Title:
RECEPTOR AGONIST
Document Type and Number:
Japanese Patent JP2004346059
Kind Code:
A
Abstract:
To provide a TGR5 (G protein-coupled receptor) receptor agonist useful for treating various diseases.
This TGR5 receptor agonist contains a fused ring compound expressed by formula (1) (wherein ring A is an aromatic ring which may be substituted; and ring B' is a 5-8-membered ring having ≥1 substituent), or its salt or its prodrug.
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Inventors:
ITO FUMIO
HINUMA KUNIJI
KANZAKI NAOYUKI
MIKI TAKASHI
KAWAMATA YUJI
OI SATORU
TAWARAISHI TAISUKE
ISHICHI YUJI
HIROHASHI MARIKO
HINUMA KUNIJI
KANZAKI NAOYUKI
MIKI TAKASHI
KAWAMATA YUJI
OI SATORU
TAWARAISHI TAISUKE
ISHICHI YUJI
HIROHASHI MARIKO
Application Number:
JP2004018643A
Publication Date:
December 09, 2004
Filing Date:
January 27, 2004
Export Citation:
Assignee:
TAKEDA CHEMICAL INDUSTRIES LTD
International Classes:
G01N33/50; A61K31/395; A61K31/4353; A61K31/5513; A61K31/553; A61P1/04; A61P1/16; A61P3/04; A61P3/10; A61P5/50; A61P9/06; A61P9/10; A61P9/12; A61P11/00; A61P13/12; A61P17/00; A61P19/02; A61P25/28; A61P29/00; A61P31/00; A61P35/00; A61P35/02; A61P37/06; A61P37/08; A61P43/00; C07D243/14; C07D267/14; C07D401/06; C07D409/06; C07D413/12; C07D417/06; C07D498/04; C07K14/705; C12N15/09; G01N33/15; (IPC1-7): C07D243/14; A61K31/395; A61K31/4353; A61K31/5513; A61K31/553; A61P1/04; A61P1/16; A61P3/04; A61P3/10; A61P5/50; A61P9/06; A61P9/10; A61P9/12; A61P11/00; A61P13/12; A61P17/00; A61P19/02; A61P25/28; A61P29/00; A61P31/00; A61P35/00; A61P35/02; A61P37/06; A61P37/08; A61P43/00; C07D267/14; C07D401/06; C07D409/06; C07D413/12; C07D417/06; C07D498/04; G01N33/15; G01N33/50
Domestic Patent References:
JPH11109356A | 1999-04-23 | |||
JPS63238069A | 1988-10-04 | |||
JP2000502356A | 2000-02-29 | |||
JP2002501944A | 2002-01-22 |
Foreign References:
WO2003002147A1 | 2003-01-09 | |||
US6150357A | 2000-11-21 | |||
WO2001055121A1 | 2001-08-02 | |||
US5324726A | 1994-06-28 | |||
WO2002099388A2 | 2002-12-12 |
Attorney, Agent or Firm:
Shuichi Takahashi
Yo Sekiguchi
Yo Sekiguchi