherein R2 is R2-- I0.394I Formu a 1.3108).

Tab e3109. Compounds o ormu a I.C, wherein R2 is R2-- I0.395I = Formu a 1.3109).

Tab e3110. Compounds o ormu a I.C, wherein R2 is R2-- I0.396I = Formu a 1.3110).

Tab e 3111. Compounds o ormu a I.C, wherein R2 is R2-- I0.397I = Formu a 1.3111).

Tab Θ3112. Compounds o ormu a I.C, wherein R2 is R2-- I0.398I = Formu a 1.3112).

Tab e3113. Compounds o ormu a I.C, wherein R2 is R2-- I0.399I = Formu a 1.3113).

Tab Θ3114. Compounds o ormu a I.C, wherein R2 is R2-- I0.400I = Formu a 1.3114).

Tab Θ3115. Compounds o ormu a I.C, wherein R2 is R2-- 10.4011 = Formu a 1.3115).

Tab e3116. Compounds o ormu a I.C, wherein R2 is R2-- 10.4021 = Formu a 1.3116).

Tab Θ3117. Compounds o ormu a I.C, wherein R2 is R2-- 10.4031 = Formu a 1.3117).

Tab e3118. Compounds o ormu a I.C, wherein R2 is R2-- 10.4041 = Formu a 1.3118).

Tab e3119. Compounds o ormu a I.C, wherein R2 is R2-- 10.4051 = Formu a 1.3119).

Tab e3120. Compounds o ormu a I.C, wherein R2 is R2-- 10.4061 = Formu a 1.3120).

Tab Θ3121. Compounds o ormu a I.C, wherein R2 is R2-- 10.4071 = Formu a 1.3121).

Tab Θ3122. Compounds o ormu a I.C, wherein R2 is R2-- 10.4081 = Formu a 1.3122).

Tab Θ3123. Compounds o ormu a I.C, wherein R2 is R2-- 10.4091 = Formu a 1.3123).

Tab Θ3124. Compounds o ormu a I.C, wherein R2 is R2-- 10.4101 = Formu a 1.3124).

Tab Θ3125. Compounds o ormu a I.C, wherein R2 is R2-- 10.4111 = Formu a 1.3125).

Tab Θ3126. Compounds o ormu a I.C, wherein R2 is R2-- 10.4121 = Formu a 1.3126).

Tab Θ3127. Compounds o ormu a I.C, wherein R2 is R2-- 10.4131 = Formu a 1.3127).

Tab Θ3128. Compounds o ormu a I.C, wherein R2 is R2-- 10.4141 = Formu a 1.3128).

Tab Θ3129. Compounds o ormu a I.C, wherein R2 is R2-- 10.4151 = Formu a 1.3129).

Tab e3130. Compounds o ormu a I.C, wherein R2 is R2-- 10.4161 = Formu a 1.3130).

Tab e3131. Compounds o ormu a I.C, wherein R2 is R2-- 10.4171 = Formu a 1.3131).

Tab e3132. Compounds o ormu a I.C, wherein R2 is R2-- 10.4181 = Formu a 1.3132).

Tab e3133. Compounds o ormu a I.C, wherein R2 is R2-- 10.4191 = Formu a 1.3133).

Tab e3134. Compounds o ormu a I.C, wherein R2 is R2-- 10.4201 = Formu a 1.3134).

Tab e3135. Compounds o ormu a I.C, wherein R2 is R2-- 10.4211 = Formu a 1.3135).

Tab e3136. Compounds o ormu a I.C, wherein R2 is R2-- 10.4221 = Formu a 1.3136).

Tab e3137. Compounds o ormu a I.C, wherein R2 is R2-- 10.4231 = Formu a 1.3137).

Tab e3138. Compounds o ormu a I.C, wherein R2 is R2-- 10.4241 = Formu a 1.3138).

Tab e3139. Compounds o ormu a I.C, wherein R2 is R2-- 10.4251 = Formu a 1.3139).

Tab e3140. Compounds o ormu a I.C, wherein R2 is R2-- 10.4261 = Formu a 1.3140).

Tab e3141. Compounds o ormu a I.C, wherein R2 is R2-- 10.4271 = Formu a 1.3141).

Tab Θ3142. Compounds o ormu a I.C, wherein R2 is R2-- 10.4281 = Formu a 1.3142).

Tab e3143. Compounds o ormu a I.C, wherein R2 is R2-- 10.4291 = Formu a 1.3143).

Tab Θ3144. Compounds o ormu a I.C, wherein R2 is R2-- 10.4301 = Formu a 1.3144).

Tab Θ3145. Compounds o ormu a I.C, wherein R2 is R2-- 10.4311 = Formu a 1.3145).

Tab Θ3146. Compounds o ormu a I.C, wherein R2 is R2-- 10.4321 = Formu a 1.3146).

Tab Θ3147. Compounds o ormu a I.C, wherein R2 is R2-- 10.4331 = Formu a 1.3147).

Tab Θ3148. Compounds o ormu a I.C, wherein R2 is R2-- 10.4341 = Formu a 1.3148).

Tab Θ3149. Compounds o ormu a I.C, wherein R2 is R2-- 10.4351 = Formu a 1.3149).

Tab Θ3150. Compounds o ormu a I.C, wherein R2 is R2-- 10.4361 = Formu a 1.3150).

Tab Θ3151. Compounds o ormu a I.C, wherein R2 is R2-- 10.4371 = Formu a 1.3151). Tab e 3- 152. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.438 ormu a 1 .3152).

Tab e 3- 153. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.439 ormu a 1 .3153).

Tab e 3' 154. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.440 ormu a 1 .3154).

Tab e 3' 155. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.441 ormu a 1 .3155).

Tab e 3' 156. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.442 ormu a 1 .3156).

Tab e 3' 157. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.443 ormu a 1 .3157).

Tab e 3' 158. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.444 ormu a 1 .3158).

Tab e 3' 159. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.445 ormu a 1 .3159).

Tab e 3' 160. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.446 ormu a 1 .3160).

Tab e 3' 161. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.447 ormu a 1 .3161 ).

Tab e 3' 162. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.448 ormu a 1 .3162).

Tab e 3' 163. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.449 ormu a 1 .3163).

Tab e 3' 164. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.450 ormu a 1 .3164).

Tab e 3' 165. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.451 ormu a 1 .3165).

Tab e 3' 166. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.452 ormu a 1 .3166).

Tab e 3' 167. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.453 ormu a 1 .3167).

Tab e 3' 168. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.454 ormu a 1 .3168).

Tab e 3' 169. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.455 ormu a 1 .3169).

Tab e 3' 170. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.456 ormu a 1 .3170).

Tab e 3' 171. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.457 ormu a 1 .3171 ).

Tab e 3' 172. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.458 ormu a 1 .3172).

Tab e 3' 173. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.459 ormu a 1 .3173).

Tab e 3' 174. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.460 ormu a 1 .3174).

Tab e 3' 175. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.461 ormu a 1 .3175).

Tab e 3' 176. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.462 ormu a 1 .3176).

Tab e 3' 177. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.463 ormu a 1 .3177).

Tab e 3' 178. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.464 ormu a 1 .3178).

Tab e 3' 179. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.465 ormu a 1 .3179).

Tab e 3' 180. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.466 ormu a 1 .3180).

Tab e 3' 181. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.467 ormu a 1 .3181 ).

Tab e 3' 182. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.468 ormu a 1 .3182).

Tab e 3' 183. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.469 ormu a 1 .3183).

Tab e 3' 184. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.470 ormu a 1 .3184).

Tab e 3' 185. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.471 ormu a 1 .3185).

Tab e 3' 186. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.472 ormu a 1 .3186).

Tab e 3' 187. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.473 ormu a 1 .3187).

Tab e 3' 188. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.474 ormu a 1 .3188).

Tab e 3' 189. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.475 ormu a 1 .3189).

Tab e 3' 190. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.476 ormu a 1 .3190).

Tab e 3' 191. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.477 ormu a 1 .3191 ).

Tab e 3' 192. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.478 ormu a 1 .3192).

Tab e 3' 193. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.479 ormu a 1 .3193).

Tab e 3' 194. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.480 ormu a 1 .3194).

Tab e 3' 195. Compounds o1 ormu a I.C wherein R 2 is R 2 -10.481 ormu a 1 .3195). Table 3196. Compounds of formu a I.C, wherein R2 is R2-- I 0.482I = Formu a 1 .3196).

Table 3197. Compounds of formu a I.C, wherein R2 is R2-- I 0.483I = Formu a 1 .3197).

Table 3198. Compounds of formu a I.C, wherein R2 is R2-- I 0.484I = Formu a 1 .3198).

Table 3199. Compounds of formu a I.C, wherein R2 is R2-- I 0.485I = Formu a 1 .3199).

Table 3200. Compounds of formu a I.C, wherein R2 is R2-- I 0.486I = Formu a 1 .3200).

Table 3201. Compounds of formu a I.C, wherein R2 is R2-- I 0.487I = Formu a 1 .3201 ).

Table 3202. Compounds of formu a I.C, wherein R2 is R2-- I 0.488I = Formu a 1 .3202).

Table 3203. Compounds of formu a I.C, wherein R2 is R2-- I 0.489I = Formu a 1 .3203).

Table 3204. Compounds of formu a I.C, wherein R2 is R2-- I 0.490I = Formu a 1 .3204).

Table 3205. Compounds of formu a I.C, wherein R2 is R2-- 10.4911 = Formu a 1 .3205).

Table 3206. Compounds of formu a I.C, wherein R2 is R2-- 10.4921 = Formu a 1 .3206).

Table 3207. Compounds of formu a I.C, wherein R2 is R2-- 10.4931 = Formu a 1 .3207).

Table 3208. Compounds of formu a I.C, wherein R2 is R2-- 10.4941 = Formu a 1 .3208).

Table 3209. Compounds of formu a I.C, wherein R2 is R2-- 10.4951 = Formu a 1 .3209).

Table 3210. Compounds of formu a I.C, wherein R2 is R2-- 10.4961 = Formu a 1 .3210).

Table 321 1. Compounds of formu a I.C, wherein R2 is R2-- 10.4971 = Formu a 1 .321 1 ).

Table 3212. Compounds of formu a I.C, wherein R2 is R2-- 10.4981 = Formu a 1 .3212).

Table 3213. Compounds of formu a I.C, wherein R2 is R2-- 10.4991 = Formu a 1 .3213).

Table 3214. Compounds of formu a I.C, wherein R2 is R2-- 10.5001 = Formu a 1 .3214).

Table 3215. Compounds of formu a I.C, wherein R2 is R2-- 10.5011 = Formu a 1 .3215).

Table 3216. Compounds of formu a I.C, wherein R2 is R2-- 10.5021 = Formu a 1 .3216).

Table 3217. Compounds of formu a I.C, wherein R2 is R2-- 10.5031 = Formu a 1 .3217).

Table 3218. Compounds of formu a I.C, wherein R2 is R2-- 10.5041 = Formu a 1 .3218).

Table 3219. Compounds of formu a I.C, wherein R2 is R2-- 10.5051 = Formu a 1 .3219).

Table 3220. Compounds of formu a I.C, wherein R2 is R2-- 10.5061 = Formu a 1 .3220).

Table 3221. Compounds of formu a I.C, wherein R2 is R2-- 10.5071 = Formu a 1 .3221 ).

Table 3222. Compounds of formu a I.C, wherein R2 is R2-- 10.5081 = Formu a 1 .3222).

Table 3223. Compounds of formu a I.C, wherein R2 is R2-- 10.5091 = Formu a 1 .3223).

Table 3224. Compounds of formu a I.C, wherein R2 is R2-- 10.5101 = Formu a 1 .3224).

Table 3225. Compounds of formu a I.C, wherein R2 is R2-- 10.51 11 = Formu a 1 .3225).

Table 3226. Compounds of formu a I.C, wherein R2 is R2-- 10.5121 = Formu a 1 .3226).

Table 3227. Compounds of formu a I.C, wherein R2 is R2-- 10.5131 = Formu a 1 .3227).

Table 3228. Compounds of formu a I.C, wherein R2 is R2-- 10.5141 = Formu a 1 .3228).

Table 3229. Compounds of formu a I.C, wherein R2 is R2-- 10.5151 = Formu a 1 .3229).

Table 3230. Compounds of formu a I.C, wherein R2 is R2-- 10.5161 = Formu a 1 .3230).

Table 3231. Compounds of formu a I.C, wherein R2 is R2-- 10.5171 = Formu a 1 .3231 ).

Table 3232. Compounds of formu a I.C, wherein R2 is R2-- 10.5181 = Formu a 1 .3232).

Table 3233. Compounds of formu a I.C, wherein R2 is R2-- 10.5191 = Formu a 1 .3233).

Table 3234. Compounds of formu a I.C, wherein R2 is R2-- 10.5201 = Formu a 1 .3234).

Table 3235. Compounds of formu a I.C, wherein R2 is R2-- 10.5211 = Formu a 1 .3235).

Table 3236. Compounds of formu a I.C, wherein R2 is R2-- 10.5221 = Formu a 1 .3236).

Table 3237. Compounds of formu a I.C, wherein R2 is R2-- 10.5231 = Formu a 1 .3237).

Table 3238. Compounds of formu a I.C, wherein R2 is R2-- 10.5241 = Formu a 1 .3238).

Table 3239. Compounds of formu a I.C, wherein R2 is R2-- 10.5251 = Formu a 1 .3239). Table 3240. Compounds of formu a I.C, wherein R2 is R2-- I 0.526I = Formu a 1 .3240).

Table 3241. Compounds of formu a I.C, wherein R2 is R2-- I 0.527I = Formu a 1 .3241 ).

Table 3242. Compounds of formu a I.C, wherein R2 is R2-- I 0.528I = Formu a 1 .3242).

Table 3243. Compounds of formu a I.C, wherein R2 is R2-- I 0.529I = Formu a 1 .3243).

Table 3244. Compounds of formu a I.C, wherein R2 is R2-- I 0.530I = Formu a 1 .3244).

Table 3245. Compounds of formu a I.C, wherein R2 is R2-- 10.5311 = Formu a 1 .3245).

Table 3246. Compounds of formu a I.C, wherein R2 is R2-- 10.5321 = Formu a 1 .3246).

Table 3247. Compounds of formu a I.C, wherein R2 is R2-- 10.5331 = Formu a 1 .3247).

Table 3248. Compounds of formu a I.C, wherein R2 is R2-- 10.5341 = Formu a 1 .3248).

Table 3249. Compounds of formu a I.C, wherein R2 is R2-- 10.5351 = Formu a 1 .3249).

Table 3250. Compounds of formu a I.C, wherein R2 is R2-- 10.5361 = Formu a 1 .3250).

Table 3251. Compounds of formu a I.C, wherein R2 is R2-- 10.5371 = Formu a 1 .3251 ).

Table 3252. Compounds of formu a I.C, wherein R2 is R2-- 10.5381 = Formu a 1 .3252).

Table 3253. Compounds of formu a I.C, wherein R2 is R2-- 10.5391 = Formu a 1 .3253).

Table 3254. Compounds of formu a I.C, wherein R2 is R2-- 10.5401 = Formu a 1 .3254).

Table 3255. Compounds of formu a I.C, wherein R2 is R2-- 10.5411 = Formu a 1 .3255).

Table 3256. Compounds of formu a I.C, wherein R2 is R2-- 10.5421 = Formu a 1 .3256).

Table 3257. Compounds of formu a I.C, wherein R2 is R2-- 10.5431 = Formu a 1 .3257).

Table 3258. Compounds of formu a I.C, wherein R2 is R2-- 10.5441 = Formu a 1 .3258).

Table 3259. Compounds of formu a I.C, wherein R2 is R2-- 10.5451 = Formu a 1 .3259).

Table 3260. Compounds of formu a I.C, wherein R2 is R2-- 10.5461 = Formu a 1 .3260).

Table 3261. Compounds of formu a I.C, wherein R2 is R2-- 10.5471 = Formu a 1 .3261 ).

Table 3262. Compounds of formu a I.C, wherein R2 is R2-- 10.5481 = Formu a 1 .3262).

Table 3263. Compounds of formu a I.C, wherein R2 is R2-- 10.5491 = Formu a 1 .3263.

Table 3264. Compounds of formu a I.C, wherein R2 is R2-- 10.5501 = Formu a 1 .3264).

Table 3265. Compounds of formu a I.C, wherein R2 is R2-- 10.5511 = Formu a 1 .3265).

Table 3266. Compounds of formu a I.C, wherein R2 is R2-- 10.5521 = Formu a 1 .3266).

Table 3267. Compounds of formu a I.C, wherein R2 is R2-- 10.5531 = Formu a 1 .3267).

Table 3268. Compounds of formu a I.C, wherein R2 is R2-- 10.5541 = Formu a 1 .3268).

Table 3269. Compounds of formu a I.C, wherein R2 is R2-- 10.5551 = Formu a 1 .3269).

Table 3270. Compounds of formu a I.C, wherein R2 is R2-- 10.5561 = Formu a 1 .3270).

Table 3271. Compounds of formu a I.C, wherein R2 is R2-- 10.5571 = Formu a 1 .3271 ).

Table 3272. Compounds of formu a I.C, wherein R2 is R2-- 10.5581 = Formu a 1 .3272).

Table 3273. Compounds of formu a I.C, wherein R2 is R2-- 10.5591 = Formu a 1 .3273).

Table 3274. Compounds of formu a I.C, wherein R2 is R2-- 10.5601 = Formu a 1 .3274).

Table 3275. Compounds of formu a I.C, wherein R2 is R2-- 10.5611 = Formu a 1 .3275).

Table 3276. Compounds of formu a I.C, wherein R2 is R2-- 10.5621 = Formu a 1 .3276).

Table 3277. Compounds of formu a I.C, wherein R2 is R2-- 10.5631 = Formu a 1 .3277).

Table 3278. Compounds of formu a I.C, wherein R2 is R2-- 10.5641 = Formu a 1 .3278).

Table 3279. Compounds of formu a I.C, wherein R2 is R2-- 10.5651 = Formu a 1 .3279).

Table 3280. Compounds of formu a I.C, wherein R2 is R2-- 10.5661 = Formu a 1 .3280).

Table 3281. Compounds of formu a I.C, wherein R2 is R2-- 10.5671 = Formu a 1 .3281 ).

Table 3282. Compounds of formu a I.C, wherein R2 is R2-- 10.5681 = Formu a 1 .3282).

Table 3283. Compounds of formu a I.C, wherein R2 is R2-- 10.5691 = Formu a 1 .3283). Table 3284. Compounds of formu a I.C, wherein R2 is R2-- I 0.570I = Formu a 1 .3284).

Table 3285. Compounds of formu a I.C, wherein R2 is R2-- 10.5711 = Formu a 1 .3285).

Table 3286. Compounds of formu a I.C, wherein R2 is R2-- 10.5721 = Formu a 1 .3286).

Table 3287. Compounds of formu a I.C, wherein R2 is R2-- 10.5731 = Formu a 1 .3287).

Table 3288. Compounds of formu a I.C, wherein R2 is R2-- 10.5741 = Formu a 1 .3288).

Table 3289. Compounds of formu a I.C, wherein R2 is R2-- 10.5751 = Formu a 1 .3289).

Table 3290. Compounds of formu a I.C, wherein R2 is R2-- 10.5761 = Formu a 1 .3290).

Table 3291. Compounds of formu a I.C, wherein R2 is R2-- 10.5771 = Formu a 1 .3291 ).

Table 3292. Compounds of formu a I.C, wherein R2 is R2-- 10.5781 = Formu a 1 .3292).

Table 3293. Compounds of formu a I.C, wherein R2 is R2-- 10.5791 = Formu a 1 .3293).

Table 3294. Compounds of formu a I.C, wherein R2 is R2-- 10.5801 = Formu a 1 .3294).

Table 3295. Compounds of formu a I.C, wherein R2 is R2-- 10.5811 = Formu a 1 .3295).

Table 3296. Compounds of formu a I.C, wherein R2 is R2-- 10.5821 = Formu a 1 .3296).

Table 3297. Compounds of formu a I.C, wherein R2 is R2-- 10.5831 = Formu a 1 .3297).

Table 3298. Compounds of formu a I.C, wherein R2 is R2-- 10.5841 = Formu a 1 .3298).

Table 3299. Compounds of formu a I.C, wherein R2 is R2-- 10.5851 = Formu a 1 .3299).

Table 3300. Compounds of formu a I.C, wherein R2 is R2-- 10.5861 = Formu a 1 .3300).

Table 3301. Compounds of formu a I.C, wherein R2 is R2-- 10.5871 = Formu a 1 .3301 ).

Table 3302. Compounds of formu a I.C, wherein R2 is R2-- 10.5881 = Formu a 1 .3302).

Table 3303. Compounds of formu a I.C, wherein R2 is R2-- 10.5891 = Formu a 1 .3303).

Table 3304. Compounds of formu a I.C, wherein R2 is R2-- 10.5901 = Formu a 1 .3304).

Table 3305. Compounds of formu a I.C, wherein R2 is R2-- 10.5911 = Formu a 1 .3305).

Table 3306. Compounds of formu a I.C, wherein R2 is R2-- 10.5921 = Formu a 1 .3306).

Table 3307. Compounds of formu a I.C, wherein R2 is R2-- 10.5931 = Formu a 1 .3307).

Table 3308. Compounds of formu a I.C, wherein R2 is R2-- 10.5941 = Formu a 1 .3308).

Table 3309. Compounds of formu a I.C, wherein R2 is R2-- 10.5951 = Formu a 1 .3309).

Table 3310. Compounds of formu a I.C, wherein R2 is R2-- 10.5961 = Formu a 1 .3310).

Table 331 1. Compounds of formu a I.C, wherein R2 is R2-- 10.5971 = Formu a 1 .331 1 ).

Table 3312. Compounds of formu a I.C, wherein R2 is R2-- 10.5981 = Formu a 1 .3312).

Table 3313. Compounds of formu a I.C, wherein R2 is R2-- 10.5991 = Formu a 1 .3313).

Table 3314. Compounds of formu a I.C, wherein R2 is R2-- 10.6001 = Formu a 1 .3314).

Table 3315. Compounds of formu a I.C, wherein R2 is R2-- 10.6011 = Formu a 1 .3315).

Table 3316. Compounds of formu a I.C, wherein R2 is R2-- 10.6021 = Formu a 1 .3316).

Table 3317. Compounds of formu a I.C, wherein R2 is R2-- 10.6031 = Formu a 1 .3317).

Table 3318. Compounds of formu a I.C, wherein R2 is R2-- 10.6041 = Formu a 1 .3318).

Table 3319. Compounds of formu a I.C, wherein R2 is R2-- 10.6051 = Formu a 1 .3319).

Table 3320. Compounds of formu a I.C, wherein R2 is R2-- 10.6061 = Formu a 1 .3320).

Table 3321. Compounds of formu a I.C, wherein R2 is R2-- 10.6071 = Formu a 1 .3321 ).

Table 3322. Compounds of formu a I.C, wherein R2 is R2-- 10.6081 = Formu a 1 .3322).

Table 3323. Compounds of formu a I.C, wherein R2 is R2-- 10.6091 = Formu a 1 .3323).

Table 3324. Compounds of formu a I.C, wherein R2 is R2-- 10.6101 = Formu a 1 .3324).

Table 3325. Compounds of formu a I.C, wherein R2 is R2-- 10.61 11 = Formu a 1 .3325).

Table 3326. Compounds of formu a I.C, wherein R2 is R2-- 10.6121 = Formu a 1 .3326).

Table 3327. Compounds of formu a I.C, wherein R2 is R2-- 10.6131 = Formu a 1 .3327). Table 3328. Compounds of formu a I.C, wherein R2 is R2-- 10.6141 = Formu a 1 .3328).

Table 3329. Compounds of formu a I.C, wherein R2 is R2-- 10.6151 = Formu a 1 .3329).

Table 3330. Compounds of formu a I.C, wherein R2 is R2-- 10.6161 = Formu a 1 .3330).

Table 3331. Compounds of formu a I.C, wherein R2 is R2-- 10.6171 = Formu a 1 .3331 ).

Table 3332. Compounds of formu a I.C, wherein R2 is R2-- 10.6181 = Formu a 1 .3332).

Table 3333. Compounds of formu a I.C, wherein R2 is R2-- 10.6191 = Formu a 1 .3333).

Table 3334. Compounds of formu a I.C, wherein R2 is R2-- 10.6201 = Formu a 1 .3334).

Table 3335. Compounds of formu a I.C, wherein R2 is R2-- 10.6211 = Formu a 1 .3335).

Table 3336. Compounds of formu a I.C, wherein R2 is R2-- 10.6221 = Formu a 1 .3336).

Table 3337. Compounds of formu a I.C, wherein R2 is R2-- 10.6231 = Formu a 1 .3337).

Table 3338. Compounds of formu a I.C, wherein R2 is R2-- 10.6241 = Formu a 1 .3338).

Table 3339. Compounds of formu a I.C, wherein R2 is R2-- 10.6251 = Formu a 1 .3339).

Table 3340. Compounds of formu a I.C, wherein R2 is R2-- 10.6261 = Formu a 1 .3340).

Table 3341. Compounds of formu a I.C, wherein R2 is R2-- 10.6271 = Formu a 1 .3341 ).

Table 3342. Compounds of formu a I.C, wherein R2 is R2-- 10.6281 = Formu a 1 .3342).

Table 3343. Compounds of formu a I.C, wherein R2 is R2-- 10.6291 = Formu a 1 .3343).

Table 3344. Compounds of formu a I.C, wherein R2 is R2-- 10.6301 = Formu a 1 .3344).

Table 3345. Compounds of formu a I.C, wherein R2 is R2-- 10.6311 = Formu a 1 .3345).

Table 3346. Compounds of formu a I.C, wherein R2 is R2-- 10.6321 = Formu a 1 .3346).

Table 3347. Compounds of formu a I.C, wherein R2 is R2-- 10.6331 = Formu a 1 .3347).

Table 3348. Compounds of formu a I.C, wherein R2 is R2-- 10.6341 = Formu a 1 .3348).

Table 3349. Compounds of formu a I.C, wherein R2 is R2-- 10.6351 = Formu a 1 .3349).

Table 3350. Compounds of formu a I.C, wherein R2 is R2-- 10.6361 = Formu a 1 .3350).

Table 3351. Compounds of formu a I.C, wherein R2 is R2-- 10.6371 = Formu a 1 .3351 ).

Table 3352. Compounds of formu a I.C, wherein R2 is R2-- 10.6381 = Formu a 1 .3352).

Table 3353. Compounds of formu a I.C, wherein R2 is R2-- 10.6391 = Formu a 1 .3353).

Table 3354. Compounds of formu a I.C, wherein R2 is R2-- 10.6401 = Formu a 1 .3354).

Table 3355. Compounds of formu a I.C, wherein R2 is R2-- 10.6411 = Formu a 1 .3355).

Table 3356. Compounds of formu a I.C, wherein R2 is R2-- 10.6421 = Formu a 1 .3356).

Table 3357. Compounds of formu a I.C, wherein R2 is R2-- 10.6431 = Formu a 1 .3357).

Table 3358. Compounds of formu a I.C, wherein R2 is R2-- 10.6441 = Formu a 1 .3358).

Table 3359. Compounds of formu a I.C, wherein R2 is R2-- 10.6451 = Formu a 1 .3359).

Table 3360. Compounds of formu a I.C, wherein R2 is R2-- 10.6461 = Formu a 1 .3360).

Table 3361. Compounds of formu a I.C, wherein R2 is R2-- 10.6471 = Formu a 1 .3361 ).

Table 3362. Compounds of formu a I.C, wherein R2 is R2-- 10.6481 = Formu a 1 .3362).

Table 3363. Compounds of formu a I.C, wherein R2 is R2-- 10.6491 = Formu a 1 .3363).

Table 3364. Compounds of formu a I.C, wherein R2 is R2-- 10.6501 = Formu a 1 .3364).

Table 3365. Compounds of formu a I.C, wherein R2 is R2-- 10.6511 = Formu a 1 .3365).

Table 3366. Compounds of formu a I.C, wherein R2 is R2-- 10.6521 = Formu a 1 .3366).

Table 3367. Compounds of formu a I.C, wherein R2 is R2-- 10.6531 = Formu a 1 .3367).

Table 3368. Compounds of formu a I.C, wherein R2 is R2-- 10.6541 = Formu a 1 .3368).

Table 3369. Compounds of formu a I.C, wherein R2 is R2-- 10.6551 = Formu a 1 .3369).

Table 3370. Compounds of formu a I.C, wherein R2 is R2-- 10.6561 = Formu a 1 .3370).

Table 3371. Compounds of formu a I.C, wherein R2 is R2-- 10.6571 = Formu a 1 .3371 ). Table 3372. Compounds of formu a I.C, wherein R2 is R2-- I0.658(=formula 1.3372).

Table 3373. Compounds of formu a I.C, wherein R2 is R2-- I0.659(=formula 1.3373).

Table 3374. Compounds of formu a I.C, wherein R2 is R2-- I0.660(=formula 1.3374).

Table 3375. Compounds of formu a I.C, wherein R2 is R2-- I0.661(=formula 1.3375).

Table 3376. Compounds of formu a I.C, wherein R2 is R2-- I0.662(=formula 1.3376).

Table 3377. Compounds of formu a I.C, wherein R2 is R2-- I0.663(=formula 1.3377).

Table 3378. Compounds of formu a I.C, wherein R2 is R2-- I0.664(=formula 1.3378).

Table 3379. Compounds of formu a I.C, wherein R2 is R2-- I0.665(=formula 1.3379).

Table 3380. Compounds of formu a I.C, wherein R2 is R2-- I0.666(=formula 1.3380).

Table 3381. Compounds of formu a I.C, wherein R2 is R2-- I0.667(=formula 1.3381).

Table 3382. Compounds of formu a I.C, wherein R2 is R2-- I0.668(=formula 1.3382).

Table 3383. Compounds of formu a I.C, wherein R2 is R2-- I0.669(=formula 1.3383).

Table 3384. Compounds of formu a I.C, wherein R2 is R2-- I0.670(=formula 1.3384).

Table 3385. Compounds of formu a I.C, wherein R2 is R2-- I0.671(=formula 1.3385).

Table 3386. Compounds of formu a I.C, wherein R2 is R2-- I0.672(=formula 1.3386).

Table 3387. Compounds of formu a I.C, wherein R2 is R2-- I0.673(=formula 1.3387).

Table 3388. Compounds of formu a I.C, wherein R2 is R2-- I0.674(=formula 1.3388).

Table 3389. Compounds of formu a I.C, wherein R2 is R2-- I0.675(=formula 1.3389).

Table 3390. Compounds of formu a I.C, wherein R2 is R2-- I0.676(=formula 1.3390).

Table 3391. Compounds of formu a I.C, wherein R2 is R2-- l5.1(=formula 1.3391).

Table 3392. Compounds of formu a I.C, wherein R2 is R2-- l5.2(=formula 1.3392).

Table 3393. Compounds of formu a I.C, wherein R2 is R2-- l5.3(=formula 1.3393).

Table 3394. Compounds of formu a I.C, wherein R2 is R2-- l5.4(=formula 1.3394).

Table 3395. Compounds of formu a I.C, wherein R2 is R2-- l5.5(=formula 1.3395).

Table 3396. Compounds of formu a I.C, wherein R2 is R2-- l5.6(=formula 1.3396).

Table 3397. Compounds of formu a I.C, wherein R2 is R2-- l5.7(=formula 1.3397).

Table 3398. Compounds of formu a I.C, wherein R2 is R2-- l5.8(=formula 1.3398).

Table 3399. Compounds of formu a I.C, wherein R2 is R2-- l5.9(=formula 1.3399).

Table 3400. Compounds of formu a I.C, wherein R2 is R2-- I5.10(=formula 1.3400).

Table 3401. Compounds of formu a I.C, wherein R2 is R2-- l5.11(=formula 1.3401).

Table 3402. Compounds of formu a I.C, wherein R2 is R2-- l5.12(=formula 1.3402).

Table 3403. Compounds of formu a I.C, wherein R2 is R2-- l5.13(=formula 1.3403).

Table 3404. Compounds of formu a I.C, wherein R2 is R2-- l5.14(=formula 1.3404).

