NOVEL METHOD FOR PRODUCING 1-(ACYLOXY)ALKYL CARBAMATE DERIVATIVE

Title:

NOVEL METHOD FOR PRODUCING 1-(ACYLOXY)ALKYL CARBAMATE DERIVATIVE

Document Type and Number:

WIPO Patent Application WO/2016/208709

Kind Code:

A1

Abstract:

A method for producing a 1-(acyloxy)alkyl carbamate derivative (III) using a fluorous alkyl carbonate derivative (I), and a fluorous alkyl carbonate derivative (I) and a method for producing the same. In the formulae: R1 represents a C1-C4 alkyl group or a C3-C6 cycloalkyl group; R2 represents a C1-C4 alkyl group or a hydrogen atom; and A represents a fluorous alkyl group (wherein a fluorous alkyl group means a C2-C11 alkyl group in which 40% or more hydrogen atoms are substituted by fluorine atoms).

More Like This:

JP3322878	[Title of Invention] Fibrinogen Receptor Antagonist
JP5397461	Compounds with S1P receptor binding ability and their uses
WO/2001/051487	NON-PEPTIDYL INHIBITORS OF VLA-4 DEPENDENT CELL BINDING USEFUL IN TREATING INFLAMMATORY, AUTOIMMUNE, AND RESPIRATORY DISEASES

Inventors:

UEDA TSUYOSHI (JP)
ABE YUZO (JP)

Application Number:

PCT/JP2016/068796

Publication Date:

December 29, 2016

Filing Date:

June 24, 2016

Export Citation:

Click for automatic bibliography generation Help

Assignee:

DAIICHI SANKYO CO LTD (JP)

International Classes:

C07D233/64; C07C68/06; C07C69/96; C12P41/00; C07B61/00

Domestic Patent References:

WO2011115064A1

2011-09-22

Foreign References:

US20140243544A1

2014-08-28

Other References:

NORIAKI HIRAYAMA: "Yuki Kagobutsu Kessho Sakusei Handbook", 25 July 2008 (2008-07-25), pages 57 - 84, XP008183996
KAZUHIDE ASHIZAWA: "Shio Kesshokei no Saitekika to Kesshoka Gijutsu", PHARM TECH JAPAN, vol. 18, no. 10, 2002, pages A1 - 96, XP008177312
LUO, Z. ET AL.: "Fluorous Boc (FBoc) Carbamates: New Amine Protecting Groups for Use in Fluorous Synthesis", JOURNAL OF ORGANIC CHEMISTRY, vol. 66, no. 12, 2001, pages 4261 - 4266, XP001061425
See also references of EP 3323808A4

Attorney, Agent or Firm:

ISHIBASHI, Koki et al. (JP)
Kimiki Ishibashi (JP)

Download PDF:

View/Download PDF PDF Help

Previous Patent: MEDIUM CONTAINING IDENTIFIER

Next Patent: LANE DEPARTURE AVOIDANCE SYSTEM