Title:
NOVEL ERYTHROMYCIN DERIVATIVES
Document Type and Number:
WIPO Patent Application WO1999035157
Kind Code:
B1
Abstract:
The invention relates to novel erythromycin derivatives, particularly ones with novel C-13 R<13> substituents, and to pharmaceutically acceptable salts thereof. The compounds of this invention are useful as antibacterial agents and antiprotozoa agents and for other applications (e.g., anticancer, atherosclerosis, gastric motility reduction, etc.) in mammals, including man, as well as in fish and birds. The invention also relates to pharmaceutical compositions containing such compounds and to methods of treating bacterial protozoa infections by administering such compounds. The invention also relates to methods of preparing such compounds and to intermediates useful in such preparation.
Inventors:
WU YONG-JIN (US)
Application Number:
PCT/IB1998/002100
Publication Date:
October 14, 1999
Filing Date:
December 21, 1998
Export Citation:
Assignee:
PFIZER PROD INC (US)
WU YONG JIN (US)
WU YONG JIN (US)
International Classes:
A61K31/7042; A61K31/7048; A61P31/04; A61P33/02; C07H17/08; (IPC1-7): C07H17/08; A61K31/70
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