Table 3405. Compounds of formu a I.C, wherein R2 is R2-- l5.15(=formula 1.3405).

Table 3406. Compounds of formu a I.C, wherein R2 is R2-- l5.16(=formula 1.3406).

Table 3407. Compounds of formu a I.C, wherein R2 is R2-- l5.17(=formula 1.3407).

Table 3408. Compounds of formu a I.C, wherein R2 is R2-- l5.18(=formula 1.3408).

Table 3409. Compounds of formu a I.C, wherein R2 is R2-- l5.19(=formula 1.3409).

Table 3410. Compounds of formu a I.C, wherein R2 is R2-- I5.20(=formula 1.3410).

Table 3411. Compounds of formu a I.C, wherein R2 is R2-- l5.21(=formula 1.3411).

Table 3412. Compounds of formu a I.C, wherein R2 is R2-- l5.22(=formula 1.3412).

Table 3413. Compounds of formu a I.C, wherein R2 is R2-- l5.23(=formula 1.3413).

Table 3414. Compounds of formu a I.C, wherein R2 is R2-- l5.24(=formula 1.3414).

Table 3415. Compounds of formu a I.C, wherein R2 is R2-- l5.25(=formula 1.3415). Tab e 3416. Compounds o ormu a I.C, wherein R2 is R2-- I 5.26( Formu a 1.3416).

Tab e 3417. Compounds o ormu a I.C, wherein R2 is R2-- I 5.27( = Formu a 1.3417).

Tab e 3418. Compounds o ormu a I.C, wherein R2 is R2-- I 5.28( = Formu a 1.3418).

Tab e 3419. Compounds o ormu a I.C, wherein R2 is R2-- I 5.29( = Formu a 1.3419).

Tab e 3420. Compounds o ormu a I.C, wherein R2 is R2-- I 5.30( = Formu a 1.3420).

Tab e 3421. Compounds o ormu a I.C, wherein R2 is R2-- I 5.31 ( = Formu a 1.3421 ).

Tab e 3422. Compounds o ormu a I.C, wherein R2 is R2-- I 5.32( = Formu a 1.3422).

Tab e 3423. Compounds o ormu a I.C, wherein R2 is R2-- I 5.33( = Formu a 1.3423).

Tab e 3424. Compounds o ormu a I.C, wherein R2 is R2-- I 5.34( = Formu a 1.3424).

Tab e 3425. Compounds o ormu a I.C, wherein R2 is R2-- I 5.35( = Formu a 1.3425).

Tab e 3426. Compounds o ormu a I.C, wherein R2 is R2-- I 5.36( = Formu a 1.3426).

Tab e 3427. Compounds o ormu a I.C, wherein R2 is R2-- I 5.37( = Formu a 1.3427).

Tab e 3428. Compounds o ormu a I.C, wherein R2 is R2-- I 5.38( = Formu a 1.3428).

Tab e 3429. Compounds o ormu a I.C, wherein R2 is R2-- I 5.39( = Formu a 1.3429).

Tab e 3430. Compounds o ormu a I.C, wherein R2 is R2-- I 5.40( = Formu a 1.3430).

Tab e 3431. Compounds o ormu a I.C, wherein R2 is R2-- I 5.41 ( = Formu a 1.3431 ).

Tab e 3432. Compounds o ormu a I.C, wherein R2 is R2-- I 5.42( = Formu a 1.3432).

Tab e 3433. Compounds o ormu a I.C, wherein R2 is R2-- I 5.43( = Formu a 1.3433).

Tab e 3434. Compounds o ormu a I.C, wherein R2 is R2-- I 5.44( = Formu a 1.3434).

Tab e 3435. Compounds o ormu a I.C, wherein R2 is R2-- I 5.45( = Formu a 1.3435).

Tab e 3436. Compounds o ormu a I.C, wherein R2 is R2-- I 5.46( = Formu a 1.3436).

Tab e 3437. Compounds o ormu a I.C, wherein R2 is R2-- I 5.47( = Formu a 1.3437).

Tab e 3438. Compounds o ormu a I.C, wherein R2 is R2-- I 5.48( = Formu a 1.3438).

Tab e 3439. Compounds o ormu a I.C, wherein R2 is R2-- I 5.49( = Formu a 1.3439).

Tab e 3440. Compounds o ormu a I.C, wherein R2 is R2-- I 5.50( = Formu a 1.3440).

Tab e 3441. Compounds o ormu a I.C, wherein R2 is R2-- I 5.51 ( = Formu a 1.3441 ).

Tab e 3442. Compounds o ormu a I.C, wherein R2 is R2-- I 5.52( = Formu a 1.3442).

Tab e 3443. Compounds o ormu a I.C, wherein R2 is R2-- I 5.53( = Formu a 1.3443).

Tab e 3444. Compounds o ormu a I.C, wherein R2 is R2-- I 5.54( = Formu a 1.3444).

Tab e 3445. Compounds o ormu a I.C, wherein R2 is R2-- I 5.55( = Formu a 1.3445).

Tab e 3446. Compounds o ormu a I.C, wherein R2 is R2-- I 5.56( = Formu a 1.3446).

Tab e 3447. Compounds o ormu a I.C, wherein R2 is R2-- I 5.57( = Formu a 1.3447).

Tab e 3448. Compounds o ormu a I.C, wherein R2 is R2-- I 5.58( = Formu a 1.3448).

Tab e 3449. Compounds o ormu a I.C, wherein R2 is R2-- I 5.59( = Formu a 1.3449).

Tab e 3450. Compounds o ormu a I.C, wherein R2 is R2-- I 5.60( = Formu a 1.3450).

Tab e 3451. Compounds o ormu a I.C, wherein R2 is R2-- I 5.61 ( = Formu a 1.3451 ).

Tab e 3452. Compounds o ormu a I.C, wherein R2 is R2-- I 5.62( = Formu a 1.3452).

Tab e 3453. Compounds o ormu a I.C, wherein R2 is R2-- I 5.63( = Formu a 1.3453).

Tab e 3454. Compounds o ormu a I.C, wherein R2 is R2-- I 5.64( = Formu a 1.3454).

Tab e 3455. Compounds o ormu a I.C, wherein R2 is R2-- I 5.65( = Formu a 1.3455).

Tab e 3456. Compounds o ormu a I.C, wherein R2 is R2-- I 5.66( = Formu a 1.3456).

Tab e 3457. Compounds o ormu a I.C, wherein R2 is R2-- I 5.67( = Formu a 1.3457).

Tab e 3458. Compounds o ormu a I.C, wherein R2 is R2-- I 5.68( = Formu a 1.3458).

Tab e 3459. Compounds o ormu a I.C, wherein R2 is R2-- I 5.69( = Formu a 1.3459). Table 3460. Compounds of formu a I.C, wherein R2 is R2 5.70(= formula 1.3460).

Table 3461. Compounds of formu a I.C, wherein R2 is R2 5.71(= formula 1 .3461).

Table 3462. Compounds of formu a I.C, wherein R2 is R2 5.72(= formula 1 .3462).

Table 3463. Compounds of formu a I.C, wherein R2 is R2 5.73(= formula 1 .3463).

Table 3464. Compounds of formu a I.C, wherein R2 is R2 5.74(= formula 1 .3464).

Table 3465. Compounds of formu a I.C, wherein R2 is R2 5.75(= formula 1 .3465).

Table 3466. Compounds of formu a I.C, wherein R2 is R2 5.76(= formula 1 .3466).

Table 3467. Compounds of formu a I.C, wherein R2 is R2 5.77(= formula 1 .3467).

Table 3468. Compounds of formu a I.C, wherein R2 is R2 5.78(= formula 1 .3468).

Table 3469. Compounds of formu a I.C, wherein R2 is R2 5.79(= formula 1 .3469).

Table 3470. Compounds of formu a I.C, wherein R2 is R2 5.80(= formula 1 .3470).

Table 3471. Compounds of formu a I.C, wherein R2 is R2 5.81(= formula 1 .3471).

Table 3472. Compounds of formu a I.C, wherein R2 is R2 5.82(= formula 1 .3472).

Table 3473. Compounds of formu a I.C, wherein R2 is R2 5.83(= formula 1 .3473).

Table 3474. Compounds of formu a I.C, wherein R2 is R2 5.84(= formula 1 .3474).

Table 3475. Compounds of formu a I.C, wherein R2 is R2 5.85(= formula 1 .3475).

Table 3476. Compounds of formu a I.C, wherein R2 is R2 5.86(= formula 1 .3476).

Table 3477. Compounds of formu a I.C, wherein R2 is R2 5.87(= formula 1 .3477).

Table 3478. Compounds of formu a I.C, wherein R2 is R2 5.88(= formula 1 .3478).

Table 3479. Compounds of formu a I.C, wherein R2 is R2 5.89(= formula 1 .3479).

Table 3480. Compounds of formu a I.C, wherein R2 is R2 5.90(= formula 1 .3480).

Table 3481. Compounds of formu a I.C, wherein R2 is R2 5.91(= formula 1 .3481).

Table 3482. Compounds of formu a I.C, wherein R2 is R2 5.92(= formula 1 .3482).

Table 3483. Compounds of formu a I.C, wherein R2 is R2 5.93(= formula 1 .3483).

Table 3484. Compounds of formu a I.C, wherein R2 is R2 5.94(= formula 1 .3484).

Table 3485. Compounds of formu a I.C, wherein R2 is R2 5.95(= formula 1 .3485).

Table 3486. Compounds of formu a I.C, wherein R2 is R2 5.96(= formula 1 .3486).

Table 3487. Compounds of formu a I.C, wherein R2 is R2 5.97(= formula 1 .3487).

Table 3488. Compounds of formu a I.C, wherein R2 is R2 5.98(= formula 1 .3488).

Table 3489. Compounds of formu a I.C, wherein R2 is R2 5.99(= formula 1 .3489).

Table 3490. Compounds of formu a I.C, wherein R2 is R2 5.100( =formula 1.3490).

Table 3491. Compounds of formu a I.C, wherein R2 is R2 5.101 ( =formula 1.3491).

Table 3492. Compounds of formu a I.C, wherein R2 is R2 5.102( =formula 1.3492).

Table 3493. Compounds of formu a I.C, wherein R2 is R2 5.103( =formula 1.3493).

Table 3494. Compounds of formu a I.C, wherein R2 is R2 5.104( =formula 1.3494).

Table 3495. Compounds of formu a I.C, wherein R2 is R2 5.105( =formula 1.3495).

Table 3496. Compounds of formu a I.C, wherein R2 is R2 5.106( =formula 1.3496).

Table 3497. Compounds of formu a I.C, wherein R2 is R2 5.107( =formula 1.3497).

Table 3498. Compounds of formu a I.C, wherein R2 is R2 5.108( =formula 1.3498).

Table 3499. Compounds of formu a I.C, wherein R2 is R2 5.109( =formula 1.3499).

Table 3500. Compounds of formu a I.C, wherein R2 is R2 5.110( =formula 1.3500).

Table 3501. Compounds of formu a I.C, wherein R2 is R2 5.111 ( =formula 1.3501).

Table 3502. Compounds of formu a I.C, wherein R2 is R2 5.112( =formula 1.3502).

Table 3503. Compounds of formu a I.C, wherein R2 is R2 5.113( =formula 1.3503). Table 3504. Compounds of formu a I.C, wherein R2 is R2-- 15.1 141 = Formu a 1 .3504).

Table 3505. Compounds of formu a I.C, wherein R2 is R2-- 15.1 151 = Formu a 1 .3505).

Table 3506. Compounds of formu a I.C, wherein R2 is R2-- 15.1 161 = Formu a 1 .3506).

Table 3507. Compounds of formu a I.C, wherein R2 is R2-- 15.1 171 = Formu a 1 .3507).

Table 3508. Compounds of formu a I.C, wherein R2 is R2-- 15.1 181 = Formu a 1 .3508).

Table 3509. Compounds of formu a I.C, wherein R2 is R2-- 15.1 191 = Formu a 1 .3509).

Table 3510. Compounds of formu a I.C, wherein R2 is R2-- 15.1201 = Formu a 1 .3510).

Table 351 1. Compounds of formu a I.C, wherein R2 is R2-- 15.1211 = Formu a 1 .351 1 ).

Table 3512. Compounds of formu a I.C, wherein R2 is R2-- 15.1221 = Formu a 1 .3512).

Table 3513. Compounds of formu a I.C, wherein R2 is R2-- 15.1231 = Formu a 1 .3513).

Table 3514. Compounds of formu a I.C, wherein R2 is R2-- 15.1241 = Formu a 1 .3514).

Table 3515. Compounds of formu a I.C, wherein R2 is R2-- 15.1251 = Formu a 1 .3515).

Table 3516. Compounds of formu a I.C, wherein R2 is R2-- 15.1261 = Formu a 1 .3516).

Table 3517. Compounds of formu a I.C, wherein R2 is R2-- 15.1271 = Formu a 1 .3517).

Table 3518. Compounds of formu a I.C, wherein R2 is R2-- 15.1281 = Formu a 1 .3518).

Table 3519. Compounds of formu a I.C, wherein R2 is R2-- 15.1291 = Formu a 1 .3519).

Table 3520. Compounds of formu a I.C, wherein R2 is R2-- 15.1301 = Formu a 1 .3520).

Table 3521. Compounds of formu a I.C, wherein R2 is R2-- 15.1311 = Formu a 1 .3521 ).

Table 3522. Compounds of formu a I.C, wherein R2 is R2-- 15.1321 = Formu a 1 .3522).

Table 3523. Compounds of formu a I.C, wherein R2 is R2-- 15.1331 = Formu a 1 .3523).

Table 3524. Compounds of formu a I.C, wherein R2 is R2-- 15.1341 = Formu a 1 .3524).

Table 3525. Compounds of formu a I.C, wherein R2 is R2-- 15.1351 = Formu a 1 .3525).

Table 3526. Compounds of formu a I.C, wherein R2 is R2-- 15.1361 = Formu a 1 .3526).

Table 3527. Compounds of formu a I.C, wherein R2 is R2-- 15.1371 = Formu a 1 .3527).

Table 3528. Compounds of formu a I.C, wherein R2 is R2-- 15.1381 = Formu a 1 .3528).

Table 3529. Compounds of formu a I.C, wherein R2 is R2-- 15.1391 = Formu a 1 .3529).

Table 3530. Compounds of formu a I.C, wherein R2 is R2-- 15.1401 = Formu a 1 .3530).

Table 3531. Compounds of formu a I.C, wherein R2 is R2-- 15.1411 = Formu a 1 .3531 ).

Table 3532. Compounds of formu a I.C, wherein R2 is R2-- 15.1421 = Formu a 1 .3532).

Table 3533. Compounds of formu a I.C, wherein R2 is R2-- 15.1431 = Formu a 1 .3533).

Table 3534. Compounds of formu a I.C, wherein R2 is R2-- 15.1441 = Formu a 1 .3534).

Table 3535. Compounds of formu a I.C, wherein R2 is R2-- 15.1451 = Formu a 1 .3535).

Table 3536. Compounds of formu a I.C, wherein R2 is R2-- 15.1461 = Formu a 1 .3536).

Table 3537. Compounds of formu a I.C, wherein R2 is R2-- 15.1471 = Formu a 1 .3537).

Table 3538. Compounds of formu a I.C, wherein R2 is R2-- 15.1481 = Formu a 1 .3538).

Table 3539. Compounds of formu a I.C, wherein R2 is R2-- 15.1491 = Formu a 1 .3539).

Table 3540. Compounds of formu a I.C, wherein R2 is R2-- 15.1501 = Formu a 1 .3540).

Table 3541. Compounds of formu a I.C, wherein R2 is R2-- 15.1511 = Formu a 1 .3541 ).

Table 3542. Compounds of formu a I.C, wherein R2 is R2-- 15.1521 = Formu a 1 .3542).

Table 3543. Compounds of formu a I.C, wherein R2 is R2-- 15.1531 = Formu a 1 .3543).

Table 3544. Compounds of formu a I.C, wherein R2 is R2-- 15.1541 = Formu a 1 .3544).

Table 3545. Compounds of formu a I.C, wherein R2 is R2-- 15.1551 = Formu a 1 .3545).

Table 3546. Compounds of formu a I.C, wherein R2 is R2-- 15.1561 = Formu a 1 .3546).

Table 3547. Compounds of formu a I.C, wherein R2 is R2-- 15.1571 = Formu a 1 .3547). Tab e 3548. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.158 ormu a 1.3548).

Tab e 3549. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.159 ormu a 1.3549).

Tab e 3550. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.160 ormu a 1.3550).

Tab e 3551. Compounds o1 ormu a I.C wherein R 2 is R2-15.161 ormu a 1.3551).

Tab e 3552. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.162 ormu a 1.3552).

Tab e 3553. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.163 ormu a 1.3553).

Tab e 3554. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.164 ormu a 1.3554).

Tab e 3555. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.165 ormu a 1.3555).

Tab e 3556. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.166 ormu a 1.3556).

Tab e 3557. Compounds o1 ormu a I.C wherein R 2 is R 2 -15.167 ormu a 1.3557).

Tab e 3558. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.168 ormu a 1.3558).

Tab e 3559. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.169 ormu a 1.3559).

Tab e 3560. Compounds o1 ormu a I.C wherein R 2 is R 2 -15.170 ormu a 1.3560).

Tab e 3561. Compounds o1 ormu a I.C wherein R 2 is R 2 -15.171 ormu a 1.3561).

Tab e 3562. Compounds o1 ormu a I.C wherein R 2 is R 2 -15.172 ormu a 1.3562).

Tab e 3563. Compounds o1 ormu a I.C wherein R 2 is R 2 -15.173 ormu a 1.3563).

Tab e 3564. Compounds o1 ormu a I.C wherein R 2 is R 2 -15.174 ormu a 1.3564).

Tab e 3565. Compounds o1 ormu a I.C wherein R 2 is R 2 -15.175 ormu a 1.3565).

Tab e 3566. Compounds o1 ormu a I.C wherein R 2 is R 2 -15.176 ormu a 1.3566).

Tab e 3567. Compounds o1 ormu a I.C wherein R 2 is R 2 -15.177 ormu a 1.3567).

Tab e 3568. Compounds o1 ormu a I.C wherein R 2 is R 2 -15.178 ormu a 1.3568).

Tab e 3569. Compounds o1 ormu a I.C wherein R 2 is R 2 -15.179 ormu a 1.3569).

Tab e 3570. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.180 ormu a 1.3570).

Tab e 3571. Compounds o1 ormu a I.C wherein R 2 is R2-15.181 ormu a 1.3571).

Tab e 3572. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.182 ormu a 1.3572).

Tab e 3573. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.183 ormu a 1.3573).

Tab e 3574. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.184 ormu a 1.3574).

Tab e 3575. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.185 ormu a 1.3575).

Tab e 3576. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.186 ormu a 1.3576).

Tab e 3577. Compounds o1 ormu a I.C wherein R 2 is R 2 -15.187 ormu a 1.3577).

Tab e 3578. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.188 ormu a 1.3578).

Tab e 3579. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.189 ormu a 1.3579).

Tab e 3580. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.190 ormu a 1.3580).

Tab e 3581. Compounds o1 ormu a I.C wherein R 2 is R2-15.191 ormu a 1.3581).

Tab e 3582. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.192 ormu a 1.3582).

Tab e 3583. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.193 ormu a 1.3583).

Tab e 3584. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.194 ormu a 1.3584).

Tab e 3585. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.195 ormu a 1.3585).

Tab e 3586. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.196 ormu a 1.3586).

Tab e 3587. Compounds o1 ormu a I.C wherein R 2 is R 2 -15.197 ormu a 1.3587).

Tab e 3588. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.198 ormu a 1.3588).

Tab e 3589. Compounds o1 ormu a I.C wherein R 2 isR 2 -15.199 ormu a 1.3589).

Tab e 3590. Compounds o1 ormu a I.C wherein R 2 is R 2 -15.200 ormu a 1.3590).

Tab e 3591. Compounds o1 ormu a I.C wherein R 2 is R 2 -15.201 ormu a 1.3591). Table 3592. Compounds of formu a I.C, wherein R2 is R2-- I 5.202I = Formu a 1 .3592).

Table 3593. Compounds of formu a I.C, wherein R2 is R2-- I 5.203I = Formu a 1 .3593).

Table 3594. Compounds of formu a I.C, wherein R2 is R2-- I 5.204I = Formu a 1 .3594).

Table 3595. Compounds of formu a I.C, wherein R2 is R2-- I 5.205I = Formu a 1 .3595).

Table 3596. Compounds of formu a I.C, wherein R2 is R2-- I 5.206I = Formu a 1 .3596).

Table 3597. Compounds of formu a I.C, wherein R2 is R2-- I 5.207I = Formu a 1 .3597).

Table 3598. Compounds of formu a I.C, wherein R2 is R2-- I 5.208I = Formu a 1 .3598).

Table 3599. Compounds of formu a I.C, wherein R2 is R2-- I 5.209I = Formu a 1 .3599).

Table 3600. Compounds of formu a I.C, wherein R2 is R2-- 15.2101 = Formu a 1 .3600).

Table 3601. Compounds of formu a I.C, wherein R2 is R2-- 15.21 11 = Formu a 1 .3601 ).

Table 3602. Compounds of formu a I.C, wherein R2 is R2-- 15.2121 = Formu a 1 .3602).

Table 3603. Compounds of formu a I.C, wherein R2 is R2-- 15.2131 = Formu a 1 .3603).

Table 3604. Compounds of formu a I.C, wherein R2 is R2-- 15.2141 = Formu a 1 .3604).

Table 3605. Compounds of formu a I.C, wherein R2 is R2-- 15.2151 = Formu a 1 .3605).

Table 3606. Compounds of formu a I.C, wherein R2 is R2-- 15.2161 = Formu a 1 .3606).

Table 3607. Compounds of formu a I.C, wherein R2 is R2-- 15.2171 = Formu a 1 .3607).

Table 3608. Compounds of formu a I.C, wherein R2 is R2-- 15.2181 = Formu a 1 .3608).

Table 3609. Compounds of formu a I.C, wherein R2 is R2-- 15.2191 = Formu a 1 .3609).

Table 3610. Compounds of formu a I.C, wherein R2 is R2-- 15.2201 = Formu a 1 .3610).

Table 361 1. Compounds of formu a I.C, wherein R2 is R2-- 15.2211 = Formu a 1 .361 1 ).

Table 3612. Compounds of formu a I.C, wherein R2 is R2-- 15.2221 = Formu a 1 .3612).

Table 3613. Compounds of formu a I.C, wherein R2 is R2-- 15.2231 = Formu a 1 .3613).

Table 3614. Compounds of formu a I.C, wherein R2 is R2-- 15.2241 = Formu a 1 .3614).

Table 3615. Compounds of formu a I.C, wherein R2 is R2-- 15.2251 = Formu a 1 .3645).

Table 3616. Compounds of formu a I.C, wherein R2 is R2-- 15.2261 = Formu a 1 .3646).

Table 3617. Compounds of formu a I.C, wherein R2 is R2-- 15.2271 = Formu a 1 .3617).

Table 3618. Compounds of formu a I.C, wherein R2 is R2-- 15.2281 = Formu a 1 .3618).

Table 3619. Compounds of formu a I.C, wherein R2 is R2-- 15.2291 = Formu a 1 .3619).

Table 3620. Compounds of formu a I.C, wherein R2 is R2-- 15.2301 = Formu a 1 .3620).

Table 3621. Compounds of formu a I.C, wherein R2 is R2-- 15.2311 = Formu a 1 .3621 ).

Table 3622. Compounds of formu a I.C, wherein R2 is R2-- 15.2321 = Formu a 1 .3622).

Table 3623. Compounds of formu a I.C, wherein R2 is R2-- 15.2331 = Formu a 1 .3623).

Table 3624. Compounds of formu a I.C, wherein R2 is R2-- 15.2341 = Formu a 1 .3624).

Table 3625. Compounds of formu a I.C, wherein R2 is R2-- 15.2351 = Formu a 1 .3625).

Table 3626. Compounds of formu a I.C, wherein R2 is R2-- 15.2361 = Formu a 1 .3626).

Table 3627. Compounds of formu a I.C, wherein R2 is R2-- 15.2371 = Formu a 1 .3627).

Table 3628. Compounds of formu a I.C, wherein R2 is R2-- 15.2381 = Formu a 1 .3628).

Table 3629. Compounds of formu a I.C, wherein R2 is R2-- 15.2391 = Formu a 1 .3629).

Table 3630. Compounds of formu a I.C, wherein R2 is R2-- 15.2401 = Formu a 1 .3630).

Table 3631. Compounds of formu a I.C, wherein R2 is R2-- 15.2411 = Formu a 1 .3631 ).

Table 3632. Compounds of formu a I.C, wherein R2 is R2-- 15.2421 = Formu a 1 .3632).

Table 3633. Compounds of formu a I.C, wherein R2 is R2-- 15.2431 = Formu a 1 .3633).

Table 3634. Compounds of formu a I.C, wherein R2 is R2-- 15.2441 = Formu a 1 .3634).

Table 3635. Compounds of formu a I.C, wherein R2 is R2-- 15.2451 = Formu a 1 .3635). Table 3636. Compounds of formu a I.C, wherein R2 is R2-- I 5.246I = Formu a 1 .3636).

Table 3637. Compounds of formu a I.C, wherein R2 is R2-- I 5.247I = Formu a 1 .3637).

Table 3638. Compounds of formu a I.C, wherein R2 is R2-- I 5.248I = Formu a 1 .3638).

Table 3639. Compounds of formu a I.C, wherein R2 is R2-- I 5.249I = Formu a 1 .3639).

Table 3640. Compounds of formu a I.C, wherein R2 is R2-- I 5.250I = Formu a 1 .3640).

Table 3641. Compounds of formu a I.C, wherein R2 is R2-- 15.2511 = Formu a 1 .3641 ).

Table 3642. Compounds of formu a I.C, wherein R2 is R2-- 15.2521 = Formu a 1 .3642).

Table 3643. Compounds of formu a I.C, wherein R2 is R2-- 15.2531 = Formu a 1 .3643).

Table 3644. Compounds of formu a I.C, wherein R2 is R2-- 15.2541 = Formu a 1 .3644).

Table 3645. Compounds of formu a I.C, wherein R2 is R2-- 15.2551 = Formu a 1 .3645).

Table 3646. Compounds of formu a I.C, wherein R2 is R2-- 15.2561 = Formu a 1 .3646).

Table 3647. Compounds of formu a I.C, wherein R2 is R2-- 15.2571 = Formu a 1 .3647).

Table 3648. Compounds of formu a I.C, wherein R2 is R2-- 15.2581 = Formu a 1 .3648).

Table 3649. Compounds of formu a I.C, wherein R2 is R2-- 15.2591 = Formu a 1 .3649).

Table 3650. Compounds of formu a I.C, wherein R2 is R2-- 15.2601 = Formu a 1 .3650).

Table 3651. Compounds of formu a I.C, wherein R2 is R2-- 15.2611 = Formu a 1 .3651 ).

Table 3652. Compounds of formu a I.C, wherein R2 is R2-- 15.2621 = Formu a 1 .3652).

Table 3653. Compounds of formu a I.C, wherein R2 is R2-- 15.2631 = Formu a 1 .3653).

Table 3654. Compounds of formu a I.C, wherein R2 is R2-- 15.2641 = Formu a 1 .3654).

Table 3655. Compounds of formu a I.C, wherein R2 is R2-- 15.2651 = Formu a 1 .3655).

Table 3656. Compounds of formu a I.C, wherein R2 is R2-- 15.2661 = Formu a 1 .3656).

Table 3657. Compounds of formu a I.C, wherein R2 is R2-- 15.2671 = Formu a 1 .3657).

Table 3658. Compounds of formu a I.C, wherein R2 is R2-- 15.2681 = Formu a 1 .3658).

Table 3659. Compounds of formu a I.C, wherein R2 is R2-- 15.2691 = Formu a 1 .3659).

Table 3660. Compounds of formu a I.C, wherein R2 is R2-- 15.2701 = Formu a 1 .3660).

Table 3661. Compounds of formu a I.C, wherein R2 is R2-- 15.2711 = Formu a 1 .3661 ).

Table 3662. Compounds of formu a I.C, wherein R2 is R2-- 15.2721 = Formu a 1 .3662).

Table 3663. Compounds of formu a I.C, wherein R2 is R2-- 15.2731 = Formu a 1 .3663).

Table 3664. Compounds of formu a I.C, wherein R2 is R2-- 15.2741 = Formu a 1 .3664).

Table 3665. Compounds of formu a I.C, wherein R2 is R2-- 15.2751 = Formu a 1 .3665).

Table 3666. Compounds of formu a I.C, wherein R2 is R2-- 15.2761 = Formu a 1 .3666).

Table 3667. Compounds of formu a I.C, wherein R2 is R2-- 15.2771 = Formu a 1 .3667).

Table 3668. Compounds of formu a I.C, wherein R2 is R2-- 15.2781 = Formu a 1 .3668).

Table 3669. Compounds of formu a I.C, wherein R2 is R2-- 15.2791 = Formu a 1 .3669).

Table 3670. Compounds of formu a I.C, wherein R2 is R2-- 15.2801 = Formu a 1 .3670).

Table 3671. Compounds of formu a I.C, wherein R2 is R2-- 15.2811 = Formu a 1 .3671 ).

Table 3672. Compounds of formu a I.C, wherein R2 is R2-- 15.2821 = Formu a 1 .3672).

Table 3673. Compounds of formu a I.C, wherein R2 is R2-- 15.2831 = Formu a 1 .3673).

Table 3674. Compounds of formu a I.C, wherein R2 is R2-- 15.2841 = Formu a 1 .3674).

Table 3675. Compounds of formu a I.C, wherein R2 is R2-- 15.2851 = Formu a 1 .3675).

Table 3676. Compounds of formu a I.C, wherein R2 is R2-- 15.2861 = Formu a 1 .3676).

Table 3677. Compounds of formu a I.C, wherein R2 is R2-- 15.2871 = Formu a 1 .3677).

Table 3678. Compounds of formu a I.C, wherein R2 is R2-- 15.2881 = Formu a 1 .3678).

Table 3679. Compounds of formu a I.C, wherein R2 is R2-- 15.2891 = Formu a 1 .3679). Table 3680. Compounds of formu a I.C, wherein R2 is R2-- I 5.290I = Formu a 1 .3680).

Table 3681. Compounds of formu a I.C, wherein R2 is R2-- 15.2911 = Formu a 1 .3681 ).

Table 3682. Compounds of formu a I.C, wherein R2 is R2-- 15.2921 = Formu a 1 .3682).

Table 3683. Compounds of formu a I.C, wherein R2 is R2-- 15.2931 = Formu a 1 .3683).

Table 3684. Compounds of formu a I.C, wherein R2 is R2-- 15.2941 = Formu a 1 .3684).

Table 3685. Compounds of formu a I.C, wherein R2 is R2-- 15.2951 = Formu a 1 .3685).

Table 3686. Compounds of formu a I.C, wherein R2 is R2-- 15.2961 = Formu a 1 .3686).

Table 3687. Compounds of formu a I.C, wherein R2 is R2-- 15.2971 = Formu a 1 .3687).

Table 3688. Compounds of formu a I.C, wherein R2 is R2-- 15.2981 = Formu a 1 .3688).

Table 3689. Compounds of formu a I.C, wherein R2 is R2-- 15.2991 = Formu a 1 .3689).

Table 3690. Compounds of formu a I.C, wherein R2 is R2-- 15.3001 = Formu a 1 .3690).

Table 3691. Compounds of formu a I.C, wherein R2 is R2-- 15.3011 = Formu a 1 .3691 ).

Table 3692. Compounds of formu a I.C, wherein R2 is R2-- 15.3021 = Formu a 1 .3692).

Table 3693. Compounds of formu a I.C, wherein R2 is R2-- 15.3031 = Formu a 1 .3693).

Table 3694. Compounds of formu a I.C, wherein R2 is R2-- 15.3041 = Formu a 1 .3694).

Table 3695. Compounds of formu a I.C, wherein R2 is R2-- 15.3051 = Formu a 1 .3695).

