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Title:
SIMPLIFIED RESINIFERATOXIN ANALOGUES AS VANILLOID RECEPTOR AGONIST SHOWING EXCELLENT ANALGESIC ACTIVITY AND THE PHARMACEUTICAL CO MPOSITIONS CONTAINING THE SAME
Document Type and Number:
WIPO Patent Application WO2003027064
Kind Code:
B1
Abstract:
The present invention is related to new vanilloid analogues containing resiniferatoxin pharmacophores, pharmaceutical compositions comprising such analogues, and their uses as vanilloid receptor agonistsand potent analgesics.The present invention provides a pharmaceutical composition for preventing, alleviating or treating pain, acute pain, chronic pain, neuropathic pain, post-operative pain, migraine, arthralgia, neutopathies, nerve injury, diabetic neuropathy, neurodegeneration, neurotic skin disorder, stroke, urinary bladder hypersensitiveness, irritable bowel syndrome, a respiratory disorder such as asthma or chronic obstructive pulmonary disease, irritation of skin, eye or mucous membrane, fervescence, stomach-duodenal ulcer, inflammatory bowel disease, inflammatory disease or urgent urinary incontinence.

Inventors:
LEE JEE-WOO (KR)
Application Number:
PCT/KR2002/001746
Publication Date:
April 08, 2004
Filing Date:
September 18, 2002
Export Citation:
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Assignee:
DIGITAL BIOTECH CO LTD (KR)
LEE JEE-WOO (KR)
International Classes:
C07C235/34; C07C275/24; C07C333/04; C07C335/18; (IPC1-7): C07C335/18
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