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Title:
凝固カスケードを選択的に阻害するのに有用な多環式アリール及びヘテロアリール置換4-ピリドン類
Document Type and Number:
Japanese Patent JP2004505013
Kind Code:
A
Abstract:
The invention relates to polycyclic aryl and heteroaryl substituted 4-pyridone compounds useful as inhibitors of serine proteases of the coagulation cascade and compounds, compositions and methods for anticoagulant therapy for the treatment and prevention of a variety of thrombotic conditions including coronary artery and cerebrovascular diseases.

Inventors:
South, Michael Es
Ma, Chun Shi
Kevin Jay, Caller
Rahman, Hayato Kay
Newman, William Elle
Application Number:
JP2001575554A
Publication Date:
February 19, 2004
Filing Date:
April 04, 2001
Export Citation:
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Assignee:
Pharmacia Corporation
International Classes:
A61K31/4418; A61K31/443; A61K31/4436; A61K31/4439; A61K31/444; A61K45/00; A61P7/00; A61P7/02; A61P9/00; A61P9/10; A61P43/00; C07D213/74; C07D213/77; C07D213/79; C07D401/12; C07D405/12; C07D409/04; C07D417/12; (IPC1-7): C07D213/74; A61K31/4418; A61K31/443; A61K31/4436; A61K31/4439; A61K31/444; A61K45/00; A61P7/02; A61P9/00; A61P9/10; A61P43/00; C07D213/77; C07D213/79; C07D401/12; C07D405/12; C07D409/04; C07D417/12
Attorney, Agent or Firm:
Kazuo Shamoto
Tadashi Masui
Yasushi Kobayashi
Akio Chiba
Hiroyuki Tomita
Hiroko Ejiri