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Patent Searching and Data


Title:
新規なキナゾリン誘導体及びそれらの使用に関連する治療方法
Document Type and Number:
Japanese Patent JP2006522109
Kind Code:
A
Abstract:
The present invention relates to novel compounds of Formula (1): which act as MCH receptor antagonists. These compositions are useful in pharmaceutical compositions whose use includes prophylaxis or treatment of improving memory function, sleeping and arousal, anxiety, depression, mood disorders, seizure, obesity, diabetes, appetite and eating disorders, cardiovascular disease, hypertension, dyslipidemia, myocardial infarction, binge eating disorders including bulimia, anorexia, mental disorders including manic depression, schizophrenia, delirium, dementia, stress, cognitive disorders, attention deficit disorder, substance abuse disorders and dyskinesias including Parkinson's disease, epilepsy, and addiction.

Inventors:
Yoshinori Sekiguchi
Kosuke Kanuma
Katsunori Omotera
Busujima Go
Trang, Thuy-Ann
Han, Sandon
Casper, Martin
Kramer, Brian, A.
Application Number:
JP2006507700A
Publication Date:
September 28, 2006
Filing Date:
March 30, 2004
Export Citation:
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Assignee:
Taisho Pharmaceutical Co., Ltd.
Arena Pharmaceuticals Incorporated
International Classes:
C07D239/95; A61K31/517; A61K31/5377; A61P3/00; A61P3/04; A61P3/06; A61P3/10; A61P9/00; A61P9/10; A61P9/12; A61P25/00; A61P25/08; A61P25/16; A61P25/18; A61P25/20; A61P25/22; A61P25/24; A61P25/28; A61P25/30; C07D401/12; C07D403/12; C07D405/12; C07D409/12; C07D413/12; C07D417/12
Foreign References:
WO1997020820A11997-06-12
WO1997020822A11997-06-12
WO1997020823A21997-06-12
US5874438A1999-02-23
Attorney, Agent or Firm:
Hideto Asamura
Hajime Asamura
Katsunori Ando
Sadafumi Kobori