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Title:
因子XAの阻害剤としてのピロリジン-2-オン誘導体
Document Type and Number:
Japanese Patent JP2005508868
Kind Code:
A
Abstract:
The invention relates to compounds of formula (Ic) processes for their preparation, pharmaceutical compositions containing them and to their use in medicine, particularly use in the amelioration of a clinical condition for which a Factor Xa inhibitor is indicated.

Inventors:
Chuen Chang
Julie Nicole Hamblin
Henry Anderson Kelly
Nigel Paul King
Andrew McMurtry Mason
Bipurkumar Canti by Patel
Stefan Senger
Jita Punjabai Shah
Nigel Stephen Watson
Helen Elizabeth Weston
Caroline Whitworth
Robert John Young
Application Number:
JP2003503652A
Publication Date:
April 07, 2005
Filing Date:
June 06, 2002
Export Citation:
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Assignee:
GLAXO GROUP LIMITED
International Classes:
C07D487/08; A61K31/4025; A61K31/407; A61K31/4365; A61K31/437; A61K31/439; A61K31/454; A61K31/496; A61K31/5377; A61K31/5386; A61K31/541; A61K31/55; A61K38/55; A61P7/02; A61P9/00; A61P9/10; A61P43/00; C07D207/273; C07D401/06; C07D401/12; C07D401/14; C07D403/06; C07D405/12; C07D409/12; C07D413/06; C07D417/14; C07D471/04; C07D471/08; C07D491/08; C07D495/04; C07D498/08; C07K5/06; C07K5/078; A61K38/00; (IPC1-7): A61K38/55; A61K31/4025; A61K31/407; A61K31/4365; A61K31/437; A61K31/439; A61K31/454; A61K31/496; A61K31/5377; A61K31/5386; A61K31/541; A61K31/55; A61P7/02; A61P9/00; A61P9/10; A61P43/00; C07D207/273; C07D401/06; C07D401/12; C07D401/14; C07D403/06; C07D405/12; C07D409/12; C07D413/06; C07D417/14; C07D471/04; C07D471/08; C07D487/08; C07D491/08; C07D495/04; C07D498/08
Attorney, Agent or Firm:
Mitsuo Tanaka
Michiko Matsutani
Tadayuki Motoyama
Kenji Tomita
Mina Shiga