Title:
OXADIAZOLE DERIVATIVE
Document Type and Number:
WIPO Patent Application WO/2021/187486
Kind Code:
A1
Abstract:
The present invention relates to the compound represented in formula (1) or a pharmaceutically acceptable salt thereof (in the formula, Q1 represents a halogen, Q2 represents a hydrogen, etc., X, Y and Z represent a nitrogen atom or an oxygen atom, and R1 represents a prescribed structure), and the present invention further relates to a therapeutic and/or prophylactic agent for disease such as epilepsy that contains these.
Inventors:
ISOBE YOSHIAKI (JP)
TANAKA TOMOYUKI (JP)
MIYACHI HIROTAKA (JP)
TANAKA TOMOYUKI (JP)
MIYACHI HIROTAKA (JP)
Application Number:
PCT/JP2021/010628
Publication Date:
September 23, 2021
Filing Date:
March 16, 2021
Export Citation:
Assignee:
SUMITOMO DAINIPPON PHARMA CO LTD (JP)
International Classes:
C07D271/06; A61K31/4245; A61K45/00; A61P21/02; A61P25/00; A61P25/04; A61P25/08; A61P25/16; A61P25/18; A61P25/22; A61P25/24; A61P25/28; A61P43/00; C07D413/04
Domestic Patent References:
| WO2015161014A1 | 2015-10-22 | |||
| WO2013062027A1 | 2013-05-02 | |||
| WO2010017132A1 | 2010-02-11 | |||
| WO2014072957A1 | 2014-05-15 | |||
| WO2006138512A2 | 2006-12-28 |
Foreign References:
| JP2014525444A | 2014-09-29 | |||
| JP2014224108A | 2014-12-04 | |||
| JP2018507886A | 2018-03-22 |
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ROBERT S. FISHER ET AL., EPILEPSIA, vol. 58, no. 4, 2017, pages 522 - 530
ANNE T. BERG ET AL., EPILEPSIA, vol. 51, no. 4, 2010, pages 676 - 85
SCHMITZ B., EPILEPSIA, 2005, pages 45 - 49
R. C. LAROCK: "Comprehensive Organic Transformations", 1999, JOHN WILEY SONS INC.
JAPAN EPILEPSY RESEARCH FOUNDATION, vol. 26, 2015, pages 69 - 76
Attorney, Agent or Firm:
YAMAO, Norihito et al. (JP)
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