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Title:
INHIBITORS OF FACTOR Xa
Document Type and Number:
WIPO Patent Application WO2000071516
Kind Code:
B1
Abstract:
Compounds, e.g. described in claim 5, formula (I) and formula (II), where A-B is (1), their salts and compositions related thereto having activity against mammalian factor Xa are disclosed. The compounds are useful in vitro or in vivo for preventing or treating coagulation disorders.

Inventors:
ZHU BING-YAN
SCARBOROUGH ROBERT M
WANG LINGYAN
Application Number:
PCT/US2000/014209
Publication Date:
March 01, 2001
Filing Date:
May 24, 2000
Export Citation:
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Assignee:
COR THERAPEUTICS INC (US)
International Classes:
A61K31/155; A61K31/18; A61K31/275; A61K31/401; A61K31/402; A61K31/451; A61P7/02; A61P9/00; A61P9/04; A61P9/10; C07C311/46; C07D207/16; C07D211/60; C07D241/04; C07D243/08; C07D401/04; C07D403/04; C07D413/04; (IPC1-7): C07D207/16; A61K31/40; A61P7/00; C07C311/39; C07D211/60; C07D241/04; C07D243/08; C07D401/04; C07D403/04; C07D413/04
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