Table 3696. Compounds of formu a I.C, wherein R2 is R2-- 15.3061 = Formu a 1 .3696).

Table 3697. Compounds of formu a I.C, wherein R2 is R2-- 15.3071 = Formu a 1 .3697).

Table 3698. Compounds of formu a I.C, wherein R2 is R2-- 15.3081 = Formu a 1 .3698).

Table 3699. Compounds of formu a I.C, wherein R2 is R2-- 15.3091 = Formu a 1 .3699).

Table 3700. Compounds of formu a I.C, wherein R2 is R2-- 15.3101 = Formu a 1 .3700).

Table 3701. Compounds of formu a I.C, wherein R2 is R2-- 15.31 11 = Formu a 1 .3701 ).

Table 3702. Compounds of formu a I.C, wherein R2 is R2-- 15.3121 = Formu a 1 .3702).

Table 3703. Compounds of formu a I.C, wherein R2 is R2-- 15.3131 = Formu a 1 .3703).

Table 3704. Compounds of formu a I.C, wherein R2 is R2-- 15.3141 = Formu a 1 .3704).

Table 3705. Compounds of formu a I.C, wherein R2 is R2-- 15.3151 = Formu a 1 .3705).

Table 3706. Compounds of formu a I.C, wherein R2 is R2-- 15.3161 = Formu a 1 .3706).

Table 3707. Compounds of formu a I.C, wherein R2 is R2-- 15.3171 = Formu a 1 .3707).

Table 3708. Compounds of formu a I.C, wherein R2 is R2-- 15.3181 = Formu a 1 .3708).

Table 3709. Compounds of formu a I.C, wherein R2 is R2-- 15.3191 = Formu a 1 .3709).

Table 3710. Compounds of formu a I.C, wherein R2 is R2-- 15.3201 = Formu a 1 .3710).

Table 371 1. Compounds of formu a I.C, wherein R2 is R2-- 15.3211 = Formu a 1 .371 1 ).

Table 3712. Compounds of formu a I.C, wherein R2 is R2-- 15.3221 = Formu a 1 .3712).

Table 3713. Compounds of formu a I.C, wherein R2 is R2-- 15.3231 = Formu a 1 .3713).

Table 3714. Compounds of formu a I.C, wherein R2 is R2-- 15.3241 = Formu a 1 .3714).

Table 3715. Compounds of formu a I.C, wherein R2 is R2-- 15.3251 = Formu a 1 .3715).

Table 3716. Compounds of formu a I.C, wherein R2 is R2-- 15.3261 = Formu a 1 .3716).

Table 3717. Compounds of formu a I.C, wherein R2 is R2-- 15.3271 = Formu a 1 .3717).

Table 3718. Compounds of formu a I.C, wherein R2 is R2-- 15.3281 = Formu a 1 .3718).

Table 3719. Compounds of formu a I.C, wherein R2 is R2-- 15.3291 = Formu a 1 .3719).

Table 3720. Compounds of formu a I.C, wherein R2 is R2-- 15.3301 = Formu a 1 .3720).

Table 3721. Compounds of formu a I.C, wherein R2 is R2-- 15.3311 = Formu a 1 .3721 ).

Table 3722. Compounds of formu a I.C, wherein R2 is R2-- 15.3321 = Formu a 1 .3722).

Table 3723. Compounds of formu a I.C, wherein R2 is R2-- 15.3331 = Formu a 1 .3723). Table 3724. Compounds of formu a I.C, wherein R2 is R2-- I 5.334I = Formu a 1 .3724).

Table 3725. Compounds of formu a I.C, wherein R2 is R2-- I 5.335I = Formu a 1 .3725).

Table 3726. Compounds of formu a I.C, wherein R2 is R2-- I 5.336I = Formu a 1 .3726).

Table 3727. Compounds of formu a I.C, wherein R2 is R2-- I 5.334I = Formu a 1 .3727).

Table 3728. Compounds of formu a I.C, wherein R2 is R2-- I 5.338I = Formu a 1 .3728).

Table 3729. Compounds of formu a I.C, wherein R2 is R2-- I 5.339I = Formu a 1 .3729).

Table 3730. Compounds of formu a I.C, wherein R2 is R2-- I 5.340I = Formu a 1 .3730).

Table 3731. Compounds of formu a I.C, wherein R2 is R2-- 15.3411 = Formu a 1 .3731 ).

Table 3732. Compounds of formu a I.C, wherein R2 is R2-- 15.3421 = Formu a 1 .3732).

Table 3733. Compounds of formu a I.C, wherein R2 is R2-- 15.3431 = Formu a 1 .3733).

Table 3734. Compounds of formu a I.C, wherein R2 is R2-- 15.3441 = Formu a 1 .3734).

Table 3735. Compounds of formu a I.C, wherein R2 is R2-- 15.3451 = Formu a 1 .3735).

Table 3736. Compounds of formu a I.C, wherein R2 is R2-- 15.3461 = Formu a 1 .3736).

Table 3737. Compounds of formu a I.C, wherein R2 is R2-- 15.3471 = Formu a 1 .3737).

Table 3738. Compounds of formu a I.C, wherein R2 is R2-- 15.3481 = Formu a 1 .3738).

Table 3739. Compounds of formu a I.C, wherein R2 is R2-- 15.3491 = Formu a 1 .3739).

Table 3740. Compounds of formu a I.C, wherein R2 is R2-- 15.3501 = Formu a 1 .3740).

Table 3741. Compounds of formu a I.C, wherein R2 is R2-- 15.3511 = Formu a 1 .3741 ).

Table 3742. Compounds of formu a I.C, wherein R2 is R2-- 15.3521 = Formu a 1 .3742).

Table 3743. Compounds of formu a I.C, wherein R2 is R2-- 15.3531 = Formu a 1 .3743).

Table 3744. Compounds of formu a I.C, wherein R2 is R2-- 15.3541 = Formu a 1 .3744).

Table 3745. Compounds of formu a I.C, wherein R2 is R2-- 15.3551 = Formu a 1 .3745).

Table 3746. Compounds of formu a I.C, wherein R2 is R2-- 15.3561 = Formu a 1 .3746).

Table 3747. Compounds of formu a I.C, wherein R2 is R2-- 15.3571 = Formu a 1 .3747).

Table 3748. Compounds of formu a I.C, wherein R2 is R2-- 15.3581 = Formu a 1 .3748).

Table 3749. Compounds of formu a I.C, wherein R2 is R2-- 15.3591 = Formu a 1 .3749).

Table 3750. Compounds of formu a I.C, wherein R2 is R2-- 15.3601 = Formu a 1 .3750).

Table 3751. Compounds of formu a I.C, wherein R2 is R2-- 15.3611 = Formu a 1 .3751 ).

Table 3752. Compounds of formu a I.C, wherein R2 is R2-- 15.3621 = Formu a 1 .3752).

Table 3753. Compounds of formu a I.C, wherein R2 is R2-- 15.3631 = Formu a 1 .3753).

Table 3754. Compounds of formu a I.C, wherein R2 is R2-- 15.3641 = Formu a 1 .3754).

Table 3755. Compounds of formu a I.C, wherein R2 is R2-- 15.3651 = Formu a 1 .3755).

Table 3756. Compounds of formu a I.C, wherein R2 is R2-- 15.3661 = Formu a 1 .3756).

Table 3757. Compounds of formu a I.C, wherein R2 is R2-- 15.3671 = Formu a 1 .3757).

Table 3758. Compounds of formu a I.C, wherein R2 is R2-- 15.3681 = Formu a 1 .3758).

Table 3759. Compounds of formu a I.C, wherein R2 is R2-- 15.3691 = Formu a 1 .3759).

Table 3760. Compounds of formu a I.C, wherein R2 is R2-- 15.3701 = Formu a 1 .3760).

Table 3761. Compounds of formu a I.C, wherein R2 is R2-- 15.3711 = Formu a 1 .3761 ).

Table 3762. Compounds of formu a I.C, wherein R2 is R2-- 15.3721 = Formu a 1 .3762).

Table 3763. Compounds of formu a I.C, wherein R2 is R2-- 15.3731 = Formu a 1 .3763).

Table 3764. Compounds of formu a I.C, wherein R2 is R2-- 15.3741 = Formu a 1 .3764).

Table 3765. Compounds of formu a I.C, wherein R2 is R2-- 15.3751 = Formu a 1 .3765).

Table 3766. Compounds of formu a I.C, wherein R2 is R2-- 15.3761 = Formu a 1 .3766).

Table 3767. Compounds of formu a I.C, wherein R2 is R2-- 15.3771 = Formu a 1 .3767). Table 3768. Compounds of formu a I.C, wherein R2 is R2-- I 5.378I = Formu a 1 .3768).

Table 3769. Compounds of formu a I.C, wherein R2 is R2-- I 5.379I = Formu a 1 .3769).

Table 3770. Compounds of formu a I.C, wherein R2 is R2-- I 5.380I = Formu a 1 .3770).

Table 3771. Compounds of formu a I.C, wherein R2 is R2-- 15.3811 = Formu a 1 .3771 ).

Table 3772. Compounds of formu a I.C, wherein R2 is R2-- 15.3821 = Formu a 1 .3772).

Table 3773. Compounds of formu a I.C, wherein R2 is R2-- 15.3831 = Formu a 1 .3773).

Table 3774. Compounds of formu a I.C, wherein R2 is R2-- 15.3841 = Formu a 1 .3774).

Table 3775. Compounds of formu a I.C, wherein R2 is R2-- 15.3851 = Formu a 1 .3775).

Table 3776. Compounds of formu a I.C, wherein R2 is R2-- 15.3861 = Formu a 1 .3776.

Table 3777. Compounds of formu a I.C, wherein R2 is R2-- 15.3871 = Formu a 1 .3777).

Table 3778. Compounds of formu a I.C, wherein R2 is R2-- 15.3881 = Formu a 1 .3778).

Table 3779. Compounds of formu a I.C, wherein R2 is R2-- 15.3891 = Formu a 1 .3779).

Table 3780. Compounds of formu a I.C, wherein R2 is R2-- 15.3901 = Formu a 1 .3780).

Table 3781. Compounds of formu a I.C, wherein R2 is R2-- 15.3911 = Formu a 1 .3781 ).

Table 3782. Compounds of formu a I.C, wherein R2 is R2-- 15.3921 = Formu a 1 .3782).

Table 3783. Compounds of formu a I.C, wherein R2 is R2-- 15.3931 = Formu a 1 .3783).

Table 3784. Compounds of formu a I.C, wherein R2 is R2-- 15.3941 = Formu a 1 .3784).

Table 3785. Compounds of formu a I.C, wherein R2 is R2-- 15.3951 = Formu a 1 .3785).

Table 3786. Compounds of formu a I.C, wherein R2 is R2-- 15.3961 = Formu a 1 .3786).

Table 3787. Compounds of formu a I.C, wherein R2 is R2-- 15.3971 = Formu a 1 .3787).

Table 3788. Compounds of formu a I.C, wherein R2 is R2-- 15.3981 = Formu a 1 .3788).

Table 3789. Compounds of formu a I.C, wherein R2 is R2-- 15.3991 = Formu a 1 .3789).

Table 3790. Compounds of formu a I.C, wherein R2 is R2-- 15.4001 = Formu a 1 .3790).

Table 3791. Compounds of formu a I.C, wherein R2 is R2-- 15.4011 = Formu a 1 .3791 ).

Table 3792. Compounds of formu a I.C, wherein R2 is R2-- 15.4021 = Formu a 1 .3792).

Table 3793. Compounds of formu a I.C, wherein R2 is R2-- 15.4031 = Formu a 1 .3793).

Table 3794. Compounds of formu a I.C, wherein R2 is R2-- 15.4041 = Formu a 1 .3794).

Table 3795. Compounds of formu a I.C, wherein R2 is R2-- 15.4051 = Formu a 1 .3795).

Table 3796. Compounds of formu a I.C, wherein R2 is R2-- 15.4061 = Formu a 1 .3796).

Table 3797. Compounds of formu a I.C, wherein R2 is R2-- 15.4071 = Formu a 1 .3797).

Table 3798. Compounds of formu a I.C, wherein R2 is R2-- 15.4081 = Formu a 1 .3798).

Table 3799. Compounds of formu a I.C, wherein R2 is R2-- 15.4091 = Formu a 1 .3799).

Table 3800. Compounds of formu a I.C, wherein R2 is R2-- 15.4101 = Formu a 1 .3800).

Table 3801. Compounds of formu a I.C, wherein R2 is R2-- 15.41 11 = Formu a 1 .3801 ).

Table 3802. Compounds of formu a I.C, wherein R2 is R2-- 15.4121 = Formu a 1 .3802).

Table 3803. Compounds of formu a I.C, wherein R2 is R2-- 15.4131 = Formu a 1 .3803).

Table 3804. Compounds of formu a I.C, wherein R2 is R2-- 15.4141 = Formu a 1 .3804).

Table 3805. Compounds of formu a I.C, wherein R2 is R2-- 15.4151 = Formu a 1 .3805).

Table 3806. Compounds of formu a I.C, wherein R2 is R2-- 15.4161 = Formu a 1 .3806).

Table 3807. Compounds of formu a I.C, wherein R2 is R2-- 15.4171 = Formu a 1 .3807).

Table 3808. Compounds of formu a I.C, wherein R2 is R2-- 15.4181 = Formu a 1 .3808).

Table 3809. Compounds of formu a I.C, wherein R2 is R2-- 15.4191 = Formu a 1 .3809).

Table 3810. Compounds of formu a I.C, wherein R2 is R2-- 15.4201 = Formu a 1 .3810).

Table 381 1. Compounds of formu a I.C, wherein R2 is R2-- 15.4211 = Formu a 1 .381 1 ). Table 3812. Compounds of formu a I.C, wherein R2 is R2-- I 5.422I = Formu a 1 .3812).

Table 3813. Compounds of formu a I.C, wherein R2 is R2-- I 5.423I = Formu a 1 .3813).

Table 3814. Compounds of formu a I.C, wherein R2 is R2-- I 5.424I = Formu a 1 .3814).

Table 3815. Compounds of formu a I.C, wherein R2 is R2-- I 5.425I = Formu a 1 .3815).

Table 3816. Compounds of formu a I.C, wherein R2 is R2-- I 5.426I = Formu a 1 .3816).

Table 3817. Compounds of formu a I.C, wherein R2 is R2-- I 5.427I = Formu a 1 .3817).

Table 3818. Compounds of formu a I.C, wherein R2 is R2-- I 5.428I = Formu a 1 .3818).

Table 3819. Compounds of formu a I.C, wherein R2 is R2-- I 5.429I = Formu a 1 .3819).

Table 3820. Compounds of formu a I.C, wherein R2 is R2-- I 5.430I = Formu a 1 .3820).

Table 3821. Compounds of formu a I.C, wherein R2 is R2-- 15.4311 = Formu a 1 .3821 ).

Table 3822. Compounds of formu a I.C, wherein R2 is R2-- 15.4321 = Formu a 1 .3822).

Table 3823. Compounds of formu a I.C, wherein R2 is R2-- 15.4331 = Formu a 1 .3823).

Table 3824. Compounds of formu a I.C, wherein R2 is R2-- 15.4341 = Formu a 1 .3824).

Table 3825. Compounds of formu a I.C, wherein R2 is R2-- 15.4351 = Formu a 1 .3825).

Table 3826. Compounds of formu a I.C, wherein R2 is R2-- 15.4361 = Formu a 1 .3826).

Table 3827. Compounds of formu a I.C, wherein R2 is R2-- 15.4371 = Formu a 1 .3827).

Table 3828. Compounds of formu a I.C, wherein R2 is R2-- 15.4381 = Formu a 1 .3828).

Table 3829. Compounds of formu a I.C, wherein R2 is R2-- 15.4391 = Formu a 1 .3829).

Table 3830. Compounds of formu a I.C, wherein R2 is R2-- 15.4401 = Formu a 1 .3830).

Table 3831. Compounds of formu a I.C, wherein R2 is R2-- 15.4411 = Formu a 1 .3831 ).

Table 3832. Compounds of formu a I.C, wherein R2 is R2-- 15.4421 = Formu a 1 .3832).

Table 3833. Compounds of formu a I.C, wherein R2 is R2-- 15.4431 = Formu a 1 .3833).

Table 3834. Compounds of formu a I.C, wherein R2 is R2-- 15.4441 = Formu a 1 .3834).

Table 3835. Compounds of formu a I.C, wherein R2 is R2-- 15.4451 = Formu a 1 .3835).

Table 3836. Compounds of formu a I.C, wherein R2 is R2-- 15.4461 = Formu a 1 .3836).

Table 3837. Compounds of formu a I.C, wherein R2 is R2-- 15.4471 = Formu a 1 .3837).

Table 3838. Compounds of formu a I.C, wherein R2 is R2-- 15.4481 = Formu a 1 .3838).

Table 3839. Compounds of formu a I.C, wherein R2 is R2-- 15.4491 = Formu a 1 .3839).

Table 3840. Compounds of formu a I.C, wherein R2 is R2-- 15.4501 = Formu a 1 .3840).

Table 3841. Compounds of formu a I.C, wherein R2 is R2-- 15.4511 = Formu a 1 .3841 ).

Table 3842. Compounds of formu a I.C, wherein R2 is R2-- 15.4521 = Formu a 1 .3842).

Table 3843. Compounds of formu a I.C, wherein R2 is R2-- 15.4531 = Formu a 1 .3843).

Table 3844. Compounds of formu a I.C, wherein R2 is R2-- 15.4541 = Formu a 1 .3844).

Table 3845. Compounds of formu a I.C, wherein R2 is R2-- 15.4551 = Formu a 1 .3845).

Table 3846. Compounds of formu a I.C, wherein R2 is R2-- 15.4561 = Formu a 1 .3846).

Table 3847. Compounds of formu a I.C, wherein R2 is R2-- 15.4571 = Formu a 1 .3847).

Table 3848. Compounds of formu a I.C, wherein R2 is R2-- 15.4581 = Formu a 1 .3848).

Table 3849. Compounds of formu a I.C, wherein R2 is R2-- 15.4591 = Formu a 1 .3849).

Table 3850. Compounds of formu a I.C, wherein R2 is R2-- 15.4601 = Formu a 1 .3850).

Table 3851. Compounds of formu a I.C, wherein R2 is R2-- 15.4611 = Formu a 1 .3851 ).

Table 3852. Compounds of formu a I.C, wherein R2 is R2-- 15.4621 = Formu a 1 .3852).

Table 3853. Compounds of formu a I.C, wherein R2 is R2-- 15.4631 = Formu a 1 .3853).

Table 3854. Compounds of formu a I.C, wherein R2 is R2-- 15.4641 = Formu a 1 .3854).

Table 3855. Compounds of formu a I.C, wherein R2 is R2-- 15.4651 = Formu a 1 .3855). Table 3856. Compounds of formu a I.C, wherein R2 is R2-- I 5.466I = Formu a 1 .3856).

Table 3857. Compounds of formu a I.C, wherein R2 is R2-- I 5.467I = Formu a 1 .3857).

Table 3858. Compounds of formu a I.C, wherein R2 is R2-- I 5.468I = Formu a 1 .3858).

Table 3859. Compounds of formu a I.C, wherein R2 is R2-- I 5.469I = Formu a 1 .3859).

Table 3860. Compounds of formu a I.C, wherein R2 is R2-- I 5.470I = Formu a 1 .3860).

Table 3861. Compounds of formu a I.C, wherein R2 is R2-- 15.4711 = Formu a 1 .3861 ).

Table 3862. Compounds of formu a I.C, wherein R2 is R2-- 15.4721 = Formu a 1 .3862).

Table 3863. Compounds of formu a I.C, wherein R2 is R2-- 15.4731 = Formu a 1 .3863).

Table 3864. Compounds of formu a I.C, wherein R2 is R2-- 15.4741 = Formu a 1 .3864).

Table 3865. Compounds of formu a I.C, wherein R2 is R2-- 15.4751 = Formu a 1 .3865).

Table 3866. Compounds of formu a I.C, wherein R2 is R2-- 15.4761 = Formu a 1 .3866).

Table 3867. Compounds of formu a I.C, wherein R2 is R2-- 15.4771 = Formu a 1 .3867).

Table 3868. Compounds of formu a I.C, wherein R2 is R2-- 15.4781 = Formu a 1 .3868).

Table 3869. Compounds of formu a I.C, wherein R2 is R2-- 15.4791 = Formu a 1 .3869).

Table 3870. Compounds of formu a I.C, wherein R2 is R2-- 15.4801 = Formu a 1 .3870).

Table 3871. Compounds of formu a I.C, wherein R2 is R2-- 15.4811 = Formu a 1 .3871 ).

Table 3872. Compounds of formu a I.C, wherein R2 is R2-- 15.4821 = Formu a 1 .3872).

Table 3873. Compounds of formu a I.C, wherein R2 is R2-- 15.4831 = Formu a 1 .3873).

Table 3874. Compounds of formu a I.C, wherein R2 is R2-- 15.4841 = Formu a 1 .3874).

Table 3875. Compounds of formu a I.C, wherein R2 is R2-- 15.4851 = Formu a 1 .3875).

Table 3876. Compounds of formu a I.C, wherein R2 is R2-- 15.4861 = Formu a 1 .3876).

Table 3877. Compounds of formu a I.C, wherein R2 is R2-- 15.4871 = Formu a 1 .3877).

Table 3878. Compounds of formu a I.C, wherein R2 is R2-- 15.4881 = Formu a 1 .3878).

Table 3879. Compounds of formu a I.C, wherein R2 is R2-- 15.4891 = Formu a 1 .3879).

Table 3880. Compounds of formu a I.C, wherein R2 is R2-- 15.4901 = Formu a 1 .3880).

Table 3881. Compounds of formu a I.C, wherein R2 is R2-- 15.4911 = Formu a 1 .3881 ).

Table 3882. Compounds of formu a I.C, wherein R2 is R2-- 15.4921 = Formu a 1 .3882).

Table 3883. Compounds of formu a I.C, wherein R2 is R2-- 15.4931 = Formu a 1 .3883).

Table 3884. Compounds of formu a I.C, wherein R2 is R2-- 15.4941 = Formu a 1 .3884).

Table 3885. Compounds of formu a I.C, wherein R2 is R2-- 15.4951 = Formu a 1 .3885).

Table 3886. Compounds of formu a I.C, wherein R2 is R2-- 15.4961 = Formu a 1 .3886).

Table 3887. Compounds of formu a I.C, wherein R2 is R2-- 15.4971 = Formu a 1 .3887).

Table 3888. Compounds of formu a I.C, wherein R2 is R2-- 15.4981 = Formu a 1 .3888).

Table 3889. Compounds of formu a I.C, wherein R2 is R2-- 15.4991 = Formu a 1 .3889).

Table 3890. Compounds of formu a I.C, wherein R2 is R2-- 15.5001 = Formu a 1 .3890).

Table 3891. Compounds of formu a I.C, wherein R2 is R2-- 15.5011 = Formu a 1 .3891 ).

Table 3892. Compounds of formu a I.C, wherein R2 is R2-- 15.5021 = Formu a 1 .3892).

Table 3893. Compounds of formu a I.C, wherein R2 is R2-- 15.5031 = Formu a 1 .3893).

Table 3894. Compounds of formu a I.C, wherein R2 is R2-- 15.5041 = Formu a 1 .3894).

Table 3895. Compounds of formu a I.C, wherein R2 is R2-- 15.5051 = Formu a 1 .3895).

Table 3896. Compounds of formu a I.C, wherein R2 is R2-- 15.5061 = Formu a 1 .3896).

Table 3897. Compounds of formu a I.C, wherein R2 is R2-- 15.5071 = Formu a 1 .3897).

Table 3898. Compounds of formu a I.C, wherein R2 is R2-- 15.5081 = Formu a 1 .3898).

Table 3899. Compounds of formu a I.C, wherein R2 is R2-- 15.5091 = Formu a 1 .3899). Table 3900. Compounds of formu a I.C, wherein R2 is R2-- 15.5101 = Formu a 1 .3900).

Table 3901. Compounds of formu a I.C, wherein R2 is R2-- 15.51 11 = Formu a 1 .3901 ).

Table 3902. Compounds of formu a I.C, wherein R2 is R2-- 15.5121 = Formu a 1 .3902).

Table 3903. Compounds of formu a I.C, wherein R2 is R2-- 15.5131 = Formu a 1 .3903).

Table 3904. Compounds of formu a I.C, wherein R2 is R2-- 15.5141 = Formu a 1 .3904).

Table 3905. Compounds of formu a I.C, wherein R2 is R2-- 15.5151 = Formu a 1 .3905).

Table 3906. Compounds of formu a I.C, wherein R2 is R2-- 15.5161 = Formu a 1 .3906).

Table 3907. Compounds of formu a I.C, wherein R2 is R2-- 15.5171 = Formu a 1 .3907).

Table 3908. Compounds of formu a I.C, wherein R2 is R2-- 15.5181 = Formu a 1 .3908).

Table 3909. Compounds of formu a I.C, wherein R2 is R2-- 15.5191 = Formu a 1 .3909).

Table 3910. Compounds of formu a I.C, wherein R2 is R2-- 15.5201 = Formu a 1 .3910).

Table 391 1. Compounds of formu a I.C, wherein R2 is R2-- 15.5211 = Formu a 1 .391 1 ).

Table 3912. Compounds of formu a I.C, wherein R2 is R2-- 15.5221 = Formu a 1 .3912).

Table 3913. Compounds of formu a I.C, wherein R2 is R2-- 15.5231 = Formu a 1 .3913).

Table 3914. Compounds of formu a I.C, wherein R2 is R2-- 15.5241 = Formu a 1 .3914).

Table 3915. Compounds of formu a I.C, wherein R2 is R2-- 15.5251 = Formu a 1 .3915).

Table 3916. Compounds of formu a I.C, wherein R2 is R2-- 15.5261 = Formu a 1 .3916).

Table 3917. Compounds of formu a I.C, wherein R2 is R2-- 15.5271 = Formu a 1 .3917).

Table 3918. Compounds of formu a I.C, wherein R2 is R2-- 15.5281 = Formu a 1 .3918).

Table 3919. Compounds of formu a I.C, wherein R2 is R2-- 15.5291 = Formu a 1 .3919).

Table 3920. Compounds of formu a I.C, wherein R2 is R2-- 15.5301 = Formu a 1 .3920).

Table 3921. Compounds of formu a I.C, wherein R2 is R2-- 15.5311 = Formu a 1 .3921 ).

Table 3922. Compounds of formu a I.C, wherein R2 is R2-- 15.5321 = Formu a 1 .3922).

Table 3923. Compounds of formu a I.C, wherein R2 is R2-- 15.5331 = Formu a 1 .3923).

Table 3924. Compounds of formu a I.C, wherein R2 is R2-- 15.5341 = Formu a 1 .3924).

Table 3925. Compounds of formu a I.C, wherein R2 is R2-- 15.5351 = Formu a 1 .3925).

Table 3926. Compounds of formu a I.C, wherein R2 is R2-- 15.5361 = Formu a 1 .3926).

Table 3927. Compounds of formu a I.C, wherein R2 is R2-- 15.5371 = Formu a 1 .3927).

Table 3928. Compounds of formu a I.C, wherein R2 is R2-- 15.5381 = Formu a 1 .3928).

Table 3929. Compounds of formu a I.C, wherein R2 is R2-- 15.5391 = Formu a 1 .3929).

Table 3930. Compounds of formu a I.C, wherein R2 is R2-- 15.5401 = Formu a 1 .3930).

Table 3931. Compounds of formu a I.C, wherein R2 is R2-- 15.5411 = Formu a 1 .3931 ).

Table 3932. Compounds of formu a I.C, wherein R2 is R2-- 15.5421 = Formu a 1 .3932).

Table 3933. Compounds of formu a I.C, wherein R2 is R2-- 15.5431 = Formu a 1 .3933).

Table 3934. Compounds of formu a I.C, wherein R2 is R2-- 15.5441 = Formu a 1 .3934).

Table 3935. Compounds of formu a I.C, wherein R2 is R2-- 15.5451 = Formu a 1 .3935).

Table 3936. Compounds of formu a I.C, wherein R2 is R2-- 15.5461 = Formu a 1 .3936).

Table 3937. Compounds of formu a I.C, wherein R2 is R2-- 15.5471 = Formu a 1 .3937).

Table 3938. Compounds of formu a I.C, wherein R2 is R2-- 15.5481 = Formu a 1 .3938).

Table 3939. Compounds of formu a I.C, wherein R2 is R2-- 15.5491 = Formu a 1 .3939).

Table 3940. Compounds of formu a I.C, wherein R2 is R2-- 15.5501 = Formu a 1 .3940).

Table 3941. Compounds of formu a I.C, wherein R2 is R2-- 15.5511 = Formu a 1 .3941 ).

Table 3942. Compounds of formu a I.C, wherein R2 is R2-- 15.5521 = Formu a 1 .3942).

Table 3943. Compounds of formu a I.C, wherein R2 is R2-- 15.5531 = Formu a 1 .3943). Table 3944. Compounds of formu a I.C, wherein R2 is R2-- I 5.554I = Formu a 1 .3944).

Table 3945. Compounds of formu a I.C, wherein R2 is R2-- I 5.555I = Formu a 1 .3945).

Table 3946. Compounds of formu a I.C, wherein R2 is R2-- I 5.556I = Formu a 1 .3946).

Table 3947. Compounds of formu a I.C, wherein R2 is R2-- I 5.557I = Formu a 1 .3947).

Table 3948. Compounds of formu a I.C, wherein R2 is R2-- I 5.558I = Formu a 1 .3948).

Table 3949. Compounds of formu a I.C, wherein R2 is R2-- I 5.559I = Formu a 1 .3949).

Table 3950. Compounds of formu a I.C, wherein R2 is R2-- I 5.560I = Formu a 1 .3950).

Table 3951. Compounds of formu a I.C, wherein R2 is R2-- 15.5611 = Formu a 1 .3951 ).

Table 3952. Compounds of formu a I.C, wherein R2 is R2-- 15.5621 = Formu a 1 .3952).

Table 3953. Compounds of formu a I.C, wherein R2 is R2-- 15.5631 = Formu a 1 .3953).

Table 3954. Compounds of formu a I.C, wherein R2 is R2-- 15.5641 = Formu a 1 .3954).

Table 3955. Compounds of formu a I.C, wherein R2 is R2-- 15.5651 = Formu a 1 .3955).

Table 3956. Compounds of formu a I.C, wherein R2 is R2-- 15.5661 = Formu a 1 .3956).

Table 3957. Compounds of formu a I.C, wherein R2 is R2-- 15.5671 = Formu a 1 .3957).

Table 3958. Compounds of formu a I.C, wherein R2 is R2-- 15.5681 = Formu a 1 .3958).

Table 3959. Compounds of formu a I.C, wherein R2 is R2-- 15.5691 = Formu a 1 .3959).

Table 3960. Compounds of formu a I.C, wherein R2 is R2-- 15.5701 = Formu a 1 .3960).

Table 3961. Compounds of formu a I.C, wherein R2 is R2-- 15.5711 = Formu a 1 .3961 ).

Table 3962. Compounds of formu a I.C, wherein R2 is R2-- 15.5721 = Formu a 1 .3962).

Table 3963. Compounds of formu a I.C, wherein R2 is R2-- 15.5731 = Formu a 1 .3963).

Table 3964. Compounds of formu a I.C, wherein R2 is R2-- 15.5741 = Formu a 1 .3964).

Table 3965. Compounds of formu a I.C, wherein R2 is R2-- 15.5751 = Formu a 1 .3965).

Table 3966. Compounds of formu a I.C, wherein R2 is R2-- 15.5761 = Formu a 1 .3966).

Table 3967. Compounds of formu a I.C, wherein R2 is R2-- 15.5771 = Formu a 1 .3967).

Table 3968. Compounds of formu a I.C, wherein R2 is R2-- 15.5781 = Formu a 1 .3968).

Table 3969. Compounds of formu a I.C, wherein R2 is R2-- 15.5791 = Formu a 1 .3969).

Table 3970. Compounds of formu a I.C, wherein R2 is R2-- 15.5801 = Formu a 1 .3970).

