Title:
【発明の名称】エストロゲン-β受容体リガンド
Document Type and Number:
Japanese Patent JP2002542187
Kind Code:
A
Abstract:
A method for treating a disease associated with the estrogen receptor-beta, comprising the step of administering a therapeutically-effective amount of a compound that satisfies the equation: (KialphaA/KibetaA)/(KialphaE/KibetaE)>1, optionally having the general structure (I).
Inventors:
Bernard Christoph Burream
Timothy Martin Piecer
Timothy Martin Piecer
Application Number:
JP2000611902A
Publication Date:
December 10, 2002
Filing Date:
April 11, 2000
Export Citation:
Assignee:
ASTRAZENECA AKTIEBOLAG
International Classes:
A61K31/00; A61K31/122; A61K31/35; A61K31/352; A61K31/37; A61K31/381; A61K31/4709; A61K45/00; A61P9/00; A61P19/02; A61P19/10; A61P25/22; A61P25/24; A61P25/28; A61P35/00; C07D311/18; C07D311/30; C07D311/36; C07D311/16; C07D311/58; C07D405/04; C07D409/04; (IPC1-7): A61K45/00; A61K31/352; A61K31/381; A61K31/4709; A61P9/00; A61P19/02; A61P19/10; A61P25/22; A61P25/24; A61P25/28; A61P35/00
Domestic Patent References:
| JPS6048924A | 1985-03-16 | |||
| JPS63107971A | 1988-05-12 | |||
| JPH0753554A | 1995-02-28 | |||
| JPH05112552A | 1993-05-07 | |||
| JPH08268890A | 1996-10-15 | |||
| JPH06321752A | 1994-11-22 | |||
| JPH0428592A | 1992-01-31 | |||
| JPS5257182A | 1977-05-11 | |||
| JPH09505801A | 1997-06-10 | |||
| JPS4954371A | 1974-05-27 | |||
| JPH07500316A | 1995-01-12 |
Foreign References:
| WO1998050026A1 | 1998-11-12 | |||
| WO1998044920A1 | 1998-10-15 | |||
| WO1998025588A1 | 1998-06-18 | |||
| WO1998008503A1 | 1998-03-05 |
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Attorney, Agent or Firm:
Chika Takagi (2 outside)