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Title:
PYRAZOLE COMPOUND AND USE THEREOF FOR MEDICAL PURPOSES
Document Type and Number:
WIPO Patent Application WO/2013/031922
Kind Code:
A1
Abstract:
A compound represented by general formula [Ib] or a pharmaceutically acceptable salt thereof. [In the formula, each symbol is as defined in the description.]

Inventors:
MIURA TOMOYA (JP)
OGOSHI YOSUKE (JP)
UEYAMA KAZUHITO (JP)
MOTODA DAI (JP)
IWAYAMA TOSHIHIKO (JP)
SUZAWA KOICHI (JP)
NAGAMORI HIRONOBU (JP)
UENO HIROSHI (JP)
TAKAHASHI AKIHIKO (JP)
SUGIMOTO KAZUYUKI (JP)
Application Number:
PCT/JP2012/072066
Publication Date:
March 07, 2013
Filing Date:
August 30, 2012
Export Citation:
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Assignee:
JAPAN TOBACCO INC (JP)
MIURA TOMOYA (JP)
OGOSHI YOSUKE (JP)
UEYAMA KAZUHITO (JP)
MOTODA DAI (JP)
IWAYAMA TOSHIHIKO (JP)
SUZAWA KOICHI (JP)
NAGAMORI HIRONOBU (JP)
UENO HIROSHI (JP)
TAKAHASHI AKIHIKO (JP)
SUGIMOTO KAZUYUKI (JP)
International Classes:
C07D401/12; A61K31/4155; A61K31/4178; A61K31/454; A61P3/10; A61P43/00; C07D403/12; C07D405/12; C07D405/14
Domestic Patent References:
WO2007034279A22007-03-29
Foreign References:
JP2008285481A2008-11-27
JP2010222298A2010-10-07
JP2009517388A2009-04-30
JP2008024693A2008-02-07
JP2008520642A2008-06-19
JP2006514942A2006-05-18
JP2008501745A2008-01-24
Other References:
AM J PHYSIOL GASTROINTEST LIVER PHYSIOL., vol. 282, no. 2, 2002, pages G241 - 8
NATURE, vol. 3 5 0, no. 6316, 1991, pages 354 - 6
J MOL CELL CARDIOL, vol. 49, no. 4, 2010, pages 683 - 92
CARDIOVASC RES., vol. 84, no. 1, 2009, pages 111 - 8
CANCER CELL, vol. 13, 2008, pages 385 - 93
PHAMNACOL THER., vol. 121, 2009, pages 29 - 40
TETRAHEDRON: ASYMMETLY, vol. 12, 2001, pages 3241 - 3249
See also references of EP 2784074A4
Attorney, Agent or Firm:
SAMEJIMA, Mutsumi et al. (JP)
Mutsumi Sameshima (JP)
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Claims: