Title:
VASOPRESSIN V1A ANTAGONISTS
Document Type and Number:
WIPO Patent Application WO2006021213
Kind Code:
A3
Abstract:
The present invention concerns compounds inter alia according to general formula: (1a). Compounds according to the invention are vasopressin V1a receptor antagonists. Pharmaceutical compositions of the compounds are useful as treatment of dysmenorrhoea.
Inventors:
ANDRZEJ ROMAN BATT (GB)
BAXTER ANDREW JOHN (GB)
HEENEY CELINE (GB)
STOCKLEY MARTIN LEE (GB)
BRYAN ROE MICHAEL (GB)
HUDSON PETER (DK)
HANDY RACHEL (GB)
BAXTER ANDREW JOHN (GB)
HEENEY CELINE (GB)
STOCKLEY MARTIN LEE (GB)
BRYAN ROE MICHAEL (GB)
HUDSON PETER (DK)
HANDY RACHEL (GB)
Application Number:
PCT/DK2005/000540
Publication Date:
August 17, 2006
Filing Date:
August 24, 2005
Export Citation:
Assignee:
FERRING BV (NL)
ANDRZEJ ROMAN BATT (GB)
BAXTER ANDREW JOHN (GB)
HEENEY CELINE (GB)
STOCKLEY MARTIN LEE (GB)
BRYAN ROE MICHAEL (GB)
HUDSON PETER (DK)
HANDY RACHEL (GB)
ANDRZEJ ROMAN BATT (GB)
BAXTER ANDREW JOHN (GB)
HEENEY CELINE (GB)
STOCKLEY MARTIN LEE (GB)
BRYAN ROE MICHAEL (GB)
HUDSON PETER (DK)
HANDY RACHEL (GB)
International Classes:
C07D487/04; A61K31/38; A61K31/495; A61K31/55; A61K31/5517; A61K31/553; C07D215/08; C07D223/16; C07D231/38; C07D231/42; C07D265/36; C07D267/14; C07D267/16; C07D333/44; C07D417/10; C07D498/14; C07D513/14
Domestic Patent References:
WO2002000626A1 | 2002-01-03 | |||
WO2001029005A1 | 2001-04-26 | |||
WO2002004403A1 | 2002-01-17 | |||
WO1995034540A1 | 1995-12-21 | |||
WO2004037788A1 | 2004-05-06 | |||
WO2003016316A1 | 2003-02-27 |
Foreign References:
US5760031A | 1998-06-02 | |||
EP0620216A1 | 1994-10-19 | |||
EP1449844A1 | 2004-08-25 | |||
US6583141B1 | 2003-06-24 | |||
US3987108A | 1976-10-19 | |||
EP0186817A1 | 1986-07-09 | |||
US5968930A | 1999-10-19 | |||
US5843952A | 1998-12-01 |
Other References:
POCIECHA D ET AL: "NEW MESOGENIC COMPOUNDS HAVING FORK-LIKE OR CYCLIC AMIDE TERMINAL GROUPS", LIQUID CRYSTALS, TAYLOR AND FRANCIS, ABINGDON, GB, vol. 29, no. 5, May 2002 (2002-05-01), pages 663 - 667, XP001102373, ISSN: 0267-8292
DATABASE BEILSTEIN BEILSTEIN INSTITUTE FOR ORGANIC CHEMISTRY, FRANKFURT-MAIN, DE; XP002357863, Database accession no. BRN: 2173418
DATABASE BEILSTEIN BEILSTEIN INSTITUTE FOR ORGANIC CHEMISTRY, FRANKFURT-MAIN, DE; XP002383169, Database accession no. BRN:2886892
DATABASE BEILSTEIN BEILSTEIN INSTITUTE FOR ORGANIC CHEMISTRY, FRANKFURT-MAIN, DE; XP002383170, Database accession no. BRN:2131233
DATABASE BEILSTEIN BEILSTEIN INSTITUTE FOR ORGANIC CHEMISTRY, FRANKFURT-MAIN, DE; XP002357863, Database accession no. BRN: 2173418
DATABASE BEILSTEIN BEILSTEIN INSTITUTE FOR ORGANIC CHEMISTRY, FRANKFURT-MAIN, DE; XP002383169, Database accession no. BRN:2886892
DATABASE BEILSTEIN BEILSTEIN INSTITUTE FOR ORGANIC CHEMISTRY, FRANKFURT-MAIN, DE; XP002383170, Database accession no. BRN:2131233
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