Title:
アスパルチルプロテアーゼ阻害因子である酸素化複素環含有スルホンアミド類
Document Type and Number:
Japanese Patent JP4240532
Kind Code:
B2
Abstract:
The present invention relates to a novel class of sulfonamides which are aspartyl protease inhibitors. This invention also relates to pharmaceutical compositions comprising these compounds. The compounds and pharmaceutical compositions of this invention are particularly well suited for inhibiting HIV-1 and HIV-2 protease activity and consequently, may be advantageously used as anti-viral agents against the HIV-1 and HIV-2 viruses. This invention also relates to methods for inhibiting the activity of HIV aspartyl protease using the compounds of this invention.
Inventors:
Toon, Roger Di
Bisetti, Govinda Lao
Bisetti, Govinda Lao
Application Number:
JP53195396A
Publication Date:
March 18, 2009
Filing Date:
April 18, 1996
Export Citation:
Assignee:
Vertex Pharmaceuticals, Inc.
International Classes:
C07D319/06; A61K31/335; A61K31/34; A61K31/341; A61K31/357; A61P31/12; A61P31/18; A61P43/00; C07D307/20; C07D309/12; C07D317/24; C07D493/04
Domestic Patent References:
| JP5345775A |
Foreign References:
| WO1994005639A1 | ||||
| WO1995006030A1 |
Attorney, Agent or Firm:
Aoyama Aoi
Shoji Nakajima
Shoji Nakajima
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