Title:
【発明の名称】置換〔1,4〕ジアゼピノ〔6,7,1-hi〕インドール-4-オンの製造方法
Document Type and Number:
Japanese Patent JP2003503498
Kind Code:
A
Abstract:
Method for the preparation of enantiomerically pure diazepino-indolone of formulawhich comprises the intramolecular cyclization of a product of formulawhere A, B, X<1>, X<2>, Z, Z<1>, Z<2 >and R are as defined in the description, in the presence of a weak Lewis acid catalyst.
Inventors:
Bernard Deli, Patrick
Application Number:
JP2001507839A
Publication Date:
January 28, 2003
Filing Date:
June 29, 2000
Export Citation:
Assignee:
Warner-Lambert Company
International Classes:
A61K31/5517; A61P11/00; C07D487/16; A61P29/00; C07B61/00; C07D209/00; C07D243/00; C07D471/00; C07D487/00; C07D487/04; C07D487/06; C07D519/00; A61K; A61P; C07D; (IPC1-7): C07D487/16; C07D519/00
Attorney, Agent or Firm:
Kazuo Shamoto (5 outside)