Title:
BENZENE RING-CONDENSED LACTAM USEFUL AS ANTIHYPERTENSIVE ANDCHOLECYSTOKININ ANTAGONIST
Document Type and Number:
Japanese Patent JPS6115874
Kind Code:
A
Abstract:
Compounds of the formula: wherein R<1> is, e.g., hydrogen or hydrocarbon of from 1 to 12 carbon atoms; R<2> is, e.g., hydroxy; loweralkoxy; amino; loweralkylamino or diloweralkylamino; m is 1-3; R<3> is loweralkyl or substituted loweralkyl wherein the substituents are hydrogen, loweralkyl, or aryl; R<4> is hydroxy; loweralkanoyloxy; arloweralkanoyloxy; R<5> is hydrogen; halo; hydroxy; loweralkyl; or loweralkoxy; and pharmaceutically acceptable salts thereof are inhibitors of angiotensin I converting enzyme and are useful as antihypertensive agents and are also useful as cholecystokinin antagonists.
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Inventors:
UIRIAMU ETSUCHI PAASONZU
Application Number:
JP13708885A
Publication Date:
January 23, 1986
Filing Date:
June 25, 1985
Export Citation:
Assignee:
MERCK & CO INC
International Classes:
A61K31/395; A61K31/47; A61K31/55; A61P1/00; A61P9/12; A61P25/00; A61P43/00; C07D215/38; C07D223/16; C07D225/06; (IPC1-7): A61K31/395; A61K31/47; A61K31/55; C07D215/38; C07D223/16; C07D225/06
Attorney, Agent or Firm:
Masao Okabe
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