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Title:
グルコース感知タンパク質に結合することができる薬剤および部分のコンジュゲート
Document Type and Number:
Japanese Patent JP2019520342
Kind Code:
A
Abstract:
本発明は、グルコース濃度に応じて薬剤の可逆的放出を可能にするグルコース感知タンパク質に結合することができる薬剤および部分の式(I)の新規コンジュゲートを述べる。

Inventors:
Stephan petry
Oliver Plettenburg
Norbert Tenagels
Ulrich Werner
Application Number:
JP2018563040A
Publication Date:
July 18, 2019
Filing Date:
June 02, 2017
Export Citation:
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Assignee:
SANOFI
International Classes:
C07K14/62; A61K47/54; A61P3/10; C07H5/04; C07H7/02; C07H9/04; C07H13/06; C07H13/08; C07H15/04; C07H15/10; C07H19/04; C07H19/056; C07H23/00
Domestic Patent References:
JP2012516342A2012-07-19
Foreign References:
WO2015051052A22015-04-09
Other References:
BIOORGANIC & MEDICINAL CHEMISTRY, vol. 18, JPN6021023673, 2010, pages 2412 - 2427, ISSN: 0004803358
JOURNAL OF LABELLED COMPOUNDS AND RADIOPHARMACEUTICALS, vol. VOL:55, NR:7,, JPN5019004827, 25 May 2012 (2012-05-25), pages 274 - 280, ISSN: 0004803359
BIOCONJUGATE CHEMISTRY, vol. 8, JPN6021023672, 1997, pages 664 - 672, ISSN: 0004803360
JOURNAL OF CONTROLLED RELEASE, vol. 1, JPN6021023671, 1984, pages 57 - 66, ISSN: 0004803361
Attorney, Agent or Firm:
Junji Yuda
Noriyuki Takebayashi