Title:
ARYL-SUBSTITUTED PYRAZOLE, IMIDAZOLE, OXAZOLE, THIAZOLE, AND PYRROLE, AND USE THEREOF
Document Type and Number:
Japanese Patent JP2011021028
Kind Code:
A
Abstract:
To provide a sodium (Na+) channel blocker.
This invention relates to a compound having the formula (I) or a pharmaceutically acceptable salt thereof, a prodrug, or a solvate thereof, and also relates to the use of the compound of the formula (I) for the treatment of neuronal damage following systemic and local ischemia, for the treatment or prevention of neurodegenerative conditions, and for the treatment, prevention, or amelioration of both acute and chronic pain, as an anti-tinnitus agent, as an anticonvulsant, and an antimanic depressant, as a local anesthetic, as an antiarrhythmic, and for the treatment or prevention of diabetic neuropathy.
Inventors:
HOGENKAMP DERK J
UPASANI RAVINDRA
NGUYEN PHONG
UPASANI RAVINDRA
NGUYEN PHONG
Application Number:
JP2010220062A
Publication Date:
February 03, 2011
Filing Date:
September 29, 2010
Export Citation:
Assignee:
EURO CELTIQUE SA
International Classes:
C07D207/34; A61K31/40; C07D233/64; A61K31/415; A61K31/4164; A61K31/4184; A61K31/421; A61K31/426; A61K31/497; A61K31/506; A61K31/5377; A61P9/06; A61P9/10; A61P21/02; A61P23/02; A61P25/06; A61P25/16; A61P25/22; A61P25/24; A61P25/28; A61P27/06; A61P27/16; A61P29/00; A61P43/00; C07D207/416; C07D231/12; C07D231/18; C07D233/54; C07D235/18; C07D263/34; C07D277/20; C07D277/32; C07D277/56; C07D403/04; A61P25/04; C07D207/40
Attorney, Agent or Firm:
Hidesaku Yamamoto
Takaaki Yasumura
Natsuki Morishita
Takaaki Yasumura
Natsuki Morishita