Title:
【発明の名称】4”(R)NH2のアザ-マクロライドの製造方法
Document Type and Number:
Japanese Patent JP2003505340
Kind Code:
A
Abstract:
The subject-matter of the invention is a process for the stereoselective preparation of a compound of general formula I by stereoselective displacement by a nitrogenous nucleophilic compound of the activated alcohol functional group present at this 4'' position in a corresponding derivative of formula II.
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Inventors:
Leon, patrick
Lermit, Frederik
Gevel, Ronan
Poise, Duni
Garrel, Loran
Odon, Jill
Lermit, Frederik
Gevel, Ronan
Poise, Duni
Garrel, Loran
Odon, Jill
Application Number:
JP2000593623A
Publication Date:
February 12, 2003
Filing Date:
January 17, 2000
Export Citation:
Assignee:
Merial
International Classes:
A61K31/70; A61P31/00; C07B61/00; C07H17/08; (IPC1-7): C07H17/08
Domestic Patent References:
JPS55151598A | 1980-11-26 | |||
JPH05255375A | 1993-10-05 | |||
JPH05255374A | 1993-10-05 | |||
JP2003512290A | 2003-04-02 |
Attorney, Agent or Firm:
Takashi Koshiba
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