チアジアジン誘導体及びポジティブAMPA受容体モジュレーターとしてのそれらの使用

Title:

チアジアジン誘導体及びポジティブAMPA受容体モジュレーターとしてのそれらの使用

Document Type and Number:

Japanese Patent JP4461139

Kind Code:

B2

Abstract:

Compounds of formula (I): wherein: A represents thienyl, furyl, pyrrolyl, oxathiol, thiazole, isothiazole, oxazole or imidazole, custom character

represents a single bond or a double bond, R1 represents hydrogen, linear or branched (C1-C6)alkyl optionally substituted by one or more groups selected from halogen or (C1-C6)alkoxy-(C1-C6)alkyl, R2 represents hydrogen or linear or branched (C1-C6)alkyl group optionally substituted by one or more halogen, R3 represents hydrogen or a group selected from linear or branched (C1-C6)alkyl, CONHR' and SO2NHR' wherein R' represents linear or branched (C1-C6)alkyl, its enantiomers and diastereoisomers, and addition salts thereof with a pharmaceutically acceptable acid or base. Medicinal products containing the same, which are useful as AMPA inhibitors.

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Inventors:

Grande Rouge, Emmanuel
Francotte, Pierre
Bovry, Stephane
De turio, pascal
Pilot, Bernard
Lestage, Pierre
Lawrence Danobel
Renard, Pierre
Canary, Daniel-Henri

Application Number:

JP2006505830A

Publication Date:

May 12, 2010

Filing Date:

May 04, 2004

Export Citation:

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