Title:
ANDROGEN RECEPTOR MODULATOR COMPOUNDS AND METHODS
Document Type and Number:
WIPO Patent Application WO2001016139
Kind Code:
A9
Abstract:
Compounds, pharmaceutical compositions, and methods for modulating processes mediated by steroid receptors. In particular, preparation and methods of use of non-steroidal compounds and compositions that are agonists, partial agonists, and antagonists for the androgen receptor (AR) are described. Further, described are the methods of making and use of critical intermediates including a stereoselective synthetic route to intermediates for the AR modulators.
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Inventors:
HIGUCHI ROBERT (US)
ARIENTI KRISTEN L (US)
NEELAKANDHA MANI (CA)
PIO BARBARA (US)
ZHI LIN (CA)
CHEN PENGHUI (CA)
CAFERRO THOMAS R (US)
ARIENTI KRISTEN L (US)
NEELAKANDHA MANI (CA)
PIO BARBARA (US)
ZHI LIN (CA)
CHEN PENGHUI (CA)
CAFERRO THOMAS R (US)
Application Number:
PCT/US2000/023520
Publication Date:
September 19, 2002
Filing Date:
August 25, 2000
Export Citation:
Assignee:
LIGAND PHARM INC (US)
HIGUCHI ROBERT (US)
ARIENTI KRISTEN L (US)
NEELAKANDHA MANI (CA)
PIO BARBARA (US)
ZHI LIN (CA)
CHEN PENGHUI (CA)
CAFERRO THOMAS R (US)
HIGUCHI ROBERT (US)
ARIENTI KRISTEN L (US)
NEELAKANDHA MANI (CA)
PIO BARBARA (US)
ZHI LIN (CA)
CHEN PENGHUI (CA)
CAFERRO THOMAS R (US)
International Classes:
A61K31/4985; A61K31/5383; A61K31/542; A61P5/00; A61P5/24; A61P5/26; A61P5/28; A61P7/00; A61P7/06; A61P13/08; A61P15/08; A61P15/10; A61P15/16; A61P17/10; A61P17/14; A61P19/10; A61P35/00; C07D471/04; C07D498/04; C07D498/14; C07D513/04; (IPC1-7): C07D498/04; C07D471/04; C07D513/04; A61K31/538; A61K31/5415; A61K31/502; A61P5/26; A61P5/28
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