Title:
新規アリールスルホンアミド誘導体及び治療用剤としてのその使用
Document Type and Number:
Japanese Patent JP4411204
Kind Code:
B2
Abstract:
N-((N-(4-Amidinobenzyl)-N-methylcarbamoyl)-alkyl)-arylsulfonamides (I) are new. Aryl sulfonamide derivatives of formula (I) and their acid addition salts are new. R1 = aromatic nucleus (optionally substituted by one or more of halo, 1-3C alkyl, 1-3C alkoxy, NO2, CN, CF3 or OCF3); R2 = H or 1-4C alkyl (optionally substituted by phenyl, CONH2 or one or more F); R3 = H or OH; R4 = H; or R3 + R4 = -CH=N- or 2-4C alkylene; R5 = H or 1-3C alkyl; R6 = H or halo; Y = optionally unsaturated 2-4C alkylene (optionally interrupted by O). An Independent claim is included for the preparation of (I).
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Inventors:
Martin, Baltic
Bondeau, michelle
Dodey, Pierre
Massardier, Christine
Luccarini, Jean-Michel
Bondeau, michelle
Dodey, Pierre
Massardier, Christine
Luccarini, Jean-Michel
Application Number:
JP2004513261A
Publication Date:
February 10, 2010
Filing Date:
June 12, 2003
Export Citation:
Assignee:
Labortoire Fourniers S.A.
International Classes:
C07C311/19; A61K31/18; A61K31/4164; A61K31/4178; A61K31/551; A61P3/06; A61P9/10; A61P9/12; A61P25/04; A61P25/22; A61P25/24; A61P29/00; A61P37/08; C07D233/24; C07D233/54; C07D233/64; C07D239/06; C07D243/04; C07D249/08; C07D409/12
Domestic Patent References:
| JP2004525936A | ||||
| JP2003501413A | ||||
| JP2000514818A |
Attorney, Agent or Firm:
Atomi International Patent Office
Yasuo Yasutomi
Yasuo Yasutomi