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Title:
INHIBITORS OF FACTOR Xa
Document Type and Number:
WIPO Patent Application WO2000071515
Kind Code:
A3
Abstract:
Compounds, e.g. described in Table (1), their salts and compositions related thereto having activity against mammalian factor Xa are disclosed. The compounds are useful in vitro or in vivo for preventing or treating coagulation disorders.

Inventors:
ZHU BING-YAN
SCARBOROUGH ROBERT M
Application Number:
PCT/US2000/014193
Publication Date:
January 25, 2001
Filing Date:
May 24, 2000
Export Citation:
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Assignee:
COR THERAPEUTICS INC (US)
International Classes:
A61K31/155; A61K31/18; A61K31/275; A61K31/401; A61K31/402; A61K31/451; A61P7/02; A61P9/00; A61P9/04; A61P9/10; C07C311/46; C07D207/16; C07D211/60; C07D241/04; C07D243/08; C07D401/04; C07D403/04; C07D413/04; (IPC1-7): C07D207/16; A61K31/40; A61P7/00; C07C311/39; C07D211/60; C07D241/04; C07D243/08; C07D401/04; C07D403/04; C07D413/04
Domestic Patent References:
WO1998006694A11998-02-19
WO1998028269A11998-07-02
Other References:
WALLIS R B: "INHIBITORS OF COAGULATION FACTOR XA: FROM MACROMOLECULAR BEGINNINGS TO SMALL MOLECULES", CURRENT OPINION IN THERAPEUTIC PATENTS,, 1 August 1993 (1993-08-01), pages 1173 - 1179, XP000653726, ISSN: 0962-2594
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