Table 3971. Compounds of formu a I.C, wherein R2 is R2-- 15.5811 = Formu a 1 .3971 ).

Table 3972. Compounds of formu a I.C, wherein R2 is R2-- 15.5821 = Formu a 1 .3972).

Table 3973. Compounds of formu a I.C, wherein R2 is R2-- 15.5831 = Formu a 1 .3973).

Table 3974. Compounds of formu a I.C, wherein R2 is R2-- 15.5841 = Formu a 1 .3974).

Table 3975. Compounds of formu a I.C, wherein R2 is R2-- 15.5851 = Formu a 1 .3975).

Table 3976. Compounds of formu a I.C, wherein R2 is R2-- 15.5861 = Formu a 1 .3976).

Table 3977. Compounds of formu a I.C, wherein R2 is R2-- 15.5871 = Formu a 1 .3977).

Table 3978. Compounds of formu a I.C, wherein R2 is R2-- 15.5881 = Formu a 1 .3978).

Table 3979. Compounds of formu a I.C, wherein R2 is R2-- 15.5891 = Formu a 1 .3979).

Table 3980. Compounds of formu a I.C, wherein R2 is R2-- 15.5901 = Formu a 1 .3980).

Table 3981. Compounds of formu a I.C, wherein R2 is R2-- 15.5911 = Formu a 1 .3981 ).

Table 3982. Compounds of formu a I.C, wherein R2 is R2-- 15.5921 = Formu a 1 .3982).

Table 3983. Compounds of formu a I.C, wherein R2 is R2-- 15.5931 = Formu a 1 .3983).

Table 3984. Compounds of formu a I.C, wherein R2 is R2-- 15.5941 = Formu a 1 .3984).

Table 3985. Compounds of formu a I.C, wherein R2 is R2-- 15.5951 = Formu a 1 .3985).

Table 3986. Compounds of formu a I.C, wherein R2 is R2-- 15.5961 = Formu a 1 .3986).

Table 3987. Compounds of formu a I.C, wherein R2 is R2-- 15.5971 = Formu a 1 .3987). Table 3988. Compounds of formu a I.C, wherein R2 is R2-- I 5.598I = Formu a 1 .3988).

Table 3989. Compounds of formu a I.C, wherein R2 is R2-- I 5.599I = Formu a 1 .3989).

Table 3990. Compounds of formu a I.C, wherein R2 is R2-- I 5.600I = Formu a 1 .3990).

Table 3991. Compounds of formu a I.C, wherein R2 is R2-- 15.6011 = Formu a 1 .3991 ).

Table 3992. Compounds of formu a I.C, wherein R2 is R2-- 15.6021 = Formu a 1 .3992).

Table 3993. Compounds of formu a I.C, wherein R2 is R2-- 15.6031 = Formu a 1 .3993).

Table 3994. Compounds of formu a I.C, wherein R2 is R2-- 15.6041 = Formu a 1 .3994).

Table 3995. Compounds of formu a I.C, wherein R2 is R2-- 15.6051 = Formu a 1 .3995).

Table 3996. Compounds of formu a I.C, wherein R2 is R2-- 15.6061 = Formu a 1 .3996).

Table 3997. Compounds of formu a I.C, wherein R2 is R2-- 15.6071 = Formu a 1 .3997).

Table 3998. Compounds of formu a I.C, wherein R2 is R2-- 15.6081 = Formu a 1 .3998).

Table 3999. Compounds of formu a I.C, wherein R2 is R2-- 15.6091 = Formu a 1 .3999).

Table 4000. Compounds of formu a I.C, wherein R2 is R2-- 15.6101 = Formu a 1 .4000).

Table 4001. Compounds of formu a I.C, wherein R2 is R2-- 15.61 11 = Formu a 1 .4001 ).

Table 4002. Compounds of formu a I.C, wherein R2 is R2-- 15.6121 = Formu a 1 .4002).

Table 4003. Compounds of formu a I.C, wherein R2 is R2-- 15.6131 = Formu a 1 .4003).

Table 4004. Compounds of formu a I.C, wherein R2 is R2-- 15.6141 = Formu a 1 .4004).

Table 4005. Compounds of formu a I.C, wherein R2 is R2-- 15.6151 = Formu a 1 .4005).

Table 4006. Compounds of formu a I.C, wherein R2 is R2-- 15.6161 = Formu a 1 .4006).

Table 4007. Compounds of formu a I.C, wherein R2 is R2-- 15.6171 = Formu a 1 .4007).

Table 4008. Compounds of formu a I.C, wherein R2 is R2-- 15.6181 = Formu a 1 .4008).

Table 4009. Compounds of formu a I.C, wherein R2 is R2-- 15.6191 = Formu a 1 .4009).

Table 4010. Compounds of formu a I.C, wherein R2 is R2-- 15.6201 = Formu a 1 .4010).

Table 401 1. Compounds of formu a I.C, wherein R2 is R2-- 15.6211 = Formu a 1 .401 1 ).

Table 4012. Compounds of formu a I.C, wherein R2 is R2-- 15.6221 = Formu a 1 .4012).

Table 4013. Compounds of formu a I.C, wherein R2 is R2-- 15.6231 = Formu a 1 .4013).

Table 4014. Compounds of formu a I.C, wherein R2 is R2-- 15.6241 = Formu a 1 .4014).

Table 4015. Compounds of formu a I.C, wherein R2 is R2-- 15.6251 = Formu a 1 .4015).

Table 4016. Compounds of formu a I.C, wherein R2 is R2-- 15.6261 = Formu a 1 .4016).

Table 4017. Compounds of formu a I.C, wherein R2 is R2-- 15.6271 = Formu a 1 .4017).

Table 4018. Compounds of formu a I.C, wherein R2 is R2-- 15.6281 = Formu a 1 .4018).

Table 4019. Compounds of formu a I.C, wherein R2 is R2-- 15.6291 = Formu a 1 .4019).

Table 4020. Compounds of formu a I.C, wherein R2 is R2-- 15.6301 = Formu a 1 .4020).

Table 4021. Compounds of formu a I.C, wherein R2 is R2-- 15.6311 = Formu a 1 .4021 ).

Table 4022. Compounds of formu a I.C, wherein R2 is R2-- 15.6321 = Formu a 1 .4022).

Table 4023. Compounds of formu a I.C, wherein R2 is R2-- 15.6331 = Formu a 1 .4023).

Table 4024. Compounds of formu a I.C, wherein R2 is R2-- 15.6341 = Formu a 1 .4024).

Table 4025. Compounds of formu a I.C, wherein R2 is R2-- 15.6351 = Formu a 1 .4025).

Table 4026. Compounds of formu a I.C, wherein R2 is R2-- 15.6361 = Formu a 1 .4026).

Table 4027. Compounds of formu a I.C, wherein R2 is R2-- 15.6371 = Formu a 1 .4027).

Table 4028. Compounds of formu a I.C, wherein R2 is R2-- 15.6381 = Formu a 1 .4028).

Table 4029. Compounds of formu a I.C, wherein R2 is R2-- 15.6391 = Formu a 1 .4029).

Table 4030. Compounds of formu a I.C, wherein R2 is R2-- 15.6401 = Formu a 1 .4030). Table 4031. Compounds of formu a I.C, wherein R2 is R2-- 15.6411 = Formu a 1 .4031 ). Table 4032. Compounds of formu a I.C, wherein R2 is R2- 15.642(=formula 1.4032).

Table 4033. Compounds of formu a I.C, wherein R2 is R2- 15.643(=formula 1.4033).

Table 4034. Compounds of formu a I.C, wherein R2 is R2- 15.644(=formula 1.4034).

Table 4035. Compounds of formu a I.C, wherein R2 is R2- 15.645(=formula 1.4035).

Table 4036. Compounds of formu a I.C, wherein R2 is R2- 15.646(=formula 1.4036).

Table 4037. Compounds of formu a I.C, wherein R2 is R2- 15.647(=formula 1.4037).

Table 4038. Compounds of formu a I.C, wherein R2 is R2- 15.648(=formula 1.4038).

Table 4039. Compounds of formu a I.C, wherein R2 is R2- 15.649(=formula 1.4039).

Table 4040. Compounds of formu a I.C, wherein R2 is R2- 15.650(=formula 1.4040).

Table 4041. Compounds of formu a I.C, wherein R2 is R2- 15.651 (=formula 1.4041).

Table 4042. Compounds of formu a I.C, wherein R2 is R2- 15.652(=formula 1.4042).

Table 4043. Compounds of formu a I.C, wherein R2 is R2- 15.653(=formula 1.4043).

Table 4044. Compounds of formu a I.C, wherein R2 is R2- 15.654(=formula 1.4044).

Table 4045. Compounds of formu a I.C, wherein R2 is R2- 15.655(=formula 1.4045).

Table 4046. Compounds of formu a I.C, wherein R2 is R2- 15.656(=formula 1.4046).

Table 4047. Compounds of formu a I.C, wherein R2 is R2- 15.657(=formula 1.4047).

Table 4048. Compounds of formu a I.C, wherein R2 is R2- 15.658(=formula 1.4048).

Table 4049. Compounds of formu a I.C, wherein R2 is R2- 15.659(=formula 1.4049).

Table 4050. Compounds of formu a I.C, wherein R2 is R2- 15.660(=formula 1.4050).

Table 4051. Compounds of formu a I.C, wherein R2 is R2- 15.661 (=formula 1.4051).

Table 4052. Compounds of formu a I.C, wherein R2 is R2- 15.662(=formula 1.4052).

Table 4053. Compounds of formu a I.C, wherein R2 is R2- 15.663(=formula 1.4053).

Table 4054. Compounds of formu a I.C, wherein R2 is R2- 15.664(=formula 1.4054).

Table 4055. Compounds of formu a I.C, wherein R2 is R2- 15.665(=formula 1.4055).

Table 4056. Compounds of formu a I.C, wherein R2 is R2- 15.666(=formula 1.4056).

Table 4057. Compounds of formu a I.C, wherein R2 is R2- 15.667(=formula 1.4057).

Table 4058. Compounds of formu a I.C, wherein R2 is R2- 15.668(=formula 1.4058).

Table 4059. Compounds of formu a I.C, wherein R2 is R2- 15.669(=formula 1.4059).

Table 4060. Compounds of formu a I.C, wherein R2 is R2- 15.670(=formula 1.4060).

Table 4061. Compounds of formu a I.C, wherein R2 is R2- 15.671 (=formula 1.4061).

Table 4062. Compounds of formu a I.C, wherein R2 is R2- 15.672(=formula 1.4062).

Table 4063. Compounds of formu a I.C, wherein R2 is R2- 15.673(=formula 1.4063).

Table 4064. Compounds of formu a I.C, wherein R2 is R2- 15.674(=formula 1.4064).

Table 4065. Compounds of formu a I.C, wherein R2 is R2- 15.675(=formula 1.4065).

Table 4066. Compounds of formu a I.C, wherein R2 is R2- 15.676(=formula 1.4066).

Table 4067. Compounds of formu a I.C, wherein R2 is R2- 9.1(=formula 1.4067).

Table 4068. Compounds of formu a I.C, wherein R2 is R2- 9.2(=formula 1.4068).

Table 4069. Compounds of formu a I.C, wherein R2 is R2- 9.3(=formula 1.4069).

Table 4070. Compounds of formu a I.C, wherein R2 is R2- 9.4(=formula 1.4070).

Table 4071. Compounds of formu a I.C, wherein R2 is R2- 9.5(=formula 1.4071).

Table 4072. Compounds of formu a I.C, wherein R2 is R2- 9.6(=formula 1.4072).

Table 4073. Compounds of formu a I.C, wherein R2 is R2- 9.7(=formula 1.4073).

Table 4074. Compounds of formu a I.C, wherein R2 is R2- 9.8(=formula 1.4074).

Table 4075. Compounds of formu a I.C, wherein R2 is R2- 9.9(=formula 1.4075). Table 4076 Compounds of formula I.C, wherein R 2 R 2 -9.10(=formula 1.4076). Table 4077 Compounds of formula I.C, wherein R 2 R 2 -9.11 (=formula 1.4077). Table 4078 Compounds of formula I.C, wherein R 2 R 2 -9.12(=formula 1.4078). Table 4079 Compounds of formula I.C, wherein R 2 R 2 -9.13(=formula 1.4079). Table 4080 Compounds of formula I.C, wherein R 2 R 2 -9.14(=formula 1.4080). Table 4081 Compounds of formula I.C, wherein R 2 R 2 -9.15(=formula 1.4081). Table 4082 Compounds of formula I.C, wherein R 2 R 2 -9.16(=formula 1.4082). TableA2:

The specific number for each single compound is deductible as follows:

Compound 1.2055.1-392 e.g. comprises the compound of formula 1.2055 from Table 2055 and line I-392 from Table A2; To widen the spectrum of action and to achieve synergistic effects, the pyrimidine compounds of formula (I) may be mixed with a large number of representatives of other herbicidal or growth- regulating active ingredient groups and then applied concomitantly. Suitable components for mixtures are, e.g., herbicides from the classes of the acetamides, amides,

aryloxyphenoxypropionat.es, benzamides, benzofuran, benzoic acids, benzothiadiazinones, bipyridylium, carbamates, chloroacetamides, chlorocarboxylic acids, cyclohexanediones, dinitroanilines, dinitrophenol, diphenyl ether, glycines, imidazolinones, isoxazoles,

isoxazolidinones, nitriles, N-phenylphthalimides, oxadiazoles, oxazolidinediones,

oxyacetamides, phenoxycarboxylic acids, phenylcarbamates, phenylpyrazoles,

phenylpyrazolines, phenylpyridazines, phosphinic acids, phosphoroamidates,

phosphorodithioates, phthalamates, pyrazoles, pyridazinones, pyridines, pyridinecarboxylic acids, pyridinecarboxamides, pyrimidinediones, pyrimidinyl(thio)benzoates, quinolinecarboxylic acids, semicarbazones, sulfonylaminocarbonyltriazolinones, sulfonylureas, tetrazolinones, thiadiazoles, thiocarbamates, triazines, triazinones, triazoles, triazolinones,

triazolocarboxamides, triazolopyrimidines, triketones, uracils, or ureas.

It may furthermore be beneficial to apply the pyrimidine compounds of formula (I) alone or in combination with other herbicides, or else in the form of a mixture with other crop protection agents, e.g. together with agents for controlling pests or phytopathogenic fungi or bacteria. Also of interest is the miscibility with mineral salt solutions, which are employed for treating nutritional and trace element deficiencies. Other additives such as non-phytotoxic oils and oil concentrates may also be added.

In one embodiment of the present invention the compositions according to the present invention comprise at least one pyrimidine compound of formula (I) (compound A) and at least one further active compound selected from herbicides B, preferably herbicides B of class b1) to b15), and safeners C (compound C).

In a preferred embodiment of the invention, the composition comprises as active compound A or component A at least one, preferably exactly one, pyrimidine compound of formula (1.1) (corresponds to pyrimidine compound of formula (I)), as defined herein;

In another preferred embodiment of the invention, the composition comprises as active compound A or component A at least one, preferably exactly one, pyrimidine compound of formula (1.2) (corresponds to pyrimidine compound of formula (I)), as defined herein;

In another preferred embodiment of the invention, the composition comprises as active compound A or component A at least one, preferably exactly one, pyrimidine compound of formula (1.3) (corresponds to pyrimidine compound of formula (I)), as defined herein;

In another preferred embodiment of the invention, the composition comprises as active compound A or component A at least one, preferably exactly one, pyrimidine compound of formula (1.4) (corresponds to pyrimidine compound of formula (I)), as defined herein;

In another preferred embodiment of the invention, the composition comprises as active compound A or component A at least one, preferably exactly one, pyrimidine compound of formula (1.5) (corresponds to pyrimidine compound of formula (I)), as defined herein; In another preferred embodiment of the invention, the composition comprises as active compound A or component A at least one, preferably exactly one, pyrimidine compound of formula (1.6) (corresponds to pyrimidine compound of formula (I)), as defined herein;

In another preferred embodiment of the invention, the composition comprises as active compound A or component A at least one, preferably exactly one, pyrimidine compound of formula (1.7) (corresponds to pyrimidine compound of formula (I)), as defined herein;

In another preferred embodiment of the invention, the composition comprises as active compound A or component A at least one, preferably exactly one, pyrimidine compound of formula (1.8) (corresponds to pyrimidine compound of formula (I)), as defined herein;

In another preferred embodiment of the invention, the composition comprises as active compound A or component A at least one, preferably exactly one, pyrimidine compound of formula (1.9) (corresponds to pyrimidine compound of formula (I)), as defined herein;

In another preferred embodiment of the invention, the composition comprises as active compound A or component A at least one, preferably exactly one, pyrimidine compound of formula (1.10) (corresponds to pyrimidine compound of formula (I)), as defined herein;

Preferred compounds of the formula (I) which, as component A, are constituent of the composition according to the invention are the compounds 1.1 to 1.10, as defined above;

In another embodiment of the present invention the compositions according to the present invention comprise at least one pyrimidine compound of formula (I) and at least one further active compound B (herbicide B).

The further herbicidal compound B (component B) is preferably selected from the herbicides of class b1) to b15):

Mixing partners for the composition can be selected from below herbicides B as defined below: B) herbicides of class b1) to b15):

b1) lipid biosynthesis inhibitors;

b2) acetolactate synthase inhibitors (ALS inhibitors);

b3) photosynthesis inhibitors;

b4) protoporphyrinogen-IX oxidase inhibitors (PPO inhibitors);

b5) bleacher herbicides;

b6) enolpyruvyl shikimate 3-phosphate synthase inhibitors (EPSP inhibitors);

b7) glutamine synthetase inhibitors;

b8) 7,8-dihydropteroate synthase inhibitors (DHP inhibitors);

b9) mitosis inhibitors;

b10) inhibitors of the synthesis of very long chain fatty acids (VLCFA inhibitors);

b11) cellulose biosynthesis inhibitors;

b12) decoupler herbicides;

b13) auxinic herbicides;

b14) auxin transport inhibitors; and

b15) other herbicides selected from the group consisting of bromobutide, chlorflurenol, chlorflurenol-methyl, cinmethylin, cumyluron, dalapon, dazomet, difenzoquat, difenzoquat- metilsulfate, dimethipin, DSMA, dymron, endothal and its salts, etobenzanid, flamprop, flamprop-isopropyl, flamprop-methyl, flamprop-M-isopropyl, flamprop-M-methyl, flurenol, flurenol-butyl, flurprimidol, fosamine, fosamine-ammonium, indanofan, indaziflam, maleic hydrazide, mefluidide, metam, methiozolin (CAS 403640-27-7), methyl azide, methyl bromide, methyl-dymron, methyl iodide, MSMA, oleic acid, oxaziclomefone, pelargonic acid, pyributicarb, quinoclamine, triaziflam, tridiphane and 6-chloro-3-(2-cyclopropyl-6-methylphenoxy)-4- pyridazinol (CAS 499223-49-3) and its salts and esters;

including their agriculturally acceptable salts or derivatives;

In one embodiment of the invention, the compositions contain at least one inhibitor of the lipid biosynthesis (herbicide b1). These compounds inhibit lipid biosynthesis. Inhibition of the lipid biosynthesis can be affected either through inhibition of acetylCoA carboxylase (hereinafter- termed ACCase herbicides) or through a different mode of action (hereinafter termed non- ACCase herbicides). The ACCase herbicides belong to the group A of the HRAC classification system whereas the non-ACCase herbicides belong to the group N of the HRAC classification. In another embodiment of the invention, the compositions contain at least one ALS inhibitor (herbicide b2). The herbicidal activity of these compounds is based on the inhibition of acetolactate synthase and thus on the inhibition of the branched chain amino acid biosynthesis. These inhibitors belong to the group B of the HRAC classification system.

In another embodiment of the invention, the compositions contain at least one inhibitor of photosynthesis (herbicide b3). The herbicidal activity of these compounds is based either on the inhibition of the photosystem II in plants (so-called PSII inhibitors, groups C1 , C2 and C3 of HRAC classification) or on diverting the electron transfer in photosystem I in plants (so-called PSI inhibitors, group D of HRAC classification) and thus on an inhibition of photosynthesis. Amongst these, PSII inhibitors are preferred.

In another embodiment of the invention, the compositions contain at least one inhibitor of protoporphyrinogen-IX-oxidase (herbicide b4). The herbicidal activity of these compounds is based on the inhibition of the protoporphyrinogen-IX-oxidase. These inhibitors belong to the group E of the HRAC classification system.

In another embodiment of the invention, the compositions contain at least one bleacher- herbicide (herbicide b5). The herbicidal activity of these compounds is based on the inhibition of the carotenoid biosynthesis. These include compounds which inhibit carotenoid biosynthesis by inhibition of phytoene desaturase (so-called PDS inhibitors, group F1 of HRAC classification), compounds that inhibit the 4-hydroxyphenylpyruvate-dioxygenase (HPPD inhibitors, group F2 of HRAC classification), compounds that inhibit DOXsynthase (group F4 of HRAC class) and compounds which inhibit carotenoid biosynthesis by an unknown mode of action (bleacher - unknown target, group F3 of HRAC classification).

In another embodiment of the invention, the compositions contain at least one EPSP synthase inhibitor (herbicide b6). The herbicidal activity of these compounds is based on the inhibition of enolpyruvyl shikimate 3-phosphate synthase, and thus on the inhibition of the amino acid biosynthesis in plants. These inhibitors belong to the group G of the HRAC classification system.

In another embodiment of the invention, the compositions contain at least one glutamine synthetase inhibitor (herbicide b7). The herbicidal activity of these compounds is based on the inhibition of glutamine synthetase, and thus on the inhibition of the aminoacid biosynthesis in plants. These inhibitors belong to the group H of the HRAC classification system.

In another embodiment of the invention, the compositions contain at least one DHP synthase inhibitor (herbicide b8). The herbicidal activity of these compounds is based on the inhibition of 7,8-dihydropteroate synthase. These inhibitors belong to the group I of the HRAC classification system.

In another embodiment of the invention, the compositions contain at least one mitosis inhibitor (herbicide b9). The herbicidal activity of these compounds is based on the disturbance or inhibition of microtubule formation or organization, and thus on the inhibition of mitosis. These inhibitors belong to the groups K1 and K2 of the HRAC classification system. Among these, compounds of the group K1 , in particular dinitroanilines, are preferred.

In another embodiment of the invention, the compositions contain at least one VLCFA inhibitor (herbicide b10). The herbicidal activity of these compounds is based on the inhibition of the synthesis of very long chain fatty acids and thus on the disturbance or inhibition of cell division in plants. These inhibitors belong to the group K3 of the HRAC classification system.

In another embodiment of the invention, the compositions contain at least one cellulose biosynthesis inhibitor (herbicide b11). The herbicidal activity of these compounds is based on the inhibition of the biosynthesis of cellulose and thus on the inhibition of the synthesis of cell walls in plants. These inhibitors belong to the group L of the HRAC classification system.

In another embodiment of the invention, the compositions contain at least one decoupler herbicide (herbicide b12). The herbicidal activity of these compounds is based on the disruption of the cell membrane. These inhibitors belong to the group M of the HRAC classification system.

In another embodiment of the invention, the compositions contain at least one auxinic herbicide (herbicide b13). These include compounds that mimic auxins, i.e. plant hormones, and affect the growth of the plants. These compounds belong to the group O of the HRAC classification system.

In another embodiment of the invention, the compositions contain at least one auxin transport inhibitor (herbicide b14). The herbicidal activity of these compounds is based on the inhibition of the auxin transport in plants. These compounds belong to the group P of the HRAC

classification system.

As to the given mechanisms of action and classification of the active substances, see e.g. "HRAC, Classification of Herbicides According to Mode of Action",

http://www.plantprotection.org/hrac/MOA.html).

Preference is given to those compositions according to the present invention comprising at least one herbicide B selected from herbicides of class b1 , b2, b3, b4, b5, b6, b9, b10, b13, and b14.

Specific preference is given to those compositions according to the present invention which comprise at least one herbicide B selected from the herbicides of class b1 , b2, b4, b5, b9, b10, b13, and b14.

Particular preference is given to those compositions according to the present invention which comprise at least one herbicide B selected from the herbicides of class b1 , b2, b4, b5, b9, b10, and b13

Examples of herbicides B which can be used in combination with the compound of formula (I) according to the present invention are:

b1) from the group of the lipid biosynthesis inhibitors:

ACC-herbicides such as alloxydim, alloxydim-sodium, butroxydim, clethodim, clodinafop, clodinafop-propargyl, cycloxydim, cyhalofop, cyhalofop-butyl, diclofop, diclofop-methyl, fenoxaprop, fenoxaprop-ethyl, fenoxaprop-P, fenoxaprop-P-ethyl, fluazifop, fluazifop-butyl, fluazifop-P, fluazifop-P-butyl, haloxyfop, haloxyfop-methyl, haloxyfop-P, haloxyfop-P-methyl, metamifop, pinoxaden, profoxydim, propaquizafop, quizalofop, quizalofop-ethyl, quizalofop- tefuryl, quizalofop-P, quizalofop-P-ethyl, quizalofop-P-tefuryl, sethoxydim, tepraloxydim, tralkoxydim,

4-(4'-Chloro-4-cyclopropyl-2'-fluoro[1 ,1 '-biphenyl]-3-yl)-5-hydroxy-2,2,6,6-tetramethyl-2H- pyran-3(6H)-one (CAS 1312337-72-6); 4-(2',4 , -Dichloro-4-cyclopropyl[1 ,1 , -biphenyl]-3-yl)-5- hydroxy-2,2,6,6-tetramethyl-2H-pyran-3(6H)-one (CAS 1312337-45-3); 4-(4'-Chloro-4-ethyl-2'- fluoro[1 ,1'-biphenyl]-3-yl)-5-hydroxy-2,2,6,6-tetramethyl-2H-pyran-3 (6H)-one (CAS 1033757-93- 5); 4-(2\4 , -Dichloro-4-ethyl[1 ,1 , -biphenyl]-3-yl)-2,2,6,6-tetramethyl-2H-pyran-3,5(4H,6 H)^^ (CAS 1312340-84-3); 5-(Acetyloxy)-4-(4'-chloro-4-cyclopropyl-2'-fluoro[1 ,1'-biphenyl]-3-yl)-3,6- dihydro-2,2,6,6-tetramethyl-2H-pyran-3-one (CAS 1312337-48-6); 5-(Acetyloxy)-4-(2 ' ,4'- dichloro-4-cyclopropyl- [1 ,1 '-biphenyl]-3-yl)-S.e-dihydro-2,2 e.e-tetramethyl-2H-pyran-3-one; 5- (Acetyloxy)-4-(4'-chloro-4-ethyl-2 , -fluoro[1 ,1 , -biphenyl]-3-yl)-3,6-dihydro-2,2,6,6-tetramethyl-2H- pyran-3-one (CAS 1312340-82-1); 5-(Acetyloxy)-4-(2',4'-dichloro-4-ethyl[1 ,1'-biphenyl]-3-yl)-3,6- dihydro-2,2,6,6-tetramethyl-2H-pyran-3-one (CAS 1033760-55-2); 4-(4'-Chloro-4-cyclopropyl-2'- fluoro[1 ,1 '-biphenyl]-3-yl)-5,6-dihydro-2,2 6.6-tetramethyl-3-oxo-2H-pyran-3-yl carbonic acid methyl ester (CAS 1312337-51-1); 4-(2 ' ,4'-Dichloro -4-cyclopropyl- [1 ,1'-biphenyl]-3-yl)-5,6- dihydro-2,2,6,6-tetramethyl-5-oxo-2H-pyran-3-yl carbonic acid methyl ester; 4-(4'-Chloro-4- ethyl-2'-fluorotl .l'-biphenyll-3-yl)-5,6-dihydro-2,2 e.e-tetramethyl-S-oxo-2H-pyran-3-yl carbonic acid methyl ester (CAS 1312340-83-2); 4-(2',4'-Dichloro-4-ethyl[1 ,1'-biphenyl]-3-yl)-5,6-dihydro- 2,2,6,6-tetramethyl-5-oxo-2H-pyran-3-yl carbonic acid methyl ester (CAS 1033760-58-5); and non ACC herbicides such as benfuresate, butylate, cycloate, dalapon, dimepiperate, EPTC, esprocarb, ethofumesate, flupropanate, molinate, orbencarb, pebulate, prosulfocarb, TCA, thiobencarb, tiocarbazil, triallate and vernolate;

b2) from the group of the ALS inhibitors:

sulfonylureas such as amidosulfuron, azimsulfuron, bensulfuron, bensulfuron-methyl, chlorimuron, chlorimuron-ethyl, chlorsulfuron, cinosulfuron, cyclosulfamuron, ethametsulfuron, ethametsulfuron-methyl, ethoxysulfuron, flazasulfuron, flucetosulfuron, flupyrsulfuron, flupyrsulfuron-methyl-sodium, foramsulfuron, halosulfuron, halosulfuron-methyl, imazosulfuron, iodosulfuron, iodosulfuron-methyl-sodium, iofensulfuron, iofensulfuron-sodium, mesosulfuron, metazosulfuron, metsulfuron, metsulfuron-methyl, nicosulfuron, orthosulfamuron, oxasulfuron, primisulfuron, primisulfuron-methyl, propyrisulfuron, prosulfuron, pyrazosulfuron,

pyrazosulfuron-ethyl, rimsulfuron, sulfometuron, sulfometuron-methyl, sulfosulfuron,

thifensulfuron, thifensulfuron-methyl, triasulfuron, tribenuron, tribenuron-methyl, trifloxysulfuron, triflusulfuron, triflusulfuron-methyl and tritosulfuron,

imidazolinones such as imazamethabenz, imazamethabenz-methyl, imazamox, imazapic, imazapyr, imazaquin and imazethapyr, triazolopyrimidine herbicides and sulfonanilides such as cloransulam, cloransulam-methyl, diclosulam, flumetsulam, florasulam, metosulam,

penoxsulam, pyrimisulfan and pyroxsulam,

pyrimidinylbenzoates such as bispyribac, bispyribac-sodium, pyribenzoxim, pyriftalid, pyriminobac, pyriminobac-methyl, pyrithiobac, pyrithiobac-sodium, 4-[[[2-[(4,6-dimethoxy-2- pyrimidinyl)oxy]phenyl]methyl]amino]-benzoic acid-1-methylethyl ester (CAS 420138-41-6), 4- [[[2-[(4,6-dimethoxy-2-pyrimidinyl)oxy]phenyl]methyl]amino]- benzoic acid propyl ester (CAS 420138-40-5), N-(4-bromophenyl)-2-[(4,6-dimethoxy-2-pyrimidinyl)oxy]benzen emethanamine (CAS 420138-01-8),

sulfonylaminocarbonyl-triazolinone herbicides such as flucarbazone, flucarbazone-sodium, propoxycarbazone, propoxycarbazone-sodium, thiencarbazone and thiencarbazone-methyl; and triafamone;

among these, a preferred embodiment of the invention relates to those compositions comprising at least one imidazolinone herbicide;

b3) from the group of the photosynthesis inhibitors:

