Title:
エスシタロプラムの製造に使用することができる中間体の分離方法
Document Type and Number:
Japanese Patent JP5520077
Kind Code:
B2
Abstract:
The present invention relates to a novel method for the preparation of diol intermediates useful for the preparation of escitalopram involving selective enzymatic acylation or deacylation.
Inventors:
Naoaki Taoka
Takahisa Kato
Shogo Yamamoto
Takashi Yoshida
Toshihiro Takeda
Yasuyoshi Ueda
Petersen Hans
Dansea Roberto
Armaian Halley
Lings larse ole
Takahisa Kato
Shogo Yamamoto
Takashi Yoshida
Toshihiro Takeda
Yasuyoshi Ueda
Petersen Hans
Dansea Roberto
Armaian Halley
Lings larse ole
Application Number:
JP2010032381A
Publication Date:
June 11, 2014
Filing Date:
February 17, 2010
Export Citation:
Assignee:
Her Lundbeck Actiezer Scabet
International Classes:
C07C253/34; C07B57/00; C12P13/00; C07C253/30; C07C255/34; C07C255/53; C07C255/59; C07D307/87; C12P41/00
Domestic Patent References:
JP2036177A | ||||
JP61087654A | ||||
JP2002509864A | ||||
JP2005513069A | ||||
JP2004538276A | ||||
JP2004536093A |
Attorney, Agent or Firm:
Hiroshi Kobayashi
Eiji Katayama
Norio Omori
Yasuhito Suzuki
Eiji Katayama
Norio Omori
Yasuhito Suzuki