STABLE ORAL FORMULATION CONTAINING 1-(3-CYANO-1-ISOPROPYL-INDOL-5-YL)PYRAZOLE-4-CARBOXYLIC ACID

Title:

STABLE ORAL FORMULATION CONTAINING 1-(3-CYANO-1-ISOPROPYL-INDOL-5-YL)PYRAZOLE-4-CARBOXYLIC ACID

Document Type and Number:

WIPO Patent Application WO/2022/119269

Kind Code:

A1

Abstract:

The present invention relates to a stable oral formulation containing 1-(3-cyano-1-isopropyl-indol-5-yl)pyrazole-4-carboxylic acid or a pharmaceutically acceptable salt thereof as an API. Being characterized by the maintenance of stability even though containing no stabilizers as excipients, the stable oral formulation according to the present invention contains an increased content of API in place of the inclusion of a stabilizer and as such, can be improved in terms of dose convenience.

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Inventors:

YOO SEOK CHEOL (KR)
LEE SUN (KR)
YUN DUCK IL (KR)
PARK JUNGHONG (KR)
SUN HYUN JI (KR)

Application Number:

PCT/KR2021/017842

Publication Date:

June 09, 2022

Filing Date:

November 30, 2021

Export Citation:

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Assignee:

LG CHEMICAL LTD (KR)

International Classes:

A61K9/20; A61K31/4155; A61P19/06

Domestic Patent References:

WO2004010973A2

2004-02-05

Foreign References:

KR20120114174A	2012-10-16
JP2008523109A	2008-07-03
KR20110037883A	2011-04-13
KR20090128488A	2009-12-15
KR200166051A
KR101751325B1	2017-06-27
KR101424013B1	2014-08-18

Attorney, Agent or Firm:

KIM, Sung Ho (KR)

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