amicarbazone, inhibitors of the photosystem II, e.g. 1-(6-tert-butylpyrimidin-4-yl)-2-hydroxy-4- methoxy-3-methyl-2H-pyrrol-5-one (CAS 1654744-66-7), 1-(5-tert-butylisoxazol-3-yl)-2-hydroxy- 4-methoxy-3-methyl-2H-pyrrol-5-one (CAS 1637455-12-9), 1-(5-tert-butylisoxazol-3-yl)-4-chloro- 2-hydroxy-3-methyl-2H-pyrrol-5-one (CAS 1637453-94-1), 1-(5-tert-butyl-1-methyl-pyrazol-3-yl)- 4-chloro-2-hydroxy-3-methyl-2H-pyrrol-5-one (CAS 1654057-29-0), 1-(5-tert-butyl-1-methyl- pyrazol-3-yl)-3-chloro-2-hydroxy-4-methyl-2H-pyrrol-5-one (CAS 1654747-80-4), 4-hydroxy-1- methoxy-5-methyl-3-[4-(trifluoromethyl)-2-pyridyl]imidazolid in-2-one; (CAS 2023785-78-4), 4- hydroxy-1 ,5-dimethyl-3-[4-(trifluoromethyl)-2-pyridyl]imidazolidin-2- one (CAS 2023785-79-5), 5- ethoxy-4-hydroxy-1 -methyl-3-[4-(trifluoromethyl)-2-pyridyl]imidazolidin-2-one (CAS 1701416-69- 4), 4-hydroxy-1-methyl-3-[4-(trifluoromethyl)-2-pyridyl]imidazol idin-2-one (CAS 1708087-22-2), 4-hydroxy-1 ,5-dimethyl-3-[1 -methyl-5-(trifluoromethyl)pyrazol-3-yl]imidazolidin-2-one (CAS 2023785-80-8), 1-(5-tert-butylisoxazol-3-yl)-4-ethoxy-5-hydroxy-3-methyl-im idazolidin-2-one (CAS 1844836-64-1), triazine herbicides, including of chlorotriazine, triazinones, triazindiones, methylthiotriazines and pyridazinones such as ametryn, atrazine, chloridazone, cyanazine, des- metryn, dimethametryn.hexazinone, metribuzin, prometon, prometryn, propazine, simazine, simetryn, terbumeton, terbuthylazin, terbutryn and trietazin, aryl urea such as chlorobromuron, chlorotoluron, chloroxuron, dimefuron, diuron, fluometuron, isoproturon, isouron, linuron, metamitron, methabenzthiazuron, metobenzuron, metoxuron, monolinuron, neburon, siduron, tebuthiuron and thiadiazuron, phenyl carbamates such as desmedipham, karbutilat,

phenmedipham, phenmedipham-ethyl, nitrile herbicides such as bromofenoxim, bromoxynil and its salts and esters, ioxynil and its salts and esters, uraciles such as bromacil, lenacil and terbacil, and bentazon and bentazon-sodium, pyridate, pyridafol, pentanochlor and propanil and inhibitors of the photosystem I such as diquat, diquat-dibromide, paraquat, paraquat-dichloride and paraquat-dimetilsulfate. Among these, a preferred embodiment of the invention relates to those compositions comprising at least one aryl urea herbicide. Among these, likewise a preferred embodiment of the invention relates to those compositions comprising at least one triazine herbicide. Among these, likewise a preferred embodiment of the invention relates to those compositions comprising at least one nitrile herbicide;

b4) from the group of the protoporphyrinogen-IX oxidase inhibitors:

acifluorfen, acifluorfen-sodium, azafenidin, bencarbazone, benzfendizone, bifenox, butafenacil, carfentrazone, carfentrazone-ethyl, chlomethoxyfen, chlorphthalim, cinidon-ethyl, fluazolate, flufenpyr, flufenpyr-ethyl, flumiclorac, flumiclorac-pentyl, flumioxazin, fluoroglycofen,

fluoroglycofen-ethyl, fluthiacet, fluthiacet-methyl, fomesafen, halosafen, lactofen, oxadiargyl, oxadiazon, oxyfluorfen, pentoxazone, profluazol, pyraclonil, pyraflufen, pyraflufen-ethyl, saflufenacil, sulfentrazone, thidiazimin, tiafenacil, trifludimoxazin, ethyl [3-[2-chloro-4-fluoro-5-(1- methyl-6-trifluoromethyl-2,4-dioxo-1 ,2,3,4-tetrahydropyrimidin-3-yl)phenoxy]-2- pyridyloxy]acetate (CAS 353292-31-6; S-3100), N-ethyl-3-(2,6-dichloro-4-trifluoro- methylphenoxy)-5-methyl-1 H-pyrazole-1-carboxamide (CAS 452098-92-9), N-tetrahydrofurfuryl- 3-(2,6-dichloro-4-trifluoromethylphenoxy)-5-methyl-1 H-pyrazole-1-carboxamide (CAS 915396- 43-9), N-ethyl-3-(2-chloro-6-fluoro-4-trifluoromethylphenoxy)-5-meH t-hyl-1 pyrazole-1- carboxamide (CAS 452099-05-7), N-tetrahydrofurfuryl-3-(2-chloro-6-fluoro-4-trifluoro- methylphenoxy)-5-methyl-1 H-pyrazole-1-carboxamide (CAS 452100-03-7), 3-[7-fluoro-3-oxo-4- (prop-2-ynyl)-3,4-dihydro-2H-benzo[1 ,4]oxazin-6-yl]-1 ,5-dimethyl-6-thioxo-[1 ,3,5]triazinan-2,4- dione (CAS 451484-50-7), 2-(2,2,7-trifluoro-3-oxo-4-prop-2-ynyl-3,4-dihydro-2H- benzo[1 ,4]oxazin-6-yl)-4,5,6,7-tetrahydro-isoindole-1 ,3-dione (CAS 1300118-96-0), 1 -methyl-6- trifluoromethyl-3-(2,2,7-trifluoro-3-oxo-4-prop-2-ynyl-3,4-d ihydro-2H-benzo[1 ,4]oxazin-6-yl)-1 H- pyrimidine-2,4-dione (CAS 1304113-05-0), methyl (E)-4-[2-chloro-5-[4-chloro-5- (difluoromethoxy)H--1 methyl-pyrazol-3-yl]-4-fluoro-phenoxy]-3-methoxy-but-2-enoat e (CAS 948893-00-3), and 3-[7-chloro-5-fluoro-2-(trifluoromethyl)-1 H-benzimidazol-4-yl]-1-methyl-6- (trifluoromethyl)-1 H-pyrimidine-2,4-dione (CAS 212754-02-4);

b5) from the group of the bleacher herbicides:

PDS inhibitors: beflubutamid, diflufenican, fluridone, flurochloridone, flurtamone, norflurazon, picolinafen, and 4-(3-trifluoromethylphenoxy)-2-(4-trifluoromethylphenyl)pyri midine (CAS 180608-33-7), HPPD inhibitors: benzobicyclon, benzofenap, bicyclopyrone, clomazone, fenquinotrione, isoxaflutole, mesotrione, oxotrione (CAS 1486617-21-3), pyrasulfotole, pyrazolynate, pyrazoxyfen, sulcotrione, tefuryltrione, tembotrione, tolpyralate, topramezone , bleacher, unknown target: aclonifen, amitrole flumeturon,2-chloro-3-methylsulfanyl-N-(1- methyltetrazol-5-yl)-4-(trifluoromethyl)benzamide (CAS 1361139-71-0), 2-(2,4- dichlorophenyl)methyl-4,4-dimethyl-3-isoxazolidone (CAS 81777-95-9) and 2-(2,5- dichlorophenyl)methyl-4,4-dimethyl-3-isoxazolidinone (CAS 81778-66-7);

b6) from the group of the EPSP synthase inhibitors: glyphosate, glyphosate- isopropylammonium, glyposate-potassium and glyphosate-trimesium (sulfosate);

b7) from the group of the glutamine synthase inhibitors: bilanaphos (bialaphos), bilanaphos- sodium, glufosinate, glufosinate-P and glufosinate-ammonium;

b8) from the group of the DHP synthase inhibitors: asulam;

b9) from the group of the mitosis inhibitors:

compounds of group K1 : dinitroanilines such as benfluralin, butralin, dinitramine, ethalfluralin, fluchloralin, oryzalin, pendimethalin, prodiamine and trifluralin, phosphoramidates such as amiprophos, amiprophos-methyl, and butamiphos, benzoic acid herbicides such as chlorthal, chlorthal-dimethyl, pyridines such as dithiopyr and thiazopyr, benzamides such as propyzamide and tebutam; compounds of group K2: carbetamide, chlorpropham, flamprop, flamprop- isopropyl, flam prop-methyl, flamprop-M-isopropyl, flamprop-M-methyl and propham ; among these, compounds of group K1 , in particular dinitroanilines are preferred;

b10) from the group of the VLCFA inhibitors:

chloroacetamides such as acetochlor, alachlor, amidochlor, butachlor, dimethachlor, dimethenamid, dimethenamid-P, metazachlor, metolachlor, metolachlor-S, pethoxamid, pretilachlor, propachlor, propisochlor and thenylchlor, oxyacetanilides such as flufenacet and mefenacet, acetanilides such as diphenamid, naproanilide, napropamide and napropamide-M, tetrazolinones such fentrazamide, and other herbicides such as anilofos, cafenstrole, fenoxasulfone, ipfencarbazone, piperophos, pyroxasulfone and isoxazoline compounds of the formulae 11.1 , II.2, II.3, II.4, II.5, II.6, II.7, II .8 and II.9

the isoxazoline compounds are known in the art, e.g. from WO 2006/024820, WO

2006/037945, WO 2007/071900 and WO 2007/096576;

among the VLCFA inhibitors, preference is given to chloroacetamides and oxyacetamides; b11) from the group of the cellulose biosynthesis inhibitors: chlorthiamid, dichlobenil, flupoxam, indaziflam, isoxaben, triaziflam and 1-cyclohexyl-5-pentafluorphenyloxy-1 4 - [1 ,2,4,6]thiatriazin-3-ylamine (CAS 175899-01-1);

b12) from the group of the decoupler herbicides: dinoseb, dinoterb and DNOC and its salts; b13) from the group of the auxinic herbicides:

2,4-D and its salts and esters such as clacyfos, 2,4-DB and its salts and esters,

aminocyclopyrachlor and its salts and esters, aminopyralid and its salts such as aminopyralid- dimethylammonium, aminopyralid-tris(2-hydroxypropyl)ammonium and its esters, benazolin, benazolin-ethyl, chloramben and its salts and esters, clomeprop, clopyralid and its salts and esters, dicamba and its salts and esters, dichlorprop and its salts and esters, dichlorprop-P and its salts and esters, flopyrauxifen, fluroxypyr, fluroxypyr-butometyl, fluroxypyr-meptyl, halauxifen and its salts and esters (CAS 943832-60-8); MCPA and its salts and esters, MCPA-thioethyl, MCPB and its salts and esters, mecoprop and its salts and esters, mecoprop-P and its salts and esters, picloram and its salts and esters, quinclorac, quinmerac, TBA (2,3,6) and its salts and esters, triclopyr and its salts and esters, florpyrauxifen, florpyrauxifen-benzyl (CAS 1390661-72- 9) and 4-amino-3-chloro-5-fluoro-6-(7-fluoro-1 H-indol-6-yl)picolinic acid (CAS 1629965-65-6); b14) from the group of the auxin transport inhibitors: diflufenzopyr, diflufenzopyr-sodium, naptalam and naptalam-sodium;

b15) from the group of the other herbicides: bromobutide, chlorflurenol, chlorflurenol-methyl, cinmethylin, cumyluron, cyclopyrimorate (CAS 499223-49-3 and its salts and esters, dalapon, dazomet, difenzoquat, difenzoquat-metilsulfate, dimethipin, DSMA, dymron, endothal and its salts, etobenzanid, flurenol, flurenol-butyl, flurprimidol, fosamine, fosamine-ammonium, indanofan, maleic hydrazide, mefluidide, metam, methiozolin (CAS 403640-27-7), methyl azide, methyl bromide, methyl-dymron, methyl iodide, MSMA, oleic acid, oxaziclomefone, pelargonic acid, pyributicarb, quinoclamine and tridiphane.

Preferred herbicides B that can be used in combination with the pyrimidine compounds of the formula (I) according to the present invention are:

b1) from the group of the lipid biosynthesis inhibitors:

clethodim, clodinafop-propargyl, cycloxydim, cyhalofop-butyl, diclofop-methyl, fenoxaprop-P- ethyl, fluazifop-P-butyl, haloxyfop-P-methyl, metamifop, pinoxaden, profoxydim, propaquizafop, quizalofop-P-ethyl, quizalofop-P-tefuryl, sethoxydim, tepraloxydim, tralkoxydim, 4-(4'-Chloro-4- cyclopropyl-2'-fluoro[1 ,1'-biphenyl]-3-yl)-5-hydroxy-2,2,6,6-tetramethyl-2H-pyran-3 (6H)-one (CAS 1312337-72-6); 4-(2',4'-Dichloro-4-cyclopropyl[1 ,1'-biphenyl]-3-yl)-5-hydroxy-2,2,6,6- tetramethyl-2H-pyran-3(6H)-one (CAS 1312337-45-3); 4-(4 , -Chloro-4-ethyl-2 , -fluoro[1 ,1'- biphenyl]-3-yl)-5-hydroxy-2,2,6,6-tetramethyl-2H-pyran-3(6H) -one (CAS 1033757-93-5); 4-(2',4'- Dichloro-4-ethyl[1 ,1'-biphenyl]-3-yl)-2,2,6,6-tetramethyl-2H-pyran-3,5(4H,6H)- dione (CAS 1312340-84-3); 5-(Acetyloxy)-4-(4'-chloro-4-cyclopropyl-2'-fluoro[1 ,1 '-biphenyl]-3-yl)-3,6- dihydro-2,2,6,6-tetramethyl-2H-pyran-3-one (CAS 1312337-48-6); 5-(Acetyloxy)-4-(2 ' ,4'- dichloro-4-cyclopropyl- [1 ,1 '-biphenyl]-3-yl)-3,6-dihydro-2,2,6,6-tetramethyl-2H-pyran-3 -one; 5- (Acetyloxy)-4-(4'-chloro-4-ethyl-2 , -fluoro[1 ,1'-biphenyl]-3-yl)-3,6-dihydro-2,2,6,6-tetramethyl-2H- pyran-3-one (CAS 1312340-82-1); 5-(Acetyloxy)-4-(2',4'-dichloro-4-ethyl[1 ,1'-biphenyl]-3-yl)-3,6- dihydro-2,2,6,6-tetramethyl-2H-pyran-3-one (CAS 1033760-55-2); 4-(4'-Chloro-4-cyclopropyl-2'- fluoro[1 ,1 '-biphenyl]-3-yl)-5,6-dihydro-2,2,6,6-tetramethyl-5-oxo-2H-p yran-3-yl carbonic acid methyl ester (CAS 1312337-51-1); 4-(2 ' ,4'-Dichloro -4-cyclopropyl- [1 ,1'-biphenyl]-3-yl)-5,6- dihydro-2,2,6,6-tetramethyl-5-oxo-2H-pyran-3-yl carbonic acid methyl ester; 4-(4'-Chloro-4- ethyl-2'-fluoro[1 ,1 '-biphenyl]-3-yl)-5,6-dihydro-2,2,6,6-tetramethyl-5-oxo-2H-p yran-3-yl carbonic acid methyl ester (CAS 1312340-83-2); 4-(2',4 , -Dichloro-4-ethyl[1 ,1 , -biphenyl]-3-yl)-5,6-dihydro- 2,2,6,6-tetramethyl-5-oxo-2H-pyran-3-yl carbonic acid methyl ester (CAS 1033760-58-5);

benfuresate, dimepiperate, EPTC, esprocarb, ethofumesate, molinate, orbencarb, prosulfocarb, thiobencarb and triallate;

b2) from the group of the ALS inhibitors:

amidosulfuron, azimsulfuron, bensulfuron-methyl, bispyribac-sodium, chlorimuron-ethyl, chlorsulfuron, cloransulam-methyl, cyclosulfamuron, diclosulam, ethametsulfuron-methyl, ethoxysulfuron, flazasulfuron, florasulam, flucarbazone-sodium, flucetosulfuron, flumetsulam, flupyrsulfuron-methyl-sodium, foramsulfuron, halosulfuron-methyl, imazamethabenz-methyl, imazamox, imazapic, imazapyr, imazaquin, imazethapyr, imazosulfuron, iodosulfuron, iodosulfuron-methyl-sodium, iofensulfuron, iofensulfuron-sodium, mesosulfuron,

metazosulfuron, metosulam, metsulfuron-methyl, nicosulfuron, orthosulfamuron, oxasulfuron, penoxsulam, primisulfuron-methyl, propoxycarbazon-sodium, propyrisulfuron, prosulfuron, pyrazosulfuron-ethyl, pyribenzoxim, pyrimisulfan, pyriftalid, pyriminobac-methyl, pyrithiobac- sodium, pyroxsulam, rimsulfuron, sulfometuron-methyl, sulfosulfuron, thiencarbazone-methyl, thifensulfuron-methyl, triasulfuron, tribenuron-methyl, trifloxysulfuron, triflusulfuron-methyl, tritosulfuron and triafamone;

b3) from the group of the photosynthesis inhibitors: ametryn, amicarbazone, atrazine, bentazone, bentazone-sodium, bromoxynil and its salts and esters, chloridazone, chlorotoluron, cyanazine, desmedipham, diquat-dibromide, diuron, fluometuron, hexazinone, ioxynil and its salts and esters, isoproturon, lenacil, linuron, metamitron, methabenzthiazuron, metribuzin, paraquat, paraquat-dichloride, phenmedipham, propanil, pyridate, simazine, terbutryn, terbuthylazine, thidiazuron, 1-(6-tert-butylpyrimidin-4-yl)-

2- hydroxy-4-methoxy-3-methyl-2H-pyrrol-5-one (CAS 1654744-66-7), 1-(5-tert-butylisoxazol-3- yl)-2-hydroxy-4-methoxy-3-methyl-2H-pyrrol-5-one (CAS 1637455-12-9), 1-(5-tert-butylisoxazol-

3- yl)-4-chloro-2-hydroxy-3-methyl-2H-pyrrol-5-one (CAS 1637453-94-1), 1-(5-tert-butyl-1- methyl-pyrazol-3-yl)-4-chloro-2-hydroxy-3-methyl-2H-pyrrol-5 -one (CAS 1654057-29-0), 1-(5- tert-butyl-1-methyl-pyrazol-3-yl)-3-chloro-2-hydroxy-4-methy l-2H-pyrrol-5-one (CAS 1654747- 80-4), 4-hydroxy-1 -methoxy-5-methyl-3-[4-(trifluoromethyl)-2-pyridyl]imidazoli din-2-one; (CAS 2023785-78-4), 4-hydroxy-1 ,5-dimethyl-3-[4-(trifluoromethyl)-2-pyridyl]imidazolidin-2- one (CAS 2023785-79-5), 5-ethoxy-4-hydroxy-1-methyl-3-[4-(trifluoromethyl)-2-pyridyl ]imidazolidin-2-one (CAS 1701416-69-4), 4-hydroxy-1-methyl-3-[4-(trifluoromethyl)-2-pyridyl]imidazol idin-2-one (CAS 1708087-22-2), 4-hydroxy-1 ,5-dimethyl-3-[1-methyl-5-(trifluoromethyl)pyrazol-3- yl]imidazolidin-2-one (CAS 2023785-80-8) and 1-(5-tert-butylisoxazol-3-yl)-4-ethoxy-5-hydroxy- 3-methyl-imidazolidin-2-one (CAS 1844836-64-1);

b4) from the group of the protoporphyrinogen-IX oxidase inhibitors:

acifluorfen-sodium, bencarbazone, benzfendizone, butafenacil, carfentrazone-ethyl, cinidon- ethyl, flufenpyr-ethyl, flumiclorac-pentyl, flumioxazin, fluoroglycofen-ethyl, fomesafen, lactofen, oxadiargyl, oxadiazon, oxyfluorfen, pentoxazone, pyraflufen, pyraflufen-ethyl, saflufenacil, sulfentrazone, tiafenacil, trifludimoxazin, ethyl [3-[2-chloro-4-fluoro-5-(1-methyl-6-trifluoromethyl- 2,4-dioxo-1 ,2,3,4-tetrahydropyrimidin-3-yl)phenoxy]-2-pyridyloxy]acetat e (CAS 353292-31-6; S- 3100), N-ethyl-3-(2,6-dichloro-4-trifluoromethylphenoxy)-5-methyl-1 H-pyrazole-1-carboxamide (CAS 452098-92-9), N-tetrahydrofurfuryl-3-(2,6-dichloro-4-trifluoromethylphenox y)-5-methyl-1 H- pyrazole-1-carboxamide (CAS 915396-43-9), N-ethyl-3-(2-chloro-6-fluoro-4-trifluoro- methylphenoxy)-5-methyl-1H- pyrazole-1-carboxamide (CAS 452099-05-7), N-tetrahydrofurfuryl- 3-(2-chloro-6-fluoro-4-trifluoromethylphenoxy)-5-methyl-1 H-pyrazole-1-carboxamide (CAS 452100-03-7), 3-[7-fluoro-3-oxo-4-(prop-2-ynyl)-3,4-dihydro-2H-benzo[1 ,4]oxazin-6-yl]-1 ,5- dimethyl-6-thioxo-[1 ,3,5]triazinan-2,4-dione (CAS 451484-50-7), 2-(2,2,7-trifluoro-3-oxo-4-prop- 2-ynyl-3,4-dihydro-2H-benzo[1 ,4]oxazin-6-yl)-4,5,6,7-tetrahydro-isoindole-1 ,3-dione (CAS 1300118-96-0); 1-methyl-6-trifluoromethyl-3-(2,2,7-trifluoro-3-oxo-4-prop-2 -ynyl-3,4-dihydro-2H- benzo[1 ,4]oxazin-6-yl)-1 H-pyrimidine-2,4-dione (CAS 1304113-05-0), and 3-[7-chloro-5-fluoro- 2-(trifluoromethyl)-1 H-benzimidazol-4-yl]-1 -methyl-6-(trifluoromethyl)-1 H-pyrimidine-2,4-dione (CAS 212754-02-4);

b5) from the group of the bleacher herbicides:

aclonifen, amitrole, beflubutamid, benzobicyclon, bicyclopyrone, clomazone, diflufenican, fenquinotrione, flumeturon, flurochloridone, flurtamone, isoxaflutole, mesotrione, oxotrione (CAS 1486617-21-3), norflurazon, picolinafen, pyrasulfotole, pyrazolynate, sulcotrione, tefuryltrione, tembotrione, tolpyralate, topramezone, 4-(3-trifluoromethylphenoxy)-2-(4-trifluoromethylphenyl)- pyrimidine (CAS 180608-33-7), 2-chloro-3-methylsulfanyl-N-(1-methyltetrazol-5-yl)-4- (trifluoromethyl)benzamide (CAS 1361139-71-0, 2-(2,4-dichlorophenyl)methyl-4,4-dimethyl-3- isoxazolidone (CAS 81777-95-9) and 2-(2,5-dichlorophenyl)methyl-4,4-dimethyl-3- isoxazolidinone (CAS 81778-66-7); b6) from the group of the EPSP synthase inhibitors:

glyphosate, glyphosate-isopropylammonium, glyphosate-potassium and glyphosate-trimesium (sulfosate);

b7) from the group of the glutamine synthase inhibitors:

glufosinate, glufosinate-P, glufosinate-ammonium;

b8) from the group of the DHP synthase inhibitors: asulam;

b9) from the group of the mitosis inhibitors:

benfluralin, dithiopyr, ethalfluralin, flamprop, flamprop-isopropyl, flamprop-methyl, flamprop-M- isopropyl, flamprop-M-methyl, oryzalin, pendimethalin, thiazopyr and trifluralin;

b10) from the group of the VLCFA inhibitors: acetochlor, alachlor, amidochlor, anilofos, buta- chlor, cafenstrole, dimethenamid, dimethenamid-P, fentrazamide, flufenacet, mefenacet, metazachlor, metolachlor, S-metolachlor, naproanilide, napropamide, napropamide-M, pretilachlor, fenoxasulfone, ipfencarbazone, pyroxasulfone thenylchlor and isoxazoline- compounds of the formulae 11.1 , II.2, II.3, II.4, II.5, II.6, II.7, II.8 and II.9 as mentioned above; b11) from the group of the cellulose biosynthesis inhibitors: dichlobenil, flupoxam, indaziflam, isoxaben, triaziflam and 1-cyclohexyl-5-pentafluorphenyloxy-1 4 -[1 ,2,4,6]thiatriazin-3-ylamine (CAS 175899-01-1);

b13) from the group of the auxinic herbicides:

2,4-D and its salts and esters, aminocyclopyrachlor and its salts and esters, aminopyralid and its salts such as aminopyralid-dimethylammonium, aminopyralid-tris(2-hydroxypropyl)ammoni- um and its esters, clopyralid and its salts and esters, dicamba and its salts and esters, dichlorprop-P and its salts and esters, flopyrauxifen, fluroxypyr-meptyl, halauxifen and its salts and esters (CAS 943832-60-8), MCPA and its salts and esters, MCPB and its salts and esters, mecoprop-P and its salts and esters, picloram and its salts and esters, quinclorac, quinmerac, triclopyr and its salts and esters, florpyrauxifen, florpyrauxifen-benzyl (CAS 1390661-72-9) and 4-amino-3-chloro-5-fluoro-6-(7-fluoro-1 H-indol-6-yl)picolinic acid (CAS 1629965-65-6);

b14) from the group of the auxin transport inhibitors: diflufenzopyr and diflufenzopyr-sodium; b15) from the group of the other herbicides: bromobutide, cinmethylin, cumyluron,

cyclopyrimorate (CAS 499223-49-3) and its salts and esters, dalapon, difenzoquat, difenzoquat- metilsulfate, DSMA, dymron (= daimuron), indanofan, metam, methylbromide, MSMA, oxaziclomefone, pyributicarb and tridiphane.

Particularly preferred herbicides B that can be used in combination with the pyrimidine compounds of the formula (I) according to the present invention are:

b1) from the group of the lipid biosynthesis inhibitors: clodinafop-propargyl, cycloxydim, cyha- lofop-butyl, fenoxaprop-P-ethyl, pinoxaden, profoxydim, tepraloxydim, tralkoxydim, 4-(4'-Chloro- 4-cyclopropyl-2'-fluoro[1 ,1'-biphenyl]-3-yl)-5-hydroxy-2,2,6,6-tetramethyl-2H-pyran-3 (6H)-one (CAS 1312337-72-6); 4-(2',4'-Dichloro-4-cyclopropyl[1 ,1'-biphenyl]-3-yl)-5-hydroxy-2,2,6,6- tetramethyl-2H-pyran-3(6H)-one (CAS 1312337-45-3); 4-(4 , -Chloro-4-ethyl-2 , -fluoro[1 ,1'- biphenyl]-3-yl)-5-hydroxy-2,2,6,6-tetramethyl-2H-pyran-3(6H) -one (CAS 1033757-93-5); 4-(2',4'- Dichloro-4-ethyl[1 ,1'-biphenyl]-3-yl)-2,2,6,6-tetramethyl-2H-pyran-3,5(4H,6H)- dione (CAS 1312340-84-3); 5-(Acetyloxy)-4-(4'-chloro-4-cyclopropyl-2'-fluoro[1 ,1 '-biphenyl]-3-yl)-3,6- dihydro-2,2,6,6-tetramethyl-2H-pyran-3-one (CAS 1312337-48-6); 5-(Acetyloxy)-4-(2 ' ,4'- dichloro-4-cyclopropyl- [1 ,1 '-biphenyl]-3-yl)-3,6-dihydro-2,2,6,6-tetramethyl-2H-pyran-3 -one; 5- (Acetyloxy)-4-(4'-chloro-4-ethyl-2 , -fluoro[1 ,1'-biphenyl]-3-yl)-3,6-dihydro-2,2,6,6-tetramethyl-2H- pyran-3-one (CAS 1312340-82-1); 5-(Acetyloxy)-4-(2',4 , -dichloro-4-ethyl[1 ,1'-biphenyl]-3-yl)-3,6- dihydro-2,2,6,6-tetramethyl-2H-pyran-3-one (CAS 1033760-55-2); 4-(4'-Chloro-4-cyclopropyl-2'- fluoro[1 ,1 '-biphenyl]-3-yl)-5,6-dihydro-2,2 6.6-tetramethyl-S-oxo-2H-pyran-3-yl carbonic acid methyl ester (CAS 1312337-51-1); 4-(2 ' ,4'-Dichloro -4-cyclopropyl- [1 ,1'-biphenyl]-3-yl)-5,6- dihydro-2,2,6,6-tetramethyl-5-oxo-2H-pyran-3-yl carbonic acid methyl ester; 4-(4'-Chloro-4- ethyl-2'-fluorotl .l'-biphenyll-3-yl)-5,6-dihydro-2,2 6.6-tetramethyl-S-oxo-2H-pyran-3-yl carbonic acid methyl ester (CAS 1312340-83-2); 4-(2 , ,4'-Dichloro-4-ethyl[1 ,1 , -biphenyl]-3-yl)-5,6-dihydro- 2,2,6,6-tetramethyl-5-oxo-2H-pyran-3-yl carbonic acid methyl ester (CAS 1033760-58-5);

esprocarb, prosulfocarb, thiobencarb and triallate;

b2) from the group of the ALS inhibitors: bensulfuron-methyl, bispyribac-sodium,

cyclosulfamuron, diclosulam, flumetsulam, flupyrsulfuron-methyl-sodium, foramsulfuron, imazamox, imazapic, imazapyr, imazaquin, imazethapyr, imazosulfuron, iodosulfuron, iodosulfuron-methyl-sodium, iofensulfuron, iofensulfuron-sodium, mesosulfuron,

metazosulfuron, nicosulfuron, penoxsulam, propoxycarbazon-sodium, propyrisulfuron, pyrazosulfuron-ethyl, pyroxsulam, rimsulfuron, sulfosulfuron, thiencarbazon-methyl, tritosulfuron and triafamone;

b3) from the group of the photosynthesis inhibitors: ametryn, atrazine, diuron, fluometuron, hexazinone, isoproturon, linuron, metribuzin, paraquat, paraquat-dichloride, propanil, terbutryn, terbuthylazine, 1-(5-tert-butylisoxazol-3-yl)-2-hydroxy-4-methoxy-3-methyl-2 H-pyrrol-5-one (CAS 1637455-12-9), 1-(5-tert-butylisoxazol-3-yl)-4-chloro-2-hydroxy-3-methyl-2H -pyrrol-5-one (CAS 1637453-94-1), 1-(5-tert-butylisoxazol-3-yl)-4-ethoxy-5-hydroxy-3-methyl-im idazolidin-2- one (CAS 1844836-64-1);

b4) from the group of the protoporphyrinogen-IX oxidase inhibitors: flumioxazin, oxyfluorfen, pyraflufen, pyraflufen-ethyl, saflufenacil, sulfentrazone, trifludimoxazin, ethyl [3-[2-chloro-4-flu- oro-5-(1-methyl-6-trifluoromethyl-2,4-dioxo-1 ,2,3,4-tetrahydropyrimidin-3-yl)phenoxy]-2-pyridyl- oxy]acetate (CAS 353292-31-6; S-3100, 3-[7-fluoro-3-oxo-4-(prop-2-ynyl)-3,4-dihydro-2H-ben- zo[1 ,4]oxazin-6-yl]-1 ,5-dimethyl-6-thioxo-[1 ,3,5]triazinan-2,4-dione (CAS 451484-50-7), 2-(2,2,7- trifluoro-3-oxo-4-prop-2-ynyl-3,4-dihydro-2H-benzo[1 ,4]oxazin-6-yl)-4,5,6,7-tetrahydro-isoindole- 1 ,3-dione (CAS 1300118-96-0), and 1-methyl-6-trifluoromethyl-3-(2,2,7-trifluoro-3-oxo-4-prop-2 - ynyl-3,4-dihydro-2H-benzo[1 ,4]oxazin-6-yl)-1 H-pyrimidine-2,4-dione (CAS 1304113-05-0);

b5) from the group of the bleacher herbicides: amitrole, bicyclopyrone, clomazone,

diflufenican, fenquinotrione, flumeturon, flurochloridone, isoxaflutole, mesotrione, oxotrione (CAS 1486617-21-3), picolinafen, sulcotrione, tefuryltrione, tembotrione, tolpyralate,

topramezone, 2-chloro-3-methylsulfanyl-N-(1-methyltetrazol-5-yl)-4-(trifl uoromethyl)benzamide (CAS 1361139-71-0), 2-(2,4-dichlorophenyl)methyl-4,4-dimethyl-3-isoxazolidone (CAS 81777- 95-9); and 2-(2,5-dichlorophenyl)methyl-4,4-dimethyl-3-isoxazolidinone (CAS 81778-66-7); b6) from the group of the EPSP synthase inhibitors: glyphosate, glyphosate- isopropylammonium and glyphosate-trimesium (sulfosate);

b7) from the group of the glutamine synthase inhibitors: glufosinate, glufosinate-P and glufosinate-ammonium;

b9) from the group of the mitosis inhibitors: pendimethalin and trifluralin;

b10) from the group of the VLCFA inhibitors: acetochlor, cafenstrole, dimethenamid-P, fentrazamide, flufenacet, mefenacet, metazachlor, metolachlor, S-metolachlor, fenoxasulfone, ipfencarbazone and pyroxasulfone; likewise, preference is given to isoxazoline compounds of the formulae 11.1 , II.2, II.3, II.4, II.5, II.6, II.7, II.8 and II.9 as mentioned above;

b1 1 ) from the group of the cellulose biosynthesis inhibitors: indaziflam, isoxaben and triaziflam;

b13) from the group of the auxinic herbicides: 2,4-D and its salts and esters such as clacyfos, and aminocyclopyrachlor and its salts and esters, aminopyralid and its salts and its esters, clopyralid and its salts and esters, dicamba and its salts and esters, flopyrauxifen, fluroxypyr- meptyl, halauxifen, halauxifen-methyl, quinclorac, quinmerac, florpyrauxifen, florpyrauxifen- benzyl (CAS 1390661-72-9) and 4-amino-3-chloro-5-fluoro-6-(7-fluoro-1 H-indol-6-yl)picolinic acid (CAS 1629965-65-6);

b14) from the group of the auxin transport inhibitors: diflufenzopyr and diflufenzopyr-sodium, b15) from the group of the other herbicides: cinmethylin, dymon (= daimuron), indanofan, oxaziclomefone.

