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Title:
キナーゼ阻害のためのヘテロアリール化合物
Document Type and Number:
Japanese Patent JP7212733
Kind Code:
B2
Abstract:
Compounds and pharmaceutical compositions that modulate kinase activity, including mutant EGFR and mutant HER2 kinase activity, and compounds, pharmaceutical compositions, and methods of treatment of diseases and conditions associated with kinase activity, including mutant EGFRand mutant HER2 activity, are described herein.

Inventors:
Wei-Sheng Huang
Gon Youngjin
Li Feng
Nicholas E. Bencivenga
David C. Dalgarno
Anna Coleman
William See. Shakespeare
Lanny M. Thomas
Angela buoy. Waist
Wilmen Youngsay
Zhang Yun
tianjun elephant
Xiaotian Zoo
Application Number:
JP2021131767A
Publication Date:
January 25, 2023
Filing Date:
August 12, 2021
Export Citation:
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Assignee:
Takeda GmbH
International Classes:
C07D401/14; C07D403/04; C07D405/14; C07D471/04
Domestic Patent References:
JP2013544273A
JP2012526113A
JP2011526299A
JP6230205B2
JP6546630B2
Foreign References:
US20110263541
WO2013169401A1
WO2015195228A1
WO2015175632A1
Attorney, Agent or Firm:
Shusaku Yamamoto
Takatoshi Iida
Daisuke Ishikawa
Kensaku Yamamoto