Title:
【発明の名称】リード又は活性化合物の同定方法
Document Type and Number:
Japanese Patent JP2003524144
Kind Code:
A
Abstract:
The invention relates to methods of selection of leads or active compounds from libraries. More specifically, the invention provides methods of selection of leads or compounds which are active and selective towards a desired target. In particular, the invention provides a screening method for the identification of leads from a library of compounds, said method comprising the steps of : (a) screening a library of compounds for activity against a desired target, to obtain potent hits; (b) profiling the potent hits of step (a) to obtain potent and selective leads. The instant invention can be used for instance in drug discovery processes.
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Inventors:
Jean, Thierry
Chaplain, Beatrice
Chaplain, Beatrice
Application Number:
JP2000513141A
Publication Date:
August 12, 2003
Filing Date:
September 25, 1998
Export Citation:
Assignee:
CEREP
International Classes:
A61K31/27; A61K31/40; A61K31/421; A61K31/438; A61K31/454; A61P39/06; A61P43/00; C07C271/16; C07D207/14; C07D241/04; C07D263/58; C07D295/205; C07D401/04; C07D401/14; C07D405/14; C07D413/12; C07D471/10; C12Q1/34; C12Q1/48; G01N33/15; G01N33/53; G01N33/50; G01N33/566; G01N33/94; G01N37/00; C07B61/00; (IPC1-7): G01N33/50; A61K31/27; A61K31/40; A61K31/421; A61K31/438; A61K31/454; A61P39/06; A61P43/00; C07C271/16; C07D207/14; C07D241/04; C07D263/58; C07D401/04; C07D401/14; C07D405/14; C07D413/12; C07D471/10; C12Q1/34; C12Q1/48; G01N33/15; G01N33/566; G01N37/00
Attorney, Agent or Firm:
Hajime Tsukuni (1 person outside)