Title:
FATTY ACID AMIDE HYDROLASE INHIBITORS
Document Type and Number:
Japanese Patent JP2016128472
Kind Code:
A
Abstract:
PROBLEM TO BE SOLVED: To provide inhibitors of fatty acid amide hydrolase (FAAH) being endogenous membrane protein contributing to hydrolysis of endogenous neuromodulating fatty acid amides (FAAs).SOLUTION: There is provided a crystalline compound represented by the formula (1) or an anhydrous trimer of a compound represented by the formula (1).SELECTED DRAWING: Figure 1
Inventors:
BRIAN C AUSTAD
LOUIS GRENIER
MICHAEL J GROGAN
LIU TAO
LO CHING KAM
THEODORE A MARTINOT
YU LIN-CHEN
LOUIS GRENIER
MICHAEL J GROGAN
LIU TAO
LO CHING KAM
THEODORE A MARTINOT
YU LIN-CHEN
Application Number:
JP2016012894A
Publication Date:
July 14, 2016
Filing Date:
January 27, 2016
Export Citation:
Assignee:
INFINITY PHARMACEUTICALS INC
International Classes:
A61K31/69; A61P1/02; A61P1/04; A61P1/08; A61P3/00; A61P3/04; A61P9/00; A61P9/10; A61P9/12; A61P13/10; A61P15/00; A61P17/02; A61P17/04; A61P19/02; A61P21/00; A61P25/00; A61P25/08; A61P25/20; A61P25/28; A61P25/36; A61P27/06; A61P29/00; A61P37/02; A61P43/00; C07C17/269; C07C25/18; C07F5/02; C07F5/05
Domestic Patent References:
| JPH10152491A | 1998-06-09 | |||
| JP2001039975A | 2001-02-13 |
Foreign References:
| WO2008063300A2 | 2008-05-29 |
Other References:
平山令明, 有機化合物結晶作製ハンドブック, JPN6016041143, 2008, pages 17 - 23, ISSN: 0003427990
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"新医薬品の規格及び試験方法の設定について", 医薬審発第５６８号, JPN6016041145, 2001, ISSN: 0003427992
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小嶌隆史: "医薬品開発における結晶性選択の効率化を目指して", 薬剤学, vol. 68, no. 5, JPN6016041144, 1 September 2008 (2008-09-01), pages 344 - 349, ISSN: 0003427991
"新医薬品の規格及び試験方法の設定について", 医薬審発第５６８号, JPN6016041145, 2001, ISSN: 0003427992
川口洋子ら: "医薬品と結晶多形", 生活工学研究, vol. 4, no. 2, JPN6016041146, 2002, pages 310 - 317, ISSN: 0003427993
大島寛: "結晶多形・擬多形の析出挙動と制御", PHARM STAGE, vol. 6, no. 10, JPN6016041147, 15 January 2007 (2007-01-15), pages 48 - 53, ISSN: 0003427994
Attorney, Agent or Firm:
Toru Ishikawa