Title:
CRYSTAL FORM OF ANACETRAPIB AND PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USE THEREOF
Document Type and Number:
WIPO Patent Application WO/2015/106674
Kind Code:
A1
Abstract:
The present invention relates to a crystal form 1 of anacetrapib. Compared with the prior art, the crystal form 1 of anacetrapib of the present invention has a better crystal form stability, is easily stored, and is suitable for use as a solid preparation. The present invention also relates to a method for preparing the crystal form 1, a pharmaceutical composition thereof and the use thereof in the preparation of drugs for treating and/or preventing diseases such as atherosclerosis, hyperlipidemia, and the like.
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Inventors:
ZHU TAO (CN)
SHENG XIAOXIA (CN)
SHENG XIAOHONG (CN)
JIA QIANG (CN)
SHENG XIAOXIA (CN)
SHENG XIAOHONG (CN)
JIA QIANG (CN)
Application Number:
PCT/CN2015/070597
Publication Date:
July 23, 2015
Filing Date:
January 13, 2015
Export Citation:
Assignee:
HANGZHOU PUSHAI PHARMACEUTICAL TECHNOLOGY CO LTD (CN)
International Classes:
C07D263/20; A61K31/4174; A61P3/04; A61P3/06; A61P7/00; A61P9/00; A61P9/10; A61P9/12
Domestic Patent References:
| WO2013064188A1 | 2013-05-10 | |||
| WO2007005572A1 | 2007-01-11 | |||
| WO2006014413A1 | 2006-02-09 |
Foreign References:
| EP2397473A1 | 2011-12-21 |
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