Title:
NITROGEN-CONTAINING FUSED HETEROCYCLIC COMPOUND
Document Type and Number:
WIPO Patent Application WO/2013/051632
Kind Code:
A1
Abstract:
The present invention provides a novel compound which has excellent activity as an ERRα modulator and is useful as a therapeutic or prophylactic agent for ERRα-related diseases such as cancers, or the like. The present invention relates to a compound represented by formula (I) or a salt thereof. (In formula (I), A represents an optionally substituted cyclic group; La represents a bonding hand or the like; Lb represents a C1-3 alkylene group or the like; Lc represents a bonding hand or the like; G represents a group represented by formula Ga or Gb (wherein each of Z1, Z2, Z3 and Z4 independently represents a nitrogen atom, a carbon atom, -CH- or the like; R4 represents a hydrogen atom or the like; and R5 represents a hydrogen atom or the like); and E represents a group represented by formula Ea or Eb (wherein X represents -S- or the like; and each of R1, R2 and R3 independently represents a hydrogen atom or the like).)
Inventors:
TOMINARI YUSUKE (JP)
ONO KOJI (JP)
MATSUMOTO SHIGEMITSU (JP)
KATOH TAISUKE (JP)
HASUOKA ATSUSHI (JP)
IMAMURA SHINICHI (JP)
ONO KOJI (JP)
MATSUMOTO SHIGEMITSU (JP)
KATOH TAISUKE (JP)
HASUOKA ATSUSHI (JP)
IMAMURA SHINICHI (JP)
Application Number:
PCT/JP2012/075721
Publication Date:
April 11, 2013
Filing Date:
October 03, 2012
Export Citation:
Assignee:
TAKEDA PHARMACEUTICAL (JP)
International Classes:
C07D401/14; A61K31/4178; A61K31/427; A61K31/437; A61K31/438; A61K31/4439; A61K31/454; A61K31/496; A61K31/506; A61K31/519; A61K31/5377; A61K31/541; A61K31/55; A61K31/551; A61P3/00; A61P3/04; A61P3/06; A61P3/10; A61P9/10; A61P9/12; A61P19/00; A61P19/02; A61P19/06; A61P25/16; A61P25/18; A61P25/22; A61P25/24; A61P25/28; A61P25/30; A61P29/00; A61P35/00; A61P35/02; A61P43/00; C07D403/06; C07D403/14; C07D405/14; C07D417/06; C07D417/14; C07D471/04; C07D471/10; C07D487/04; C07D487/10
Domestic Patent References:
WO2011016501A1 | 2011-02-10 | |||
WO2011075565A1 | 2011-06-23 | |||
WO2011103130A1 | 2011-08-25 | |||
WO2011103134A1 | 2011-08-25 |
Attorney, Agent or Firm:
TAKASHIMA, HAJIME (JP)
Takashima 1 (JP)
Takashima 1 (JP)
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Claims: