Title:
NEW FATTY ACID DERIVATIVE
Document Type and Number:
Japanese Patent JP2009280583
Kind Code:
A
Abstract:
To provide a method for improving the actions of many biologically active compounds such as drugs and agrochemicals by a chemical derivatization method.
The properties of biologically active compounds such as drugs and agrochemicals containing in their molecular structure one or more functional groups selected from an alcohol, ether, phenyl, amino, amide, thiol, carboxylic acid and carboxylic acid ester groups are modified by replacing one or more of these functional groups by a lipophilic group selected from those of formula: RCOO-, RCONH-, RCOS-, RCH2O-, RCH2NH-, -COOCH2R and -SCH2R, wherein R is a lipophilic moiety selected from cis-8-heptadecenyl, trans-8-heptadecenyl, cis-10-nonadecenyl and trans-10-nonadecenyl.
Inventors:
MYHREN FINN
DALEN ARE
BORRETZEN BERNT
SANDVOLD MARIT LILAND
DALEN ARE
BORRETZEN BERNT
SANDVOLD MARIT LILAND
Application Number:
JP2009141714A
Publication Date:
December 03, 2009
Filing Date:
June 12, 2009
Export Citation:
Assignee:
CLAVIS PHARMA ASA
International Classes:
C07D251/70; A01N25/00; C07J5/00; A01N37/34; A01N37/40; A01N47/24; A01N57/28; A01N61/00; A61K31/00; A61K31/165; A61K31/192; A61K31/196; A61K31/216; A61K31/231; A61K31/235; A61K31/337; A61K31/37; A61K31/405; A61K31/416; A61K31/426; A61K31/43; A61K31/431; A61K31/4439; A61K31/4706; A61K31/505; A61K31/519; A61K31/52; A61K31/53; A61K31/565; A61K31/567; A61K31/57; A61K31/573; A61K31/675; A61K31/704; A61K31/7042; A61K47/48; A61P7/00; A61P9/00; A61P11/00; A61P25/00; A61P29/00; A61P31/00; A61P31/04; A61P33/00; A61P35/00; A61P43/00; C07C43/00; C07C53/00; C07C57/00; C07C59/64; C07C65/28; C07C69/00; C07C69/72; C07C69/734; C07C69/84; C07C69/86; C07C69/88; C07C219/00; C07C229/42; C07C229/64; C07C233/00; C07C233/18; C07C233/49; C07C233/55; C07C235/34; C07D209/28; C07D211/00; C07D211/88; C07D215/46; C07D231/56; C07D233/90; C07D239/42; C07D277/16; C07D305/14; C07D311/56; C07D317/70; C07D417/12; C07D473/24; C07D473/38; C07D475/08; C07D487/04; C07D499/00; C07D499/893; C07D499/897; C07H5/06; C07H15/252; C07H17/04; C07J1/00; C07J3/00; C07J7/00; C07J71/00; A61K
Domestic Patent References:
| JPH0381286A | 1991-04-05 | |||
| JPS61204197A | 1986-09-10 | |||
| JPS6143110A | 1986-03-01 | |||
| JPS5982399A | 1984-05-12 |
Other References:
JPN6007012129; Ｉｎｔｅｒｎａｔｉｏｎａｌ Ｊｏｕｒｎａｌ ｏｆ Ｐｈａｒｍａｃｅｕｔｉｃｓ ２４, 1985, １７３-１８４
Attorney, Agent or Firm:
Michiharu Soga
Hidetoshi Furukawa
Suzuki Kenchi
Kajinami order
Kazuhiro Oyaku
Hidetoshi Furukawa
Suzuki Kenchi
Kajinami order
Kazuhiro Oyaku