Particularly preferred herbicides B are the herbicides B as defined above; in particular, the herbicides B.1 - B.202 listed below in table B:

Table B

In another embodiment of the present invention the compositions according to the present invention comprise at least one pyrimidine compound of formula (I) and at least one safener C.

Safeners are chemical compounds which prevent or reduce damage on useful plants without having a major impact on the herbicidal action of the herbicidal active components of the present compositions towards unwanted plants. They can be applied either before sowings (e.g. on seed treatments, shoots or seedlings) or in the pre-emergence application or post- emergence application of the useful plant. The safeners and the pyrimidine compounds of formula (I) and/or the herbicides B can be applied simultaneously or in succession.

Suitable safeners are e.g. (quinolin-8-oxy)acetic acids, 1-phenyl-5-haloalkyl-1 H-1 ,2,4-triazol-3- carboxylic acids, 1-phenyl-4,5-dihydro-5-alkyl-1 H-pyrazol-3,5-dicarboxylic acids, 4,5-dihydro- 5,5-diaryl-3-isoxazol carboxylic acids, dichloroacetamides, alpha-oximinophenylacetonitriles, acetophenonoximes, 4,6-dihalo-2-phenylpyrimidines, N-[[4-(aminocarbonyl)phenyl]sulfonyl]-2- benzoic amides, 1 ,8-naphthalic anhydride, 2-halo-4-(haloalkyl)-5-thiazol carboxylic acids, phosphorthiolates and N-alkyl-O-phenylcarbamates and their agriculturally acceptable salts and their agriculturally acceptable derivatives such amides, esters, and thioesters, provided they have an acid group.

Examples of preferred safeners C are benoxacor, cloquintocet, cyometrinil, cyprosulfamide, dichlormid, dicyclonon, dietholate, fenchlorazole, fenclorim, flurazole, fluxofenim, furilazole, isoxadifen, mefenpyr, mephenate, naphthalic anhydride, oxabetrinil, 4-(dichloroacetyl)-1-oxa-4- azaspiro[4.5]decane (MON4660, CAS 71526-07-3), 2,2,5-trimethyl-3-(dichloroacetyl)-1 ,3- oxazolidine (R-29148, CAS 52836-31-4), metcamifen and BPCMS (CAS 54091-06-4).

Especially preferred safeners C are benoxacor, cloquintocet, cyprosulfamide, dichlormid, fenchlorazole, fenclorim, flurazole, fluxofenim, furilazole, isoxadifen, mefenpyr, naphthalic anhydride, oxabetrinil, 4-(dichloroacetyl)-1-oxa-4-azaspiro[4.5]decane (MON4660, CAS 71526- 07-3), 2,2,5-trimethyl-3-(dichloroacetyl)-1 ,3-oxazolidine (R-29148, CAS 52836-31-4) and metcamifen.

Particularly preferred safeners C are benoxacor, cloquintocet, cyprosulfamide, dichlormid, fenchlorazole, fenclorim, furilazole, isoxadifen, mefenpyr, naphtalic anhydride, 4-(dichloro- acetyl)-1-oxa-4-azaspiro[4.5]decane (MON4660, CAS 71526-07-3), 2,2,5-trimethyl-3- (dichloroacetyl)-l ,3-oxazolidine (R-29148, CAS 52836-31-4) and metcamifen.

Particularly preferred safeners C, which, as component C, are constituent of the composition according to the invention are the safeners C as defined above; in particular the safeners C.1 - C.17 listed below in table C:

Table C:

The active compounds B of groups b1) to b15) and the active compounds C are known herbicides and safeners, see, e.g., The Compendium of Pesticide Common Names

(http://www.alanwood.net/pesticides/); Farm Chemicals Handbook 2000 volume 86, Meister Publishing Company, 2000; B. Hock, C. Fedtke, R. R. Schmidt, Herbizide [Herbicides], Georg Thieme Verlag, Stuttgart 1995; W. H. Ahrens, Herbicide Handbook, 7th edition, Weed Science Society of America, 1994; and K. K. Hatzios, Herbicide Handbook, Supplement for the 7th edition, Weed Science Society of America, 1998. 2,2,5-Trimethyl-3-(dichloroacetyl)-1 ,3- oxazolidine [CAS No. 52836-31-4] is also referred to as R-29148. 4-(Dichloroacetyl)-1-oxa-4- azaspiro[4.5]decane [CAS No. 71526-07-3] is also referred to as AD-67 and MON 4660.

The assignment of the active compounds to the respective mechanisms of action is based on current knowledge. If several mechanisms of action apply to one active compound, this substance was only assigned to one mechanism of action.

Active compounds B and C having a carboxyl group can be employed in the form of the acid, in the form of an agriculturally suitable salt as mentioned above or else in the form of an agriculturally acceptable derivative in the compositions according to the invention.

In the case of dicamba, suitable salts include those, where the counterion is an agriculturally acceptable cation. E.g., suitable salts of dicamba are dicamba-sodium, dicamba-potassium, dicamba-methylammonium, dicamba-dimethylammonium, dicamba-isopropylammonium, dicamba-diglycolamine, dicamba-olamine, dicamba-diolamine, dicamba-trolamine, dicamba- N,N-bis-(3-aminopropyl)methylamine and dicamba-diethylenetriamine. Examples of a suitable ester are dicamba-methyl and dicamba-butotyl.

Suitable salts of 2,4-D are 2,4-D-ammonium, 2,4-D-dimethylammonium, 2,4-D-diethylammoni- um, 2,4-D-diethanolammonium (2,4-D-diolamine), 2,4-D-triethanolammonium, 2,4-D- isopropylammonium, 2,4-D-triisopropanolammonium, 2,4-D-heptylammonium, 2,4-D- dodecylammonium, 2,4-D-tetradecylammonium, 2,4-D-triethylammonium, 2,4-D-tris(2- hydroxypropyl)ammonium, 2,4-D-tris(isopropyl)ammonium, 2,4-D-trolamine, 2,4-D-lithium, 2,4- D-sodium. Examples of suitable esters of 2,4-D are 2,4-D-butotyl, 2,4-D-2-butoxypropyl, 2,4-D- 3-butoxypropyl, 2,4-D-butyl, 2,4-D-ethyl, 2,4-D-ethylhexyl, 2,4-D-isobutyl, 2,4-D-isooctyl, 2,4-D- isopropyl, 2,4-D-meptyl, 2,4-D-methyl, 2,4-D-octyl, 2,4-D-pentyl, 2,4-D-propyl, 2,4-D-tefuryl and clacyfos.

Suitable salts of 2,4-DB are e.g. 2,4-DB-sodium, 2,4-DB-potassium and 2,4-DB-dimethyl- ammonium. Suitable esters of 2,4-DB are e.g. 2,4-DB-butyl and 2,4-DB-isoctyl. Suitable salts of dichlorprop are e.g. dichlorprop-sodium, dichlorprop-potassium and dichlorprop-dimethylammonium. Examples of suitable esters of dichlorprop are dichlorprop- butotyl and dichlorprop-isoctyl.

Suitable salts and esters of MCPA include MCPA-butotyl, MCPA-butyl, MCPA-dimethyl- ammonium, MCPA-diolamine, M CPA-ethyl, MCPA-thioethyl, MCPA-2-ethylhexyl, MCPA- isobutyl, MCPA-isoctyl, MCPA-isopropyl, MCPA-isopropylammonium, MCPA-methyl, MCPA- olamine, MCPA-potassium, MCPA-sodium and MCPA-trolamine.

A suitable salt of MCPB is MCPB sodium. A suitable ester of MCPB is MCPB-ethyl.

Suitable salts of clopyralid are clopyralid-potassium, clopyralid-olamine and clopyralid-tris-(2- hydroxypropyl)ammonium. Example of suitable esters of clopyralid is clopyralid-methyl.

Examples of a suitable ester of fluroxypyr are fluroxypyr-meptyl and fluroxypyr-2-butoxy-1- methylethyl, wherein fluroxypyr-meptyl is preferred.

Suitable salts of picloram are picloram-dimethylammonium, picloram-potassium, picloram- triisopropanolammonium, picloram-triisopropylammonium and picloram-trolamine. A suitable ester of picloram is picloram-isoctyl.

A suitable salt of triclopyr is triclopyr-triethylammonium. Suitable esters of triclopyr are e.g. triclopyr-ethyl and triclopyr-butotyl.

Suitable salts and esters of chloramben include chloramben-ammonium, chloramben- diolamine, chloramben-methyl, chloramben-methylammonium and chloramben-sodium. Suitable salts and esters of 2,3,6-TBA include 2,3,6-TBA-dimethylammonium, 2,3,6-TBA-lithium, 2,3,6- TBA-potassium and 2,3,6-TBA-sodium.

Suitable salts and esters of aminopyralid include aminopyralid-potassium, aminopyralid- dimethylammonium, and aminopyralid-tris(2-hydroxypropyl)ammonium.

Suitable salts of glyphosate are e.g. glyphosate-ammonium, glyphosate-diammonium, glyphoste-dimethylammonium, glyphosate-isopropylammonium, glyphosate-potassium, glyphosate-sodium, glyphosate-trimesium as well as the ethanolamine and diethanolamine salts, preferably glyphosate-diammonium, glyphosate-isopropylammonium and glyphosate- trimesium (sulfosate).

A suitable salt of glufosinate is e.g. glufosinate-ammonium.

A suitable salt of glufosinate-P is e.g. glufosinate-P-ammonium.

Suitable salts and esters of bromoxynil are e.g. bromoxynil-butyrate, bromoxynil-heptanoate, bromoxynil-octanoate, bromoxynil-potassium and bromoxynil-sodium.

Suitable salts and esters of ioxonil are e.g. ioxonil-octanoate, ioxonil-potassium and ioxonil- sodium.

Suitable salts and esters of mecoprop include mecoprop-butotyl, mecoprop- dimethylammonium, mecoprop-diolamine, mecoprop-ethadyl, mecoprop-2-ethylhexyl, mecoprop-isoctyl, mecoprop-methyl, mecoprop-potassium, mecoprop-sodium and mecoprop- trolamine.

Suitable salts of mecoprop-P are e.g. mecoprop-P-butotyl, mecoprop-P-dimethylammonium, mecoprop-P-2-ethylhexyl, mecoprop-P-isobutyl, mecoprop-P-potassium and mecoprop-P- sodium.

A suitable salt of diflufenzopyr is e.g. diflufenzopyr-sodium.

A suitable salt of naptalam is e.g. naptalam-sodium. Suitable salts and esters of aminocyclopyrachlor are e.g. aminocyclopyrachlor- dimethylammonium, aminocyclopyrachlor-methyl, aminocyclopyrachlor- triisopropanolammonium, aminocyclopyrachlor-sodium and aminocyclopyrachlor-potassium.

A suitable salt of quinclorac is e.g. quinclorac-dimethylammonium.

A suitable salt of quinmerac is e.g. quinmerac-dimethylammonium.

A suitable salt of imazamox is e.g. imazamox-ammonium.

Suitable salts of imazapic are e.g. imazapic-ammonium and imazapic-isopropylammonium. Suitable salts of imazapyr are e.g. imazapyr-ammonium and imazapyr-isopropylammonium. A suitable salt of imazaquin is e.g. imazaquin-ammonium.

Suitable salts of imazethapyr are e.g. imazethapyr-ammonium and imazethapyr- isopropylammonium.

A suitable salt of topramezone is e.g. topramezone-sodium.

According to a preferred embodiment of the invention, the composition comprises as herbicidal active compound B or component B at least one, preferably exactly one herbicide B.

According to another preferred embodiment of the invention, the composition comprises as herbicidal active compounds B or component B at least two, preferably exactly two herbicides B different from each other.

According to another preferred embodiment of the invention, the composition comprises as herbicidal active compounds B or component B at least three, preferably exactly three herbicides B different from each other.

According to another preferred embodiment of the invention, the composition comprises as safening component C or component C at least one, preferably exactly one safener C.

According to another preferred embodiment of the invention, the composition comprises as component B at least one, preferably exactly one herbicide B, and as component C at least one, preferably exactly one, safener C.

According to another preferred embodiment of the invention, the composition comprises at least two, preferably exactly two, herbicides B different from each other, and as component C at least one, preferably exactly one, safener C.

According to another preferred embodiment of the invention, the composition comprises at least three, preferably exactly three, herbicides B different from each other, and as component C at least one, preferably exactly one, safener C.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.1), especially preferred the compound (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1-25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1-59), (1.1.1-60), (1.1.1-66), or (1.1.1-67), and as component B at least one, preferably exactly one, herbicide B.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.1), especially preferred the compound (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1-25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1-59), (1.1.1-60), (1.1.1-66), or (1.1.1-67), and at least two, preferably exactly two, herbicides B different from each other. According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.1), especially preferred the compound (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1-25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1-59), (1.1.1-60), (1.1.1-66), or (1.1.1-67), and at least three, preferably exactly three, herbicides B different from each other.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.1), especially preferred the compound (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1-25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1-59), (1.1.1-60), (1.1.1-66), or (1.1.1-67), and as component C at least one, preferably exactly one, safener C.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.1), especially preferred the compound (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1-25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1-59), (1.1.1-60), (1.1.1-66), or (1.1.1-67), as component B at least one, preferably exactly one, herbicide B, and as component C at least one, preferably exactly one safener C.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly pyrimidine compound of formula (I), preferably of formula (1.1), especially preferred the compound (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1- 17), (1.1.1-18), (1.1.1-24), (1.1.1-25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1- 46), (1.1.1-52), (1.1.1-53), (1.1.1-59), (1.1.1-60), (1.1.1-66), or (1.1.1-67), at least two, preferably exactly two herbicides B different from each other, and as component C at least one, preferably exactly one, safener C.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.1), especially preferred the compound (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1-25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1-59), (1.1.1-60), (1.1.1-66), or (1.1.1-67), at least three, preferably exactly three herbicides B different from each other, and as component C at least one, preferably exactly one, safener C.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.2), especially preferred the compound (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), or (1.2.1-67), and as component B at least one, preferably exactly one, herbicide B.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.2), especially preferred the compound (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), or (1.2.1-67), and at least two, preferably exactly two, herbicides B different from each other.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.2), especially preferred the compound (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11 ), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), or (1.2.1-67), and at least three, preferably exactly three, herbicides B different from each other.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.2), especially preferred the compound (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), or (1.2.1-67), and as component C at least one, preferably exactly one, safener C.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.2), especially preferred the compound (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), or (1.2.1-67), as component B at least one, preferably exactly one, herbicide B, and as component C at least one, preferably exactly one safener C.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly pyrimidine compound of formula (I), preferably of formula (1.2), especially preferred the compound (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1- 17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1- 46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), or (1.2.1-67), at least two, preferably exactly two herbicides B different from each other, and as component C at least one, preferably exactly one, safener C.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.2), especially preferred the compound (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), or (1.2.1-67), at least three, preferably exactly three herbicides B different from each other, and as component C at least one, preferably exactly one, safener C.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.5), especially preferred the compound (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), or (1.5.1-67), and as component B at least one, preferably exactly one, herbicide B.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.5), especially preferred the compound (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), or (1.5.1-67), and at least two, preferably exactly two, herbicides B different from each other.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.5), especially preferred the compound (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), or (1.5.1-67), and at least three, preferably exactly three, herbicides B different from each other.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.5), especially preferred the compound (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), or (1.5.1-67), and as component C at least one, preferably exactly one, safener C.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.5), especially preferred the compound (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), or (1.5.1-67), as component B at least one, preferably exactly one, herbicide B, and as component C at least one, preferably exactly one safener C.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly pyrimidine compound of formula (I), preferably of formula (1.5), especially preferred the compound (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1- 17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1- 46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), or (1.5.1-67), at least two, preferably exactly two herbicides B different from each other, and as component C at least one, preferably exactly one, safener C.

According to another preferred embodiment of the invention, the composition comprises as component A at least one, preferably exactly one pyrimidine compound of formula (I), preferably of formula (1.5), especially preferred the compound (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), or (1.5.1-67), at least three, preferably exactly three herbicides B different from each other, and as component C at least one, preferably exactly one, safener C.

According to another preferred embodiment of the invention, the composition comprises, in addition to a pyrimidine compounds of formula (I), especially an active compound from the group consisting of (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1- 25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1- 59), (1.1.1-60), (1.1.1-66), (1.1.1-67), (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), (1.2.1-67), (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), and (1.5.1-67), at least one and especially exactly one herbicidally active compound from group b1), in particular selected from the group consisting of clethodim, clodinafop-propargyl, cycloxydim, cyhalofop-butyl, fenoxaprop-ethyl, fenoxaprop-P-ethyl, metamifop, pinoxaden, profoxydim, sethoxydim, tepraloxydim, tralkoxydim, esprocarb, ethofumesate, molinate, prosulfocarb, thiobencarb and triallate.

According to another preferred embodiment of the invention, the composition comprises, in addition to a pyrimidine compounds of formula (I), especially an active compound from the group consisting of (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1- 25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1- 59), (1.1.1-60), (1.1.1-66), (1.1.1-67), (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), (1.2.1-67), (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), and (1.5.1-67), at least one and especially exactly one herbicidally active compound from group b2), in particular selected from the group consisting of bensulfuron-methyl, bispyribac-sodium, cloransulam-methyl,

chlorsulfuron, clorimuron, cyclosulfamuron, diclosulam, florasulam, flumetsulam, flupyrsulfuron- methyl-sodium, foramsulfuron, imazamox, imazamox-ammonium, imazapic, imazapic- ammonium, imazapic-isopropylammonium, imazapyr, imazapyr-ammonium, imazethapyr- isopropylammonium, imazaquin, imazaquin-ammonium, imazethapyr, imazethapyr-ammonium, imazethapyr-isopropylammonium, imazosulfuron, iodosulfuron-methyl-sodium, iofensulfuron, iofensulfuron-sodium, mesosulfuron-methyl, metazosulfuron, metsulfuron-methyl, metosulam, nicosulfuron, penoxsulam, propoxycarbazon-sodium, pyrazosulfuron-ethyl, pyribenzoxim, pyriftalid, pyroxsulam, propyrisulfuron, rimsulfuron, sulfosulfuron, thiencarbazon-methyl, thifensulfuron-methyl, tribenuron-methyl, tritosulfuron and triafamone.

According to another preferred embodiment of the invention, the composition comprises, in addition to a pyrimidine compounds of formula (I), especially an active compound from the group consisting (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1- 25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1- 59), (1.1.1-60), (1.1.1-66), (1.1.1-67), (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), (1.2.1-67), (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), and (1.5.1-67), at least one and especially exactly one herbicidally active compound from group b3), in particular selected from the group consisting of ametryn, atrazine, bentazon, bromoxynil, bromoxynil-octanoate, bromoxynil-heptanoate, bromoxynil-potassium, diuron, fluometuron, hexazinone, isoproturon, linuron, metamitron, metribuzin, paraquat-dichloride, propanil, simazin, terbutryn and

terbuthylazine.

According to another preferred embodiment of the invention, the composition comprises, in addition to a pyrimidine compounds of formula (I), especially an active compound from the group consisting of (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1- 25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1- 59), (1.1.1-60), (1.1.1-66), (1.1.1-67), (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), (1.2.1-67), (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), and (1.5.1-67), at least one and especially exactly one herbicidally active compound from group b4), in particular selected from the group consisting of acifluorfen, butafencil, carfenetrazone-ethyl, flumioxazin, fomesafen, oxadiargyl, oxyfluorfen, pyraflufen, pyraflufen-ethyl, saflufenacil, sulfentrazone, trifludimoxazin , ethyl [3-[2-chloro-4-fluoro-5-(1-methyl-6-trifluoromethyl-2,4-diox o-1,2,3,4-tetrahydropyrimidin-3- yl)phenoxy]-2-pyridyloxy]acetate (CAS 353292-31-6; S-3100).

According to another preferred embodiment of the invention, the composition comprises, in addition to a pyrimidine compounds of formula (I), especially an active compound from the group consisting of (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1- 25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1- 59), (1.1.1-60), (1.1.1-66), (1.1.1-67), (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), (1.2.1-67), (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), and (1.5.1-67), at least one and especially exactly one herbicidally active compound from group b5), in particular selected from the group consisting of amitrole, benzobicyclon, bicyclopyrone, clomazone, diflufenican, fenquintrone, fluometuron, flurochloridone, isoxaflutole, mesotrione, norflurazone, oxotrione (CAS 1486617-21-3), picolinafen, sulcotrione, tefuryltrione, tembotrione, tolpyralate,

topramezone, topramezone-sodium and 2-chloro-3-methylsulfanyl-N-(1-methyltetrazol-5-yl)-4- (trifluoromethyl)benzamide (CAS 1361139-71-0) .

According to another preferred embodiment of the invention, the composition comprises, in addition to a pyrimidine compounds of formula (I), especially an active compound from the group consisting of (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1- 25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1- 59), (1.1.1-60), (1.1.1-66), (1.1.1-67), (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), (1.2.1-67), (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), and (1.5.1-67), at least one and especially exactly one herbicidally active compound from group b6), in particular selected from the group consisting of glyphosate, glyphosate-ammonium, glyphosate-dimethylammonium , glyphosate-isopropylammonium and glyphosate-trimesium (sulfosate) and glyphosate- potassium.

According to another preferred embodiment of the invention, the composition comprises, in addition to a pyrimidine compounds of formula (I), especially an active compound from the group consisting of (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1- 25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1- 59), (1.1.1-60), (1.1.1-66), (1.1.1-67), (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), (1.2.1-67), (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), and (1.5.1-67), at least one and especially exactly one herbicidally active compound from group b7), in particular selected from the group consisting of glufosinate, glufosinate-ammonium, glufosinate-P and glufosinate-P- ammonium.

According to another preferred embodiment of the invention, the composition comprises, in addition to a pyrimidine compounds of formula (I), especially an active compound from the group consisting of (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1- 25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1- 59), (1.1.1-60), (1.1.1-66), (1.1.1-67), (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), (1.2.1-67), (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), and (1.5.1-67), at least one and especially exactly one herbicidally active compound from group b9), in particular selected from the group consisting of pendimethalin and trifluralin.

According to another preferred embodiment of the invention, the composition comprises, in addition to a pyrimidine compounds of formula (I), especially an active compound from the group consisting of (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1- 25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1- 59), (1.1.1-60), (1.1.1-66), (1.1.1-67), (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), (1.2.1-67), (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), and (1.5.1-67), at least one and especially exactly one herbicidally active compound from group b10), in particular selected from the group consisting of acetochlor, butachlor, cafenstrole, dimethenamid-P, fentrazamide, flufenacet, mefenacet, metazachlor, metolachlor, S-metolachlor, fenoxasulfone, ipfencarbazone and pyroxasulfone. Likewise, preference is given to compositions comprising in addition to a pyrimidine compounds of formula (I), especially an active compound from the group consisting of (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1-25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1-59), (1.1.1-60), (1.1.1-66), (1.1.1-67), (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31 ), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), (1.2.1-67), (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), and (1.5.1-67), at least one and especially exactly one herbicidally active compound from group b10), in particular selected from the group consisting of isoxazoline compounds of the formulae 11.1, II.2, II.3, II.4, II.5, II.6, II.7, II.8 and II.9, as defined above.

According to another preferred embodiment of the invention, the composition comprises, in addition to a pyrimidine compounds of formula (I), especially an active compound from the group consisting of (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1- 25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1- 59), (1.1.1-60), (1.1.1-66), (1.1.1-67), (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), (1.2.1-67), (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), and (1.5.1-67), at least one and especially exactly one herbicidally active compound from group b11), in particular indaziflam, isoxaben and triaziflam.

According to another preferred embodiment of the invention, the composition comprises, in addition to a pyrimidine compounds of formula (I), especially an active compound from the group consisting of (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1- 25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1- 59), (1.1.1-60), (1.1.1-66), (1.1.1-67), (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), (1.2.1-67), (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), and (1.5.1-67), at least one and especially exactly one herbicidally active compound from group b13), in particular selected from the group consisting of 2,4-D, 2,4-D-isobutyl, 2,4-D-dimethylammonium, 2,4-D-N,N,N- trimethylethanolammonium, aminocyclopyrachlor, aminocyclopyrachlor-potassium,

aminocyclopyrachlor-methyl, aminopyralid, aminopyralid-methyl, aminopyralid- dimethylammonium, aminopyralid-tris(2-hydroxypropyl)ammonium, clopyralid, clopyralid-methyl, clopyralid-olamine, dicamba, dicamba-butotyl, dicamba-diglycolamine, dicamba- dimethylammonium, dicamba-diolamine, dicamba-isopropylammonium, dicamba-potassium, dicamba-sodium, dicamba-trolamine, dicamba-N,N-bis-(3-aminopropyl)methylamine, dicamba- diethylenetriamine, flopyrauxifen, fluroxypyr, fluroxypyr-meptyl, halauxifen, halauxifen-methyl, MCPA, MCPA-2-ethylhexyl, MCPA-dimethylammonium, quinclorac, quinclorac- dimethylammonium, quinmerac, quinmerac-dimethylammonium, florpyrauxifen , florpyrauxifen- benzyl (CAS 1390661-72-9), and 4-amino-3-chloro-5-fluoro-6-(7-fluoro-1H-indol-6-yl)picolini c acid (CAS 1629965-65-6) .

According to another preferred embodiment of the invention, the composition comprises, in addition to a pyrimidine compounds of formula (I), especially an active compound from the group consisting of (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1- 25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1- 59), (1.1.1-60), (1.1.1-66), (1.1.1-67), (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), (1.2.1-67), (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), and (1.5.1-67), at least one and especially exactly one herbicidally active compound from group b14), in particular selected from the group consisting of diflufenzopyr, diflufenzopyr-sodium, dymron, indanofan and

diflufenzopyr-sodium.

According to another preferred embodiment of the invention, the composition comprises, in addition to a pyrimidine compounds of formula (I), especially an active compound from the group consisting of (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1- 25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1- 59), (1.1.1-60), (1.1.1-66), (1.1.1-67), (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), (1.2.1-67), (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), and (1.5.1-67), at least one and especially exactly one herbicidally active compound from group b15), in particular selected from the group consisting of cinmethylin, dymron (= daimuron), indanofan and oxaziclomefone.

According to another preferred embodiment of the invention, the composition comprises, in addition to a pyrimidine compounds of formula (I), especially an active compound from the group consisting of (1.1.1-3), (1.1.1-4), (1.1.1-10), (1.1.1-11), (1.1.1-17), (1.1.1-18), (1.1.1-24), (1.1.1- 25), (1.1.1-31), (1.1.1-32), (1.1.1-38), (1.1.1-39), (1.1.1-45), (1.1.1-46), (1.1.1-52), (1.1.1-53), (1.1.1- 59), (1.1.1-60), (1.1.1-66), (1.1.1-67), (1.2.1-3), (1.2.1-4), (1.2.1-10), (1.2.1-11), (1.2.1-17), (1.2.1-18), (1.2.1-24), (1.2.1-25), (1.2.1-31), (1.2.1-32), (1.2.1-38), (1.2.1-39), (1.2.1-45), (1.2.1-46), (1.2.1-52), (1.2.1-53), (1.2.1-59), (1.2.1-60), (1.2.1-66), (1.2.1-67), (1.5.1-3), (1.5.1-4), (1.5.1-10), (1.5.1-11), (1.5.1-17), (1.5.1-18), (1.5.1-24), (1.5.1-25), (1.5.1-31), (1.5.1-32), (1.5.1-38), (1.5.1-39), (1.5.1-45), (1.5.1-46), (1.5.1-52), (1.5.1-53), (1.5.1-59), (1.5.1-60), (1.5.1-66), and (1.5.1-67), at least one and especially exactly one safener C, in particular selected from the group consisting of benoxacor, cloquintocet, cyprosulfamide, dichlormid, fenchlorazole, fenclorim, furilazole, isoxadifen, mefenpyr, 4-(dichloroacetyl)-1-oxa-4-azaspiro[4.5]decane (MON4660, CAS 71526-07-3) and 2,2,5-trimethyl-3-(dichloroacetyl)-1 ,3-oxazolidine (R-29148, CAS 52836-31-4).

Here and below, the term "binary compositions" includes compositions comprising one or more, e.g. 1 , 2 or 3, active compounds of the formula (I) and either one or more, e.g. 1 , 2 or 3, herbicides B or one or more safeners C.

Correspondingly, the term "ternary compositions" includes compositions comprising one or more, e.g. 1 , 2 or 3, active compounds of the formula (I), one or more, e.g. 1 , 2 or 3, herbicides B and one or more, e.g. 1 , 2 or 3, safeners C.

In binary compositions comprising at least one pyrimidine of formula (I) as component A and at least one herbicide B, the weight ratio of the active compounds A:B is generally in the range of from 1 :1000 to 1000:1 , preferably in the range of from 1 :500 to 500:1 , in particular in the range of from 1 :250 to 250:1 and particularly preferably in the range of from 1 :75 to 75:1.

In binary compositions comprising at least one pyrimidine of formula (I) as component A and at least one safener C, the weight ratio of the active compounds A:C is generally in the range of from 1 :1000 to 1000:1 , preferably in the range of from 1 :500 to 500:1 , in particular in the range of from 1 :250 to 250:1 and particularly preferably in the range of from 1 :75 to 75:1.

In ternary compositions comprising at least one pyrimidine of formula (I) as component A, at least one herbicide B and at least one safener C, the relative proportions by weight of the components A:B are generally in the range of from 1 :1000 to 1000:1 , preferably in the range of from 1 :500 to 500:1 , in particular in the range of from 1 :250 to 250:1 and particularly preferably in the range of from 1 :75 to 75:1 , the weight ratio of the components A:C is generally in the range of from 1 :1000 to 1000:1 , preferably in the range of from 1 :500 to 500:1 , in particular in the range of from 1 :250 to 250:1 and particularly preferably in the range of from 1 :75 to 75:1 , and the weight ratio of the components B:C is generally in the range of from 1 :1000 to 1000:1 , preferably in the range of from 1 :500 to 500:1 , in particular in the range of from 1 :250 to 250:1 and particularly preferably in the range of from 1 :75 to 75:1 . The weight ratio of components A + B to component C is preferably in the range of from 1 :500 to 500:1 , in particular in the range of from 1 :250 to 250:1 and particularly preferably in the range of from 1 :75 to 75:1 .

The weight ratios of the individual components in the preferred mixtures mentioned below are within the limits given above, in particular within the preferred limits.

Particularly preferred are the compositions mentioned below comprising the pyrimidine compounds of formula I as defined and the substance(s) as defined in the respective row of table T;

especially preferred comprising as only herbicidal active compounds the pyrimidine compounds of formula I as defined and the substance(s) as defined in the respective row of table T;

most preferably comprising as only active compounds the pyrimidine compounds of formula I as defined and the substance(s) as defined in the respective row of table T.

