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Title:
SIX-MEMBERED ARYL OR HETEROARYL AMIDES, AND COMPOSITION AND USE THEREOF
Document Type and Number:
WIPO Patent Application WO/2023/279986
Kind Code:
A1
Abstract:
A compound of formula I and a use thereof as an MALT1 inhibitor, and a pharmaceutical composition containing the compound. The compound can be used to treat diseases or disorders such as cancer.

Inventors:
FU BANG (CN)
LI YINLONG (CN)
REN WEI (CN)
SHEN QICHAO (CN)
DU GUOLONG (CN)
ZHOU XIAOJUN (CN)
SUN YUN (CN)
ZHOU YUZHEN (CN)
SUN XIAO (CN)
CAI WEIDONG (CN)
LIU XIANGYONG (CN)
DING LIEMING (CN)
WANG JIABING (CN)
Application Number:
PCT/CN2022/101146
Publication Date:
January 12, 2023
Filing Date:
June 24, 2022
Export Citation:
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Assignee:
BETTA PHARMACEUTICALS CO LTD (CN)
International Classes:
C07D401/04; A61K31/165; A61K31/4192; A61P35/00; C07D401/12; C07D401/14; C07D403/12; C07D409/14; C07D413/14
Domestic Patent References:
WO2021138298A12021-07-08
Foreign References:
CN111171020A2020-05-19
CN110214136A2019-09-06
CN1805923A2006-07-19
Other References:
DATABASE REGISTRY 23 June 2022 (2022-06-23), ANONYMOUS: "/1 -(C) FILE REGISTRY RN -2776345-09-4 REGISTRY ED -Entered STN: 23 Jun 2022 CN -Benzamide, 4-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)-N-[4-(2H-1,2,3- triazol-2-yl)phenyl]-(CA INDEX NAME)", XP093021706, retrieved from STN Database accession no. 2776345-09-4
DATABASE REGISTRY 23 April 2021 (2021-04-23), ANONYMOUS: "/1 -(C) FILE REGISTRY RN -2637183-50-5 REGISTRY ED -Entered STN: 23 Apr 2021 CN -Benzamide, 4-(4-pyridinyl)-N-[3-(2H-1,2,3-triazol-2-yl)phenyl]- (CA INDEX NAME)", XP093021720, retrieved from STN Database accession no. 2637183-50-5
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