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Title:
10A-AZALIDE COMPOUND CROSSLINKED AT POSITION-10A AND POSITION-12
Document Type and Number:
WIPO Patent Application WO/2009/019868
Kind Code:
A1
Abstract:
Disclosed is a novel 10a-azalide compound crosslinked at position-10a and position-12, which is represented by the formula shown below and is effective against an influenza bacterium or an erythromycin-resistant bacterium (e.g., an erythromycin-resistant pneumococcal or streptococcal bacterium).

Inventors:
SUGIMOTO TOMOHIRO (JP)
YAMAMOTO KANAKO (JP)
KUROSAKA JUN (JP)
SASAMOTO NAOKI (JP)
KASHIMURA MASATO (JP)
MIURA TOMOAKI (JP)
KANEMOTO KENICHI (JP)
OZAWA TOMOHIRO (JP)
CHIKAUCHI KEN (JP)
SHITARA EIKI (JP)
Application Number:
PCT/JP2008/002129
Publication Date:
February 12, 2009
Filing Date:
August 06, 2008
Export Citation:
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Assignee:
TAISHO PHARMACEUTICAL CO LTD (JP)
MEIJI SEIKA KAISHA (JP)
SUGIMOTO TOMOHIRO (JP)
YAMAMOTO KANAKO (JP)
KUROSAKA JUN (JP)
SASAMOTO NAOKI (JP)
KASHIMURA MASATO (JP)
MIURA TOMOAKI (JP)
KANEMOTO KENICHI (JP)
OZAWA TOMOHIRO (JP)
CHIKAUCHI KEN (JP)
SHITARA EIKI (JP)
International Classes:
C07H17/08; A61K31/7056; A61P31/04
Domestic Patent References:
WO2005019238A12005-03-03
WO2007091393A12007-08-16
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WO2005019238A12005-03-03
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WO2001077134A22001-10-18
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JP2002530422A2002-09-17
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See also references of EP 2177526A4
Attorney, Agent or Firm:
SIKs & Co. (Kyobashi-Nisshoku Bldg.8-7, Kyobashi, 1-chome, Chuo-k, Tokyo 31, JP)
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