Title:
METHOD FOR PRODUCING HETEROCYCLIDENE ACETAMIDE DERIVATIVES
Document Type and Number:
WIPO Patent Application WO/2021/039023
Kind Code:
A1
Abstract:
The present invention provides, inter alia, a novel method for producing a compound represented by formula (I) and a novel method for producing a compound represented by formula (B) or a salt thereof, which are intermediates in the production of formula (I).
Inventors:
UCHIDA HIDEHARU (JP)
SATOH TSUTOMU (JP)
SUN BAOQUAN (CN)
SHA CHUNBO (CN)
LIN JINGUANG (CN)
GE YONGHUI (CN)
CHEN YANLIANG (CN)
ZHAO BIN (CN)
GU XIAOMIN (CN)
LUO JIAN (CN)
CHEN CHUAN (CN)
CAI XIAOFEI (CN)
YE JIAJIE (CN)
LI JIE (CN)
SUN FENGLAI (CN)
SATOH TSUTOMU (JP)
SUN BAOQUAN (CN)
SHA CHUNBO (CN)
LIN JINGUANG (CN)
GE YONGHUI (CN)
CHEN YANLIANG (CN)
ZHAO BIN (CN)
GU XIAOMIN (CN)
LUO JIAN (CN)
CHEN CHUAN (CN)
CAI XIAOFEI (CN)
YE JIAJIE (CN)
LI JIE (CN)
SUN FENGLAI (CN)
Application Number:
PCT/JP2020/022827
Publication Date:
March 04, 2021
Filing Date:
June 10, 2020
Export Citation:
Assignee:
MOCHIDA PHARM CO LTD (JP)
International Classes:
C07B53/00; C07C29/143; C07C35/52; C07C209/10; C07C215/70; C07D311/58; C12P7/02; C07B61/00
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"Experimental Chemistry Course", vol. 22, 1992, pages: 193 - 309
"The Fourth Series of Experimental Chemistry Lecture 26: Organic Synthesis 8", 30 November 1991, CHEMICAL SOCIETY OF JAPAN, Japan, ISBN: 4-621-03702-1, article "Passage", pages: 33, XP009533910
CAS , no. 1823929-47-0
ADVANCED SYNTHESIS & CATALYSIS, vol. 350, 2008, pages 2322 - 2328
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 18, no. 6, 2008, pages l830 - 1834
JOURNAL OF MEDICINAL CHEMISTRY, vol. 36, no. 17, 1993, pages 2485 - 93
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 28, no. 9, 1993, pages 693 - 701
ANGEW. CHEM. INT. ED., vol. 41, 2002, pages l020
J. AM. CHEM. SOC., vol. 129, no. 34, 2007, pages 10354 - 10355
J. AM. CHEM. SOC., vol. 110, 1988, pages 629
J. AM. CHEM. SOC., vol. 109, 1987, pages 5551
FLOW CHEMISTRY, 13 February 2012 (2012-02-13), pages 213 - 439
J. AM. CHEM. SOC., vol. 128, no. 31, 2006, pages l0028 - 10029
CHEM. COMMUN., vol. 26, 2008, pages 3052 - 3054
J. ORG. CHEM., vol. 74, no. 12, 2009, pages 4542 - 4546
ANGEW. CHEM. INT. ED., vol. 48, no. 2, 2009, pages 337 - 339
UKRAINSKII KHIMICHE SKII ZHURNAL, vol. 53, no. 12, 1987, pages 1299 - 302
"Experimental Chemistry Course", vol. 22, 1992, pages: 193 - 309
Attorney, Agent or Firm:
KOBAYASHI Hiroshi et al. (JP)
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