10A-AZALIDE COMPOUND HAVING 4-MEMBERED RING STRUCTURE

Title:

10A-AZALIDE COMPOUND HAVING 4-MEMBERED RING STRUCTURE

Document Type and Number:

WIPO Patent Application WO/2009/139181

Kind Code:

A1

Abstract:

Disclosed is a 10a-azalide compound which is effective against a bacterium Haemophilus influenzae (an influenza bacterium) or an erythromycin-resistant bacterium (e.g., resistant pneumococcus or streptococcus) and has a novel structure. The 10a-azalide compound is represented by formula (I) and has a 4-membered ring structure cross-linked at position-10a and position-12.

Inventors:

SUGIMOTO TOMOHIRO (JP)
YAMAMOTO KANAKO (JP)
KUROSAKA JUN (JP)
SASAMOTO NAOKI (JP)
KASHIMURA MASATO (JP)
MIURA TOMOAKI (JP)
KANEMOTO KENICHI (JP)
YOSHIDA SATOSHI (JP)
KUMURA KOU (JP)
AJITO KEIICHI (JP)

Application Number:

PCT/JP2009/002135

Publication Date:

November 19, 2009

Filing Date:

May 15, 2009

Export Citation:

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Assignee:

TAISHO PHARMACEUTICAL CO LTD (JP)
MEIJI SEIKA KAISHA (JP)
SUGIMOTO TOMOHIRO (JP)
YAMAMOTO KANAKO (JP)
KUROSAKA JUN (JP)
SASAMOTO NAOKI (JP)
KASHIMURA MASATO (JP)
MIURA TOMOAKI (JP)
KANEMOTO KENICHI (JP)
YOSHIDA SATOSHI (JP)
KUMURA KOU (JP)
AJITO KEIICHI (JP)

International Classes:

C07H17/00; A61K31/7052; A61P31/04

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