Title:
有機化合物
Document Type and Number:
Japanese Patent JP4065399
Kind Code:
B2
Abstract:
Compounds of formula (I), where R is a monovalent cyclic organic group having from 3 to 15 atoms in the ring system, useful as pharmaceuticals
More Like This:
Inventors:
Bernard Queneu
David Beatty
Thomas Hugo Keller
Gainer Elizabeth Pilgrim
David Andrew Sandham
Simon James Watson
David Beatty
Thomas Hugo Keller
Gainer Elizabeth Pilgrim
David Andrew Sandham
Simon James Watson
Application Number:
JP2002505801A
Publication Date:
March 26, 2008
Filing Date:
June 26, 2001
Export Citation:
Assignee:
NOVARTIS AG
International Classes:
A61K31/56; A61K31/569; C07J3/00; A61K31/58; A61P11/08; A61P29/00; A61P43/00; C07C401/00; C07J17/00; C07J33/00; C07J41/00; C07J43/00; C07J71/00
Domestic Patent References:
| JP8291073A | ||||
| JP8291072A | ||||
| JP60058999A | ||||
| JP52102264A | ||||
| JP56011720B1 | ||||
| JP49080058A | ||||
| JP57146800A |
Foreign References:
| US3828080 |
Other References:
Isogai M. 等,Binding Affinites of Mometasone Furoate and Related Compounds Including Its Metabolites for the Glucocorticoid Receptor of Rat Skin Tissue,Journal of Biochemistry and Molecular Biology,1993年,vol. 44, no. 2,pages 141-145
Shapiro, Elliot L.; Gentles, Margaret J.; Tiberi, Robert L.; Popper, Thomas L.; Berkenkopf, Joseph; Lutsky, Barry; Watnick, Arthur S,17-Heteroaroyl esters of corticosteroids. 2. 11?-Hydroxy series,Journal of Medicinal Chemistry,1987年,30(9),1581-8
Shapiro, Elliot L.; Gentles, Margaret J.; Tiberi, Robert L.; Popper, Thomas L.; Berkenkopf, Joseph; Lutsky, Barry; Watnick, Arthur S,Synthesis and structure-activity studies of corticosteroid 17-heterocyclic aromatic esters. 1. 9?,11?-Dichloro series,Journal of Medicinal Chemistry,1987年,30(6),1068-73
Ueno, Hiroaki; Maruyama, Akira; Miyake, Motoyoshi; Nakao, Etsuko; Nakao, Kenichiro; Umezu, Kohei; Nitta, Issei,Synthesis and evaluation of antiinflammatory activities of a series of corticosteroid 17?-esters containing a functional group ,Journal of Medicinal Chemistry,1991年,34(8),2468-73
Shapiro, Elliot L.; Gentles, Margaret J.; Tiberi, Robert L.; Popper, Thomas L.; Berkenkopf, Joseph; Lutsky, Barry; Watnick, Arthur S,17-Heteroaroyl esters of corticosteroids. 2. 11?-Hydroxy series,Journal of Medicinal Chemistry,1987年,30(9),1581-8
Shapiro, Elliot L.; Gentles, Margaret J.; Tiberi, Robert L.; Popper, Thomas L.; Berkenkopf, Joseph; Lutsky, Barry; Watnick, Arthur S,Synthesis and structure-activity studies of corticosteroid 17-heterocyclic aromatic esters. 1. 9?,11?-Dichloro series,Journal of Medicinal Chemistry,1987年,30(6),1068-73
Ueno, Hiroaki; Maruyama, Akira; Miyake, Motoyoshi; Nakao, Etsuko; Nakao, Kenichiro; Umezu, Kohei; Nitta, Issei,Synthesis and evaluation of antiinflammatory activities of a series of corticosteroid 17?-esters containing a functional group ,Journal of Medicinal Chemistry,1991年,34(8),2468-73
Attorney, Agent or Firm:
Aoyama Aoi
Kazuaki Kojima
Mitsutaka Iwasaki
Kazuaki Kojima
Mitsutaka Iwasaki