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Title:
ピモベンダン及びシクロデキストリンの錯体を含む液体製剤
Document Type and Number:
Japanese Patent JP5565794
Kind Code:
B2
Abstract:
The invention relates to novel liquid preparation comprising a substituted benzimidazol, preferably pimobendan as pharmaceutically active compound. In particular, the present invention relates to liquid preparation comprising an etherified cyclodextrin derivative, preferably in a concentration of about 20 to 70% (w/v) and said substituted benzimidazol, preferably in a concentration of about 0.005 to 0.15 % (w/w).

Inventors:
Folger Martin A
Lener stephan
Application Number:
JP2009535699A
Publication Date:
August 06, 2014
Filing Date:
November 05, 2007
Export Citation:
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Assignee:
Boehringer Ingelheim Fethmedika Gesellschaft Mitt Beschlenktel Haftung
International Classes:
A61K31/501; A61K9/08; A61K47/40; A61P1/00; A61P9/00; A61P9/04; A61P9/10; A61P13/12; A61P43/00
Domestic Patent References:
JP61500788A
JP2009825A
JP5070612A
JP11228302A
JP2005281283A
Foreign References:
WO2006022562A1
Other References:
MENARD,F. et al,Drug Development and Industrial Pharmacy,1990年,Vol.16, No.1,p.91-113
BASSINI,V.L. et al,Journal of Inclusion Phenomena and Molecular Recognition in Chemistry,1996年,Vol.25, No.1-3,p.149-152
LOFTSSON,T. et al,Journal of pharmaceutical sciences,1996年,Vol.85, No.10,p.1017-25
遠藤政夫,週刊医学のあゆみ,1998年,Vol.187, No.10,p.827-831
PIEL,G. et al,S.T.P. Pharma Sciences,1999年,Vol.9, No.3,p.257-260
Attorney, Agent or Firm:
Sadao Kumakura
Nobuo Ogawa
Atsushi Hakoda
Kenji Asai
Kazuo Yamazaki
Hironobu Hattori