Particularly preferred are compositions 1 .1 to 1.3653, comprising the compound 1.3.1-3 and the substance(s) as defined in the respective row of table T:

The specific number for each single composition is deductible as follows:

Composition 1.203 e.g. comprises the compound (1.1.1-25), clethodim (B.1) and benoxacor (C.1) (see table B, entry B.1 and table C, entry C.1).

Also especially preferred are compositions 2.1 to 2.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.1.1-4) in place of the compound (1.1.1-3).

Also especially preferred are compositions 3.1 to 3.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.2 as further herbicide B.

Also especially preferred are compositions 4.1 to 4.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.8 as further herbicide B. Also especially preferred are compositions 5.1 to 5.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.30 as further herbicide B. Also especially preferred are compositions 6.1 to 6.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.32 as further herbicide B.

Also especially preferred are compositions 7.1 to 7.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.35 as further herbicide B. Also especially preferred are compositions 8.1 to 8.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.38 as further herbicide B.

Also especially preferred are compositions 9.1 to 9.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.40 as further herbicide B. Also especially preferred are compositions 10.1 to 10.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.51 as further herbicide B.

Also especially preferred are compositions 11.1 to 11.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.55 as further herbicide B.

Also especially preferred are compositions 12.1 to 12.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.56 as further herbicide B.

Also especially preferred are compositions 13.1 to 13.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.64 as further herbicide B.

Also especially preferred are compositions 14.1 to 14.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.66 as further herbicide B. Also especially preferred are compositions 15.1 o 15.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.67 as further herbicide B.

Also especially preferred are compositions 16.1 :o 16.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.68 as further herbicide B.

Also especially preferred are compositions 17.1 :o 17.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.69 as further herbicide B.

Also especially preferred are compositions 18.1 :o 18.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.73 as further herbicide B.

Also especially preferred are compositions 19.1 :o 19.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.76 as further herbicide B.

Also especially preferred are compositions 20.1 :o 20.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.81 as further herbicide B.

Also especially preferred are compositions 21.1 :o 21.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.82 as further herbicide B.

Also especially preferred are compositions 22.1 :o 22.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.85 as further herbicide B.

Also especially preferred are compositions 23.1 :o 23.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.88 as further herbicide B.

Also especially preferred are compositions 24.1 :o 24.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.89 as further herbicide B.

Also especially preferred are compositions 25.1 :o 25.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.94 as further herbicide B.

Also especially preferred are compositions 26.1 :o 26.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.95 as further herbicide B.

Also especially preferred are compositions 27.1 :o 27.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.98 as further herbicide B.

Also especially preferred are compositions 28.1 :o 28.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.100 as further herbicide B.

Also especially preferred are compositions 29.1 :o 29.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.103 as further herbicide B.

Also especially preferred are compositions 30.1 to 30.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.103 and B.67 as further herbicides B.

Also especially preferred are compositions 31.1 to 31.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.103 and B.76 as further herbicides B.

Also especially preferred are compositions 32.1 to 32.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.103 and B.82 as further herbicides B.

Also especially preferred are compositions 33.1 to 33.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.104 as further herbicide B.

Also especially preferred are compositions 34.1 to 34.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.104 and B.67 as further herbicides B.

Also especially preferred are compositions 35.1 to 35.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.104 and B.76 as further herbicides B.

Also especially preferred are compositions 36.1 to 36.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.104 and B.82 as further herbicides B.

Also especially preferred are compositions 37.1 to 37.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.106 as further herbicide B.

Also especially preferred are compositions 38.1 to 38.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.107 as further herbicide B.

Also especially preferred are compositions 39.1 to 39.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B. 107 and B.67 as further herbicides B.

Also especially preferred are compositions 40.1 to 40.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B. 107 and B.76 as further herbicides B.

Also especially preferred are compositions 41.1 to 41 .3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B. 107 and B.82 as further herbicides B.

Also especially preferred are compositions 42.1 to 42.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.109 as further herbicide B.

Also especially preferred are compositions 43.1 to 43.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.1 1 1 as further herbicide B.

Also especially preferred are compositions 44.1 to 44.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.111 and B.67 as further herbicides B.

Also especially preferred are compositions 45.1 to 45.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.111 and B.76 as further herbicides B.

Also especially preferred are compositions 46.1 to 46.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.111 and B.82 as further herbicides B.

Also especially preferred are compositions 47.1 to 47.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B. 116 as further herbicide B.

Also especially preferred are compositions 48.1 to 48.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.116 and B.67 as further herbicides B.

Also especially preferred are compositions 49.1 to 49.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.116 and B.94 as further herbicides B.

Also especially preferred are compositions 50.1 to 50.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.116 and B.103 as further herbicides B.

Also especially preferred are compositions 51.1 to 51.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.116 and B.128 as further herbicides B.

Also especially preferred are compositions 52.1 to 52.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.116 and B.104 as further herbicides B.

Also especially preferred are compositions 53.1 to 53.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.116 and B.107 as further herbicides B.

Also especially preferred are compositions 54.1 to 54.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.116 and B.111 as further herbicides B.

Also especially preferred are compositions 55.1 to 55.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.122 as further herbicide B.

Also especially preferred are compositions 56.1 to 56.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.126 as further herbicide B.

Also especially preferred are compositions 57.1 to 57.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.128 as further herbicide B.

Also especially preferred are compositions 58.1 to 58.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they additionally comprise B.131 as further herbicide B. Also especially preferred are compositions 59.1 o 59.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.132 as further herbicide B.

Also especially preferred are compositions 60.1 :o 60.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.133 as further herbicide B.

Also especially preferred are compositions 61.1 :o 61.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.135 as further herbicide B.

Also especially preferred are compositions 62.1 :o 62.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.137 as further herbicide B.

Also especially preferred are compositions 63.1 :o 63.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.138 as further herbicide B.

Also especially preferred are compositions 64.1 :o 64.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.140 as further herbicide B.

Also especially preferred are compositions 65.1 :o 65.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.145 as further herbicide B.

Also especially preferred are compositions 66.1 :o 66.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.153 as further herbicide B.

Also especially preferred are compositions 67.1 :o 67.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.156 as further herbicide B.

Also especially preferred are compositions 68.1 :o 68.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.171 as further herbicide B.

Also especially preferred are compositions 69.1 :o 69.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they additionally comprise B.174 as further herbicide B.

Also especially preferred are compositions 70.1 :o 70.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they comprise the compound (1.1.1-10) place of the compound (1.1.1-3).

Also especially preferred are compositions 71.1 :o 71.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they comprise the compound (1.1.1-11) place of the compound (1.1.1-3).

Also especially preferred are compositions 72.1 :o 72.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they comprise the compound (1.1.1-17) place of the compound (1.1.1-3).

Also especially preferred are compositions 73.1 :o 73.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in hat they comprise the compound (1.1.1-18) place of the compound (1.1.1-3).

Also especially preferred are compositions 74.1 to 74.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.1.1-24) in place of the compound (1.1.1-3).

Also especially preferred are compositions 75.1 to 75.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.1.1-25) in place of the compound (1.1.1-3).

Also especially preferred are compositions 76.1 to 76.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.1.1-31) in place of the compound (1.1.1-3).

Also especially preferred are compositions 77.1 to 77.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.1.1-32) in place of the compound (1.1.1-3).

Also especially preferred are compositions 78.1 to 78.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.1.1-38) in place of the compound (1.1.1-3).

Also especially preferred are compositions 79.1 to 79.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.1.1-39) in place of the compound (1.1.1-3).

Also especially preferred are compositions 80.1 to 80.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.1.1-45) in place of the compound (1.1.1-3).

Also especially preferred are compositions 81.1 to 81.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.1.1-46) in place of the compound (1.1.1-3).

Also especially preferred are compositions 82.1 to 82.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.1.1-52) in place of the compound (1.1.1-3).

Also especially preferred are compositions 83.1 to 83.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.1.1-53) in place of the compound (1.1.1-3).

Also especially preferred are compositions 84.1 to 84.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.1.1-59) in place of the compound (1.1.1-3).

Also especially preferred are compositions 85.1 to 85.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.1.1-60) in place of the compound (1.1.1-3).

Also especially preferred are compositions 86.1 to 86.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.1.1-66) in place of the compound (1.1.1-3).

Also especially preferred are compositions 87.1 to 87.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.1.1-67) in place of the compound (1.1.1-3).

Also especially preferred are compositions 88.1 to 88.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-3) in place of the compound (1.1.1-3).

Also especially preferred are compositions 89.1 to 89.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-4) in place of the compound (1.1.1-3).

Also especially preferred are compositions 90.1 to 90.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-10) in place of the compound (1.1.1-3).

Also especially preferred are compositions 91.1 to 91.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-11) in place of the compound (1.1.1-3).

Also especially preferred are compositions 92.1 to 92.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-17) in place of the compound (1.1.1-3).

Also especially preferred are compositions 93.1 to 93.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-24) in place of the compound (1.1.1-3).

Also especially preferred are compositions 94.1 to 94.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-25) in place of the compound (1.1.1-3).

Also especially preferred are compositions 95.1 to 95.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-31) in place of the compound (1.1.1-3).

Also especially preferred are compositions 96.1 to 96.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-32) in place of the compound (1.1.1-3).

Also especially preferred are compositions 97.1 to 97.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-38) in place of the compound (1.1.1-3).

Also especially preferred are compositions 98.1 to 98.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-39) in place of the compound (1.1.1-3).

Also especially preferred are compositions 99.1 to 99.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-45) in place of the compound (1.1.1-3).

Also especially preferred are compositions 100.1 to 100.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-46) in place of the compound (1.1.1-3).

Also especially preferred are compositions 101.1 to 101.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-52) in place of the compound (1.1.1-3).

Also especially preferred are compositions 102.1 to 102.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-53) in place of the compound (1.1.1-3). Also especially preferred are compositions 103.1 to 103.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-59) in place of the compound (1.1.1-3).

Also especially preferred are compositions 104.1 to 104.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-60) in place of the compound (1.1.1-3).

Also especially preferred are compositions 105.1 to 105.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-66) in place of the compound (1.1.1-3).

Also especially preferred are compositions 106.1 to 106.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-67) in place of the compound (1.1.1-3).

Also especially preferred are compositions 107.1 to 107.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-3) in place of the compound (1.1.1-3).

Also especially preferred are compositions 108.1 to 108.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-4) in place of the compound (1.1.1-3).

Also especially preferred are compositions 109.1 to 109.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-10) in place of the compound (1.1.1-3).

Also especially preferred are compositions 110.1 to 110.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-11) in place of the compound (1.1.1-3).

Also especially preferred are compositions 111.1 to 111.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-17) in place of the compound (1.1.1-3).

Also especially preferred are compositions 112.1 to 112.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-18) in place of the compound (1.1.1-3).

Also especially preferred are compositions 113.1 to 113.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-24) in place of the compound (1.1.1-3).

Also especially preferred are compositions 114.1 to 114.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-25) in place of the compound (1.1.1-3).

Also especially preferred are compositions 115.1 to 115.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-31) in place of the compound (1.1.1-3).

Also especially preferred are compositions 116.1 to 116.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-32) in place of the compound (1.1.1-3).

Also especially preferred are compositions 117.1 to 117.3653 which differ from the corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-38) in place of the compound (1.1.1-3).

Also especially preferred are compositions 118.1 to 118.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-39) in place of the compound (1.1.1-3).

Also especially preferred are compositions 119.1 to 119.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-45) in place of the compound (1.1.1-3).

Also especially preferred are compositions 120.1 to 120.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-46) in place of the compound (1.1.1-3).

Also especially preferred are compositions 121.1 to 121.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-52) in place of the compound (1.1.1-3).

Also especially preferred are compositions 122.1 to 122.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-53) in place of the compound (1.1.1-3).

Also especially preferred are compositions 123.1 to 123.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-59) in place of the compound (1.1.1-3).

Also especially preferred are compositions 124.1 to 124.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-60) in place of the compound (1.1.1-3).

Also especially preferred are compositions 125.1 to 125.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-66) in place of the compound (1.1.1-3).

Also especially preferred are compositions 126.1 to 126.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.5.1-67) in place of the compound (1.1.1-3).

Also especially preferred are compositions 127.1 to 127.3653 which differ from the

corresponding compositions 1.1 to 1.3653 only in that they comprise the compound (1.2.1-18) in place of the compound (1.1.1-3).

The invention also relates to agrochemical compositions comprising at least an auxiliary and at least one pyrimidine compound of formula (I) according to the invention.

An agrochemical composition comprises a pesticidal effective amount of a pyrimidine compound of formula (I). The term "effective amount" denotes an amount of the composition or of the compounds I, which is sufficient for controlling unwanted plants, especially for controlling unwanted plants in cultivated plants and which does not result in a substantial damage to the treated plants. Such an amount can vary in a broad range and is dependent on various factors, such as the plants to be controlled, the treated cultivated plant or material, the climatic conditions and the specific pyrimidine compound of formula (I) used.

The pyrimidine compounds of formula (I), their N-oxides, salts or derivatives can be converted into customary types of agrochemical compositions, e. g. solutions, emulsions, suspensions, dusts, powders, pastes, granules, pressings, capsules, and mixtures thereof. Examples for agrochemical composition types are suspensions (e.g. SC, OD, FS), emulsifiable concentrates (e.g. EC), emulsions (e.g. EW, EO, ES, ME), capsules (e.g. CS, ZC), pastes, pastilles, wettable powders or dusts (e.g. WP, SP, WS, DP, DS), pressings (e.g. BR, TB, DT), granules (e.g. WG, SG, GR, FG, GG, MG), insecticidal articles (e.g. LN), as well as gel formulations for the treatment of plant propagation materials such as seeds (e.g. GF). These and further

agrochemical compositions types are defined in the "Catalogue of pesticide formulation types and international coding system", Technical Monograph No. 2, 6 th Ed. May 2008, CropLife International.

The agrochemical compositions are prepared in a known manner, such as described by Mollet and Grubemann, Formulation technology, Wiley VCH, Weinheim, 2001 ; or Knowles, New developments in crop protection product formulation, Agrow Reports DS243, T&F Informa, London, 2005.

Suitable auxiliaries are solvents, liquid carriers, solid carriers or fillers, surfactants,

dispersants, emulsifiers, wetters, adjuvants, solubilizers, penetration enhancers, protective colloids, adhesion agents, thickeners, humectants, repellents, attractants, feeding stimulants, compatibilizers, bactericides, anti-freezing agents, anti-foaming agents, colorants, tackifiers and binders.

Suitable solvents and liquid carriers are water and organic solvents, such as mineral oil fractions of medium to high boiling point, e.g. kerosene, diesel oil; oils of vegetable or animal origin; aliphatic, cyclic, and aromatic hydrocarbons, e. g. toluene, paraffin,

tetrahydronaphthalene, alkylated naphthalenes; alcohols, e.g. ethanol, propanol, butanol, benzylalcohol, cyclohexanol; glycols; DMSO; ketones, e.g. cyclohexanone; esters, e.g. lactates, carbonates, fatty acid esters, gamma-butyrolactone; fatty acids; phosphonates; amines; amides, e.g. N-methylpyrrolidone, fatty acid dimethylamides; and mixtures thereof.

Suitable solid carriers or fillers are mineral earths, e.g. silicates, silica gels, talc, kaolins, limestone, lime, chalk, clays, dolomite, diatomaceous earth, bentonite, calcium sulfate, magnesium sulfate, magnesium oxide; polysaccharides, e.g. cellulose, starch; fertilizers, e.g. ammonium sulfate, ammonium phosphate, ammonium nitrate, ureas; products of vegetable origin, e.g. cereal meal, tree bark meal, wood meal, nutshell meal, and mixtures thereof.

Suitable surfactants are surface-active compounds, such as anionic, cationic, non-ionic, and amphoteric surfactants, block polymers, polyelectrolytes, and mixtures thereof. Such surfactants can be used as emulsifier, dispersant, solubilizer, wetter, penetration enhancer, protective colloid, or adjuvant. Examples of surfactants are listed in McCutcheon's, Vol.1 : Emulsifiers & Detergents, McCutcheon's Directories, Glen Rock, USA, 2008 (International Ed. or North American Ed.).

Suitable anionic surfactants are alkali, alkaline earth or ammonium salts of sulfonates, sulfates, phosphates, carboxylates, and mixtures thereof. Examples of sulfonates are alkylarylsulfonates, diphenylsulfonates, alpha-olefin sulfonates, lignine sulfonates, sulfonates of fatty acids and oils, sulfonates of ethoxylated alkylphenols, sulfonates of alkoxylated

arylphenols, sulfonates of condensed naphthalenes, sulfonates of dodecyl- and

tridecylbenzenes, sulfonates of naphthalenes and alkylnaphthalenes, sulfosuccinates or sulfosuccinamates. Examples of sulfates are sulfates of fatty acids and oils, of ethoxylated alkylphenols, of alcohols, of ethoxylated alcohols, or of fatty acid esters. Examples of phosphates are phosphate esters. Examples of carboxylates are alkyl carboxylates, and carboxylated alcohol or alkylphenol ethoxylates.

Suitable nonionic surfactants are alkoxylates, N-substituted fatty acid amides, amine oxides, esters, sugar-based surfactants, polymeric surfactants, and mixtures thereof. Examples of alkoxylates are compounds such as alcohols, alkylphenols, amines, amides, a ryl phenols, fatty acids, or fatty acid esters which have been alkoxylated with 1 to 50 equivalents. Ethylene oxide and/or propylene oxide may be employed for the alkoxylation, preferably ethylene oxide.

Examples of N-substituted fatty acid amides are fatty acid glucamides or fatty acid

alkanolamides. Examples of esters are fatty acid esters, glycerol esters, or monoglycerides. Examples of sugar-based surfactants are sorbitans, ethoxylated sorbitans, sucrose, and glucose esters, or alkylpoly-glucosides. Examples of polymeric surfactants are home- or copolymers of vinylpyrrolidone, vinylalcohols, or vinylacetate.

Suitable cationic surfactants are quaternary surfactants, e.g. quaternary ammonium compounds with one or two hydrophobic groups, or salts of long-chain primary amines. Suitable amphoteric surfactants are alkylbetains and imidazolines. Suitable block polymers are block polymers of the A-B or A-B-A type comprising blocks of polyethylene oxide and polypropylene oxide, or of the A-B-C type comprising alkanol, polyethylene oxide and polypropylene oxide. Suitable polyelectrolytes are polyacids or polybases. Examples of polyacids are alkali salts of polyacrylic acid or polyacid comb polymers. Examples of polybases are polyvinylamines or polyethyleneamines.

Suitable adjuvants are compounds, which have a neglectable or even no pesticidal activity themselves, and which improve the biological performance of the pyrimidine compounds of formula (I) on the target. Examples are surfactants, mineral or vegetable oils, and other auxiliaries. Further examples are listed by Knowles, Adjuvants, and additives, Agrow Reports DS256, T&F Informa UK, 2006, chapter 5.

Suitable thickeners are polysaccharides (e.g. xanthan gum, carboxymethylcellulose), inorganic clays (organically modified or unmodified), polycarboxylates, and silicates.

Suitable bactericides are bronopol and isothiazolinone derivatives such as

alkylisothiazolinones and benzisothiazolinones.

Suitable anti-freezing agents are ethylene glycol, propylene glycol, urea, and glycerin.

Suitable anti-foaming agents are silicones, long chain alcohols, and salts of fatty acids.

Suitable colorants (e.g. in red, blue, or green) are pigments of low water solubility and water- soluble dyes. Examples are inorganic colorants (e.g. iron oxide, titan oxide, iron

hexacyanoferrate) and organic colorants (e.g. alizarin-, azo-, and phthalocyanine colorants). Suitable tackifiers or binders are polyvinylpyrrolidons, polyvinylacetates, polyvinyl alcohols, polyacrylates, biological or synthetic waxes, and cellulose ethers.

Examples for agrochemical composition types and their preparation are:

i) Water-soluble concentrates (SL, LS)

10-60 wt% of a pyrimidine compound of formula (I) according to the invention and 5-15 wt% wetting agent (e.g. alcohol alkoxylates) are dissolved in water and/or in a water-soluble solvent (e.g. alcohols) ad 100 wt%. The active substance dissolves upon dilution with water.

ii) Dispersible concentrates (DC)

5-25 wt% of a pyrimidine compound of formula (I) according to the invention and 1-10 wt% dispersant (e. g. polyvinylpyrrolidone) are dissolved in organic solvent (e.g. cyclohexanone) ad 100 wt%. Dilution with water gives a dispersion.

iii) Emulsifiable concentrates (EC)

15-70 wt% of a pyrimidine compound of formula (I) according to the invention and 5-10 wt% emulsifiers (e.g. calcium dodecylbenzenesulfonate and castor oil ethoxylate) are dissolved in water-insoluble organic solvent (e.g. aromatic hydrocarbon) ad 100 wt%. Dilution with water gives an emulsion.

iv) Emulsions (EW, EO, ES)

5-40 wt% of a pyrimidine compound of formula (I) according to the invention and 1-10 wt% emulsifiers (e.g. calcium dodecylbenzenesulfonate and castor oil ethoxylate) are dissolved in 20-40 wt% water-insoluble organic solvent (e.g. aromatic hydrocarbon). This mixture is introduced into water ad 100 wt% by means of an emulsifying machine and made into a homogeneous emulsion. Dilution with water gives an emulsion.

v) Suspensions (SC, OD, FS)

In an agitated ball mill, 20-60 wt% of a pyrimidine compound of formula (I) according to the invention are comminuted with addition of 2-10 wt% dispersants and wetting agents (e.g.

sodium lignosulfonate and alcohol ethoxylate), 0,1-2 wt% thickener (e.g. xanthan gum) and water ad 100 wt% to give a fine active substance suspension. Dilution with water gives a stable suspension of the active substance. For FS type composition up to 40 wt% binder (e.g.

polyvinylalcohol) is added.

vi) Water-dispersible granules and water-soluble granules (WG, SG)

50-80 wt% of a pyrimidine compound of formula (I) according to the invention are ground finely with addition of dispersants and wetting agents (e.g. sodium lignosulfonate and alcohol ethoxylate) ad 100 wt% and prepared as water-dispersible or water-soluble granules by means of technical appliances (e. g. extrusion, spray tower, fluidized bed). Dilution with water gives a stable dispersion or solution of the active substance.

vii) Water-dispersible powders and water-soluble powders (WP, SP, WS)

50-80 wt% of a pyrimidine compound of formula (I) according to the invention are ground in a rotor-stator mill with addition of 1-5 wt% dispersants (e.g. sodium lignosulfonate), 1-3 wt% wetting agents (e.g. alcohol ethoxylate) and solid carrier (e.g. silica gel) ad 100 wt%. Dilution with water gives a stable dispersion or solution of the active substance.

viii) Gel (GW, GF)

In an agitated ball mill, 5-25 wt% of a pyrimidine compound of formula (I) according to the invention are comminuted with addition of 3-10 wt% dispersants (e.g. sodium lignosulfonate), 1- 5 wt% thickener (e.g. carboxymethylcellulose) and water ad 100 wt% to give a fine suspension of the active substance. Dilution with water gives a stable suspension of the active substance. iv) Microemulsion (ME)

5-20 wt% of a pyrimidine compound of formula (I) according to the invention are added to 5-30 wt% organic solvent blend (e.g. fatty acid dimethylamide and cyclohexanone), 10-25 wt% surfactant blend (e.g. alcohol ethoxylate and arylphenol ethoxylate), and water ad 100 %. This mixture is stirred for 1 h to produce spontaneously a thermodynamically stable microemulsion. iv) Microcapsules (CS)

An oil phase comprising 5-50 wt% of a pyrimidine compound of formula (I) according to the invention, 0-40 wt% water insoluble organic solvent (e.g. aromatic hydrocarbon), 2-15 wt% acrylic monomers (e.g. methylmethacrylate, methacrylic acid, and a di- or triacrylate) are dispersed into an aqueous solution of a protective colloid (e.g. polyvinyl alcohol). Radical polymerization initiated by a radical initiator results in the formation of poly(meth)acrylate microcapsules. Alternatively, an oil phase comprising 5-50 wt% of a pyrimidine compound of formula (I) according to the invention, 0-40 wt% water insoluble organic solvent (e.g. aromatic hydrocarbon), and an isocyanate monomer (e.g. diphenylmethene-4,4'-diisocyanate) are dispersed into an aqueous solution of a protective colloid (e.g. polyvinyl alcohol). The addition of a polyamine (e.g. hexamethylenediamine) results in the formation of polyurea microcapsules. The monomers amount to 1-10 wt%. The wt% relate to the total CS composition.

ix) Dustable powders (DP, DS)

1-10 wt% of a pyrimidine compound of formula (I) according to the invention are ground finely and mixed intimately with solid carrier (e.g. finely divided kaolin) ad 100 wt%.

x) Granules (GR, FG)

0.5-30 wt% of a pyrimidine compound of formula (I) according to the invention is ground finely and associated with solid carrier (e.g. silicate) ad 100 wt%. Granulation is achieved by extrusion, spray-drying or the fluidized bed.

xi) Ultra-low volume liquids (UL)

1-50 wt% of a pyrimidine compound of formula (I) according to the invention are dissolved in organic solvent (e.g. aromatic hydrocarbon) ad 100 wt%.

The agrochemical compositions types i) to xi) may optionally comprise further auxiliaries, such as 0,1-1 wt% bactericides, 5-15 wt% anti-freezing agents, 0,1-1 wt% anti-foaming agents, and 0,1-1 wt% colorants.

The agrochemical compositions comprising generally comprise between 0.01 and 95%, preferably between 0.1 and 90%, and in particular between 0.5 and 75%, by weight of the pyrimidine compound of formula (I). The pyrimidine compounds of formula (I) are employed in a purity of from 90% to 100%, preferably from 95% to 100% (according to NMR spectrum).

Solutions for seed treatment (LS), suspoemulsions (SE), flowable concentrates (FS), powders for dry treatment (DS), water-dispersible powders for slurry treatment (WS), water-soluble powders (SS), emulsions (ES), emulsifiable concentrates (EC) and gels (GF) are usually employed for the purposes of treatment of plant propagation materials, particularly seeds. The agrochemical compositions in question give, after two-to-tenfold dilution, active substance concentrations of from 0.01 to 60% by weight, preferably from 0.1 to 40% by weight, in the ready-to-use preparations. Application can be carried out before or during sowing.

Methods for applying pyrimidine compounds of formula (I) and agrochemical compositions thereof, on to plant propagation material, especially seeds, include dressing, coating, pelleting, dusting, soaking and in-furrow application methods of the propagation material. Preferably, pyrimidine compounds of formula (I) and agrochemical compositions thereof, are applied on to the plant propagation material by a method such that germination is not induced, e. g. by seed dressing, pelleting, coating and dusting.

Various types of oils, wetters, adjuvants, fertilizer, or micronutrients, and further pesticides (e.g. herbicides, insecticides, fungicides, growth regulators, safeners) may be added to the pyrimidine compounds of formula (I) and the agrochemical compositions comprising them as premix or, if appropriate not until immediately prior to use (tank mix). These agents can be admixed with the agrochemical compositions according to the invention in a weight ratio of 1 :100 to 100:1 , preferably 1 :10 to 10:1. The user applies the pyrimidine compound of formula (I) according to the invention and the agrochemical compositions comprising them usually from a pre-dosage device, a knapsack sprayer, a spray tank, a spray plane, or an irrigation system. Usually, the agrochemical composition is made up with water, buffer, and/or further auxiliaries to the desired application concentration and the ready-to-use spray liquor or the agrochemical composition according to the invention is thus obtained. Usually, 20 to 2000 liters, preferably 50 to 400 liters, of the ready- to-use spray liquor are applied per hectare of agricultural useful area.

According to one embodiment, either individual components of the agrochemical composition according to the invention or partially premixed components, e. g. components comprising pyrimidine compounds of formula (I) may be mixed by the user in a spray tank and further auxiliaries and additives may be added, if appropriate.

In a further embodiment, individual components of the agrochemical composition according to the invention such as parts of a kit or parts of a binary or ternary mixture may be mixed by the user himself in a spray tank and further auxiliaries may be added, if appropriate.

In a further embodiment, either individual components of the agrochemical composition according to the invention or partially premixed components, e. g components comprising pyrimidine compounds of formula (I) can be applied jointly (e.g. after tank mix) or consecutively.

The pyrimidine compounds of formula (I), are suitable as herbicides. They are suitable as such or as an appropriately formulated composition (agrochemical composition).

The pyrimidine compounds of formula (I), or the agrochemical compositions comprising the pyrimidine compounds of formula (I), control vegetation on non-crop areas very efficiently, especially at high rates of application. They act against broad-leaved weeds and grass weeds in crops such as wheat, rice, maize, soya, and cotton without causing any significant damage to the crop plants. This effect is mainly observed at low rates of application.

The pyrimidine compounds of formula (I), or the agrochemical compositions comprising them, are applied to the plants mainly by spraying the leaves. Here, the application can be carried out using, e.g., water as carrier by customary spraying techniques using spray liquor amounts of from about 100 to 1000 l/ha (e.g. from 300 to 400 l/ha). The pyrimidine compounds of formula (I), or the agrochemical compositions comprising them, may also be applied by the low-volume or the ultra-low-volume method, or in the form of micro granules.

Application of the pyrimidine compounds of formula (I), or the agrochemical compositions comprising them, can be done before, during, and/or after, preferably during and/or after, the emergence of the undesirable plants.

The pyrimidine compounds of formula (I), or the agrochemical compositions comprising them, can be applied pre-, post-emergence or pre-plant, or together with the seed of a crop plant. It is also possible to apply the pyrimidine compounds of formula (I), or the agrochemical

compositions comprising them, by applying seed, pretreated with the pyrimidine compounds of formula (I), or the agrochemical compositions comprising them, of a crop plant. If the active ingredients are less well tolerated by certain crop plants, application techniques may be used in which the herbicidal compositions are sprayed, with the aid of the spraying equipment, in such a way that as far as possible they do not come into contact with the leaves of the sensitive crop plants, while the active ingredients reach the leaves of undesirable plants growing underneath, or the bare soil surface (post-directed, lay-by).

In a further embodiment, the pyrimidine compounds of formula (I), or the agrochemical compositions comprising them, can be applied by treating seed. The treatment of seeds comprises essentially all procedures familiar to the person skilled in the art (seed dressing, seed coating, seed dusting, seed soaking, seed film coating, seed multilayer coating, seed

encrusting, seed dripping and seed pelleting) based on the pyrimidine compounds of formula (I), or the agrochemical compositions prepared therefrom. Here, the herbicidal compositions can be applied diluted or undiluted.

The term "seed" comprises seed of all types, such as, e.g., corns, seeds, fruits, tubers, seedlings and similar forms. Here, preferably, the term seed describes corns and seeds. The seed used can be seed of the useful plants mentioned above, but also the seed of transgenic plants or plants obtained by customary breeding methods.

When employed in plant protection, the amounts of active substances applied, i.e. the pyrimidine compounds of formula (I) without formulation auxiliaries, are, depending on the kind of effect desired, from 0.001 to 2 kg per ha, preferably from 0.005 to 2 kg per ha, more preferably from 0.05 to 0.9 kg per ha and in particular from 0.1 to 0.75 kg per ha.

In another embodiment of the invention, the application rate of the pyrimidine compounds of formula (I) is from 0.001 to 3 kg/ha, preferably from 0.005 to 2.5 kg/ha and in particular from 0.01 to 2 kg/ha of active substance (a.s.).

In another preferred embodiment of the invention, the rates of application of the pyrimidine compounds of formula (I) according to the present invention (total amount of pyrimidine compounds of formula (I)) are from 0.1 g/ha to 3000 g/ha, preferably 10 g/ha to 1000 g/ha, depending on the control target, the season, the target plants and the growth stage.

In another preferred embodiment of the invention, the application rates of the pyrimidine compounds of formula (I) are in the range from 0.1 g/ha to 5000 g/ha and preferably in the range from 1 g/ha to 2500 g/ha or from 5 g/ha to 2000 g/ha.

In another preferred embodiment of the invention, the application rate of the pyrimidine compounds of formula (I) is 0.1 to 1000 g/ha, preferablyl to 750 g/ha, more preferably 5 to 500 g/ha.

