Title:
NOVEL AMINE DERIVATIVE OR SALT THEREOF
Document Type and Number:
WIPO Patent Application WO/2014/069510
Kind Code:
A1
Abstract:
A novel amine derivative expressed by general formula (1) (in the formula: G1, G2, and G3 are the same or different and represent CH or a nitrogen atom; R1 represents a chlorine atom, an optionally-substituted C3-8 cycloalkyl group, or the like; R2 represents -COOR5 (in the formula, R5 represents a hydrogen atom or a carboxyl protective group), or the like; R3 represents a hydrogen atom, or the like; and R4 represents an optionally-substituted condensed bicyclic hydrocarbon group, an optionally-substituted bicyclic heterocyclic group, or the like), or a salt thereof is useful in procedures such as the treatment or prevention of conditions related to excessive keratinocyte proliferation.
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Inventors:
TANAKA TADASHI (JP)
KONISHI YOSHITAKE (JP)
KUBO DAISUKE (JP)
FUJINO MASATAKA (JP)
DOI ISSEI (JP)
NAKAGAWA DAISUKE (JP)
MURAKAMI TATSUYA (JP)
YAMAKAWA TAKAYUKI (JP)
KONISHI YOSHITAKE (JP)
KUBO DAISUKE (JP)
FUJINO MASATAKA (JP)
DOI ISSEI (JP)
NAKAGAWA DAISUKE (JP)
MURAKAMI TATSUYA (JP)
YAMAKAWA TAKAYUKI (JP)
Application Number:
PCT/JP2013/079364
Publication Date:
May 08, 2014
Filing Date:
October 30, 2013
Export Citation:
Assignee:
TOYAMA CHEMICAL CO LTD (JP)
FUJIFILM CORP (JP)
FUJIFILM CORP (JP)
International Classes:
C07D209/08; A61K31/4035; A61K31/404; A61K31/416; A61K31/4184; A61K31/423; A61K31/427; A61K31/428; A61K31/437; A61K31/4439; A61K31/454; A61K31/455; A61K31/4709; A61K31/4725; A61K31/497; A61K31/498; A61K31/501; A61K31/506; A61K31/517; A61K31/5377; A61K31/538; A61P17/00; A61P17/06; A61P35/00; A61P37/08; A61P43/00; C07D209/12; C07D209/34; C07D209/38; C07D209/42; C07D209/46; C07D209/48; C07D213/80; C07D215/38; C07D217/24; C07D231/56; C07D235/08; C07D235/26; C07D241/44; C07D263/58; C07D277/68; C07D401/04; C07D401/06; C07D401/12; C07D401/14; C07D403/04; C07D403/12; C07D405/14; C07D413/12; C07D417/04; C07D417/06; C07D417/12; C07D471/04
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Other References:
MEESALA, R. ET AL.: "A short route to the synthesis of pyrroloacridines via Ullmann- Goldberg condensation", TETRAHEDRON LETTERS, vol. 51, no. 2, 2010, pages 422 - 424, XP027259074
BALDWIN, R. W. ET AL.: "Further studies on the influence of peripheral ring substitution on the carcinogenicity of tricycloquinazoline", BIOCHEMICAL PHARMACOLOGY, vol. 14, no. 3, 1965, pages 323 - 331, XP023746009
BUNKER, A. M. ET AL.: "1,3-Diaryl-2- carboxyindoles as potent non-peptide endothelin antagonists", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 6, no. 9, 1996, pages 1061 - 1066, XP004134909
See also references of EP 2915804A4
N ENGL J MED, vol. 352, 2005, pages 1899 - 18912
BIOCHEM. BIOPHYS. RES. COMMUN, vol. 166, 1990, pages 916 - 923
W GREENE ET AL.: "Protective Groups in Organic Synthesis", 2007, JOHN WILEY & SONS, INC, pages: 696 - 926
W. GREENE ET AL.: "Protective Groups in Organic Synthesis", 2007, JOHN WILEY & SONS, INC, pages: 16 - 366
W. GREENE ET AL.: "Protective Groups in Organic Synthesis", 2007, JOHN WILEY & SONS, INC, pages: 533 - 646
W GREENE ET AL.: "Protective Groups in Organic Synthesis", 2007, JOHN WILEY & SONS, INC., pages: 533 - 646
M. WUTS; W. GREENE: "Protective Groups in Organic Synthesis", 2006, JOHN WILEY & SONS, INC., pages: 696 - 926
RICHARD C. LAROCK ET AL.: "Comprehensive Organic Transformations", 1999, JOHN WILEY & SONS, INC., pages: 823 - 827
BALDWIN, R. W. ET AL.: "Further studies on the influence of peripheral ring substitution on the carcinogenicity of tricycloquinazoline", BIOCHEMICAL PHARMACOLOGY, vol. 14, no. 3, 1965, pages 323 - 331, XP023746009
BUNKER, A. M. ET AL.: "1,3-Diaryl-2- carboxyindoles as potent non-peptide endothelin antagonists", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 6, no. 9, 1996, pages 1061 - 1066, XP004134909
See also references of EP 2915804A4
N ENGL J MED, vol. 352, 2005, pages 1899 - 18912
BIOCHEM. BIOPHYS. RES. COMMUN, vol. 166, 1990, pages 916 - 923
W GREENE ET AL.: "Protective Groups in Organic Synthesis", 2007, JOHN WILEY & SONS, INC, pages: 696 - 926
W. GREENE ET AL.: "Protective Groups in Organic Synthesis", 2007, JOHN WILEY & SONS, INC, pages: 16 - 366
W. GREENE ET AL.: "Protective Groups in Organic Synthesis", 2007, JOHN WILEY & SONS, INC, pages: 533 - 646
W GREENE ET AL.: "Protective Groups in Organic Synthesis", 2007, JOHN WILEY & SONS, INC., pages: 533 - 646
M. WUTS; W. GREENE: "Protective Groups in Organic Synthesis", 2006, JOHN WILEY & SONS, INC., pages: 696 - 926
RICHARD C. LAROCK ET AL.: "Comprehensive Organic Transformations", 1999, JOHN WILEY & SONS, INC., pages: 823 - 827
Attorney, Agent or Firm:
ASAMURA PATENT OFFICE, p. c. (JP)
Patent business corporation Asamura patent firm (JP)
Patent business corporation Asamura patent firm (JP)
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