Title:
It is a terrorism atomic compound to the fourth class of Including .
Document Type and Number:
Japanese Patent JP6061923
Kind Code:
B2
Abstract:
A compound useful for the preparation of building blocks for the manufacture of various compounds is represented by Formula 2a:
Inventors:
Douglas Sea Behena
Brian M Stoltz
Scott Sea Vergil
David E White
Yurino Taiga
Eyan Riu
Douglas Duquette
Christian Adam Schauss
Brian M Stoltz
Scott Sea Vergil
David E White
Yurino Taiga
Eyan Riu
Douglas Duquette
Christian Adam Schauss
Application Number:
JP2014517239A
Publication Date:
January 18, 2017
Filing Date:
June 23, 2012
Export Citation:
Assignee:
The Regents of The University of California
International Classes:
C07C33/035; C07C29/147; C07D207/06; C07D207/08; C07D207/16; C07D207/27; C07D207/46; C07D211/12; C07D211/16; C07D211/76; C07D211/94; C07D211/96; C07D223/04; C07D223/10; C07D241/04; C07D241/08; C07D265/30; C07D265/32; C07D309/04; C07F7/10
Domestic Patent References:
| JP2005524628A | ||||
| JP2007516172A | ||||
| JP4264068A |
Foreign References:
| WO2009153178A1 | ||||
| DE668489B | ||||
| US20060084820 | ||||
| WO2011153509A1 |
Other References:
Johnson, Timothy A.; Jang, Doo Ok; et.al.,Asymmetric Carbon-Carbon Bond Formations in Conjugate Additions of Lithiated N-Boc Allylic and Benzylic Amines to Nitroalkenes,Journal of the American Chemical Society,2002年,124(39),11689-11698
Amat, Mercedes; Lozano, Oscar; Escolano, Carmen; et.al.,Enantioselective Synthesis of 3,3-Disubstituted Piperidine Derivatives by Enolate Dialkylation of Phenylglycinol-Derived Oxazolopiperidone Lactams,Journal of Organic Chemistry,2007年,72(12),4431-4439
Horrillo-Martinez, Patricia; Hultzsch, Kai C.; Hampel, Frank,Base-catalyzed asymmetric hydroamination/cyclization of aminoalkenes utilizing a dimeric chiral diamidobinaphthyl dilithium salt,Chemical Communications (Cambridge, United Kingdom),2006年,(21),2221-2223
Enders, Dieter; Teschner, Pascal; Raabe, Gerhard; Runsink, Jan,Asymmetric electrophilic substitutions at the α-position of γ-and δ-lactams,European Journal of Organic Chemistry,2001年,(23),4463-4477
Phillip C.Bulman Page; A. Sazali Hamzah;et.al.,Short and Versatile Route to Key intermediate for Lactacystin Synthesis,Organic Letters,2003年,5(3),353-355
Marc Rodriguez; Annie Heitz;et.al.,“Carba” peptide bond surrogates Different approaches to Gly-ψ(CH2-CH2)-D,L-Xaa pseudo-dipeptide units,International Journal of Peptide & Protein Research,1992年,39(3),273-277
Yendapally, Raghunandan; Lee, Richard E.,Design, synthesis, and evaluation of novel ethambutol analogues,Bioorganic & Medicinal Chemistry Letters,2008年,18(5),1607-1611
Zawisza, Anna; Fenet, Bernard; Sinou, Denis,Palladium-catalyzed formation of cyclic ethers - regio-, stereo- and enantioselectivity of the reaction,European Journal of Organic Chemistry,2007年,(14),2296-2309
Bell, Mark; Frisch, Kim; Jorgensen, Karl Anker,Organocatalytic Asymmetric Deconjugative Michael Additions,Journal of Organic Chemistry,2006年,71(14),5407-5410
Zawisza, Anna; Sinou, Denis,An unexpected palladium-catalyzed cyclization of bis-hydroxy allylic alcohols to dioxabicyclo[2.2.2]octanes,Tetrahedron Letters,2006年,47(19),3271-3274
Thorsten Bach; Frank Eilers ;Kristian Kather,Regioselective Reductive Ring Opening of 2-(2-Hydroxyphenyl)-3-[(trimethylsilyl)oxy]oxetanes at the More Substituted C-2 Position,Liebigs Ann,1997年,(7),1529-1536
ORGANIC LETTERS,2010年,Vol. 12, No. 13,3042-3045
NATURE CHEMISTRY,2012年,Vol. 4, Issue 2,130-133
Amat, Mercedes; Lozano, Oscar; Escolano, Carmen; et.al.,Enantioselective Synthesis of 3,3-Disubstituted Piperidine Derivatives by Enolate Dialkylation of Phenylglycinol-Derived Oxazolopiperidone Lactams,Journal of Organic Chemistry,2007年,72(12),4431-4439
Horrillo-Martinez, Patricia; Hultzsch, Kai C.; Hampel, Frank,Base-catalyzed asymmetric hydroamination/cyclization of aminoalkenes utilizing a dimeric chiral diamidobinaphthyl dilithium salt,Chemical Communications (Cambridge, United Kingdom),2006年,(21),2221-2223
Enders, Dieter; Teschner, Pascal; Raabe, Gerhard; Runsink, Jan,Asymmetric electrophilic substitutions at the α-position of γ-and δ-lactams,European Journal of Organic Chemistry,2001年,(23),4463-4477
Phillip C.Bulman Page; A. Sazali Hamzah;et.al.,Short and Versatile Route to Key intermediate for Lactacystin Synthesis,Organic Letters,2003年,5(3),353-355
Marc Rodriguez; Annie Heitz;et.al.,“Carba” peptide bond surrogates Different approaches to Gly-ψ(CH2-CH2)-D,L-Xaa pseudo-dipeptide units,International Journal of Peptide & Protein Research,1992年,39(3),273-277
Yendapally, Raghunandan; Lee, Richard E.,Design, synthesis, and evaluation of novel ethambutol analogues,Bioorganic & Medicinal Chemistry Letters,2008年,18(5),1607-1611
Zawisza, Anna; Fenet, Bernard; Sinou, Denis,Palladium-catalyzed formation of cyclic ethers - regio-, stereo- and enantioselectivity of the reaction,European Journal of Organic Chemistry,2007年,(14),2296-2309
Bell, Mark; Frisch, Kim; Jorgensen, Karl Anker,Organocatalytic Asymmetric Deconjugative Michael Additions,Journal of Organic Chemistry,2006年,71(14),5407-5410
Zawisza, Anna; Sinou, Denis,An unexpected palladium-catalyzed cyclization of bis-hydroxy allylic alcohols to dioxabicyclo[2.2.2]octanes,Tetrahedron Letters,2006年,47(19),3271-3274
Thorsten Bach; Frank Eilers ;Kristian Kather,Regioselective Reductive Ring Opening of 2-(2-Hydroxyphenyl)-3-[(trimethylsilyl)oxy]oxetanes at the More Substituted C-2 Position,Liebigs Ann,1997年,(7),1529-1536
ORGANIC LETTERS,2010年,Vol. 12, No. 13,3042-3045
NATURE CHEMISTRY,2012年,Vol. 4, Issue 2,130-133
Attorney, Agent or Firm:
Kenji Sugimura
Kazuyuki Tomita
Hiroshi Ikeda
Kazuyuki Tomita
Hiroshi Ikeda