In treatment of plant propagation materials such as seeds, e. g. by dusting, coating or drenching seed, amounts of active substance of from 0.1 to 1000 g, preferably from 1 to 1000 g, more preferably from 1 to 100 g, and most preferably from 5 to 100 g, per 100 kilogram of plant propagation material (preferably seeds) are generally required.

In another embodiment of the invention, to treat the seed, the amounts of active substances applied, i.e. the pyrimidine compounds of formula (I) are generally employed in amounts of from

0.001 to 10 kg per 100 kg of seed.

When used in the protection of materials or stored products, the amount of active substance applied depends on the kind of application area and on the desired effect. Amounts customarily applied in the protection of materials are 0.001 g to 2 kg, preferably 0.005 g to 1 kg, of active substance per cubic meter of treated material.

Depending on the application method in question, the pyrimidine compounds of formula (I), or the agrochemical compositions comprising them, can additionally be employed in a further number of crop plants for eliminating undesirable plants. Examples of suitable crops are the following:

Allium cepa, Ananas comosus, Arachis hypogaea, Asparagus officinalis, Avena sativa, Beta vulgaris spec, altissima, Beta vulgaris spec, rapa, Brassica napus var. napus, Brassica napus var. napobrassica, Brassica rapa var. silvestris, Brassica oleracea, Brassica nigra, Camellia sinensis, Carthamus tinctorius, Carya illinoinensis, Citrus limon, Citrus sinensis, Coffea arabica (Coffea canephora, Coffea liberica), Cucumis sativus, Cynodon dactylon, Daucus carota, Elaeis guineensis, Fragaria vesca, Glycine max, Gossypium hirsutum, (Gossypium arboreum,

Gossypium herbaceum, Gossypium vitifolium), Helianthus annuus, Hevea brasiliensis, Hordeum vulgare, Humulus lupulus, Ipomoea batatas, Juglans regia, Lens culinaris, Linum usitatissimum, Lycopersicon lycopersicum, Malus spec, Manihot esculenta, Medicago sativa, Musa spec, Nicotiana tabacum (N.rustica), Olea europaea, Oryza sativa, Phaseolus lunatus, Phaseolus vulgaris, Picea abies, Pinus spec, Pistacia vera, Pisum sativum, Prunus avium, Prunus persica, Pyrus communis, Prunus armeniaca, Prunus cerasus, Prunus dulcis and Prunus domestica, Ribes sylvestre, Ricinus communis, Saccharum officinarum, Secale cereale, Sinapis alba, Solanum tuberosum, Sorghum bicolor (s. vulgare), Theobroma cacao, Trifolium pratense, Triticum aestivum, Triticale, Triticum durum, Vicia faba, Vitis vinifera, and Zea mays.

Preferred crops are Arachis hypogaea, Beta vulgaris spec, altissima, Brassica napus var. napus, Brassica oleracea, Citrus limon, Citrus sinensis, Coffea arabica (Coffea canephora, Coffea liberica), Cynodon dactylon, Glycine max, Gossypium hirsutum, (Gossypium arboreum, Gossypium herbaceum, Gossypium vitifolium), Helianthus annuus, Hordeum vulgare, Juglans regia, Lens culinaris, Linum usitatissimum, Lycopersicon lycopersicum, Malus spec, Medicago sativa, Nicotiana tabacum (N.rustica), Olea europaea, Oryza sativa , Phaseolus lunatus, Phaseolus vulgaris, Pistacia vera, Pisum sativum, Prunus dulcis, Saccharum officinarum,

Secale cereale, Solanum tuberosum, Sorghum bicolor (s. vulgare), Triticale, Triticum aestivum, Triticum durum, Vicia faba, Vitis vinifera, and Zea mays.

Especially preferred crops are crops of cereals, corn, soybeans, rice, oilseed rape, cotton, potatoes, peanuts, or permanent crops.

The pyrimidine compounds of formula (I) according to the invention, or the agrochemical compositions comprising them, can also be used in genetically modified plants. The term "genetically modified plants" is to be understood as plants whose genetic material has been modified by the use of recombinant DNA techniques to include an inserted sequence of DNA that is not native to that plant species' genome or to exhibit a deletion of DNA that was native to that species' genome, wherein the modification(s) cannot readily be obtained by cross breeding, mutagenesis or natural recombination alone. Often, a particular genetically modified plant will be one that has obtained its genetic modification(s) by inheritance through a natural breeding or propagation process from an ancestral plant whose genome was the one directly treated by use of a recombinant DNA technique. Typically, one or more genes have been integrated into the genetic material of a genetically modified plant in order to improve certain properties of the plant. Such genetic modifications also include but are not limited to targeted post-translational modification of protein(s), oligo- or polypeptides, e. g., by inclusion therein of amino acid mutation(s) that permit, decrease, or promote glycosylation or polymer additions such as prenylation, acetylation farnesylation, or PEG moiety attachment.

Plants that have been modified by breeding, mutagenesis or genetic engineering, e.g. have been rendered tolerant to applications of specific classes of herbicides, such as auxin herbicides such as dicamba or 2,4-D; bleacher herbicides such as hydroxyphenylpyruvate dioxygenase (HPPD) inhibitors or phytoene desaturase (PDS) inhibitors; acetolactate synthase (ALS) inhibitors such as sulfonyl ureas or imidazolinones; enolpyruvyl shikimate 3-phosphate synthase (EPSP) inhibitors such as glyphosate; glutamine synthetase (GS) inhibitors such as glufosinate; protoporphyrinogen-IX oxidase inhibitors; lipid biosynthesis inhibitors such as acetyl CoA carboxylase (ACCase) inhibitors; or oxynil (i. e. bromoxynil or ioxynil) herbicides as a result of conventional methods of breeding or genetic engineering; furthermore, plants have been made resistant to multiple classes of herbicides through multiple genetic modifications, such as resistance to both glyphosate and glufosinate or to both glyphosate and a herbicide from another class such as ALS inhibitors, HPPD inhibitors, auxin herbicides, or ACCase inhibitors. These herbicide resistance technologies are, e.g., described in Pest Management Science 61 , 2005, 246; 61 , 2005, 258; 61 , 2005, 277; 61 , 2005, 269; 61 , 2005, 286; 64, 2008, 326; 64, 2008, 332; Weed Science 57, 2009, 108; Australian Journal of Agricultural Research 58, 2007, 708; Science 316, 2007, 1185; and references quoted therein. Several cultivated plants have been rendered tolerant to herbicides by mutagenesis and conventional methods of breeding, e. g., Clearfield® summer rape (Canola, BASF SE, Germany) being tolerant to imidazolinones, e. g., imazamox, or ExpressSun® sunflowers (DuPont, USA) being tolerant to sulfonyl ureas, e. g., tribenuron. Genetic engineering methods have been used to render cultivated plants such as soybean, cotton, corn, beets and rape, tolerant to herbicides such as glyphosate,

imidazolinones, and glufosinate, some of which are under development or commercially available under the brands or trade names RoundupReady® (glyphosate tolerant, Monsanto, USA), Cultivance® (imidazolinone tolerant, BASF SE, Germany), and LibertyLink® (glufosinate tolerant, Bayer CropScience, Germany).

Furthermore, plants are also covered that are by the use of recombinant DNA techniques capable to synthesize one or more insecticidal proteins, especially those known from the bacterial genus Bacillus, particularly from Bacillus thuringiensis, such as delta-endotoxins, e. g., CrylA(b), CrylA(c), CrylF, CrylF(a2), CryllA(b), CrylllA, CrylllB(bl) or Cry9c; vegetative insecticidal proteins (VIP), e. g., VIP1 , VIP2, VIP3, or VIP3A; insecticidal proteins of bacteria colonizing nematodes, e. g., Photorhabdus spp. or Xenorhabdus spp.; toxins produced by animals, such as scorpion toxins, arachnid toxins, wasp toxins, or other insect-specific neurotoxins; toxins produced by fungi, such as Streptomycetes toxins, plant lectins, such as pea or barley lectins; agglutinins; proteinase inhibitors, such as trypsin inhibitors, serine protease inhibitors, patatin, cystatin or papain inhibitors; ribosome-inactivating proteins (RIP), such as ricin, maize-RIP, abrin, luffin, saporin or bryodin; steroid metabolism enzymes, such as 3- hydroxy-steroid oxidase, ecdysteroid-IDP-glycosyl-transferase, cholesterol oxidases, ecdysone inhibitors or HMG-CoA-reductase; ion channel blockers, such as blockers of sodium or calcium channels; juvenile hormone esterase; diuretic hormone receptors (helicokinin receptors);

stilbene synthase, bibenzyl synthase, chitinases or glucanases. In the context of the present invention these insecticidal proteins or toxins are to be understood expressly also as including pre-toxins, hybrid proteins, truncated or otherwise modified proteins. Hybrid proteins are characterized by a new combination of protein domains, (see, e. g., WO 02/015701). Further examples of such toxins or genetically modified plants capable of synthesizing such toxins are disclosed, e. g., in EP-A 374 753, WO 93/007278, WO 95/34656, EP-A 427 529, EP-A 451 878, WO 03/18810, and WO 03/52073. The methods for producing such genetically modified plants are generally known to the person skilled in the art and are described, e. g., in the publications mentioned above. These insecticidal proteins contained in the genetically modified plants impart to the plants producing these proteins tolerance to harmful pests from all taxonomic groups of arthropods, especially to beetles (Coeloptera), two-winged insects (Diptera), and moths (Lepidoptera) and to nematodes (Nematoda). Genetically modified plants capable to synthesize one or more insecticidal proteins are, e. g., described in the publications mentioned above, and some of which are commercially available such as YieldGard® (corn cultivars producing the CrylAb toxin), YieldGard® Plus (corn cultivars producing CrylAb and Cry3Bb1 toxins),

Starlink® (corn cultivars producing the Cry9c toxin), Herculex® RW (corn cultivars producing Cry34Ab1 , Cry35Ab1 and the enzyme Phosphinothricin-N-Acetyltransferase [PAT]); NuCOTN® 33B (cotton cultivars producing the CrylAc toxin), Bollgard® I (cotton cultivars producing the CrylAc toxin), Bollgard® II (cotton cultivars producing CrylAc and Cry2Ab2 toxins); VIPCOT® (cotton cultivars producing a VIP-toxin); NewLeaf® (potato cultivars producing the Cry3A toxin); Bt-Xtra®, NatureGard®, KnockOut®, BiteGard®, Protecta®, Bt11 (e. g., Agrisure® CB) and Bt176 from Syngenta Seeds SAS, France, (corn cultivars producing the CrylAb toxin and PAT enzyme), MIR604 from Syngenta Seeds SAS, France (corn cultivars producing a modified version of the Cry3A toxin, c.f. WO 03/018810), MON 863 from Monsanto Europe S.A., Belgium (corn cultivars producing the Cry3Bb1 toxin), IPC 531 from Monsanto Europe S.A., Belgium (cotton cultivars producing a modified version of the CrylAc toxin) and 1507 from Pioneer Overseas Corporation, Belgium (corn cultivars producing the Cry1 F toxin and PAT enzyme).

Furthermore, plants are also covered that are by the use of recombinant DNA techniques capable to synthesize one or more proteins to increase the resistance or tolerance of those plants to bacterial, viral or fungal pathogens. Examples of such proteins are the so-called

"pathogenesis-related proteins" (PR proteins, see, e.g., EP-A 392 225), plant disease resistance genes (e. g., potato culti-vars, which express resistance genes acting against Phytophthora infestans derived from the Mexican wild potato, Solanum bulbocastanum) or T4-lyso-zym (e.g., potato cultivars capable of synthesizing these proteins with increased resistance against bacteria such as Erwinia amylovora). The methods for producing such genetically modi-fied plants are generally known to the person skilled in the art and are described, e.g., in the publications mentioned above.

Furthermore, plants are also covered that are by the use of recombinant DNA techniques capable to synthesize one or more proteins to increase the productivity (e.g., bio-mass production, grain yield, starch content, oil content or protein content), tolerance to drought, salinity or other growth-limiting environmental factors or tolerance to pests and fungal, bacterial or viral pathogens of those plants.

Furthermore, plants are also covered that contain by the use of recombinant DNA techniques a modified amount of ingredients or new ingredients, specifically to improve human or animal nutrition, e. g., oil crops that produce health-promoting long-chain omega-3 fatty acids or unsaturated omega-9 fatty acids (e. g., Nexera® rape, Dow AgroSciences, Canada).

Furthermore, plants are also covered that contain by the use of recombinant DNA techniques a modified amount of ingredients or new ingredients, specifically to improve raw material production, e.g., potatoes that produce increased amounts of amylopectin (e.g. Amflora® potato, BASF SE, Germany).

The preparation of the pyrimidine compounds of formula (I) is illustrated by the following examples.

A Preparation examples Example 1 : [5-(3-Chloro-2-pyridyl)-2-cyclopropyl-pyrimidin-4-yl]methano l

1.1 5-Bromo-2-cyclopropyl-pyrimidine-4-carboxylic acid:

NaH (60% purity, 41.9 g) is added in portions to EtOH (800 mL) at 0 °C. The resulting mixture is warmed to ambient temperature and the cyclopropanecarboxamidine hydrochlorid (93.5 g) is added in portions. The reaction is warmed to 50 °C and maintained at this temperature for 0.5 h and then cooled to ambient temperature before mucobromic acid (100 g) is added in EtOH while keeping the internal temperature below 55 °C. The mixture is allowed to cool to ambient temperature and stirred for additional 16 h. All solid components are removed by filtration and the resulting solution is concentrated under reduced pressure. Aq. HCI (1 mol/L) is added, the aqueous phase is washed with EtOAc (3x), the combined organic extracts are dried over MgSO 4 and the solid parts removed by filtration. The residue is concentrated under reduced pressure and the resulting solid titrated with ('Pr)20. The solids are collected by filtration and dried yielding the title compound (68.0 g, yield 72 %) as a colorless solid.

1H NMR (400 MHz, CDCI 3 ): δ = 8.91 (s, 1 H), 2.38 - 2.26 (m, 1 H), 1.34 - 1.14 (m, 4H) ppm; MS (ESI) m/z 244.9 [M + H + ].

1.2 Methyl 5-bromo-2-cyclopropyl-pyrimidine-4-carboxylate:

5-Bromo-2-cyclopropyl-pyrimidine-4-carboxylic acid (91.0 g) is dissolved in MeOH (1200 mL) and cone, sulfuric acid (20 mL) is added dropwise at ambient temperature. The reaction is heated to reflux and stirred for 16 h. The resulting mixture is cooled to ambient temperature and neutralized with aq. sat. NaHCO 3 . The residue is parted between EtOAc and aq. sat. NaHCO 3 , the phases are separated, the aq. phase is extracted with EtOAc and the combined organics are dried over MgSO 4 . Solid parts are removed by filtration and the organic phase is

concentrated under reduced pressure. Column chromatography of the resulting crude product (ISCO-CombiFlash Rf, cyclohexane/EtOAc) yields the title compound (81.0 g, yield 84%) as a colorless solid.

H NMR (400 MHz, CDCI3): δ = 8.74 (s, 1 H), 4.01 (s, 3H), 2.33 - 2.22 (m, 1 H), 1.21 - 1.06 (m, 4H) ppm; MS (ESI) m/z 246.9 [M + H + ].

1.3 Methyl 2-cyclopropyl-5-(4,4,5,5-tetramethyl-1 ,3,2-dioxaborolan-2-yl)pyrimidine-4- carboxylate:

A mixture of methyl 2-cyclopropyl-5-(4,4,5,5-tetramethyl-1 ,3,2-dioxaborolan-2-yl)pyrimidine-4- carboxylate (1.00 g), 2,3-dibromopyridine (1.56 g), CsF (1.25 g) and PdCI2dppf (403 mg) in toluene (20 mL) is heated under reflux under an atmosphere of argon for 3 h. The volatiles are removed under reduced pressure and column chromatography of the crude product

(cyclohexane/EtOAc) yields the title compound (300 mg, yield 27%) as a colorless solid.

1 H NMR (400 MHz, CDCI3): δ 8.78 (s, 1 H), 8.62 (dd, J = 4.7, 1.5 Hz, 1 H), 7.99 (dd, J = 8.1 , 1.5 Hz, 1 H), 7.23 (dd, J = 8.1 , 4.7 Hz, 1 H), 3.82 (s, 3H), 2.47 - 2.41 (m, 1 H), 1.39 - 1.25 (m, 2H), 1.20 - 1.15 (m, 2H) ppm; MS (ESI) m/z 336.0 [M + H + ].

1.4 Methyl 5-(3-chloro-2-pyridyl)-2-cyclopropyl-pyrimidine-4-carboxylat e:

A mixture of methyl 2-cyclopropyl-5-(4,4,5,5-tetramethyl-1 ,3,2-dioxaborolan-2-yl)pyrimidine-4- carboxylate (33.0 g), 2-Bromo-3-chloropyridine (22.7 g), CsF (41.2 g) and PdCI 2 dppf (13.3 g) in toluene (350 mL) is heated under reflux under an atmosphere of argon for 3 h. The volatiles are removed under reduced pressure and column chromatography of the crude product

(cyclohexane/EtOAc) yields the title compound (10.0 g, yield 32%) as a colorless solid. H NMR (400 MHz, CDCI 3 ): δ 8.81 (s, 1 H), 8.58 (dd, J = 4.8, 1.1 Hz, 1 H), 7.81 (dd, J = 8.1 , 1.3 Hz, 1 H), 7.31 (dd, J = 8.2, 4.7 Hz, 1 H), 3.82 (s, 3H), 2.47 - 2.40 (m, 1 H), 1.29 - 1.23 (m, 2H), 1.20 - 1.15 (m, 2H) ppm; MS (ESI) m/z 290.0 [M + H + ].

1.5 5-(3-Chloro-2-pyridyl)-2-cyclopropyl-pyrimidine-4-carboxylic acid:

Methyl 5-(3-chloro-2-pyridyl)-2-cyclopropyl-pyrimidine-4-carboxylat e (1.30 g) is dissolved in a mixture THF/water (vol/vol = 1/1 ; 50 mL) and lithiumhydroxid (215 mg) is added as a solution in water. The resulting mixture is stirred for 20 hours at ambient temperature and then acidified to pH = 2 - 3 with aqueous hydrochloric acid (2 mol/L). The aq. phase is extracted with EtOAc (3 x) and the combined organics are dried over Na2SO 4 . Solid parts are removed by filtration and the organic phase is concentrated under reduced pressure and the residues are triturated with CH2CI2 yielding the title compound (850 mg, 69%) as a colorless solid.

H NMR (400 MHz, CDCI3): δ 8.79 (s, 1 H), 8.59 (dd, J = 4.8, 1.4 Hz, 1 H), 7.83 (dd, J = 8.1 , 1.3 Hz, 1 H), 7.36 (dd, J = 8.2, 4.7 Hz, 1 H), 2.46 - 2.40 (m, 1 H), 1.32 - 1.23 (m, 4H) ppm; MS (ESI) m/z 275.9 [M + H + ].

1.6 [5-(3-Chloro-2-pyridyl)-2-cyclopropyl-pyrimidin-4-yl]methano l:

To a solution of 5-(3-Chloro-2-pyridyl)-2-cyclopropyl-pyrimidine-4-carboxylic acid (15.0 g) in THF (20 mL) CDI (10.0 g) is added in small portions. The resulting mixture is stirred for 1 h at ambient temperature and cooled to 0°C before NaBH 4 (4.11 g) in ice-cold water (10 mL) is added. After stirring for two additional hours at ambient temperature, EtOAc is added and the phases are separated. The aq. phase is extracted with EtOAc (2x), the combined organics are washed with water and dried over Na2SO 4 . Solid parts are removed by filtration, the remaining solution is concentrated under reduced pressure and column chromatography of the crude product (cyclohexane/EtOAc) yields the title compound (5.00 g, yield 33%).

H NMR (400 MHz, CDCI3): δ 8.61 (s, 1 H), 8.60 (dd, J = 4.7, 1.5Hz, 1 H), 7.87 (dd, J = 8.2, 1.5 Hz, 1 H), 7.34 (dd, J = 8.2, 4.7 Hz, 1 H), 4.56 (s, 2H), 2.40 - 2.34 (m, 1 H), 1.28 - 1.24 (m, 2H), 1.19 - 1.14 (m, 2H) ppm; MS (ESI) m/z 262.0 [M + H + ].

Example 2: 5-(3-Bromo-2-pyridyl)-2-cyclopropyl-4-(3-furyl)pyrimidine:

2.1 2-(3-Bromo-2-pyridyl)-1-(3-furyl)ethanone:LHMDS (1.06 mol/L in THF, 300 mL) is added to a solution of 3-bromo-2-methyl-pyridine (50.0 g) in dry THF (500 mL) maintained at 0 °C, followed by the dropwise addition of ethyl furan-3-carboxylate (45.0 g) in THF. The reaction mixture is warmed to ambient temperature and stirred for 16 h. Citric acid (15% m/m) is added and the mixture is extracted with EtOAc (3x). The combined organics are dried over Na2SO 4 , solid parts are removed by filtration and the remaining solution is concentrated under reduced pressure. The resulting crude product (87.0 g) is used directly in the next step. MS (ESI) m/z 265.9 [M + H + ].

2.2 2-(3-Bromo-2-pyridyl)-3-(dimethylamino)-1-(3-furyl)prop-2-en -1-one:The resulting crude product (87.0 g, see above) containing 2-(3-bromo-2-pyridyl)-1-(3-furyl)ethanone is stirred in N,N- DMF dimethyl acetal (550 mL) for 3 h at 75 °C. Volatiles are removed under reduced pressure. Purification by column chromatography (gradient from EtOAc to EtOAc/MeOH = 4/1) yields the desired product (29.0 g, 28%). MS (ESI) m/z 322.9 [M + H + ].

2.3 5-(3-Bromo-2-pyridyl)-2-cyclopropyl-4-(3-furyl)pyrimidine:

To a solution of 2-(3-bromo-2-pyridyl)-3-(dimethylamino)-1-(3-furyl)prop-2-en -1-one (29.0 g) in EtOH (500 mL) was added cyclopropanecarboxamidine hydrochloride (10.9 g) and NaOEt (20%, 30.7 g). The mixture is refluxed for 4 h, cooled to ambient temperature and filtered. Volatiles are removed under reduced pressure and the crude product is purified by column chromatography (cyclohexane/EtOAc) to yield the title compound (21.2 g, 69 %) as a yellow oil. H NMR (400 MHz, CDCI 3 ): δ 8.70 (dd, J = 4.7, 1.5 Hz, 1 H), 8.46 (s, 1 H), 8.01 (dd, J = 8.1 , 1.5 Hz, 1 H), 7.31 - 7.28 (m, 2H), 7.23 (dd, J = 1 .6, 0.8 Hz, 1 H), 6.37 (dd, J = 1 .9, 0.8 Hz, 1 H), 2.38 - 2.31 (m, 1 H), 1.27 - 1 .23 (m, 2H), 1 .14 - 1.10 (m, 2H) ppm; MS (ESI) m/z 343.9 [M + H + ].

With appropriate modification of the starting materials, the procedures given in the synthesis examples below were used to obtain further compounds of formula I. The compounds obtained in this manner are listed in the table that follows, together with physical data.

The products shown below were characterized by melting point determination, by the masses ([m/z]) or retention time (RT; [min.]) determined by HPLC-MS or HPLC spectrometry.

HPLC-MS = high performance liquid chromatography-coupled mass spectrometry; HPLC methods:

Method: Column: Phenomenex Kinetex 1 .7 μιη XB-C18 100A; 50 x 2.1 mm; mobile phase: A: water + 0.1 % trifluoroacetic acid (TFA); B: acetonitrile + 0.1 % TFA; gradient: 5-100% B in 1 .50 minutes; 100% B 0.25 min; flow: 0.8-1.Oml/min in 1.51 minutes at 60°C.MS: quadrupole electrospray ionization, 80 V (positive mode).

Table 1 : # denotes point of attachment to the pyrimidine ring.

B Use examples

The herbicidal activity of the pyrimidine compounds of formula (I) was demonstrated by the following greenhouse experiments:

The culture containers used were plastic flowerpots containing loamy sand with approximately 3.0% of humus as the substrate. The seeds of the test plants were sown separately for each species.

For the pre-emergence treatment, the active ingredients, which had been suspended or emulsified in water, were applied directly after sowing by means of finely distributing nozzles. The containers were irrigated gently to promote germination and growth and subsequently covered with transparent plastic hoods until the plants had rooted. This cover caused uniform germination of the test plants, unless this had been impaired by the active ingredients.

For the post-emergence treatment, the test plants were first grown to a height of 3 to 15 cm, depending on the plant habit, and only then treated with the active ingredients which had been suspended or emulsified in water. For this purpose, the test plants were either sown directly and grown in the same containers, or they were first grown separately as seedlings and transplanted into the test containers a few days prior to treatment.

Depending on the species, the plants were kept at 10 - 25°C or 20 - 35°C, respectively.

The test period extended over 2 to 4 weeks. During this time, the plants were tended, and their response to the individual treatments was evaluated.

Evaluation was carried out using a scale from 0 to 100. 100 means no emergence of the plants, or complete destruction of at least the aerial moieties, and 0 means no damage, or normal course of growth. A good herbicidal activity is given at values of at least 70 and a very good herbicidal activity is given at values of at least 85.

The plants used in the greenhouse experiments were of the following species:

At an application rate of 1000 g/ha, Ex.6 applied by the post-emergence method showed very good herbicidal activity against SETVI.

At an application rate of 2000 g/ha, Ex.8 applied by the pre-emergence method showed very good herbicidal activity against APESV.

At an application rate of 2000 g/ha, Ex.9 applied by the post-emergence method showed good herbicidal activity against ECHCG.

At an application rate of 2000 g/ha, Ex.10 applied by the post-emergence method showed good herbicidal activity against ALOMY.

At an application rate of 1000 g/ha, Ex.11 applied by the post-emergence method showed good herbicidal activity against ECHCG.

At an application rate of 2000 g/ha, Ex.12 applied by the post-emergence method showed good herbicidal activity against AVEFA, ECHCG and ALOMY, and applied by the pre- emergence method showed very good herbicidal activity against APESV.

At an application rate of 2000 g/ha, Ex.13 applied by the post-emergence method showed good herbicidal activity against ECHCG and SETVI. At an application rate of 2000 g/ha, Ex.17 applied by the post-emergence method showed very good herbicidal activity against AVEFA, and applied by the pre-emergence method showed very good herbicidal activity against APESV and ECHCG.

At an application rate of 2000 g/ha, Ex.18 applied by the post-emergence method showed very good herbicidal activity against AFEVA, good herbicidal activity against and ECHCG.

At an application rate of 2000 g/ha, Ex.01 applied by the post-emergence method showed very good herbicidal activity against MATIN and AMARE.

At an application rate of 2000 g/ha, Ex. 14 applied by the post-emergence method showed very good herbicidal activity against SETVI.

At an application rate of 500 g/ha, Ex.15 applied by the pre-emergence method showed good herbicidal activity against ECHCG.

At an application rate of 2000 g/ha, Ex.20 applied by the post-emergence method showed very good herbicidal activity against AVEFA, ECHCG and ALOMY, and applied by the pre- emergence method showed very good herbicidal activity against ECHCG.

At an application rate of 2000 g/ha, Ex.21 applied by the post-emergence method showed very good herbicidal activity against ECHCG, and good herbicidal activity against AMARE, and applied by the pre-emergence method showed good herbicidal activity against APESV.

At an application rate of 2000 g/ha, Ex.22 applied by the post-emergence method showed very good herbicidal activity against AMARE.

At an application rate of 2000 g/ha, Ex.23 applied by the post-emergence method showed very good herbicidal activity against SETVI, ALOMY and AMARE.

At an application rate of 2000 g/ha, Ex.24 applied by the post-emergence method showed very good herbicidal activity against ALOMY, and good herbicidal activity against AVEFA and SETVI, and applied by the pre-emergence method showed very good herbicidal activity against APESV and ECHCG.

At an application rate of 2000 g/ha, Ex.25 applied by the post-emergence method showed very good herbicidal activity against ALOMY, SETVI and ECHCG, and applied by the pre-emergence method showed very good herbicidal activity against APESV and ECHCG.

At an application rate of 2000 g/ha, Ex.26 applied by the post-emergence method showed very good herbicidal activity against SETVI.

At an application rate of 2000 g/ha, Ex.27 applied by the post-emergence method showed very good herbicidal activity against ALOMY, AVEFA and ECHCG, and applied by the pre- emergence method showed very good herbicidal activity against APESV and ECHCG.

At an application rate of 2000 g/ha, Ex.28 applied by the post-emergence method showed very good herbicidal activity against ALOMY and ECHCG, and good herbicidal activity against

AVEFA, and applied by the pre-emergence method showed very good herbicidal activity against APESV and ECHCG.

At an application rate of 2000 g/ha, Ex.29 applied by the post-emergence method showed very good herbicidal activity against SETVI, and good herbicidal activity against ABUTH, and applied by the pre-emergence method showed very good herbicidal activity against APESV and

ECHCG.

At an application rate of 2000 g/ha, Ex.30 applied by the post-emergence method showed very good herbicidal activity against ALOMY, and good herbicidal activity against ECHCG, and applied by the pre-emergence method showed very good herbicidal activity against APESV and ECHCG.

At an application rate of 2000 g/ha, Ex.31 applied by the post-emergence method showed very good herbicidal activity against ALOMY, SETVI and ECHCG, and applied by the pre-emergence method showed very good herbicidal activity against APESV and ECHCG.

At an application rate of 2000 g/ha, Ex.32 applied by the post-emergence method showed very good herbicidal activity against ALOMY and AMARE, and good herbicidal activity against AVEFA, and applied by the pre-emergence method showed very good herbicidal activity against APESV.

At an application rate of 2000 g/ha, Ex.33 applied by the post-emergence method showed very good herbicidal activity against AMARE, and good herbicidal activity against ECHCG.

At an application rate of 2000 g/ha, Ex.34 applied by the post-emergence method showed very good herbicidal activity against ALOMY and AMARE, and good herbicidal activity against AVEFA, and applied by the pre-emergence method showed very good herbicidal activity against APESV and ECHCG.

At an application rate of 2000 g/ha, Ex.35 applied by the post-emergence method showed very good herbicidal activity against ALOMY and SETVI, and good herbicidal activity against AVEFA, and applied by the pre-emergence method showed very good herbicidal activity against APESV and ECHCG.

At an application rate of 2000 g/ha, Ex.36 applied by the post-emergence method showed very good herbicidal activity against ALOMY, ECHCG and SETVI.

At an application rate of 2000 g/ha, Ex.37 applied by the post-emergence method showed very good herbicidal activity against ABUTH, AMARE and SETVI.

At an application rate of 2000 g/ha, Ex.38 applied by the post-emergence method showed very good herbicidal activity against ECHCG, and applied by the pre-emergence method showed very good herbicidal activity against and ECHCG.

At an application rate of 2000 g/ha, Ex.39 applied by the post-emergence method showed good herbicidal activity against ALOMY, and very good herbicidal activity against ECHCG, and applied by the pre-emergence method showed very good herbicidal activity against APESV and ECHCG.

At an application rate of 2000 g/ha, Ex.41 applied by the post-emergence method showed good herbicidal activity against ECHCG, and applied by the pre-emergence method showed very good herbicidal activity against APESV and ECHCG.

At an application rate of 2000 g/ha, Ex.42 applied by the post-emergence method showed good herbicidal activity against ECHCG.

At an application rate of 2000 g/ha, Ex.44 applied by the post-emergence method showed very good herbicidal activity against ALOMY and good herbicidal activity against AMARE, and applied by the pre-emergence method showed very good herbicidal activity against APESV and ECHCG.

At an application rate of 2000 g/ha, Ex.45 applied by the post-emergence method showed good herbicidal activity against ALOMY, and applied by the pre-emergence method showed very good herbicidal activity against ECHCG and good herbicidal activity against APESV. At an application rate of 2000 g/ha, Ex.46 applied by the post-emergence method showed very good herbicidal activity against AVEFA, SETVI and ECHCG, and applied by the pre-emergence method showed very good herbicidal activity against APESV and ECHCG.