Title:
3-アルキルピペラジン誘導体及びその使用
Document Type and Number:
Japanese Patent JP2011512340
Kind Code:
A
Abstract:
Compounds of formula I: or pharmaceutically acceptable salts thereof, wherein Ar is indolyl, indazolyl or dihydroindolyl, and R1, R2, R3 and R4 are as defined herein. Also provided are pharmaceutical compositions, methods of using the compounds in the treatment of depressive, anxiolytic and other disorders associated with inhibition of the reuptake of norepinephrine, serotonin, and dopamine, and methods of preparing the compounds.
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Inventors:
Carter, david scott
Lucas, Matthew Sea
Schoenfeld, Ryan Craig
Weikart, Robert James
Lucas, Matthew Sea
Schoenfeld, Ryan Craig
Weikart, Robert James
Application Number:
JP2010546289A
Publication Date:
April 21, 2011
Filing Date:
February 05, 2009
Export Citation:
Assignee:
F. HOFFMANN-LA ROCHE AKTIENGESELLSCHAFT
International Classes:
C07D403/04; A61K31/496; A61K31/499; A61K31/4995; A61P1/14; A61P3/04; A61P3/06; A61P3/10; A61P13/02; A61P13/08; A61P19/02; A61P19/06; A61P25/00; A61P25/02; A61P25/04; A61P25/08; A61P25/14; A61P25/18; A61P25/20; A61P25/22; A61P25/24; A61P25/28; A61P25/30; A61P29/00; A61P29/02; A61P37/02; A61P43/00; C07D401/14; C07D405/14; C07D409/04; C07D487/08
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Attorney, Agent or Firm:
Hajime Tsukuni
Fusayuki Saito
Fusayuki Saito