Title:
一置換及び二置換のオキシコドン化合物及び組成物
Document Type and Number:
Japanese Patent JP2009533443
Kind Code:
A
Abstract:
The invention relates to pharmaceutical compounds and compositions comprised of a chemical moiety attached to oxycodone in a manner that substantially decreases the potential for overdose. When delivered at the proper dosage the pharmaceutical composition provides therapeutic activity similar to that of oxycodone and may also provide sustained release characteristics and/or reduced side-effects. Further the compounds and compositions of the invention are useful in preventing addiction and susceptibility to addiction of oxycodone.
Inventors:
Mickle, Travis
Krishnan, Zuma
James Scott, Montcryv
Loader back, Christopher
Bella, sanjib
Krishnan, Zuma
James Scott, Montcryv
Loader back, Christopher
Bella, sanjib
Application Number:
JP2009505431A
Publication Date:
September 17, 2009
Filing Date:
April 10, 2007
Export Citation:
Assignee:
Shire LRC
International Classes:
C07K5/08; A61K31/485; A61K47/48; A61P25/04; A61P25/36; C07D489/08; C07K5/06; C07K5/10; C07K7/00; C07K14/00
Attorney, Agent or Firm:
Mamoru Ushiki
Masayoshi Yoshida
Shimizu Sakaematsu
Soichi Kogo
Masayoshi Yoshida
Shimizu Sakaematsu
Soichi Kogo
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