Title:
PHARMACEUTICAL DRUG CONTAINING HETEROCYCLIDENE ACETAMIDE DERIVATIVE
Document Type and Number:
WIPO Patent Application WO/2021/066144
Kind Code:
A1
Abstract:
This disclosure provides a means for treating dry eye. This disclosure can provide: a composition for treating dry eye; and a use thereof. The composition includes (E) -2-(7-trifluoromethyl-chroman-4-yllidene)-N-(7-hydroxy-5,6,7,8-tetrahydronaphthalene-1-yl)acetamide, a pharmaceutically acceptable salt thereof, or a solvate thereof. This disclosure can provide: a composition for treating dry eye; and a use thereof. The composition includes a Vi/Vc zone inhibitor.
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Inventors:
TARUI TAKESHI (JP)
KOBAYASHI SHINYA (JP)
KOBAYASHI SHINYA (JP)
Application Number:
PCT/JP2020/037548
Publication Date:
April 08, 2021
Filing Date:
October 02, 2020
Export Citation:
Assignee:
SENJU PHARMA CO (JP)
MOCHIDA PHARM CO LTD (JP)
MOCHIDA PHARM CO LTD (JP)
International Classes:
A61K31/353; A61K9/10; A61P27/04; A61P43/00
Domestic Patent References:
WO2007010383A1 | 2007-01-25 | |||
WO2018221543A1 | 2018-12-06 | |||
WO2007010383A1 | 2007-01-25 | |||
WO2018221543A1 | 2018-12-06 |
Foreign References:
US20090131449A1 | 2009-05-21 | |||
JP4754566B2 | 2011-08-24 | |||
JPS6230743B2 | 1987-07-03 | |||
JP2019184053A | 2019-10-24 |
Other References:
"2016 Result Report for Collaborative Research* Result Report for encouragement research of KANAZAWA MEDICAL UNIVERSITY", 30 November 2017, KANAZAWA MEDICAL UNIVERSITY, JP, article MASUOKA, TAKAYOSHI: "Role of neurotrophic factors in corneal dysesthesia in dry eye", pages: 35 - 37, XP009536140
BELMONTE CARLOS,: "TFOS DEWS II pain and sensation report", THE OCULAR SURFACE, vol. 15, no. 3, 2017, pages 404 - 437, XP055811111
FARUMASHIA, vol. 50, no. 3, 2014, pages 201 - 206
THE JOURNAL OF JAPANESE BIOCHEMICAL SOCIETY, vol. 85, no. 7, pages 561 - 565
"Understand from reading! Change from understanding! Dry eye diagnosis and treatment", 1 October 2017, MEDICAL VIEW CO., LTD., pages: 46 - 58
"Qualification for ophthalmic diagnosis and treatment for specialists 19 Road to dry eye specialist", 5 November 2013, NAKAYAMA SHOTEN CO., LTD, pages: 103 - 106
REVISED DEFINITION AND DIAGNOSTIC CRITERIA OF DRY EYE, 2016
THE JOURNAL OF NEUROSCIENCE, vol. 24, no. 17, 28 April 2004 (2004-04-28), pages 4224 - 4232
NEUROSCIENCE, vol. 290, 2015, pages 204 - 213
J NEUROPHYSIOL, vol. 77, no. 1, January 1997 (1997-01-01), pages 43 - 56
HEADACHE, vol. 52, no. 2, February 2012 (2012-02-01), pages 262 - 273
SNINSKY, J. J. ET AL.: "Short Protocols in Molecular Biology: A Compendium of Methods from Current Protocols in Molecular Biology", 1999, GREENE PUB. ASSOCIATES AND WILEY-INTERSCIENCE
AUSUBEL, F.M.: "Current Protocols in Molecular Biology", 1987, GREENE PUB. ASSOCIATES AND WILEY-INTERSCIENCE
INNIS, M. A.: "PCR Protocols: A Guide to Methods and Applications", 1990, ACADEMIC PRESS
GAIT, M. J.: "Oligonucleotide Synthesis: A Practical Approach", 1985, IRL PRESS
ECKSTEIN, F.: "Oligonucleotides and Analogues: A Practical Approach", 1991, IRL PRESS
ADAMS, R. L. ET AL.: "The Biochemistry of the Nucleic Acids", 1992, CHAPMAN & HALL
SHABAROVA, Z. ET AL.: "Advanced Organic Chemistry of Nucleic Acids", 1994, WEINHEIM
BLACKBURN, G. M. ET AL.: "Nucleic Acids in Chemistry and Biology", 1996, OXFORD UNIVERSITY PRESS
EXPERIMENTAL MEDICINE
YODOSHA, EXPERIMENTAL METHODS FOR TRANSGENESIS & EXPRESSION ANALYSIS, 1997
BELMONTE CARLOS,: "TFOS DEWS II pain and sensation report", THE OCULAR SURFACE, vol. 15, no. 3, 2017, pages 404 - 437, XP055811111
FARUMASHIA, vol. 50, no. 3, 2014, pages 201 - 206
THE JOURNAL OF JAPANESE BIOCHEMICAL SOCIETY, vol. 85, no. 7, pages 561 - 565
"Understand from reading! Change from understanding! Dry eye diagnosis and treatment", 1 October 2017, MEDICAL VIEW CO., LTD., pages: 46 - 58
"Qualification for ophthalmic diagnosis and treatment for specialists 19 Road to dry eye specialist", 5 November 2013, NAKAYAMA SHOTEN CO., LTD, pages: 103 - 106
REVISED DEFINITION AND DIAGNOSTIC CRITERIA OF DRY EYE, 2016
THE JOURNAL OF NEUROSCIENCE, vol. 24, no. 17, 28 April 2004 (2004-04-28), pages 4224 - 4232
NEUROSCIENCE, vol. 290, 2015, pages 204 - 213
J NEUROPHYSIOL, vol. 77, no. 1, January 1997 (1997-01-01), pages 43 - 56
HEADACHE, vol. 52, no. 2, February 2012 (2012-02-01), pages 262 - 273
SNINSKY, J. J. ET AL.: "Short Protocols in Molecular Biology: A Compendium of Methods from Current Protocols in Molecular Biology", 1999, GREENE PUB. ASSOCIATES AND WILEY-INTERSCIENCE
AUSUBEL, F.M.: "Current Protocols in Molecular Biology", 1987, GREENE PUB. ASSOCIATES AND WILEY-INTERSCIENCE
INNIS, M. A.: "PCR Protocols: A Guide to Methods and Applications", 1990, ACADEMIC PRESS
GAIT, M. J.: "Oligonucleotide Synthesis: A Practical Approach", 1985, IRL PRESS
ECKSTEIN, F.: "Oligonucleotides and Analogues: A Practical Approach", 1991, IRL PRESS
ADAMS, R. L. ET AL.: "The Biochemistry of the Nucleic Acids", 1992, CHAPMAN & HALL
SHABAROVA, Z. ET AL.: "Advanced Organic Chemistry of Nucleic Acids", 1994, WEINHEIM
BLACKBURN, G. M. ET AL.: "Nucleic Acids in Chemistry and Biology", 1996, OXFORD UNIVERSITY PRESS
EXPERIMENTAL MEDICINE
YODOSHA, EXPERIMENTAL METHODS FOR TRANSGENESIS & EXPRESSION ANALYSIS, 1997
Attorney, Agent or Firm:
YAMAMOTO, Shusaku et al. (JP)
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